indazoles has been researched along with gamendazole in 9 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 2 (22.22) | 29.6817 |
| 2010's | 4 (44.44) | 24.3611 |
| 2020's | 3 (33.33) | 2.80 |
| Authors | Studies |
|---|---|
| Blagg, BS; Chakrasali, R; Georg, GI; Hadden, MK; Heckert, LL; Hornbaker, K; Hughes, J; Jakkaraj, SR; Kinzy, TG; Ozturk, SB; Smith, SK; Tash, JS | 1 |
| Attardi, B; Chakrasali, R; Georg, GI; Hild, SA; Jakkaraj, SR; Tash, JS | 1 |
| Cheng, CY; Lie, PP; Lui, WY; Mok, KW; Mruk, DD | 1 |
| Amory, JK; Nya-Ngatchou, JJ | 1 |
| Bousmina, M; El Kazzouli, S; Essassi, el M; Guillaumet, G; Naas, M | 1 |
| Burglová, K; Dzubak, P; Hajduch, M; Hlavac, J; Hradil, P; Markos, A; Medvedikova, M; Petracek, M; Prichystalova, H; Rylová, G; Sopko, B; Soural, M; Tejral, G | 1 |
| Cherrington, NJ; Georg, GI; Hau, RK; Tash, JS; Wright, SH | 1 |
| Calvet, JP; Georg, GI; Jakkaraj, SR; Li, X; Magenheimer, BS; Reif, GA; Sundar, SV; Tash, JS; Wallace, DP; Yu, ASL; Zhou, JX | 1 |
| Golemis, EA; Pirestani, S | 1 |
2 review(s) available for indazoles and gamendazole
| Article | Year |
|---|---|
Adjudin, a potential male contraceptive, exerts its effects locally in the seminiferous epithelium of mammalian testes.
Topics: Animals; Cell Adhesion; Contraceptive Agents, Male; Humans; Hydrazines; Indazoles; Indenes; Male; Piperidines; Seminiferous Epithelium; Sertoli Cells; Spermatogenesis; Spermatozoa | 2011 |
New approaches to male non-hormonal contraception.
Topics: Animals; Contraception; Contraceptive Agents, Male; Diamines; Humans; Hydrazines; Indazoles; Male; Retinoids; Tretinoin | 2013 |
7 other study(ies) available for indazoles and gamendazole
| Article | Year |
|---|---|
Gamendazole, an orally active indazole carboxylic acid male contraceptive agent, targets HSP90AB1 (HSP90BETA) and EEF1A1 (eEF1A), and stimulates Il1a transcription in rat Sertoli cells.
Topics: Administration, Oral; Amino Acid Sequence; Animals; Binding Sites; Cell Line; Cell Line, Tumor; Female; HSP90 Heat-Shock Proteins; Indazoles; Interleukin-1alpha; Male; Models, Biological; Molecular Sequence Data; Ovarian Neoplasms; Peptide Elongation Factor 1; Rats; Sertoli Cells; Spermatogenesis-Blocking Agents; Testis; Transcription, Genetic | 2008 |
A novel potent indazole carboxylic acid derivative blocks spermatogenesis and is contraceptive in rats after a single oral dose.
Topics: Administration, Oral; Animals; Body Weight; Female; Fertility; Follicle Stimulating Hormone; Genitalia, Male; Hydrazines; Indazoles; Inhibins; Male; Organ Size; Pregnancy; Rats; Rats, Long-Evans; Spermatogenesis; Spermatogenesis-Blocking Agents; Testis; Time Factors | 2008 |
Palladium-Catalyzed Oxidative Direct C3- and C7-Alkenylations of Indazoles: Application to the Synthesis of Gamendazole.
Topics: Alkenes; Catalysis; Indazoles; Molecular Structure; Oxidants; Oxidation-Reduction; Palladium; Stereoisomerism | 2015 |
Identification of Eukaryotic Translation Elongation Factor 1-α 1 Gamendazole-Binding Site for Binding of 3-Hydroxy-4(1 H)-quinolinones as Novel Ligands with Anticancer Activity.
Topics: Antineoplastic Agents; Binding Sites; Cell Line, Tumor; Computational Biology; Humans; Indazoles; Ligands; Models, Molecular; Molecular Conformation; Peptide Elongation Factor 1; Quinolones; Structure-Activity Relationship | 2018 |
Physiological Characterization of the Transporter-Mediated Uptake of the Reversible Male Contraceptive H2-Gamendazole Across the Blood-Testis Barrier.
Topics: Animals; Blood-Testis Barrier; Carboxylic Acids; CHO Cells; Chromatography, Liquid; Contraceptive Agents, Male; Cricetinae; Cricetulus; Dogs; Female; HEK293 Cells; Humans; Indazoles; Male; Membrane Transport Proteins; Organic Anion Transporters; Tandem Mass Spectrometry | 2022 |
The lonidamine derivative H2-gamendazole reduces cyst formation in polycystic kidney disease.
Topics: Actins; Animals; Carboxylic Acids; Cell Proliferation; Cells, Cultured; Colforsin; Cyclin-Dependent Kinase 4; Cystic Fibrosis Transmembrane Conductance Regulator; Cysts; EGF Family of Proteins; Heat-Shock Proteins; Humans; Indazoles; Kidney; Mice; Polycystic Kidney Diseases; Polycystic Kidney, Autosomal Dominant; Proto-Oncogene Proteins c-akt; Receptors, Cell Surface | 2022 |
H2-gamendazole: a new therapeutic lead for the treatment of polycystic kidney disease.
Topics: Humans; Indazoles; Polycystic Kidney Diseases; Polycystic Kidney, Autosomal Dominant | 2022 |