Page last updated: 2024-09-04

iodoproxyfan and piperidines

iodoproxyfan has been researched along with piperidines in 4 studies

Compound Research Comparison

Studies
(iodoproxyfan)
Trials
(iodoproxyfan)
Recent Studies (post-2010)
(iodoproxyfan)
Studies
(piperidines)
Trials
(piperidines)
Recent Studies (post-2010) (piperidines)
250240,2355,22114,545

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (25.00)18.2507
2000's3 (75.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bitschnau, H; Kathmann, M; Marr, I; Reidemeister, S; Schlicker, E; Schunack, W; Stark, H1
Arrang, JM; Ganellin, CR; Gbahou, F; Ligneau, X; Morisset, S; Schunack, W; Schwartz, JC; Stark, H; Tardivel-Lacombe, J1
Arrang, JM; Cochois, V; Héron, A; Pillot, C; Rouleau, A; Schwartz, JC1
Anaclet, C; Arrang, JM; Berrebi-Bertrand, I; Bertaina-Anglade, V; Calmels, TP; Camelin, JC; d'Aniello, F; Ganellin, CR; Gbahou, F; la Rochelle, CD; Landais, L; Lecomte, JM; Ligneau, X; Lin, JS; Parmentier, R; Perrin, D; Rouleau, A; Schunack, W; Schwartz, JC; Stark, H1

Other Studies

4 other study(ies) available for iodoproxyfan and piperidines

ArticleYear
Potencies of antagonists chemically related to iodoproxyfan at histamine H3 receptors in mouse brain cortex and guinea-pig ileum: evidence for H3 receptor heterogeneity?
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:5

    Topics: Animals; Binding, Competitive; Cerebral Cortex; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine Antagonists; Histamine H2 Antagonists; Imidazoles; In Vitro Techniques; Intestine, Small; Iodine Radioisotopes; Male; Methylhistamines; Mice; Piperidines; Rats; Rats, Wistar; Structure-Activity Relationship

1996
Distinct pharmacology of rat and human histamine H(3) receptors: role of two amino acids in the third transmembrane domain.
    British journal of pharmacology, 2000, Volume: 131, Issue:7

    Topics: Amino Acid Sequence; Amino Acid Substitution; Amino Acids; Animals; Binding, Competitive; COS Cells; DNA, Complementary; Dose-Response Relationship, Drug; Histamine Antagonists; Humans; Imidazoles; Membrane Proteins; Molecular Sequence Data; Mutagenesis, Site-Directed; Mutation; Piperidines; Protein Structure, Tertiary; Radioligand Assay; Rats; Receptors, Histamine H3; Sequence Alignment; Sequence Homology, Amino Acid; Tritium

2000
Cloning and expression of the mouse histamine H3 receptor: evidence for multiple isoforms.
    Journal of neurochemistry, 2004, Volume: 90, Issue:6

    Topics: Animals; Blotting, Northern; Brain; Chlorocebus aethiops; Cloning, Molecular; Competitive Bidding; COS Cells; Gene Expression; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; In Situ Hybridization; Iodine Radioisotopes; Isoenzymes; Mice; Piperidines; Radioligand Assay; Rats; Receptors, Histamine H3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiourea; Transfection

2004
BF2.649 [1-{3-[3-(4-Chlorophenyl)propoxy]propyl}piperidine, hydrochloride], a nonimidazole inverse agonist/antagonist at the human histamine H3 receptor: Preclinical pharmacology.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 320, Issue:1

    Topics: Acetylcholine; Animals; Cats; Dopamine; Electroencephalography; Guinea Pigs; Histamine Agonists; Histamine Antagonists; Histamine Release; Humans; Imidazoles; Male; Methylhistamines; Mice; Mice, Inbred C57BL; Piperidines; Prefrontal Cortex; Receptors, Histamine H3; Scopolamine

2007