Page last updated: 2024-08-21

indazoles and tropisetron

indazoles has been researched along with tropisetron in 21 studies

Research

Studies (21)

TimeframeStudies, this research(%)All Research%
pre-19902 (9.52)18.7374
1990's15 (71.43)18.2507
2000's2 (9.52)29.6817
2010's2 (9.52)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andrews, PL; Bhandari, P1
Higgins, GA; Jones, BJ; Oakley, NR; Tyers, MB1
de Mulder, PH; Seynaeve, C; Verweij, J1
Gamse, R; Humpel, C; Javorsky, F; Saria, A2
Itoh, Z; Iwanaga, Y; Mizumoto, A; Yoshida, N1
Gandara, DR; Hesketh, PJ1
Costall, B; Domeney, AM; Naylor, RJ1
Cutler, MG1
Moss, HE; Sanger, GJ1
Brown, GW; Butcher, ME; Kidgell, AE1
Chen, HI1
Ashby, CR; Edwards, E; Harkins, K; Wang, RY1
Ito, A; Ito, T; Iwanaga, H; Karasawa, T; Mizumoto, A; Yoshida, N1
Harris, RA; Klein, RL; McQuilkin, SJ; Sanna, E; Whiting, PJ1
Grahame-Smith, DG; Leslie, RA; Pei, Q; Zetterström, T1
Barrett, JE; Critchett, D; Hu, W; Sokol, PT; Solomon, AJ; Toral, J; Ziai, MR1
Castro, G; Hilburn, C; King, GR; Konen, J; Pinto, G; Tran, S1
Berry, N; McBride, WJ; McKinzie, DL; Melendez, RI; Murphy, JM; Rodd-Henricks, ZA1
Asano, H; Funakami, Y; Ichida, S; Imanishi, T; Matsushima, K; Wada, T1
Bell, RL; Ding, ZM; Hauser, SR; McBride, WJ; Oster, SM; Rodd, ZA; Toalston, JE1

Reviews

2 review(s) available for indazoles and tropisetron

ArticleYear
5-HT3 receptor antagonists, a new approach in emesis: a review of ondansetron, granisetron and tropisetron.
    Anti-cancer drugs, 1991, Volume: 2, Issue:4

    Topics: Animals; Antiemetics; Granisetron; Humans; Imidazoles; Indazoles; Indoles; Ondansetron; Serotonin Antagonists; Tropisetron; Vomiting

1991
Antiemetic control: 5-HT3 antagonists: review of clinical results, with particular emphasis on ondansetron.
    Cancer treatment reviews, 1990, Volume: 17, Issue:2-3

    Topics: Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Cisplatin; Granisetron; Headache; Humans; Imidazoles; Indazoles; Indoles; Nausea; Ondansetron; Radiation Injuries; Radiotherapy; Serotonin Antagonists; Tropisetron; Vomiting

1990

Other Studies

19 other study(ies) available for indazoles and tropisetron

ArticleYear
Preliminary evidence for the involvement of the putative 5-HT4 receptor in zacopride- and copper sulphate-induced vomiting in the ferret.
    European journal of pharmacology, 1991, Nov-12, Volume: 204, Issue:3

    Topics: Analysis of Variance; Animals; Antiemetics; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Copper; Copper Sulfate; Female; Ferrets; Granisetron; Imidazoles; Indazoles; Indoles; Loperamide; Male; Ondansetron; Receptors, Serotonin; Serotonin Antagonists; Tropisetron; Vomiting

1991
Evidence that the amygdala is involved in the disinhibitory effects of 5-HT3 receptor antagonists.
    Psychopharmacology, 1991, Volume: 104, Issue:4

    Topics: Amygdala; Animals; Anxiety; Conflict, Psychological; Granisetron; Imidazoles; Indazoles; Indoles; Lighting; Male; Ondansetron; Raphe Nuclei; Rats; Serotonin; Serotonin Antagonists; Social Behavior; Tropanes; Tropisetron

1991
5-HT3 receptor antagonists inhibit sensory neuropeptide release from the rat spinal cord.
    Neuroreport, 1990, Volume: 1, Issue:2

    Topics: Animals; Calcitonin Gene-Related Peptide; Granisetron; In Vitro Techniques; Indazoles; Indoles; Neurokinin A; Neurons, Afferent; Neuropeptides; Potassium; Rats; Rats, Inbred Strains; Serotonin Antagonists; Spinal Cord; Substance P; Tropisetron

1990
Endogenous 5-hydroxytryptamine modulates the release of tachykinins and calcitonin gene-related peptide from the rat spinal cord via 5-HT3 receptors.
    Annals of the New York Academy of Sciences, 1991, Volume: 632

    Topics: Animals; Calcitonin Gene-Related Peptide; Granisetron; In Vitro Techniques; Indazoles; Indoles; Neurokinin A; Potassium Chloride; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spinal Cord; Substance P; Tachykinins; Tropisetron

1991
Effects of 5-hydroxytryptamine 3 receptor antagonists on gastrointestinal motor activity in conscious dogs.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 256, Issue:1

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Digestion; Dogs; Dose-Response Relationship, Drug; Female; Gastrointestinal Motility; Granisetron; Imidazoles; Indazoles; Indoles; Infusions, Intravenous; Injections, Intravenous; Male; Motilin; Motor Activity; Muscle Contraction; Muscle, Smooth; Ondansetron; Serotonin Antagonists; Time Factors; Tropisetron

1991
Serotonin antagonists: a new class of antiemetic agents.
    Journal of the National Cancer Institute, 1991, May-01, Volume: 83, Issue:9

    Topics: Antiemetics; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Granisetron; Humans; Imidazoles; Indazoles; Indoles; Metoclopramide; Ondansetron; Quinolizines; Receptors, Serotonin; Serotonin Antagonists; Tropanes; Tropisetron; Vomiting

1991
5-HT3 receptor antagonists attenuate dopamine-induced hyperactivity in the rat.
    Neuroreport, 1990, Volume: 1, Issue:1

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Dopamine; Dopamine Antagonists; Female; Granisetron; Indazoles; Indoles; Injections; Motor Activity; Nucleus Accumbens; Rats; Rats, Inbred Strains; Serotonin Antagonists; Tropisetron

1990
Behavioural effects in gerbils of the 5-HT3 receptor antagonists, BRL 43694 and ICS 205-930, under circumstances of high and low light intensity.
    Neuropharmacology, 1990, Volume: 29, Issue:6

    Topics: Animals; Behavior, Animal; Gerbillinae; Granisetron; Indazoles; Indoles; Light; Male; Pyrazoles; Serotonin Antagonists; Social Behavior; Tropisetron

1990
The effects of granisetron, ICS 205-930 and ondansetron on the visceral pain reflex induced by duodenal distension.
    British journal of pharmacology, 1990, Volume: 100, Issue:3

    Topics: Animals; Blood Pressure; Duodenum; Granisetron; Imidazoles; Indazoles; Indoles; Male; Morphine; Muscle Contraction; Muscle, Smooth; Ondansetron; Pain; Pyrazoles; Rats; Rats, Inbred Strains; Reflex; Serotonin Antagonists; Stomach; Tropisetron; Vagotomy

1990
Evidence for the presynaptic action of 5-hydroxytryptamine and the involvement of purinergic innervation in the rabbit lower urinary tract.
    British journal of pharmacology, 1990, Volume: 101, Issue:1

    Topics: Adenosine Triphosphate; Animals; Atropine; Electric Stimulation; Female; Granisetron; In Vitro Techniques; Indazoles; Indoles; Male; Muscle Contraction; Muscle, Smooth; Purines; Rabbits; Serotonin; Serotonin Antagonists; Synapses; Tropanes; Tropisetron; Urethra; Urinary Tract

1990
Characterization of 5-hydroxytryptamine3 receptors in the medial prefrontal cortex: a microiontophoretic study.
    European journal of pharmacology, 1989, Dec-07, Volume: 173, Issue:2-3

    Topics: Animals; Cerebral Cortex; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Granisetron; Indazoles; Indoles; Iontophoresis; Magnesium Chloride; Male; Metergoline; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropisetron

1989
[Effect of 5-HT3 receptor antagonists on gastrointestinal motility].
    Nihon Heikatsukin Gakkai zasshi, 1989, Volume: 25, Issue:6

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Dogs; Gastrointestinal Motility; Granisetron; Imidazoles; In Vitro Techniques; Indazoles; Indoles; Motilin; Ondansetron; Rabbits; Serotonin Antagonists; Tropisetron

1989
Effects of 5-HT3 receptor antagonists on binding and function of mouse and human GABAA receptors.
    European journal of pharmacology, 1994, Jul-15, Volume: 268, Issue:2

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Flumazenil; Flunitrazepam; Humans; Indazoles; Indoles; Male; Mice; Mice, Inbred ICR; Receptors, GABA-A; Serotonin Antagonists; Tropanes; Tropisetron; Xenopus laevis

1994
5-HT3 receptor antagonists inhibit morphine-induced stimulation of mesolimbic dopamine release and function in the rat.
    European journal of pharmacology, 1993, Jan-05, Volume: 230, Issue:1

    Topics: Animals; Behavior, Animal; Dialysis; Dopamine; Dose-Response Relationship, Drug; Granisetron; Indazoles; Indoles; Limbic System; Male; Morphine; Ondansetron; Rats; Rats, Sprague-Dawley; Serotonin Antagonists; Tropisetron

1993
5-HT3 receptor-independent inhibition of the depolarization-induced 86Rb efflux from human neuroblastoma cells, TE671, by ondansetron.
    The Journal of pharmacy and pharmacology, 1995, Volume: 47, Issue:7

    Topics: Anti-Anxiety Agents; Benzamides; Benzofurans; Biguanides; Bridged Bicyclo Compounds, Heterocyclic; Humans; Hypoglycemic Agents; Indazoles; Indoles; Neuroblastoma; Neurotoxins; Ondansetron; Potassium Channels; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Rubidium Radioisotopes; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship; Tropanes; Tropisetron; Tumor Cells, Cultured

1995
The effects of continuous 5-HT(3) receptor antagonist administration on the subsequent behavioral response to cocaine.
    European journal of pharmacology, 2002, Aug-09, Volume: 449, Issue:3

    Topics: Animals; Behavior, Animal; Cocaine; Dose-Response Relationship, Drug; Down-Regulation; Indazoles; Indoles; Infusion Pumps; Male; Motor Activity; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Stereotyped Behavior; Substance Withdrawal Syndrome; Tropanes; Tropisetron

2002
Effects of serotonin-3 receptor antagonists on the intracranial self-administration of ethanol within the ventral tegmental area of Wistar rats.
    Psychopharmacology, 2003, Volume: 165, Issue:3

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Central Nervous System Depressants; Drug Interactions; Ethanol; Female; Indazoles; Indoles; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Self Administration; Serotonin Antagonists; Stereoisomerism; Tropanes; Tropisetron; Ventral Tegmental Area

2003
Changes in characteristics of the specific binding of [3H]LY-278584, a 5-HT3-receptor antagonist, on differentiated NG108-15 cells.
    Journal of pharmacological sciences, 2010, Volume: 113, Issue:3

    Topics: Animals; Binding, Competitive; Bucladesine; Cell Differentiation; Hybrid Cells; Indazoles; Indoles; Kinetics; Mice; Nerve Tissue Proteins; Neurons; Rats; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin 5-HT3 Receptor Antagonists; Serotonin Antagonists; Tropanes; Tropisetron; Up-Regulation

2010
Synergistic self-administration of ethanol and cocaine directly into the posterior ventral tegmental area: involvement of serotonin-3 receptors.
    The Journal of pharmacology and experimental therapeutics, 2012, Volume: 340, Issue:1

    Topics: Analysis of Variance; Animals; Anti-Arrhythmia Agents; Central Nervous System Depressants; Cocaine; Conditioning, Operant; Drug Synergism; Ethanol; Female; Indazoles; Indoles; Microinjections; Rats; Rats, Wistar; Receptors, Serotonin, 5-HT3; Self Administration; Serotonin 5-HT3 Receptor Agonists; Serotonin 5-HT3 Receptor Antagonists; Stereotaxic Techniques; Tropanes; Tropisetron; Ventral Tegmental Area

2012