indole and benzofurans

indole has been researched along with benzofurans in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19901 (6.67)18.7374
1990's1 (6.67)18.2507
2000's3 (20.00)29.6817
2010's7 (46.67)24.3611
2020's3 (20.00)2.80

Authors

AuthorsStudies
Cha, YN; Heine, HS; Stoskopf, MK; Thompson, DC1
Matthews, BW; Morton, A1
Ballesteros, A; Barluenga, J; González, JM; Merino, I; Vázquez-Villa, H1
Anand, R; Christ, DD; Covington, MB; Duan, JJ; Liu, RQ; Lu, Z; Newton, RC; Ott, GR; Qian, M; Trzaskos, J; Vaddi, K1
Lautens, M; Tseng, NW1
Cacchi, S; Fabrizi, G; Goggiamani, A1
Abdayem, R; Barret, R; Colomb, E; Dubois, J; Guillaume, J; Haftek, M; Lomberget, T; Nachtergaele, L; Nguyen, TT; Thoret, S; Tran, NC1
Dong, X; Xiao, T; Zhou, L1
Chang, W; Coburn, CA; Fandozzi, CM; Graham, DJ; Hu, B; Huang, Q; Kargman, S; Kozlowski, J; Liu, R; Ludmerer, SW; McCauley, JA; Meinke, PT; Nomeir, AA; Olsen, DB; Soll, RM; Vacca, JP; Wang, D; Wu, H; Zhong, B1
Ananikov, VP; Asachenko, AF; Bush, AA; Khrustalev, VN; Lunchev, AV; Morozov, OS; Nechaev, MS; Tukov, AA; Zalesskiy, SS1
Beaud, R; Cucca, M; Denizot, N; Guillot, R; Kouklovsky, C; Pouilhès, A; Vincent, G1
Bhadbhade, M; Black, DS; Griffith, R; Kandemir, H; Kumar, N; Lewis, PJ; Ma, C; Mielczarek, M; Thomas, RV; Yang, X1
Bertrand, B; Chang, L; Dechoux, L; Fischer-Durand, N; Gontard, G; Thorimbert, S1
Kaur, N; Kaur, P; Kumar, V; Nayak, SK; Sahu, SK; Wadhwa, P1
Basilico, N; Butini, S; Campiani, G; D'Alessandro, S; Gemma, S; Ibba, R; Parapini, S; Pozzetti, L; Rossi, S; Taglialatela-Scafati, O; Taramelli, D1

Reviews

1 review(s) available for indole and benzofurans

ArticleYear
Alpha-amylase as molecular target for treatment of diabetes mellitus: A comprehensive review.
    Chemical biology & drug design, 2021, Volume: 98, Issue:4

    Topics: 1-Deoxynojirimycin; Acarbose; alpha-Amylases; Benzofurans; Blood Glucose; Diabetes Mellitus; Drug Discovery; Flavonoids; Glycoside Hydrolase Inhibitors; Humans; Hydrazones; Hypoglycemic Agents; Indoles; Inositol; Oxadiazoles; Structure-Activity Relationship

2021

Other Studies

14 other study(ies) available for indole and benzofurans

ArticleYear
Enhancement of epoxide hydrolase activity in hepatic microsomes of mice given heterocyclic compounds.
    Chemico-biological interactions, 1986, Volume: 59, Issue:2

    Topics: Animals; Benzofurans; Butylated Hydroxyanisole; Butylated Hydroxytoluene; Epoxide Hydrolases; Ethers, Cyclic; Female; Glutathione Transferase; Heterocyclic Compounds; Indoles; Mice; Mice, Inbred Strains; Microsomes, Liver; Quinone Reductases; Structure-Activity Relationship

1986
Specificity of ligand binding in a buried nonpolar cavity of T4 lysozyme: linkage of dynamics and structural plasticity.
    Biochemistry, 1995, Jul-11, Volume: 34, Issue:27

    Topics: Bacteriophage T4; Benzene Derivatives; Benzofurans; Computer Graphics; Crystallography, X-Ray; Hydrogen Bonding; Indenes; Indoles; Ligands; Models, Molecular; Muramidase; Protein Binding; Protein Conformation; Xylenes

1995
The reaction of o-alkynylarene and heteroarene carboxaldehyde derivatives with iodonium ions and nucleophiles: a versatile and regioselective synthesis of 1H-isochromene, naphthalene, indole, benzofuran, and benzothiophene compounds.
    Chemistry (Weinheim an der Bergstrasse, Germany), 2006, Jul-24, Volume: 12, Issue:22

    Topics: Aldehydes; Alkynes; Benzofurans; Benzopyrans; Heterocyclic Compounds; Indoles; Ions; Naphthalenes; Onium Compounds; Pyridines; Thiophenes

2006
Potent, selective, orally bioavailable inhibitors of tumor necrosis factor-alpha converting enzyme (TACE): discovery of indole, benzofuran, imidazopyridine and pyrazolopyridine P1' substituents.
    Bioorganic & medicinal chemistry letters, 2008, Mar-15, Volume: 18, Issue:6

    Topics: ADAM Proteins; ADAM17 Protein; Administration, Oral; Animals; Benzofurans; Biological Availability; Humans; Hydroxamic Acids; Imidazoles; Indoles; Lipopolysaccharides; Matrix Metalloproteinase Inhibitors; Molecular Structure; Protease Inhibitors; Pyrazoles; Pyridines; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship; Tumor Necrosis Factor-alpha

2008
Application of a rhodium-catalyzed addition/cyclization sequence toward the synthesis of polycyclic heteroaromatics.
    The Journal of organic chemistry, 2009, Feb-20, Volume: 74, Issue:4

    Topics: Alkenes; Benzofurans; Boronic Acids; Catalysis; Cyclization; Esters; Heterocyclic Compounds; Indoles; Polycyclic Compounds; Rhodium; Thiophenes

2009
Copper catalysis in the construction of indole and benzo[b]furan rings.
    Organic & biomolecular chemistry, 2011, Feb-07, Volume: 9, Issue:3

    Topics: Benzofurans; Catalysis; Copper; Indoles; Ligands

2011
Synthesis and biological evaluation of novel heterocyclic derivatives of combretastatin A-4.
    Bioorganic & medicinal chemistry letters, 2012, Dec-01, Volume: 22, Issue:23

    Topics: Antimitotic Agents; Benzofurans; Cell Cycle Checkpoints; Cell Line, Tumor; Cell Proliferation; Colchicine; Heterocyclic Compounds; Humans; Indoles; Microscopy, Confocal; Microtubules; Stereoisomerism; Stilbenes; Thiophenes

2012
Benzofuran and indole synthesis via Cu(I)-catalyzed coupling of N-tosylhydrazone and o-hydroxy or o-amino phenylacetylene.
    Organic & biomolecular chemistry, 2013, Mar-07, Volume: 11, Issue:9

    Topics: Acetylene; Benzofurans; Catalysis; Copper; Hydrazones; Indoles; Molecular Structure

2013
Discovery of MK-8742: an HCV NS5A inhibitor with broad genotype activity.
    ChemMedChem, 2013, Volume: 8, Issue:12

    Topics: Animals; Antiviral Agents; Benzofurans; Dogs; Drug Evaluation, Preclinical; Enzyme Inhibitors; Half-Life; Hepacivirus; Imidazoles; Indoles; Mutation; Pan troglodytes; Protein Binding; Rats; Structure-Activity Relationship; Viral Nonstructural Proteins

2013
Expanded-ring N-heterocyclic carbenes efficiently stabilize gold(I) cations, leading to high activity in π-acid-catalyzed cyclizations.
    Chemistry (Weinheim an der Bergstrasse, Germany), 2014, May-12, Volume: 20, Issue:20

    Topics: Acids; Alkynes; Benzofurans; Catalysis; Cations; Cyclization; Gold; Heterocyclic Compounds; Indoles; Methane

2014
Bioinspired direct access to benzofuroindolines by oxidative [3 + 2] annulation of phenols and indoles.
    Organic letters, 2014, Nov-07, Volume: 16, Issue:21

    Topics: Benzofurans; Catalysis; Indoles; Molecular Structure; Oxidation-Reduction; Phenols

2014
Synthesis and biological activity of novel mono-indole and mono-benzofuran inhibitors of bacterial transcription initiation complex formation.
    Bioorganic & medicinal chemistry, 2015, Apr-15, Volume: 23, Issue:8

    Topics: Anti-Bacterial Agents; Bacteria; Bacterial Infections; Benzofurans; DNA-Directed RNA Polymerases; Humans; Indoles; Models, Molecular; Structure-Activity Relationship; Transcriptional Activation

2015
A Solvent-free, Catalyst-free Formal [3+3] Cycloaddition Dearomatization Strategy: Towards New Fluorophores for Biomolecules Labelling.
    ChemSusChem, 2021, Apr-22, Volume: 14, Issue:8

    Topics: Anisoles; Benzofurans; Catalysis; Cycloaddition Reaction; Fluorescent Dyes; Heterocyclic Compounds; Hydrocarbons, Aromatic; Immunoglobulin G; Indoles; Molecular Structure; Optical Imaging; Pyrones; Pyrroles; Serum Albumin, Bovine; Solvents

2021
Total Synthesis of the Natural Chalcone Lophirone E, Synthetic Studies toward Benzofuran and Indole-Based Analogues, and Investigation of Anti-Leishmanial Activity.
    Molecules (Basel, Switzerland), 2022, Jan-11, Volume: 27, Issue:2

    Topics: Antiparasitic Agents; Benzofurans; Biflavonoids; Chalcones; Chemical Phenomena; Chemistry Techniques, Synthetic; Humans; Indoles; Leishmania infantum; Molecular Structure; Structure-Activity Relationship

2022