indole and piperazine

indole has been researched along with piperazine in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (20.00)18.2507
2000's1 (20.00)29.6817
2010's2 (40.00)24.3611
2020's1 (20.00)2.80

Authors

AuthorsStudies
Marinov, BS1
Anzali, S; Bartoszyk, GD; Böttcher, H; Gericke, R; Greiner, HE; Heinrich, T; Seyfried, CA; Van Amsterdam, C1
Caliendo, G; De Angelis, F; Esposito, A; Fiorino, F; Frecentese, F; Magli, E; Massarelli, P; Nencini, C; Perissutti, E; Santagada, V; Severino, B; Viti, B1
Cho, S; Choo, DJ; Choo, HY; Hayat, F; Indu Viswanath, AN; Lee, JY; Pae, AN; Rhim, H1
Abe, H; Asawa, Y; Katsuragi, K; Makino, K; Nakamura, H; Nomura, M; Ogino, Y; Okazawa, M; Oyama, T; Sakamoto, Y; Sato, A; Shibasaki, Y; Takahashi, H; Tanuma, N; Tanuma, SI; Uchiumi, F; Yamazaki, H; Yoshimori, A1

Other Studies

5 other study(ies) available for indole and piperazine

ArticleYear
A possible role of the redox interactions in the dual, activatory and inhibitory, action of DPI 201-106 on the potential-dependent Na+ channels.
    Membrane & cell biology, 1997, Volume: 10, Issue:6

    Topics: Allosteric Regulation; Cardiotonic Agents; Indoles; Myoglobin; NAD; Oxidants, Photochemical; Oxidation-Reduction; Piperazine; Piperazines; Sodium Channel Blockers; Sodium Channels; Stereoisomerism

1997
Synthesis and structure--activity relationship in a class of indolebutylpiperazines as dual 5-HT(1A) receptor agonists and serotonin reuptake inhibitors.
    Journal of medicinal chemistry, 2004, Sep-09, Volume: 47, Issue:19

    Topics: Animals; Biological Transport; Hippocampus; Indoles; Inhibitory Concentration 50; Molecular Structure; Piperazine; Piperazines; Rats; Receptors, Serotonin, 5-HT1; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin 5-HT1 Receptor Agonists; Structure-Activity Relationship

2004
Efficient microwave combinatorial synthesis of novel indolic arylpiperazine derivatives as serotoninergic ligands.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:2

    Topics: Animals; Combinatorial Chemistry Techniques; Drug Evaluation, Preclinical; Indoles; Ligands; Male; Microwaves; Piperazine; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin

2010
Design and synthesis of novel series of 5-HT6 receptor ligands having indole, a central aromatic core and 1-amino-4 methyl piperazine as a positive ionizable group.
    Bioorganic & medicinal chemistry, 2013, Sep-01, Volume: 21, Issue:17

    Topics: Algorithms; Drug Design; HEK293 Cells; Humans; Indoles; Ions; Ligands; Piperazine; Piperazines; Protein Binding; Quantitative Structure-Activity Relationship; Receptors, Serotonin; Recombinant Proteins; Serotonin Antagonists; Structure-Activity Relationship

2013
Structural Basis of Beneficial Design for Effective Nicotinamide Phosphoribosyltransferase Inhibitors.
    Molecules (Basel, Switzerland), 2020, Aug-10, Volume: 25, Issue:16

    Topics: Binding Sites; Catalytic Domain; Drug Design; Enzyme Inhibitors; Humans; Indoles; Kinetics; Molecular Docking Simulation; Nicotinamide Phosphoribosyltransferase; Piperazine; Piperidines

2020