iodoproxyfan has been researched along with alpha-methylhistamine in 7 studies
| Studies (iodoproxyfan) | Trials (iodoproxyfan) | Recent Studies (post-2010) (iodoproxyfan) | Studies (alpha-methylhistamine) | Trials (alpha-methylhistamine) | Recent Studies (post-2010) (alpha-methylhistamine) |
|---|---|---|---|---|---|
| 25 | 0 | 2 | 240 | 3 | 13 |
| 25 | 0 | 2 | 46 | 0 | 12 |
| Protein | Taxonomy | iodoproxyfan (IC50) | alpha-methylhistamine (IC50) |
|---|---|---|---|
| Histamine H3 receptor | Rattus norvegicus (Norway rat) | 0.0015 | |
| Histamine H3 receptor | Homo sapiens (human) | 0.0023 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 2 (28.57) | 18.2507 |
| 2000's | 3 (42.86) | 29.6817 |
| 2010's | 2 (28.57) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Garbarg, M; Hüls, A; Ligneau, X; Purand, K; Schunack, W; Schwartz, JC; Stark, H | 1 |
| Arrang, JM; Gbahou, F; Rouleau, A | 1 |
| Christiaans, JA; Gynther, J; Kotisaari, S; Kovalainen, JT; Laitinen, JT; Männistö, PT; Tuomisto, L | 1 |
| Hastrup, S; Rimvall, K; Wulff, BS | 1 |
| Arrang, JM; Fkyerat, A; Ganellin, CR; Garbarg, M; Ligneau, X; Pelloux-Léon, N; Piripitsi, A; Schunack, W; Schwartz, JC; Stark, H; Tertiuk, W | 1 |
| Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM | 1 |
| Buschauer, A; Dove, S; Igel, P | 1 |
7 other study(ies) available for iodoproxyfan and alpha-methylhistamine
| Article | Year |
|---|---|
[125I]iodoproxyfan and related compounds: a reversible radioligand and novel classes of antagonists with high affinity and selectivity for the histamine H3 receptor.
Topics: Animals; Cerebral Cortex; Guinea Pigs; Histamine Antagonists; Imidazoles; In Vitro Techniques; Iodine Radioisotopes; Methylhistamines; Radioligand Assay; Rats; Structure-Activity Relationship | 1996 |
The histamine autoreceptor is a short isoform of the H₃ receptor.
Topics: Animals; Arachidonic Acid; Autoreceptors; Brain; Calcimycin; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Guanosine 5'-O-(3-Thiotriphosphate); Histamine; Imidazoles; In Vitro Techniques; Male; Methylhistamines; Protein Isoforms; Rats; Rats, Wistar; Receptors, Histamine H3 | 2012 |
Synthesis and in vitro pharmacology of a series of new chiral histamine H3-receptor ligands: 2-(R and S)-Amino-3-(1H-imidazol-4(5)-yl)propyl ether derivatives.
Topics: Animals; Autoradiography; Binding, Competitive; Cerebral Cortex; Corpus Striatum; Histamine Agonists; Histamine Antagonists; Imidazoles; In Vitro Techniques; Ligands; Male; Propylamines; Rats; Rats, Wistar; Receptors, Histamine H3; Stereoisomerism; Structure-Activity Relationship | 1999 |
Characteristics of recombinantly expressed rat and human histamine H3 receptors.
Topics: Animals; Cell Line; Cloning, Molecular; Histamine Agonists; Histamine Antagonists; Humans; Rats; Receptors, Histamine; Receptors, Histamine H3; Recombination, Genetic | 2002 |
Meta-substituted aryl(thio)ethers as potent partial agonists (or antagonists) for the histamine H3 receptor lacking a nitrogen atom in the side chain.
Topics: Animals; Brain; Ethers; Histamine Agonists; Histamine Antagonists; Histamine Release; Imidazoles; Male; Methylhistamines; Mice; Rats; Receptors, Histamine H3; Structure-Activity Relationship; Sulfides; Synaptosomes | 2004 |
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4 | 2005 |
Histamine H4 receptor agonists.
Topics: Animals; Benzimidazoles; Binding Sites; Clozapine; Guanidines; Humans; Ligands; Mice; Oximes; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Structure-Activity Relationship | 2010 |