Page last updated: 2024-08-21

indazoles and danusertib

indazoles has been researched along with danusertib in 3 studies

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (33.33)24.3611
2020's2 (66.67)2.80

Authors

AuthorsStudies
Coumar, MS; Sarvagalla, S1
Khan, T; Prabhu, A; Sankhe, K1
He, X; Ji, X; Jiang, C; Shen, Z; Yin, L; Zhou, H; Zhu, X1

Reviews

2 review(s) available for indazoles and danusertib

ArticleYear
Structural Biology Insight for the Design of Sub-type Selective Aurora Kinase Inhibitors.
    Current cancer drug targets, 2015, Volume: 15, Issue:5

    Topics: Animals; Aurora Kinase A; Aurora Kinase B; Aurora Kinases; Benzamides; Binding Sites; Humans; Indazoles; Piperazines; Protein Kinase Inhibitors; Protein Structure, Secondary; Pyrazoles

2015
Design strategies, SAR, and mechanistic insight of Aurora kinase inhibitors in cancer.
    Chemical biology & drug design, 2021, Volume: 98, Issue:1

    Topics: Animals; Antineoplastic Agents; Aurora Kinase A; Azepines; Benzamides; Drug Approval; Drug Resistance; Drug Screening Assays, Antitumor; Flavones; Gene Expression Regulation; Humans; Indazoles; Neoplasms; Organophosphates; Protein Binding; Protein Conformation; Protein Kinase Inhibitors; Pyrazoles; Pyrimidines; Quinazolines; Structure-Activity Relationship

2021

Other Studies

1 other study(ies) available for indazoles and danusertib

ArticleYear
Combined inhibition of AURKA and HSF1 suppresses proliferation and promotes apoptosis in hepatocellular carcinoma by activating endoplasmic reticulum stress.
    Cellular oncology (Dordrecht), 2021, Volume: 44, Issue:5

    Topics: Aminopyridines; Animals; Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Aurora Kinase A; Benzamides; Carcinoma, Hepatocellular; Cell Line, Tumor; Cell Proliferation; Endoplasmic Reticulum Stress; Female; Gene Expression Regulation, Neoplastic; Heat Shock Transcription Factors; Hep G2 Cells; Humans; Indazoles; Kaplan-Meier Estimate; Liver Neoplasms; Mice, Inbred BALB C; Mice, Nude; Pyrazoles; RNA Interference; Xenograft Model Antitumor Assays

2021