iodoproxyfan has been researched along with histamine in 10 studies
*Histamine: An amine derived by enzymatic decarboxylation of HISTIDINE. It is a powerful stimulant of gastric secretion, a constrictor of bronchial smooth muscle, a vasodilator, and also a centrally acting neurotransmitter. [MeSH]
*Histamine: An amine derived by enzymatic decarboxylation of HISTIDINE. It is a powerful stimulant of gastric secretion, a constrictor of bronchial smooth muscle, a vasodilator, and also a centrally acting neurotransmitter. [MeSH]
| Studies (iodoproxyfan) | Trials (iodoproxyfan) | Recent Studies (post-2010) (iodoproxyfan) | Studies (histamine) | Trials (histamine) | Recent Studies (post-2010) (histamine) |
|---|---|---|---|---|---|
| 25 | 0 | 2 | 37,718 | 1,372 | 3,457 |
| Protein | Taxonomy | iodoproxyfan (IC50) | histamine (IC50) |
|---|---|---|---|
| Histamine H1 receptor | Rattus norvegicus (Norway rat) | 0.1585 | |
| Histamine H1 receptor | Homo sapiens (human) | 0.1585 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 1 (10.00) | 18.2507 |
| 2000's | 5 (50.00) | 29.6817 |
| 2010's | 4 (40.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Christiaans, JA; Gynther, J; Kotisaari, S; Kovalainen, JT; Laitinen, JT; Männistö, PT; Tuomisto, L | 1 |
| Hastrup, S; Rimvall, K; Wulff, BS | 1 |
| Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM | 1 |
| Buschauer, A; Dove, S; Igel, P | 1 |
| de Esch, IJ; de Graaf, C; Istyastono, EP; Kooistra, AJ; Leurs, R; Lim, HD; Nijmeijer, S; Roumen, L; van de Stolpe, A; Vischer, HF | 1 |
| Arrang, JM; Cochois, V; Heron, A; Ligneau, X; Pillot, C; Schwartz, JC; Tardivel-Lacombe, J | 1 |
| Arrang, JM; Cochois, V; Héron, A; Pillot, C; Rouleau, A; Schwartz, JC | 1 |
| Arrang, JM; Chabret, C; Gbahou, F; Humbert-Claude, M; Tardivel-Lacombe, J; Vincent, L | 1 |
| Arrang, JM; Davenas, E; Gbahou, F; Morisset, S | 1 |
| Arrang, JM; Gbahou, F; Rouleau, A | 1 |
10 other study(ies) available for iodoproxyfan and histamine
| Article | Year |
|---|---|
Synthesis and in vitro pharmacology of a series of new chiral histamine H3-receptor ligands: 2-(R and S)-Amino-3-(1H-imidazol-4(5)-yl)propyl ether derivatives.
Topics: Animals; Autoradiography; Binding, Competitive; Cerebral Cortex; Corpus Striatum; Histamine Agonists; Histamine Antagonists; Imidazoles; In Vitro Techniques; Ligands; Male; Propylamines; Rats; Rats, Wistar; Receptors, Histamine H3; Stereoisomerism; Structure-Activity Relationship | 1999 |
Characteristics of recombinantly expressed rat and human histamine H3 receptors.
Topics: Animals; Cell Line; Cloning, Molecular; Histamine Agonists; Histamine Antagonists; Humans; Rats; Receptors, Histamine; Receptors, Histamine H3; Recombination, Genetic | 2002 |
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4 | 2005 |
Histamine H4 receptor agonists.
Topics: Animals; Benzimidazoles; Binding Sites; Clozapine; Guanidines; Humans; Ligands; Mice; Oximes; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Structure-Activity Relationship | 2010 |
Molecular determinants of ligand binding modes in the histamine H(4) receptor: linking ligand-based three-dimensional quantitative structure-activity relationship (3D-QSAR) models to in silico guided receptor mutagenesis studies.
Topics: Cell Line, Tumor; Histamine Antagonists; Humans; Hydrophobic and Hydrophilic Interactions; Imidazoles; Ligands; Models, Molecular; Molecular Conformation; Molecular Dynamics Simulation; Mutagenesis, Site-Directed; Quantitative Structure-Activity Relationship; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H3; Receptors, Histamine H4; Stereoisomerism; Thiourea | 2011 |
A detailed mapping of the histamine H(3) receptor and its gene transcripts in rat brain.
Topics: Animals; Binding Sites; Brain; Brain Mapping; Gene Expression; Histamine; Imidazoles; In Situ Hybridization; Male; Neurons; Oligonucleotide Probes; Protein Isoforms; Radioligand Assay; Rats; Rats, Wistar; Receptors, Histamine H3; RNA, Messenger | 2002 |
Cloning and expression of the mouse histamine H3 receptor: evidence for multiple isoforms.
Topics: Animals; Blotting, Northern; Brain; Chlorocebus aethiops; Cloning, Molecular; Competitive Bidding; COS Cells; Gene Expression; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; In Situ Hybridization; Iodine Radioisotopes; Isoenzymes; Mice; Piperidines; Radioligand Assay; Rats; Receptors, Histamine H3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiourea; Transfection | 2004 |
Compared pharmacology of human histamine H3 and H4 receptors: structure-activity relationships of histamine derivatives.
Topics: Binding, Competitive; Colforsin; Cyclic AMP; DNA, Complementary; Histamine; Histamine H2 Antagonists; Humans; Imidazoles; In Vitro Techniques; Kidney; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H3; Receptors, Histamine H4; Recombinant Proteins; Structure-Activity Relationship; Transfection | 2006 |
Effects of betahistine at histamine H3 receptors: mixed inverse agonism/agonism in vitro and partial inverse agonism in vivo.
Topics: Administration, Oral; Animals; Arachidonic Acid; Betahistine; Brain; Brain Chemistry; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Histamine; Histamine Agonists; Histamine H2 Antagonists; Histamine H3 Antagonists; Humans; Imidazoles; Injections, Intraperitoneal; Methylhistamines; Mice; Neurons; Pertussis Toxin; Rats; Receptors, Histamine H3; Recombinant Proteins | 2010 |
The histamine autoreceptor is a short isoform of the H₃ receptor.
Topics: Animals; Arachidonic Acid; Autoreceptors; Brain; Calcimycin; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Guanosine 5'-O-(3-Thiotriphosphate); Histamine; Imidazoles; In Vitro Techniques; Male; Methylhistamines; Protein Isoforms; Rats; Rats, Wistar; Receptors, Histamine H3 | 2012 |