indole and colchicine

indole has been researched along with colchicine in 6 studies

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (16.67)29.6817
2010's4 (66.67)24.3611
2020's1 (16.67)2.80

Authors

AuthorsStudies
Bánhegyi, P; Erös, D; Hafenbradl, D; Hegymegi-Barakonyi, B; Hollósy, F; Kéri, G; Klebl, B; Mészáros, G; Obert, S; Orfi, L; Pató, J; Székelyhidi, Z; Wáczek, F1
Borges, F; Chavarria, D; Fernandes, C; Gil-Martins, E; Oliveira, PJ; Remião, F; Silva, C; Silva, R; Silva, T; Silva, V; Soares, P1
Abdayem, R; Barret, R; Colomb, E; Dubois, J; Guillaume, J; Haftek, M; Lomberget, T; Nachtergaele, L; Nguyen, TT; Thoret, S; Tran, NC1
Devambatla, RK; Dybdal-Hargreaves, NF; Gangjee, A; Hamel, E; Mooberry, SL; Raghavan, S; Westbrook, CD; Zaware, N1
Chaplin, DJ; Hall, JJ; Hamel, E; Macdonough, MT; Pinney, KG; Strecker, TE; Trawick, ML1
Chen, J; Jiang, S; Li, L; Li, X; Liu, Y; Su, J1

Reviews

1 review(s) available for indole and colchicine

ArticleYear
Recent advances in trimethoxyphenyl (TMP) based tubulin inhibitors targeting the colchicine binding site.
    European journal of medicinal chemistry, 2018, May-10, Volume: 151

    Topics: Animals; Benzene Derivatives; Binding Sites; Biological Products; Chalcone; Clinical Trials as Topic; Colchicine; Drug Discovery; Humans; Indoles; Microtubules; Molecular Docking Simulation; Stilbenes; Tubulin; Tubulin Modulators

2018

Other Studies

5 other study(ies) available for indole and colchicine

ArticleYear
Synthesis of selective SRPK-1 inhibitors: novel tricyclic quinoxaline derivatives.
    Bioorganic & medicinal chemistry letters, 2005, Jul-01, Volume: 15, Issue:13

    Topics: Antiviral Agents; Enzyme Inhibitors; Hepatitis B; Hepatitis B virus; Humans; Inhibitory Concentration 50; Protein Serine-Threonine Kinases; Quinoxalines; Structure-Activity Relationship

2005
Design of novel monoamine oxidase-B inhibitors based on piperine scaffold: Structure-activity-toxicity, drug-likeness and efflux transport studies.
    European journal of medicinal chemistry, 2020, Jan-01, Volume: 185

    Topics: Alkaloids; Benzodioxoles; Caco-2 Cells; Cell Differentiation; Cell Survival; Dose-Response Relationship, Drug; Drug Design; Humans; Ligands; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Neuroprotective Agents; Oxidative Stress; Piperidines; Polyunsaturated Alkamides; Structure-Activity Relationship; Tumor Cells, Cultured

2020
Synthesis and biological evaluation of novel heterocyclic derivatives of combretastatin A-4.
    Bioorganic & medicinal chemistry letters, 2012, Dec-01, Volume: 22, Issue:23

    Topics: Antimitotic Agents; Benzofurans; Cell Cycle Checkpoints; Cell Line, Tumor; Cell Proliferation; Colchicine; Heterocyclic Compounds; Humans; Indoles; Microscopy, Confocal; Microtubules; Stereoisomerism; Stilbenes; Thiophenes

2012
Synthesis of N(4)-(substituted phenyl)-N(4)-alkyl/desalkyl-9H-pyrimido[4,5-b]indole-2,4-diamines and identification of new microtubule disrupting compounds that are effective against multidrug resistant cells.
    Bioorganic & medicinal chemistry, 2013, Feb-15, Volume: 21, Issue:4

    Topics: Aniline Compounds; Binding Sites; Cell Line, Tumor; Cell Proliferation; Colchicine; Cyclization; Cyclohexanones; Diamines; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Humans; Indoles; Microtubules; Molecular Docking Simulation; Oxidation-Reduction; Protein Binding; Protein Structure, Tertiary; Pyrimidines; Tubulin Modulators

2013
Synthesis and biological evaluation of indole-based, anti-cancer agents inspired by the vascular disrupting agent 2-(3'-hydroxy-4'-methoxyphenyl)-3-(3″,4″,5″-trimethoxybenzoyl)-6-methoxyindole (OXi8006).
    Bioorganic & medicinal chemistry, 2013, Nov-01, Volume: 21, Issue:21

    Topics: Antineoplastic Agents; Cell Line, Tumor; Cell Survival; Colchicine; Drug Screening Assays, Antitumor; Humans; Indoles; Protein Binding; Structure-Activity Relationship; Tubulin; Tubulin Modulators

2013