Page last updated: 2024-08-21

indazoles and imidazole

indazoles has been researched along with imidazole in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (28.57)18.2507
2000's2 (28.57)29.6817
2010's3 (42.86)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lubeskie, A; Umansky, S; Wolff, DJ1
Ko, FN; Kuo, SC; Lee, FY; Teng, CM; Wu, CC1
Kitagawa, T; Li, Z; Ohta, T; Pal, B; Takenaka, S; Tsuyama, S1
Arion, VB; Eichinger, A; Guedes da Silva, MF; Keppler, BK; Kukushkin, VY; Lichtenecker, R; Pombeiro, AJ; Reisner, E1
Bylina, D; Czeczuk, A; Dziecioł, J; Grześk, E; Grześk, G; Krzyzanowski, M; Malinowski, B; Michalska, A; Sinjab, AT; Szadujkis-Szadurska, K; Wiciński, M1
Carey, LM; Franzen, S; Ghiladi, RA; Hough, MA; McCombs, NL; Moreno-Chicano, T1
Bearss, DJ; Bearss, J; Call, L; Carpenter, K; Chen, T; Choi, S; Sharma, S; Sorna, V; Vankayalapati, H; Warner, SL1

Other Studies

7 other study(ies) available for indazoles and imidazole

ArticleYear
The inhibition of the constitutive bovine endothelial nitric oxide synthase by imidazole and indazole agents.
    Archives of biochemistry and biophysics, 1994, Nov-01, Volume: 314, Issue:2

    Topics: Amino Acid Oxidoreductases; Animals; Brain; Cattle; Citrulline; Endothelium, Vascular; Imidazoles; Indazoles; Isoenzymes; Kinetics; Macrophages; Nitric Oxide Synthase; Pulmonary Artery

1994
YC-1, a novel activator of platelet guanylate cyclase.
    Blood, 1994, Dec-15, Volume: 84, Issue:12

    Topics: 1-Methyl-3-isobutylxanthine; Adenosine Triphosphate; Alprostadil; Animals; Bleeding Time; Blood Platelets; Calcium; Colforsin; Collagen; Cyclic AMP; Cyclic GMP; Drug Interactions; Enzyme Activation; Guanylate Cyclase; Imidazoles; Indazoles; Indomethacin; Methemoglobin; Mice; Molecular Structure; Nitroprusside; Phosphoric Diester Hydrolases; Platelet Aggregation Inhibitors; Prostaglandin D2; Rabbits; Superoxide Dismutase; Thromboxane A2

1994
Resonance Raman study on synergistic activation of soluble guanylate cyclase by imidazole, YC-1 and GTP.
    Journal of inorganic biochemistry, 2004, Volume: 98, Issue:5

    Topics: Animals; Cattle; Drug Synergism; Enzyme Activation; Guanosine Triphosphate; Guanylate Cyclase; Heme; Imidazoles; In Vitro Techniques; Indazoles; Solubility; Spectrum Analysis, Raman

2004
Tuning of redox potentials for the design of ruthenium anticancer drugs -- an electrochemical study of [trans-RuCl(4)L(DMSO)](-) and [trans-RuCl(4)L(2)](-) complexes, where L = imidazole, 1,2,4-triazole, indazole.
    Inorganic chemistry, 2004, Nov-01, Volume: 43, Issue:22

    Topics: Antineoplastic Agents; Dimethyl Sulfoxide; Drug Design; Electrochemistry; Imidazoles; Indazoles; Molecular Conformation; Molecular Structure; Organometallic Compounds; Oxidation-Reduction; Ruthenium; Stereoisomerism; Triazoles

2004
Imidazole-induced contractility of vascular smooth muscle cells in the presence of U-73122, ODQ, indomethacin and 7-nitroindazole.
    Polish journal of veterinary sciences, 2013, Volume: 16, Issue:2

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Enzyme Inhibitors; Estrenes; Guanylate Cyclase; Imidazoles; Indazoles; Indomethacin; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Oxadiazoles; Phosphodiesterase Inhibitors; Pyrrolidinones; Rats; Receptors, Cytoplasmic and Nuclear; Soluble Guanylyl Cyclase; Vasoconstriction

2013
Interaction of Azole-Based Environmental Pollutants with the Coelomic Hemoglobin from Amphitrite ornata: A Molecular Basis for Toxicity.
    Biochemistry, 2017, 05-02, Volume: 56, Issue:17

    Topics: Amino Acid Motifs; Animals; Benzimidazoles; Catalytic Domain; Computational Biology; Environmental Pollutants; Enzyme Inhibitors; Fungicides, Industrial; Hemoglobins; Hydrogen Bonding; Hydrophobic and Hydrophilic Interactions; Imidazoles; Indazoles; Isoenzymes; Kinetics; Ligands; Models, Molecular; Peroxidases; Pesticides; Polychaeta; Recombinant Fusion Proteins; Recombinant Proteins; Triazoles

2017
Fragment-based design, synthesis, biological evaluation, and SAR of 1H-benzo[d]imidazol-2-yl)-1H-indazol derivatives as potent PDK1 inhibitors.
    Bioorganic & medicinal chemistry letters, 2017, 12-15, Volume: 27, Issue:24

    Topics: Apoptosis; Binding Sites; Cell Line, Tumor; Down-Regulation; Drug Design; Dual Specificity Phosphatase 6; Dual-Specificity Phosphatases; Humans; Imidazoles; Indazoles; Inhibitory Concentration 50; Mitogen-Activated Protein Kinase Phosphatases; Molecular Docking Simulation; Phosphorylation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins c-akt; PTEN Phosphohydrolase; Pyruvate Dehydrogenase Acetyl-Transferring Kinase; Ribosomal Protein S6 Kinases, 70-kDa; RNA Interference; RNA, Small Interfering; Structure-Activity Relationship

2017