Page last updated: 2024-08-21

indazoles and colchicine

indazoles has been researched along with colchicine in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19901 (12.50)18.7374
1990's0 (0.00)18.2507
2000's2 (25.00)29.6817
2010's2 (25.00)24.3611
2020's3 (37.50)2.80

Authors

AuthorsStudies
Hiramoto, RN; Miller, ML; Samuelson, CO; Soong, SJ; Ward, JR1
Cai, X; Duan, JX; Hart, C; Lan, L; Matteucci, M; Meng, F1
Fayne, D; Flood, CT; Golfis, G; Knox, AJ; Lloyd, DG; Meegan, MJ; Pawlak, M; Price, T; Williams, DC1
Füessl, HS; Stiefelhagen, P1
Bharatham, N; Chattopadhaya, S; Choi, BH; Feng, L; Harikishore, A; Lim, CB; Liu, X; Nanga, RP; Nguyen, QT; Thanh, le N; Yoon, HS; Zhao, Y1
Cui, YJ; Liu, ZP; Ma, CC; Tang, LQ; Zhang, CM1
Balasaheb Nimse, S; Dashrath Warkad, S; Pal, D; Saha, S; Seong Yeom, G; Shinde, PB; Song, IH; Song, KS1
Cui, YJ; Dou, BK; Ma, CC; Zhang, J; Zhang, XW; Zhou, Y1

Reviews

1 review(s) available for indazoles and colchicine

ArticleYear
Indazole-based microtubule-targeting agents as potential candidates for anticancer drugs discovery.
    Bioorganic chemistry, 2022, Volume: 122

    Topics: Antineoplastic Agents; Binding Sites; Cell Line, Tumor; Cell Proliferation; Colchicine; Indazoles; Microtubules; Tubulin; Tubulin Modulators

2022

Other Studies

7 other study(ies) available for indazoles and colchicine

ArticleYear
Acute colchicine and vinblastine toxicity in 6-sulfanilamidoindazole-pretreated rats.
    Toxicology and applied pharmacology, 1981, Sep-30, Volume: 60, Issue:3

    Topics: Aging; Animals; Colchicine; Indazoles; Kidney; Lethal Dose 50; Male; Phenylbutazone; Rats; Rats, Inbred Strains; Shwartzman Phenomenon; Sulfanilamides; Sulfonamides; Vinblastine

1981
Potent antitubulin tumor cell cytotoxins based on 3-aroyl indazoles.
    Journal of medicinal chemistry, 2007, Mar-08, Volume: 50, Issue:5

    Topics: Acetylene; Animals; Binding Sites; Binding, Competitive; Cattle; Cell Line, Tumor; Colchicine; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Humans; Indazoles; Radioligand Assay; Stilbenes; Structure-Activity Relationship; Tubulin; Tubulin Modulators

2007
Integration of ligand and structure-based virtual screening for the identification of the first dual targeting agent for heat shock protein 90 (Hsp90) and tubulin.
    Journal of medicinal chemistry, 2009, Apr-23, Volume: 52, Issue:8

    Topics: Adenosine Triphosphate; Antineoplastic Agents; Binding Sites; Biopolymers; Cell Line, Tumor; Colchicine; Databases, Factual; Estrogen Receptor alpha; HSP90 Heat-Shock Proteins; Humans; Imidazoles; Indazoles; Ligands; Models, Molecular; Principal Component Analysis; Protein Binding; Quantitative Structure-Activity Relationship; Tubulin; Tubulin Modulators

2009
[Frequent gout attacks during therapy - what can be done?].
    MMW Fortschritte der Medizin, 2013, May-16, Volume: 155, Issue:9

    Topics: Angiogenesis Inhibitors; Carcinoma, Renal Cell; Colchicine; Drug Therapy, Combination; Gout; Gout Suppressants; Humans; Indazoles; Kidney Neoplasms; Male; Pyrimidines; Sulfonamides

2013
Suprafenacine, an indazole-hydrazide agent, targets cancer cells through microtubule destabilization.
    PloS one, 2014, Volume: 9, Issue:10

    Topics: Amino Acid Sequence; Animals; Antineoplastic Agents; Apoptosis; Binding Sites; Colchicine; G2 Phase Cell Cycle Checkpoints; HeLa Cells; Humans; Hydrazines; Indazoles; Membrane Potential, Mitochondrial; Mice; Microtubules; Molecular Sequence Data; PC12 Cells; Protein Binding; Rats; Small Molecule Libraries

2014
The discovery of novel indazole derivatives as tubulin colchicine site binding agents that displayed potent antitumor activity both in vitro and in vivo.
    European journal of medicinal chemistry, 2020, Feb-01, Volume: 187

    Topics: Animals; Antineoplastic Agents; Binding Sites; Cell Proliferation; Cells, Cultured; Colchicine; Dose-Response Relationship, Drug; Drug Discovery; Drug Screening Assays, Antitumor; Humans; Indazoles; Mice; Mice, Nude; Models, Molecular; Molecular Structure; Polymerization; Structure-Activity Relationship; Tubulin; Tubulin Modulators

2020
The discovery of water-soluble indazole derivatives as potent microtubule polymerization inhibitors.
    European journal of medicinal chemistry, 2023, Dec-15, Volume: 262

    Topics: Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Colchicine; Indazoles; Microtubules; Paclitaxel; Polymerization; Structure-Activity Relationship; Tubulin; Tubulin Modulators

2023