Page last updated: 2024-08-21

indazoles and bendazac lysine

indazoles has been researched along with bendazac lysine in 39 studies

Research

Studies (39)

TimeframeStudies, this research(%)All Research%
pre-199017 (43.59)18.7374
1990's17 (43.59)18.2507
2000's3 (7.69)29.6817
2010's2 (5.13)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chao, R; Gao, X; Ma, P; Wu, C1
Hockwin, O; Schmidt, J; Schmitt, C1
Campana, A; Caranti, S; D'Onofrio, E; Scorza Barcellona, P; Silvestrini, B1
Cedrone, C; Cerulli, L; Missiroli, A; Pocobelli, A; Ricci, F1
Blanksma, LJ; Kooijman, AC; Van den Brom, HJ1
Cupak, K; Kosanović, M1
Balfour, JA; Clissold, SP1
Baraldi, P; Benassi, B; Bocca, E; Fonda, S; Luppi, ML; Mazza, C; Penne, A; Toschi, P1
Apponi-Battini, G; Costagliola, C; Iuliano, G; Menzione, M1
Elliott, DB; Gilchrist, J; Hurst, M; Pickwell, LD; Sheridan, M; Weatherill, J; Whitaker, D1
Carrieri, MP; De Gregorio, M; Hockwin, O; Laser, H1
Hofmann, H; Schmut, O1
Campistron, G; Ego, D; Escourrou, J; Houin, G; Ribet, A; Rovei, V; Thiola, A1
Choi, O; Jung, HR; Lee, J; Rhee, SW; Youn, DH1
Catanese, B; Martinelli, B; Palmery, M; Valeri, P1
Bonacini, M; Nuzzi, G; Sarzi-Amadé, R; Venturini, I1
Campistron, G; Conte, JJ; Dueymes, JM; Ego, D; Houin, G; Rovei, V1
Bono, A; Livrea, MA; Pandolfo, L1
Barillari, G; Catanese, B; Corradino, C; Picollo, R1
Catanese, B; Durando, L; Gismondi, A; Valeri, P1
Cioli, V; Corradino, C; Mazzanti, G; Silvestrini, B1
Guarino, V; Lampa, E; Marmo, E; Matera, MG; Romano, AR; Spadaro, R1
Barillari, G; Catanese, B; Iorio, E; Silvestrini, B; Valeri, P1
Barillari, G; Catanese, B; Galli Angeli, D; Iorio, E1
Barillari, G; Catanese, B; Iorio, E; Silvestrini, B1
Benitez del Castillo, JM; Castillo, A; Diaz, D; Garcia-Sanchez, J; Jimenez-Alfaro, I; Ortega, P; Toledano, N1
Evans, TC; Levy, B; Szabocsik, J1
Marques, C; Mota, MC; Pereira, P; Ramalho, JS1
Alcalde, M; Cebria, L; Donoso, MS; Garcia-Diaz, M; Najarro, F; Pascasio, JM1
Jung, WT; Park, WC; Rho, SH1
Arsenio, L; De Gregorio, M; Maraini, G; Nuzzi, G; Venturini, I1
Arciola, CR; Caramazza, R; Cavedagna, D; Montanaro, L; Sassoli, V1
Kidane, A; Park, K; Szabocsik, JM1
Chen, XX; Pu, J; Qiu, JJ; Shen, JP; Yan, HY; Zhang, YD; Zhu, YQ1
Bianchetti, C; Delfini, M; Di Cocco, ME; Pescosolido, N; Porcelli, F; Rosa, R; Rugo, G1
Jiang, SJ; Li, LM; Qiu, J; Shen, JP; Wu, HW; Yin, XX; Zhang, YD; Zheng, XG; Zhu, X1
Jiang, SJ; Qiu, J; Shen, JP; Yin, HL; Yin, XX; Yu, JX1
Chen, X; Gou, S; Shen, H; Shen, J; Zhang, Y; Zhu, Y1
Chen, J; Cheng, Q; He, J; Hong, L; Luo, L; Yang, W; Zhu, P1

Reviews

1 review(s) available for indazoles and bendazac lysine

ArticleYear
Bendazac lysine. A review of its pharmacological properties and therapeutic potential in the management of cataracts.
    Drugs, 1990, Volume: 39, Issue:4

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Cataract; Humans; Indazoles; Pyrazoles; Rabbits

1990

Trials

5 trial(s) available for indazoles and bendazac lysine

ArticleYear
Clinical and physical measurements of the cataractous lens.
    Documenta ophthalmologica. Advances in ophthalmology, 1990, Volume: 75, Issue:3-4

    Topics: Aged; Aged, 80 and over; Cataract; Contrast Sensitivity; Female; Humans; Indazoles; Lens, Crystalline; Light; Male; Middle Aged; Photography; Scattering, Radiation; Visual Acuity

1990
Bendazac lysine in selected types of human senile cataract. A long-term double-masked placebo-controlled clinical trial with multilinear densitometric image analysis of Scheimpflug photographs.
    Ophthalmic research, 1989, Volume: 21, Issue:3

    Topics: Adult; Aged; Cataract; Clinical Trials as Topic; Densitometry; Drug Administration Schedule; Female; Humans; Image Processing, Computer-Assisted; Indazoles; Lens Capsule, Crystalline; Lens Cortex, Crystalline; Lens Nucleus, Crystalline; Male; Middle Aged; Photography; Pyrazoles; Random Allocation; Time Factors

1989
The effects of Bendaline on cataracts.
    Korean journal of ophthalmology : KJO, 1987, Volume: 1, Issue:1

    Topics: Administration, Oral; Adult; Aged; Anti-Inflammatory Agents, Non-Steroidal; Cataract; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Indazoles; Male; Middle Aged; Pyrazoles; Random Allocation; Tablets; Visual Acuity

1987
Vitreous fluorophotometry and changes in blood-retinal barrier permeability induced by bendazac lysine.
    Acta ophthalmologica Scandinavica, 1997, Volume: 75, Issue:1

    Topics: Adult; Anti-Inflammatory Agents, Non-Steroidal; Blood-Retinal Barrier; Cell Membrane Permeability; Cross-Over Studies; Diabetes Mellitus, Type 1; Double-Blind Method; Female; Fluorescein; Fluoresceins; Fluorescent Dyes; Fluorophotometry; Follow-Up Studies; Humans; Indazoles; Male; Middle Aged; Sample Size; Vitreous Body

1997
Pharmacokinetics of bendazac lysine in 10 Chinese young men.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1997, Volume: 18, Issue:2

    Topics: Adult; Anti-Inflammatory Agents, Non-Steroidal; Area Under Curve; Biological Availability; Cross-Over Studies; Humans; Indazoles; Male; Therapeutic Equivalency

1997

Other Studies

33 other study(ies) available for indazoles and bendazac lysine

ArticleYear
[Determination of bendazac lysine by RP-HPLC].
    Hua xi yi ke da xue xue bao = Journal of West China University of Medical Sciences = Huaxi yike daxue xuebao, 1992, Volume: 23, Issue:2

    Topics: Chromatography, High Pressure Liquid; Indazoles

1992
Protein profiles after UV-B irradiation and bendazac lysine (bendalina) treatment.
    Developments in ophthalmology, 1991, Volume: 21

    Topics: Animals; Crystallins; Indazoles; Lens, Crystalline; Rats; Ultraviolet Rays

1991
Pretreatment with bendazac attenuates retinal damage induced by intense light in rats.
    Pharmacological research, 1991, Volume: 24, Issue:1

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Atrophy; Eye Injuries; Indazoles; Light; Male; Rats; Rats, Inbred Strains; Retina

1991
Use of bendazac lysine to limit protein deposition on soft contact lenses in vitro.
    The CLAO journal : official publication of the Contact Lens Association of Ophthalmologists, Inc, 1991, Volume: 17, Issue:2

    Topics: Anti-Inflammatory Agents, Non-Steroidal; Colorimetry; Contact Lenses, Hydrophilic; Indazoles; Muramidase; Protein Binding

1991
Contemporary possibilities of medicamentous prevention of cataract.
    Acta medica Iugoslavica, 1990, Volume: 44, Issue:4

    Topics: Adult; Aged; Aspartic Acid; Cataract; Drug Combinations; Female; Humans; Indazoles; Inosine Monophosphate; Male; Middle Aged; Niacinamide; Parabens; Thimerosal; Visual Acuity

1990
Medical treatment of senile cataract: clinical investigation of bendazac-lysine using objective and subjective methods.
    Graefe's archive for clinical and experimental ophthalmology = Albrecht von Graefes Archiv fur klinische und experimentelle Ophthalmologie, 1990, Volume: 228, Issue:2

    Topics: Aged; Aged, 80 and over; Aging; Cataract; Contrast Sensitivity; Densitometry; Female; Follow-Up Studies; Humans; Image Processing, Computer-Assisted; Indazoles; Interferometry; Lens, Crystalline; Light; Male; Middle Aged; Pyrazoles; Visual Acuity

1990
Inhibition of rat lens aldose reductase by bendazac-L-lysine salt.
    Enzyme, 1989, Volume: 42, Issue:4

    Topics: Aldehyde Reductase; Animals; Cataract; Indazoles; Kinetics; Lens, Crystalline; Pyrazoles; Rats; Sugar Alcohol Dehydrogenases

1989
The subjective assessment of cataract.
    Ophthalmic & physiological optics : the journal of the British College of Ophthalmic Opticians (Optometrists), 1989, Volume: 9, Issue:1

    Topics: Aged; Cataract; Contrast Sensitivity; Humans; Indazoles; Macular Degeneration; Refractive Errors; Scattering, Radiation; Sensory Thresholds; Visual Acuity

1989
Studies on the activity of Bendalina (bendazac L-lysine salt) as a scavenger of hydroxyl and superoxide radicals.
    Wiener klinische Wochenschrift, 1985, Nov-08, Volume: 97, Issue:21

    Topics: Ascorbic Acid; Cysteine; Free Radicals; Hyaluronic Acid; Indazoles; Pyrazoles; Superoxides; Viscosity

1985
The pharmacokinetics of bendazac-lysine and 5-hydroxybendazac, its main metabolite, in patients with hepatic cirrhosis.
    European journal of clinical pharmacology, 1988, Volume: 35, Issue:4

    Topics: Adult; Aged; Blood Proteins; Female; Humans; Indazoles; Liver Cirrhosis; Male; Middle Aged; Protein Binding; Pyrazoles

1988
Absorption of bendazac lysine after topical application to the rabbit eye.
    Pharmacological research communications, 1987, Volume: 19, Issue:8

    Topics: Absorption; Administration, Topical; Animals; Anti-Inflammatory Agents, Non-Steroidal; Eye; Indazoles; Male; Pyrazoles; Rabbits

1987
Improvement of the blood-retinal barrier induced by bendazac lysine: preliminary clinical observation in insulin-dependent diabetics.
    Archives of ophthalmology (Chicago, Ill. : 1960), 1987, Volume: 105, Issue:9

    Topics: Adult; Blood-Retinal Barrier; Diabetes Mellitus, Type 1; Female; Humans; Indazoles; Male; Middle Aged; Pyrazoles

1987
Pharmacokinetics of bendazac-lysine and 5-hydroxybendazac in patients with renal insufficiency.
    European journal of clinical pharmacology, 1987, Volume: 33, Issue:3

    Topics: Adult; Aged; Anti-Inflammatory Agents, Non-Steroidal; Biological Availability; Blood Proteins; Female; Humans; Indazoles; Kidney Failure, Chronic; Male; Middle Aged; Protein Binding; Pyrazoles

1987
Effects of bendazac L-lysine salt on X-ray-induced cataract in the rabbit lens.
    Experimental eye research, 1986, Volume: 42, Issue:2

    Topics: Animals; Cataract; Chromatography, Gel; Crystallins; Dithiothreitol; Dose-Response Relationship, Radiation; Glutathione; Indazoles; Lens, Crystalline; Molecular Weight; Organ Size; Pyrazoles; Rabbits; Time Factors; Water

1986
Plasma levels and metabolism of bendazac lysine salt in man.
    Bollettino chimico farmaceutico, 1986, Volume: 125, Issue:8

    Topics: Chromatography, High Pressure Liquid; Humans; Indazoles; Pyrazoles

1986
Tissue distribution, urinary, fecal and biliary excretion of 14C bendazac L-lysine salt in rats.
    Pharmacological research communications, 1985, Volume: 17, Issue:5

    Topics: Animals; Anti-Inflammatory Agents; Bile; Feces; Female; Indazoles; Kinetics; Lens, Crystalline; Male; Pyrazoles; Rats; Sex Factors; Tissue Distribution

1985
General pharmacological investigations on bendazac lysine.
    Il Farmaco; edizione pratica, 1984, Volume: 39, Issue:12

    Topics: Animals; Anti-Inflammatory Agents; Bile; Biogenic Amines; Blood Sedimentation; Clofibrate; Female; Guinea Pigs; Indazoles; Lipids; Male; Mice; Pyrazoles; Rats

1984
On the hypolipemic properties of bendaline.
    Journal of medicine, 1984, Volume: 15, Issue:2

    Topics: Animals; Bile; Cholesterol, Dietary; Female; Fructose; Hyperlipidemias; Hypolipidemic Agents; Indazoles; Lipidoses; Liver Diseases, Alcoholic; Male; Malondialdehyde; Mice; Platelet Aggregation; Pyrazoles; Rabbits; Rats

1984
Basic data supporting the use of the l-lysine salt of bendazac in cataract.
    International journal of tissue reactions, 1983, Volume: 5, Issue:2

    Topics: Administration, Oral; Animals; Anti-Inflammatory Agents; Cataract; Crystallins; Indazoles; Lens, Crystalline; Microscopy, Electron; Protein Denaturation; Pyrazoles; Rats

1983
Oral absorption of bendazac lysine salt in man after repeated administrations.
    Pharmacological research communications, 1983, Volume: 15, Issue:5

    Topics: Administration, Oral; Adult; Blood Chemical Analysis; Female; Humans; Indazoles; Intestinal Absorption; Kinetics; Male; Pyrazoles; Time Factors

1983
A comparative study of the oral absorption in man of bendazac and its lysine salt.
    Bollettino chimico farmaceutico, 1982, Volume: 121, Issue:2

    Topics: Absorption; Administration, Oral; Adult; Anti-Inflammatory Agents; Female; Humans; Indazoles; Male; Pyrazoles; Tablets; Time Factors

1982
Effect of bendazac lysine on lens and retina in diabetics.
    Documenta ophthalmologica. Advances in ophthalmology, 1994, Volume: 86, Issue:4

    Topics: Administration, Oral; Anti-Inflammatory Agents, Non-Steroidal; Blood-Retinal Barrier; Capillary Permeability; Diabetes Complications; Diabetes Mellitus; Diabetic Retinopathy; Female; Fluorophotometry; Humans; Indazoles; Lens, Crystalline; Male; Middle Aged; Retina

1994
Clinical study of bendazac lysine for in vivo contact lens cleaning.
    Optometry and vision science : official publication of the American Academy of Optometry, 1993, Volume: 70, Issue:3

    Topics: Anti-Inflammatory Agents, Non-Steroidal; Contact Lenses; Disinfection; Eye Proteins; Female; Humans; Hydrogel, Polyethylene Glycol Dimethacrylate; Indazoles; Male; Ophthalmic Solutions; Placebos; Polyethylene Glycols

1993
Bendazac decreases in vitro glycation of human lens crystallins. Decrease of in vitro protein glycation by bendazac.
    Documenta ophthalmologica. Advances in ophthalmology, 1995, Volume: 90, Issue:4

    Topics: Adult; Anti-Inflammatory Agents, Non-Steroidal; Crystallins; Dose-Response Relationship, Drug; Fluorescence; Fructose; Glucose; Glycation End Products, Advanced; Glycosylation; Humans; Indazoles; Lens, Crystalline

1995
Hepatotoxicity due to lysine salt of bendazac.
    Scandinavian journal of gastroenterology, 1996, Volume: 31, Issue:2

    Topics: Aged; Aged, 80 and over; Anti-Inflammatory Agents, Non-Steroidal; Cataract; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Humans; Indazoles; Liver Function Tests

1996
Racemization of lens crystalline constituents in UV-induced cataract evaluated by chiral GC/MS spectroscopy.
    Ophthalmic research, 1996, Volume: 28 Suppl 2

    Topics: Amino Acids; Animals; Anti-Inflammatory Agents; Cataract; Crystallins; Gas Chromatography-Mass Spectrometry; Indazoles; Lens, Crystalline; Male; Radiation Injuries, Experimental; Rats; Stereoisomerism; Steroids; Ultraviolet Rays

1996
Inhibition of bacterial adherence to a high-water-content polymer by a water-soluble, nonsteroidal, anti-inflammatory drug.
    Journal of biomedical materials research, 1998, Volume: 42, Issue:1

    Topics: Anti-Inflammatory Agents, Non-Steroidal; Bacterial Adhesion; Contact Lenses; Humans; Indazoles; Polymers; Pseudomonas aeruginosa; Solubility; Staphylococcus aureus; Staphylococcus epidermidis; Water

1998
Accelerated study on lysozyme deposition on poly(HEMA) contact lenses.
    Biomaterials, 1998, Volume: 19, Issue:22

    Topics: Biocompatible Materials; Contact Lens Solutions; Contact Lenses; Indazoles; Iodine Radioisotopes; Kinetics; Muramidase; Polyhydroxyethyl Methacrylate; Temperature

1998
An NMR spectroscopy study of bendaline-albumin interactions.
    Bioorganic chemistry, 2003, Volume: 31, Issue:5

    Topics: Binding Sites; Carbon Isotopes; Dose-Response Relationship, Drug; Humans; Indazoles; Magnetic Resonance Spectroscopy; Molecular Structure; Protons; Serum Albumin

2003
Protective effects of bendazac lysine on early experimental diabetic nephropathy in rats.
    Acta pharmacologica Sinica, 2005, Volume: 26, Issue:6

    Topics: Aldehyde Reductase; Animals; Diabetic Nephropathies; Erythrocytes; Glomerular Mesangium; Glycation End Products, Advanced; Indazoles; Kidney; Laminin; Male; Oxidative Stress; Rats; Rats, Sprague-Dawley; RNA, Messenger; Transforming Growth Factor beta; Transforming Growth Factor beta1

2005
Protective effects of bendazac lysine on diabetic peripheral neuropathy in streptozotocin-induced diabetic rats.
    Clinical and experimental pharmacology & physiology, 2006, Volume: 33, Issue:12

    Topics: Aldehyde Reductase; Animals; Anti-Inflammatory Agents, Non-Steroidal; Behavior, Animal; Blood Glucose; Diabetes Mellitus, Experimental; Diabetic Neuropathies; Erythrocytes; Glutathione Peroxidase; Glycated Hemoglobin; Glycation End Products, Advanced; Indazoles; Insulin; Male; Myelin Sheath; Pain; Rats; Rats, Sprague-Dawley; Sodium-Potassium-Exchanging ATPase; Sural Nerve

2006
Synthesis and biological evaluations of novel bendazac lysine analogues as potent anticataract agents.
    Bioorganic & medicinal chemistry letters, 2010, Apr-01, Volume: 20, Issue:7

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Antioxidants; Cataract; Indazoles; Lens, Crystalline; Oxidative Stress; Rabbits; Rats; Solubility

2010
Characterization of a novel process-related impurity in commercial bendazac lysine eye drops by LC-ESI-QTOF/MS/MS and NMR.
    Journal of pharmaceutical and biomedical analysis, 2015, Mar-25, Volume: 107

    Topics: Chromatography, High Pressure Liquid; Drug Contamination; Indazoles; Magnetic Resonance Spectroscopy; Ophthalmic Solutions; Spectrometry, Mass, Electrospray Ionization; Tandem Mass Spectrometry

2015