Page last updated: 2024-08-21

indazoles and pyrimidine

indazoles has been researched along with pyrimidine in 3 studies

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (66.67)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kumar, KP; Lingaiah, BP; Murthy, US; Narsaiah, B; Yakaiah, T1
Behm, DJ; Bentley, R; Doe, CP; Dowdell, SE; Dul, E; Elkins, PA; Evans, C; Goodman, KB; Hu, E; Jolivette, LJ; Khandekar, SS; Kirkpatrick, RB; Lee, D; Sehon, CA; Semus, SF; Smith, GK; Viet, AQ; Wang, GZ; Wright, LL; Yi, T1
Kim, D; Kwon, A; Lee, BY; Min, KH; Nguyen, HK; Song, J; Suh, W; Yoo, J1

Other Studies

3 other study(ies) available for indazoles and pyrimidine

ArticleYear
GdCl(3) catalysed Grieco condensation: a facile approach for the synthesis of novel pyrimidine and annulated pyrimidine fused indazole derivatives in single pot under mild conditions and their anti-microbial activity.
    European journal of medicinal chemistry, 2008, Volume: 43, Issue:2

    Topics: Anti-Bacterial Agents; Antifungal Agents; Catalysis; Gadolinium; Indazoles; Magnetic Resonance Spectroscopy; Mass Spectrometry; Microbial Sensitivity Tests; Pyrimidines

2008
Potent, selective and orally bioavailable dihydropyrimidine inhibitors of Rho kinase (ROCK1) as potential therapeutic agents for cardiovascular diseases.
    Journal of medicinal chemistry, 2008, Nov-13, Volume: 51, Issue:21

    Topics: Adenosine Triphosphate; Administration, Oral; Aldehydes; Animals; Cardiovascular Diseases; Crystallography, X-Ray; Indazoles; Models, Molecular; Molecular Structure; Protein Kinase Inhibitors; Pyrimidines; Rats; rho-Associated Kinases; Structure-Activity Relationship

2008
Structure-Activity Relationship of Indole-Tethered Pyrimidine Derivatives that Concurrently Inhibit Epidermal Growth Factor Receptor and Other Angiokinases.
    PloS one, 2015, Volume: 10, Issue:9

    Topics: Angiogenesis Inhibitors; Carcinoma, Non-Small-Cell Lung; Cell Proliferation; ErbB Receptors; Human Umbilical Vein Endothelial Cells; Humans; Indazoles; Indoles; Inhibitory Concentration 50; Lung Neoplasms; Molecular Docking Simulation; Neovascularization, Pathologic; Protein Kinase Inhibitors; Protein Kinases; Pyrimidines; Structure-Activity Relationship; Sulfonamides; Vascular Endothelial Growth Factor A

2015