iodoproxyfan has been researched along with clobenpropit in 6 studies
| Studies (iodoproxyfan) | Trials (iodoproxyfan) | Recent Studies (post-2010) (iodoproxyfan) | Studies (clobenpropit) | Trials (clobenpropit) | Recent Studies (post-2010) (clobenpropit) |
|---|---|---|---|---|---|
| 25 | 0 | 2 | 147 | 0 | 29 |
| Protein | Taxonomy | iodoproxyfan (IC50) | clobenpropit (IC50) |
|---|---|---|---|
| Histamine H3 receptor | Mus musculus (house mouse) | 0.001 | |
| Histamine H3 receptor | Homo sapiens (human) | 0.0011 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 1 (16.67) | 18.2507 |
| 2000's | 4 (66.67) | 29.6817 |
| 2010's | 1 (16.67) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Christiaans, JA; Gynther, J; Kotisaari, S; Kovalainen, JT; Laitinen, JT; Männistö, PT; Tuomisto, L | 1 |
| Arrang, JM; Ganellin, CR; Ligneau, X; Schunack, W; Schwartz, JC; Sippl, W; Stark, H | 1 |
| De Esch, IJ; Dean, PM; Hoffmann, M; Leurs, R; Menge, WM; Mills, JE; Nederkoorn, PH; Perkins, TD; Romeo, G; Timmerman, H; Wieland, K | 1 |
| Hastrup, S; Rimvall, K; Wulff, BS | 1 |
| Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM | 1 |
| de Esch, IJ; de Graaf, C; Istyastono, EP; Kooistra, AJ; Leurs, R; Lim, HD; Nijmeijer, S; Roumen, L; van de Stolpe, A; Vischer, HF | 1 |
6 other study(ies) available for iodoproxyfan and clobenpropit
| Article | Year |
|---|---|
Synthesis and in vitro pharmacology of a series of new chiral histamine H3-receptor ligands: 2-(R and S)-Amino-3-(1H-imidazol-4(5)-yl)propyl ether derivatives.
Topics: Animals; Autoradiography; Binding, Competitive; Cerebral Cortex; Corpus Striatum; Histamine Agonists; Histamine Antagonists; Imidazoles; In Vitro Techniques; Ligands; Male; Propylamines; Rats; Rats, Wistar; Receptors, Histamine H3; Stereoisomerism; Structure-Activity Relationship | 1999 |
Different antagonist binding properties of human and rat histamine H3 receptors.
Topics: Animals; CHO Cells; Cricetinae; Female; Histamine Antagonists; Humans; Imidazoles; Models, Molecular; Protein Binding; Rats; Receptors, Histamine H3; Rhodopsin; Species Specificity | 2001 |
Development of a pharmacophore model for histamine H3 receptor antagonists, using the newly developed molecular modeling program SLATE.
Topics: Animals; Benzyl Compounds; Cerebral Cortex; Guinea Pigs; Histamine Antagonists; Histamine Release; Imidazoles; In Vitro Techniques; Intestines; Ligands; Models, Molecular; Muscle Contraction; Muscle, Smooth; Piperidines; Quantitative Structure-Activity Relationship; Radioligand Assay; Rats; Receptors, Histamine H3; Software | 2001 |
Characteristics of recombinantly expressed rat and human histamine H3 receptors.
Topics: Animals; Cell Line; Cloning, Molecular; Histamine Agonists; Histamine Antagonists; Humans; Rats; Receptors, Histamine; Receptors, Histamine H3; Recombination, Genetic | 2002 |
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4 | 2005 |
Molecular determinants of ligand binding modes in the histamine H(4) receptor: linking ligand-based three-dimensional quantitative structure-activity relationship (3D-QSAR) models to in silico guided receptor mutagenesis studies.
Topics: Cell Line, Tumor; Histamine Antagonists; Humans; Hydrophobic and Hydrophilic Interactions; Imidazoles; Ligands; Models, Molecular; Molecular Conformation; Molecular Dynamics Simulation; Mutagenesis, Site-Directed; Quantitative Structure-Activity Relationship; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H3; Receptors, Histamine H4; Stereoisomerism; Thiourea | 2011 |