iodosulpride has been researched along with sulpiride in 39 studies
Studies (iodosulpride) | Trials (iodosulpride) | Recent Studies (post-2010) (iodosulpride) | Studies (sulpiride) | Trials (sulpiride) | Recent Studies (post-2010) (sulpiride) |
---|---|---|---|---|---|
39 | 0 | 2 | 4,152 | 427 | 635 |
Protein | Taxonomy | iodosulpride (IC50) | sulpiride (IC50) |
---|---|---|---|
Carbonic anhydrase 1 | Homo sapiens (human) | 1.2 | |
Carbonic anhydrase 2 | Homo sapiens (human) | 0.04 | |
Alpha-2A adrenergic receptor | Homo sapiens (human) | 2.019 | |
D(2) dopamine receptor | Homo sapiens (human) | 0.0858 | |
D(3) dopamine receptor | Homo sapiens (human) | 0.2651 | |
D(2) dopamine receptor | Rattus norvegicus (Norway rat) | 0.2215 | |
Carbonic anhydrase 4 | Bos taurus (cattle) | 0.62 | |
D(2) dopamine receptor | Canis lupus familiaris (dog) | 0.2 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 7 (17.95) | 18.7374 |
1990's | 21 (53.85) | 18.2507 |
2000's | 8 (20.51) | 29.6817 |
2010's | 3 (7.69) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Andrieux, M; Besançon, R; Giros, B; Martres, MP; Pilon, C; Schwartz, JC; Sokoloff, P | 1 |
Kilts, CD; Lachowicz, JE; Scibilia, RJ | 1 |
Gommeren, W; Janssen, PF; Leysen, JE; Luyten, WH; Schotte, A | 1 |
Diaz, J; Giros, B; Lévesque, D; Martres, MP; Morgat, JL; Pilon, C; Schott, D; Schwartz, JC; Sokoloff, P; Souil, E | 1 |
Barton, AC; Black, LE; Sibley, DR | 1 |
Bouthenet, ML; Giros, B; Martres, MP; Schwartz, JC; Sokoloff, P; Souil, E | 1 |
Costentin, J; Mann, A; Martres, MP; Rognan, D; Schwartz, JC; Sokoloff, P; Wermuth, CG | 1 |
Denis, P; Elena, PP; Lapalus, P; Nordmann, JP; Saraux, H | 1 |
Masuo, Y; Montagne, MN; Pélaprat, D; Rostène, W; Scherman, D | 1 |
Nowak, JZ; Schorderet, M | 1 |
Bouthenet, ML; Martres, MP; Sales, N; Schwartz, JC | 3 |
Martres, MP; Riou, JF; Schwartz, JC; Sokoloff, P | 1 |
Denis, P; Elena, PP; Kosina-Boix, M; Lapalus, P | 1 |
Di Chiara, G; Mennini, T; Morelli, M | 1 |
Bouthenet, ML; Martres, MP; Sales, N; Schwartz, JC; Sokoloff, P | 1 |
De Souza, EB; Grigoriadis, DE; Levant, B | 1 |
Fuxe, K; Hedlund, PB; Li, XM | 1 |
Hedlund, PB; von Euler, G | 1 |
Booze, RM; Wallace, DR | 1 |
Emms, F; Freedman, SB; Knowles, MR; Marwood, R; McAllister, G; Patel, S; Seabrook, GR | 1 |
Audinot, V; Jacques, V; Millan, MJ; Newman-Tancredi, A; Peglion, JL | 1 |
Adair, J; Filloux, FM; Narang, N | 1 |
Andersson, K; Bjelke, B; Chen, Y; Gross, J; Herrera-Marschitz, M; Hillefors-Berglund, M; von Euler, G | 1 |
Coronas, V; Jourdan, F; Liang, JJ; Moyse, E; Srivastava, LK | 1 |
Fosbraey, P; Kitchen, I; Ridd, MJ | 1 |
Perachon, S; Schwartz, JC; Sokoloff, P | 1 |
Hillefors, M; von Euler, G | 1 |
Birnbaumer, L; Boulay, G; Jiang, M; Spicher, K; Wang, Y | 1 |
Agnati, LF; Díaz-Cabiale, Z; Ferré, S; Finnman, UB; Fuxe, K; Guidolin, D; Hurd, Y; Vanderhaeghen, JJ; Zoli, M | 1 |
Collins, SL; D'Addario, C; Izenwasser, S | 1 |
Antonelli, T; Díaz-Cabiale, Z; Ferraro, L; Finetti, S; Fuxe, K; Narváez, JA; Tanganelli, S | 1 |
Copolov, DL; Dean, B; Goeringer, K; Pavey, G; Scarr, E | 1 |
Bello, NT; Hajnal, A | 1 |
Covasa, M; Hajnal, A; Margas, WM | 1 |
Morganstern, I; Tejani-Butt, S | 1 |
Lévesque, D; Minogianis, EA; Samaha, AN | 1 |
Blanchet, PJ; Lévesque, D; Mahmoudi, S | 1 |
1 review(s) available for iodosulpride and sulpiride
Article | Year |
---|---|
Retinal dopamine D1 and D2 receptors: characterization by binding or pharmacological studies and physiological functions.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Arylamine N-Acetyltransferase; Benzazepines; Colforsin; Cyclic AMP; Dopamine; Ergolines; Light; Quinpirole; Receptors, Dopamine; Retina; Second Messenger Systems; Species Specificity; Spiperone; Sulpiride; Vertebrates | 1990 |
38 other study(ies) available for iodosulpride and sulpiride
Article | Year |
---|---|
Pharmacology of human dopamine D3 receptor expressed in a mammalian cell line: comparison with D2 receptor.
Topics: Animals; Chlorides; CHO Cells; Cricetinae; Dopamine; Dopamine Agents; Dopamine Antagonists; Guanylyl Imidodiphosphate; Humans; Lithium; Lithium Chloride; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Sodium Chloride; Sulpiride; Transfection | 1992 |
Topographic nonoverlapping distribution of D1 and D2 dopamine receptors in the amygdaloid nuclear complex of the rat brain.
Topics: Amygdala; Animals; Benzazepines; Brain Mapping; Dopamine Antagonists; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride | 1992 |
Autoradiographic evidence for the occlusion of rat brain dopamine D3 receptors in vivo.
Topics: Animals; Autoradiography; Brain; In Vitro Techniques; Iodine Radioisotopes; Radioligand Assay; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulpiride | 1992 |
Identification, characterization, and localization of the dopamine D3 receptor in rat brain using 7-[3H]hydroxy-N,N-di-n-propyl-2-aminotetralin.
Topics: Animals; Brain; Brain Mapping; Cell Membrane; Cells, Cultured; Drug Design; Gene Expression; In Vitro Techniques; Male; Nucleic Acid Hybridization; Rats; Rats, Inbred Strains; Receptors, Dopamine; RNA, Messenger; Sulpiride; Tetrahydronaphthalenes | 1992 |
Agonist-induced desensitization of D2 dopamine receptors in human Y-79 retinoblastoma cells.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Cell Differentiation; Dopamine; Dopamine Agents; Dose-Response Relationship, Drug; Down-Regulation; Humans; Pertussis Toxin; Receptors, Dopamine; Retinoblastoma; Spiperone; Sulpiride; Tumor Cells, Cultured; Virulence Factors, Bordetella | 1991 |
Localization of dopamine D3 receptor mRNA in the rat brain using in situ hybridization histochemistry: comparison with dopamine D2 receptor mRNA.
Topics: Animals; Autoradiography; Blotting, Northern; Brain; Brain Chemistry; Histocytochemistry; Male; Nucleic Acid Hybridization; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; RNA, Messenger; Sulpiride; Transcription, Genetic | 1991 |
Optically active benzamides as predictive tools for mapping the dopamine D2 receptor.
Topics: Animals; Antipsychotic Agents; Benzamides; Computer Simulation; Dopamine Antagonists; Iodine Radioisotopes; Isoquinolines; Mice; Models, Chemical; Molecular Conformation; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Stereoisomerism; Structure-Activity Relationship; Sulpiride | 1990 |
Autoradiographic localization of D1 and D2 dopamine binding sites in the human retina.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Aged; Aged, 80 and over; Autoradiography; Benzazepines; Bromocriptine; Domperidone; Dopamine Antagonists; Humans; Iodine Radioisotopes; Middle Aged; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Retina; Sulpiride | 1990 |
Regulation of neurotensin-containing neurons in the rat striatum. Effects of unilateral striatal lesions with quinolinic acid and ibotenic acid on neurotensin content and its binding site density.
Topics: Animals; Binding Sites; Biogenic Amines; Corpus Striatum; Functional Laterality; gamma-Aminobutyric Acid; Ibotenic Acid; Male; Neurons; Neurotensin; Quinolinic Acid; Quinolinic Acids; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Neurotensin; Receptors, Neurotransmitter; Reference Values; Stereotaxic Techniques; Sulpiride; Tetrabenazine | 1990 |
Ontogeny of dopaminergic D-2 receptors in the rat nervous system: characterization and detailed autoradiographic mapping with [125I]iodosulpride.
Topics: Aging; Animals; Autoradiography; Binding, Competitive; Embryonic and Fetal Development; Female; Nervous System; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Sulpiride | 1989 |
Presence of dopamine D-2 receptors in human tumoral cell lines.
Topics: Apomorphine; Breast Neoplasms; Cell Membrane; Digestive System Neoplasms; Dopamine; Humans; Iodine Radioisotopes; Leukemia; Lung Neoplasms; Neoplasms; Neuroblastoma; Phenethylamines; Receptors, Dopamine; Receptors, Dopamine D2; Sulpiride; Tumor Cells, Cultured | 1989 |
Dopamine receptors in rabbit and rat eye: characterization and localization of DA1 and DA2 binding sites.
Topics: Animals; Autoradiography; Benzazepines; Eye; In Vitro Techniques; Rabbits; Rats; Receptors, Dopamine; Retina; Sulpiride; Time Factors | 1989 |
A detailed mapping of dopamine D-2 receptors in rat central nervous system by autoradiography with [125I]iodosulpride.
Topics: Animals; Autoradiography; Brain; Densitometry; Dopamine; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Sulpiride; Tyrosine 3-Monooxygenase | 1987 |
Localisation and pharmacological characterisation of D-2 dopamine receptors in rat cerebral neocortex and cerebellum using [125I]iodosulpride.
Topics: Animals; Autoradiography; Cerebellum; Cerebral Cortex; Guanylyl Imidodiphosphate; In Vitro Techniques; Iodine Radioisotopes; Male; Membranes; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Sulpiride | 1985 |
Nigral dopamine autoreceptors are exclusively of the D2 type: quantitative autoradiography of [125I]iodosulpride and [125I]SCH 23982 in adjacent brain sections.
Topics: Animals; Autoradiography; Benzazepines; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Substantia Nigra; Sulpiride | 1988 |
Widespread distribution of brain dopamine receptors evidenced with [125I]iodosulpride, a highly selective ligand.
Topics: Animals; Autoradiography; Brain; Cerebellum; Cerebral Cortex; Hippocampus; Iodine Radioisotopes; Ligands; Motor Cortex; Rats; Receptors, Dopamine; Sulpiride | 1985 |
Relative affinities of dopaminergic drugs at dopamine D2 and D3 receptors.
Topics: Animals; Autoradiography; Binding, Competitive; Brain; Caudate Nucleus; Cerebellum; CHO Cells; Cricetinae; Dopamine Agents; Iodine Radioisotopes; Male; Putamen; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Sensitivity and Specificity; Sulpiride; Tetrahydronaphthalenes | 1995 |
Cholecystokinin octapeptide in vitro and ex vivo strongly modulates striatal dopamine D2 receptors in rat forebrain sections.
Topics: Animals; Apomorphine; Autoradiography; Dopamine; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Nucleus Accumbens; Prosencephalon; Putamen; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Sincalide; Sulpiride | 1995 |
Regional and age-dependent differences in the affinity of dopamine D2 agonist binding in the rat brain.
Topics: Aging; Analysis of Variance; Animals; Autoradiography; Brain; Iodine Radioisotopes; Male; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Regression Analysis; Sulpiride | 1995 |
Dopamine D2 and D3 receptors in the rat striatum and nucleus accumbens: use of 7-OH-DPAT and [125I]-iodosulpride.
Topics: Animals; Autoradiography; Binding, Competitive; Cell Membrane; Corpus Striatum; Dopamine Agonists; Iodine Radioisotopes; Kinetics; Male; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulpiride; Tetrahydronaphthalenes | 1995 |
Expression and pharmacological characterization of the human D3 dopamine receptor.
Topics: Animals; Binding, Competitive; Cells, Cultured; CHO Cells; Cricetinae; Dopamine; Dopamine Antagonists; GTP-Binding Proteins; Guanine Nucleotides; Humans; Potassium Channels; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Recombinant Proteins; Second Messenger Systems; Sulpiride | 1994 |
[3H](+)S 14297: a novel, selective radioligand at cloned human dopamine D3 receptors.
Topics: 2-Naphthylamine; Animals; Binding, Competitive; CHO Cells; Cricetinae; Dopamine Agents; Furans; Humans; Ligands; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulpiride; Transfection; Tritium | 1995 |
The temporal evolution of striatal dopamine receptor binding and mRNA expression following hypoxia-ischemia in the neonatal rat.
Topics: Animals; Animals, Newborn; Autoradiography; Base Sequence; Benzazepines; Brain Ischemia; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Female; Hypoxia, Brain; In Situ Hybridization; Iodine Radioisotopes; Molecular Sequence Data; Neostriatum; Neuronal Plasticity; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; RNA, Messenger; Sulpiride; Time Factors; Tritium | 1996 |
Perinatal asphyxia induces long-term changes in dopamine D1, D2, and D3 receptor binding in the rat brain.
Topics: Animals; Apomorphine; Asphyxia Neonatorum; Benzazepines; Brain; Cesarean Section; Dopamine Agonists; Female; Humans; Infant, Newborn; Iodine Radioisotopes; Organ Specificity; Pregnancy; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Spiperone; Sulpiride | 1997 |
Identification and localization of dopamine receptor subtypes in rat olfactory mucosa and bulb: a combined in situ hybridization and ligand binding radioautographic approach.
Topics: Animals; Autoradiography; Benzazepines; Binding Sites; Binding, Competitive; Domperidone; Dopamine Agonists; Dopamine Antagonists; In Situ Hybridization; Iodine Radioisotopes; Male; Olfactory Bulb; Olfactory Mucosa; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; RNA, Messenger; Sulpiride; Tetrahydronaphthalenes | 1997 |
The effect of acute kainic acid treatment on dopamine D2 receptors in rat brain.
Topics: Animals; Brain; Iodine Radioisotopes; Isotope Labeling; Kainic Acid; Male; Neurons; Protein Binding; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D2; Salicylamides; Spiperone; Sulpiride; Tritium | 1998 |
Functional potencies of new antiparkinsonian drugs at recombinant human dopamine D1, D2 and D3 receptors.
Topics: Animals; Antiparkinson Agents; Benzazepines; Binding, Competitive; CHO Cells; Cricetinae; Cyclic AMP; Dopamine; Dopamine Agonists; Dopamine Antagonists; Drug Evaluation; Humans; Hybrid Cells; Mitosis; Radioligand Assay; Receptors, Dopamine D1; Receptors, Dopamine D2; Recombinant Fusion Proteins; Sulpiride; Tumor Cells, Cultured | 1999 |
Pharmacology of [3H]R(+)-7-OH-DPAT binding in the rat caudate-putamen.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzopyrans; Binding, Competitive; Caudate Nucleus; Clozapine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Guanidines; Guanosine Triphosphate; Haloperidol; Heterotrimeric GTP-Binding Proteins; Indans; Kinetics; Magnesium; Male; Oxazines; Protein Binding; Putamen; Quinpirole; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Remoxipride; Sodium; Specific Pathogen-Free Organisms; Sulfones; Sulpiride; Tetrahydronaphthalenes | 2001 |
Most central nervous system D2 dopamine receptors are coupled to their effectors by Go.
Topics: Animals; Brain; Dopamine D2 Receptor Antagonists; GTP-Binding Protein alpha Subunits, Gi-Go; Guanosine 5'-O-(3-Thiotriphosphate); Heterotrimeric GTP-Binding Proteins; Mice; Mice, Knockout; Receptors, Dopamine D2; Sulpiride | 2001 |
Adenosine A2A agonist CGS 21680 decreases the affinity of dopamine D2 receptors for dopamine in human striatum.
Topics: Adenosine; Adult; Animals; Antihypertensive Agents; Binding, Competitive; Dopamine; Dopamine D2 Receptor Antagonists; Drug Interactions; Female; Humans; Male; Middle Aged; Neostriatum; Neurons; Nucleus Accumbens; Phenethylamines; Purinergic P1 Receptor Agonists; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2A; Receptors, Dopamine D2; Receptors, Purinergic P1; Sulpiride | 2001 |
Effects of kappa-opioid receptor agonists on long-term cocaine use and dopamine neurotransmission.
Topics: Analgesics; Animals; Autoradiography; Benzazepines; Benzeneacetamides; Benzomorphans; Binding, Competitive; Brain; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Iodine Radioisotopes; Male; Membrane Glycoproteins; Membrane Transport Proteins; Motor Activity; Nerve Tissue Proteins; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Opioid, kappa; Sulpiride; Synaptic Transmission; Time Factors; Tyrosine 3-Monooxygenase | 2001 |
Neurotensin-induced modulation of dopamine D2 receptors and their function in rat striatum: counteraction by a NTR1-like receptor antagonist.
Topics: Animals; Binding, Competitive; Dopamine; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Drug Interactions; Male; Neostriatum; Neurons; Neurotensin; Pergolide; Pyrazoles; Quinolines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Neurotensin; Sulpiride; Synaptic Transmission | 2002 |
Measurement of dopamine D2-like receptors in postmortem CNS and pituitary: differential regional changes in schizophrenia.
Topics: Adult; Aged; Antipsychotic Agents; Autopsy; Autoradiography; Case-Control Studies; Caudate Nucleus; Female; Humans; Iodine Radioisotopes; Male; Middle Aged; Pituitary Gland; Putamen; Receptors, Dopamine D2; Schizophrenia; Spiperone; Sulpiride | 2004 |
Acute methylphenidate treatments reduce sucrose intake in restricted-fed bingeing rats.
Topics: Analysis of Variance; Animals; Behavior, Animal; Body Weight; Bulimia; Central Nervous System Stimulants; Cocaine; Dose-Response Relationship, Drug; Drinking; Drug Interactions; Eating; Energy Intake; Food Deprivation; Insulin; Male; Methylphenidate; Protein Binding; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Sucrose; Sulpiride | 2006 |
Altered dopamine D2 receptor function and binding in obese OLETF rat.
Topics: Analysis of Variance; Animals; Behavior, Animal; Brain; Conditioning, Operant; Disease Models, Animal; Dopamine Agonists; Dose-Response Relationship, Drug; Glucose Tolerance Test; Iodine Radioisotopes; Male; Motor Activity; Obesity; Protein Binding; Quinpirole; Rats; Rats, Inbred OLETF; Receptors, Dopamine D2; Sucrose; Sulpiride | 2008 |
Differential patterns of alcohol consumption and dopamine-2 receptor binding in Wistar-Kyoto and Wistar rats.
Topics: Alcohol Drinking; Animals; Depressive Disorder; Male; Models, Animal; Rats; Rats, Inbred WKY; Rats, Wistar; Receptors, Dopamine D2; Sulpiride | 2010 |
The speed of cocaine delivery determines the subsequent motivation to self-administer the drug.
Topics: Analysis of Variance; Animals; Cocaine; Conditioning, Operant; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Administration Schedule; Guanosine 5'-O-(3-Thiotriphosphate); Iodine Radioisotopes; Male; Motivation; Protein Binding; Rats; Rats, Wistar; Receptors, Dopamine D2; Self Administration; Sulpiride; Time Factors | 2013 |
Upregulation of dopamine D3, not D2, receptors correlates with tardive dyskinesia in a primate model.
Topics: Animals; Antipsychotic Agents; Brain; Cebus; Clozapine; Disease Models, Animal; Dopamine Antagonists; Enkephalins; Female; Haloperidol; Iodine Radioisotopes; Movement Disorders; Neurons; Ovariectomy; Protein Binding; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulpiride; Tetrahydronaphthalenes; Up-Regulation | 2014 |