Page last updated: 2024-09-03

iodobolpyramine and pyrilamine

iodobolpyramine has been researched along with pyrilamine in 6 studies

Compound Research Comparison

Studies
(iodobolpyramine)
Trials
(iodobolpyramine)
Recent Studies (post-2010)
(iodobolpyramine)
Studies
(pyrilamine)
Trials
(pyrilamine)
Recent Studies (post-2010) (pyrilamine)
6001,86026116

Protein Interaction Comparison

ProteinTaxonomyiodobolpyramine (IC50)pyrilamine (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)1.13
Alpha-2A adrenergic receptorHomo sapiens (human)2.976
Cytochrome P450 2D6Homo sapiens (human)0.3
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.997
5-hydroxytryptamine receptor 2CHomo sapiens (human)1.13
Histamine H1 receptorCavia porcellus (domestic guinea pig)0.0015
Histamine H1 receptorRattus norvegicus (Norway rat)0.0126
Sodium-dependent serotonin transporterHomo sapiens (human)0.047
Histamine H1 receptorHomo sapiens (human)0.0166
5-hydroxytryptamine receptor 2BHomo sapiens (human)2.788
Sodium-dependent dopamine transporter Homo sapiens (human)0.879
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1.1
Sigma non-opioid intracellular receptor 1Homo sapiens (human)1.558

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19902 (33.33)18.7374
1990's4 (66.67)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bouthenet, ML; Hirschfeld, J; Martinez-Mir, I; Moreau, J; Palacios, JM; Pollard, H; Ruat, M; Schwartz, JC; Souil, E; Traiffort, E1
Bach, JF; Chatenoud, LM; Villemain, FM1
Arrang, JM; Martinez-Mir, MI; Moreau, J; Palacios, JM; Pollard, H; Ruat, M; Schwartz, JC; Traiffort, E1
Bouthenet, ML; Ganellin, CR; Ruat, M; Schwartz, JC1
Bouthenet, ML; Garbarg, M; Ruat, M; Sales, N; Schwartz, JC1
Bouthenet, ML; Ganellin, CR; Garbarg, M; Gros, C; Ife, RJ; Korner, M; Sales, N; Schwartz, JC1

Reviews

1 review(s) available for iodobolpyramine and pyrilamine

ArticleYear
Reversible and irreversible labelling of H1- and H2 -receptors using novel [125I] probes.
    Agents and actions. Supplements, 1991, Volume: 33

    Topics: Affinity Labels; Animals; Guanidines; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Iodine Radioisotopes; Myocardium; Photochemistry; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Succinimides

1991

Other Studies

5 other study(ies) available for iodobolpyramine and pyrilamine

ArticleYear
Characterization of histamine H1 binding sites on human T lymphocytes by means of 125I-iodobolpyramine. Preferential expression of H1 receptors on CD8 T lymphocytes.
    Journal of immunology (Baltimore, Md. : 1950), 1990, Feb-15, Volume: 144, Issue:4

    Topics: Aminopyridines; Animals; Antigens, Differentiation, T-Lymphocyte; CD4-Positive T-Lymphocytes; CD8 Antigens; Cell Membrane; Cerebellum; Guinea Pigs; Humans; Kinetics; Pyrilamine; Receptors, Histamine H1; Succinimides; T-Lymphocytes; T-Lymphocytes, Helper-Inducer; T-Lymphocytes, Regulatory

1990
Three histamine receptors (H1, H2 and H3) visualized in the brain of human and non-human primates.
    Brain research, 1990, Sep-03, Volume: 526, Issue:2

    Topics: Adult; Aged; Aged, 80 and over; Animals; Autoradiography; Brain Chemistry; Female; Guanidines; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Iodine Radioisotopes; Macaca mulatta; Male; Methylhistamines; Middle Aged; Pyrilamine; Radioligand Assay; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Succinimides

1990
Histamine H1-receptor in heart: unique electrophoretic mobility and autoradiographic localization.
    Journal of neurochemistry, 1990, Volume: 55, Issue:2

    Topics: Affinity Labels; Animals; Autoradiography; Cell Membrane; Cerebellum; Chlorpheniramine; Electrophoresis, Polyacrylamide Gel; Guinea Pigs; Heart Atria; Ileum; Iodine Radioisotopes; Lung; Male; Mianserin; Molecular Weight; Myocardium; Photochemistry; Pyrilamine; Receptors, Histamine H1; Succinimides

1990
A detailed mapping of histamine H1-receptors in guinea-pig central nervous system established by autoradiography with [125I]iodobolpyramine.
    Neuroscience, 1988, Volume: 26, Issue:2

    Topics: Aminopyridines; Animals; Autoradiography; Brain; Brain Mapping; Guinea Pigs; Pyrilamine; Receptors, Histamine; Spinal Cord; Succinimides

1988
[125I]Iodobolpyramine, a highly sensitive probe for histamine H1-receptors in guinea-pig brain.
    European journal of pharmacology, 1986, Jan-21, Volume: 120, Issue:2

    Topics: Aminopyridines; Animals; Autoradiography; Brain; Cerebellum; Guinea Pigs; In Vitro Techniques; Indicators and Reagents; Iodine Radioisotopes; Kinetics; Male; Membranes; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Succinimides

1986