Page last updated: 2024-08-21

indazoles and gsk2292767

indazoles has been researched along with gsk2292767 in 2 studies

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Amour, A; Baldwin, IR; Cooper, AW; Deakin, AM; Down, K; Felton, LM; Guntrip, SB; Hamblin, JN; Hardy, C; Harrison, ZA; Jones, KL; Jones, P; Keeling, SE; Le, J; Livia, S; Lucas, F; Lunniss, CJ; Parr, NJ; Robinson, E; Rowland, P; Smith, S; Thomas, DA; Vitulli, G; Washio, Y1
Begg, M; Cahn, A; Clark, J; Edwards, CD; Ehtesham, F; Fernando, D; Gilbert, J; Hamblin, JN; Harrell, A; Hessel, EM; Hingle, MI; Mallett, D; Marotti, M; Morrell, J; Newman, CF; Pefani, E; Uddin, S; Vitulli, G; Wilson, R1

Trials

1 trial(s) available for indazoles and gsk2292767

ArticleYear
Translation of Inhaled Drug Optimization Strategies into Clinical Pharmacokinetics and Pharmacodynamics Using GSK2292767A, a Novel Inhaled Phosphoinositide 3-Kinase
    The Journal of pharmacology and experimental therapeutics, 2019, Volume: 369, Issue:3

    Topics: Administration, Inhalation; Adult; Animals; Bronchoalveolar Lavage; Eosinophilia; Female; Humans; Indazoles; Lung; Male; Mice; Middle Aged; Permeability; Phosphoinositide-3 Kinase Inhibitors; Safety; Solubility; Sputum; Sulfonamides; Translational Research, Biomedical

2019

Other Studies

1 other study(ies) available for indazoles and gsk2292767

ArticleYear
Optimization of Novel Indazoles as Highly Potent and Selective Inhibitors of Phosphoinositide 3-Kinase δ for the Treatment of Respiratory Disease.
    Journal of medicinal chemistry, 2015, Sep-24, Volume: 58, Issue:18

    Topics: Administration, Inhalation; Animals; Asthma; Female; Humans; Indazoles; Indoles; Isoenzymes; Male; Microsomes; Molecular Docking Simulation; Ovalbumin; Oxazoles; Phosphoinositide-3 Kinase Inhibitors; Piperazines; Pneumonia; Pulmonary Disease, Chronic Obstructive; Rabbits; Rats; Rats, Sprague-Dawley; Respiratory Tract Diseases; Stereoisomerism; Structure-Activity Relationship; Sulfonamides; Th2 Cells

2015