Page last updated: 2024-09-03

ips 339 and isoproterenol

ips 339 has been researched along with isoproterenol in 9 studies

Compound Research Comparison

Studies
(ips 339)
Trials
(ips 339)
Recent Studies (post-2010)
(ips 339)
Studies
(isoproterenol)
Trials
(isoproterenol)
Recent Studies (post-2010) (isoproterenol)
260030,7808032,640

Protein Interaction Comparison

ProteinTaxonomyips 339 (IC50)isoproterenol (IC50)
Beta-2 adrenergic receptorHomo sapiens (human)0.246
Beta-1 adrenergic receptorHomo sapiens (human)0.333
Beta-2 adrenergic receptorRattus norvegicus (Norway rat)0.2125
Polyunsaturated fatty acid lipoxygenase ALOX15Oryctolagus cuniculus (rabbit)1.77
Beta-1 adrenergic receptorRattus norvegicus (Norway rat)0.2125
Beta-3 adrenergic receptorRattus norvegicus (Norway rat)0.2125
Beta-2 adrenergic receptorCanis lupus familiaris (dog)0.6667

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19909 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Nathanson, JA1
Bjellin, LA; Ek, BA; Lundgren, BT1
Dattel, BJ; Lam, F; Roberts, JM1
Clerici, C; Harf, A; Macquin-Mavier, I1
Kanda, A; Kimura, T; Satoh, S; Yorikane, R1
Himori, N; Ishimori, T; Izumi, A1
Ek, B; Lundgren, B1
Gerber, JG; Nies, AS; Olson, RD1
Carlsson, E; Hedberg, A; Mattsson, H1

Other Studies

9 other study(ies) available for ips 339 and isoproterenol

ArticleYear
Differential inhibition of beta adrenergic receptors in human and rabbit ciliary process and heart.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 232, Issue:1

    Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Adult; Aged; Animals; Ciliary Body; Dose-Response Relationship, Drug; Heart Rate; Humans; Isoproterenol; Kinetics; Male; Methylation; Middle Aged; Myocardium; Propanolamines; Propranolol; Rabbits; Receptors, Adrenergic, beta; Timolol

1985
Beta-adrenergic control of motility in the rat colon. I. Evidence for functional separation of the beta 1- and beta 2-adrenoceptor-mediated inhibition of colon activity.
    Gastroenterology, 1986, Volume: 90, Issue:2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colon; Gastrointestinal Motility; Isoproterenol; Male; Metoprolol; Muscle, Smooth; Practolol; Prenalterol; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Sympathectomy; Terbutaline; Tetrodotoxin

1986
Failure to demonstrate decreased beta-adrenergic receptor concentration or decreased agonist efficacy in term or preterm human parturition.
    American journal of obstetrics and gynecology, 1986, Volume: 154, Issue:2

    Topics: Adrenergic beta-Agonists; Binding, Competitive; Female; Humans; Iodocyanopindolol; Isoproterenol; Labor, Obstetric; Myometrium; Obstetric Labor, Premature; Pindolol; Pregnancy; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta

1986
Effects of cardioselective beta blockade on the peripheral lung in guinea pigs.
    The European respiratory journal, 1988, Volume: 1, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Atenolol; Bronchi; Dose-Response Relationship, Drug; Drug Synergism; Guinea Pigs; Heart Rate; Histamine; Isoproterenol; Lung; Lung Compliance; Propanolamines; Propranolol

1988
Effects of epinephrine, isoproterenol and IPS-339 on sympathetic transmission to the dog heart: evidence against the facilitatory role of presynaptic beta adrenoceptors.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:1

    Topics: Animals; Blood Pressure; Coronary Circulation; Dogs; Electric Stimulation; Epinephrine; Female; Heart Conduction System; Heart Rate; Isoproterenol; Male; Propanolamines; Receptors, Adrenergic, beta; Regional Blood Flow; Sympathetic Nervous System; Synaptic Transmission

1986
Analysis of beta-adrenoceptors mediating renin release produced by isoproterenol in conscious dogs.
    The American journal of physiology, 1980, Volume: 238, Issue:5

    Topics: Adrenergic beta-Antagonists; Angiotensin II; Animals; Blood Pressure; Dogs; Female; Heart Rate; Isoproterenol; Kidney; Male; Propanolamines; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, beta; Renin

1980
Characterization of the beta-adrenergic inhibition of motility in cat colon strips.
    European journal of pharmacology, 1982, Jan-08, Volume: 77, Issue:1

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cats; Colon; Female; Gastrointestinal Motility; In Vitro Techniques; Isoproterenol; Male; Metoprolol; Practolol; Prenalterol; Propanolamines; Receptors, Adrenergic; Receptors, Adrenergic, beta; Terbutaline; Tetrodotoxin

1982
Beta adrenergically mediated release of renin in the dog is not confined to either beta-1 or beta-2 adrenoceptors.
    The Journal of pharmacology and experimental therapeutics, 1982, Volume: 222, Issue:3

    Topics: Adrenergic beta-Antagonists; Albuterol; Animals; Atenolol; Dogs; Female; Indomethacin; Isoproterenol; Kidney; Male; Propanolamines; Receptors, Adrenergic; Receptors, Adrenergic, beta; Renin; Sotalol; Stimulation, Chemical

1982
Basic pharmacological properties of prenalterol.
    Acta medica Scandinavica. Supplementum, 1982, Volume: 659

    Topics: Adrenergic beta-Agonists; Animals; Blood Pressure; Cats; Cyclic AMP; Dose-Response Relationship, Drug; Epinephrine; Guinea Pigs; Heart Rate; In Vitro Techniques; Isoproterenol; Metoprolol; Myocardial Contraction; Papillary Muscles; Phentolamine; Practolol; Prenalterol; Propanolamines; Rabbits; Receptors, Adrenergic, beta; Terbutaline; Vascular Resistance

1982