Page last updated: 2024-08-21

indazoles and 1H-indazol-3-amine

indazoles has been researched along with 1H-indazol-3-amine in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's4 (80.00)24.3611
2020's1 (20.00)2.80

Authors

AuthorsStudies
Bamborough, P; Brown, MJ; Christopher, JA; Chung, CW; Mellor, GW1
Dong, J; Dong, Y; Pan, X; Shan, Y; Wang, M; Zhang, J; Zhang, L1
Ai, J; Cui, J; Dai, Y; Gao, D; Li, Y; Peng, X1
Li, C; Pan, X; Shan, Y; Si, R; Sun, Y; Wang, B; Zhang, J1
Abarbri, M; El Qami, A; Frlan, R; Gobec, S; Jismy, B; Knez, D; Kos, J; Pišlar, A1

Other Studies

5 other study(ies) available for indazoles and 1H-indazol-3-amine

ArticleYear
Selectivity of kinase inhibitor fragments.
    Journal of medicinal chemistry, 2011, Jul-28, Volume: 54, Issue:14

    Topics: Adenine; Adenosine Triphosphate; Aniline Compounds; Binding Sites; Enzyme Inhibitors; High-Throughput Screening Assays; Indazoles; Indoles; Isoenzymes; Models, Molecular; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphotransferases; Protein Binding; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-pim-1; Pyridines; Pyrimidines; Quantitative Structure-Activity Relationship; Small Molecule Libraries

2011
Expanding the structural diversity of Bcr-Abl inhibitors: Dibenzoylpiperazin incorporated with 1H-indazol-3-amine.
    European journal of medicinal chemistry, 2015, Nov-02, Volume: 104

    Topics: Antineoplastic Agents; Cell Proliferation; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Fusion Proteins, bcr-abl; Humans; Indazoles; K562 Cells; Molecular Docking Simulation; Molecular Structure; Piperazines; Protein Kinase Inhibitors; Structure-Activity Relationship

2015
Optimization of 1H-indazol-3-amine derivatives as potent fibroblast growth factor receptor inhibitors.
    Bioorganic & medicinal chemistry letters, 2017, 08-15, Volume: 27, Issue:16

    Topics: Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Humans; Indazoles; Models, Molecular; Molecular Structure; Receptor, Fibroblast Growth Factor, Type 1; Receptor, Fibroblast Growth Factor, Type 2; Structure-Activity Relationship

2017
Discovery of novel anti-angiogenesis agents. Part 8: Diaryl thiourea bearing 1H-indazole-3-amine as multi-target RTKs inhibitors.
    European journal of medicinal chemistry, 2017, Dec-01, Volume: 141

    Topics: Angiogenesis Inhibitors; Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Cell Survival; Dose-Response Relationship, Drug; Drug Discovery; Drug Screening Assays, Antitumor; Human Umbilical Vein Endothelial Cells; Humans; Indazoles; Molecular Docking Simulation; Molecular Structure; Neovascularization, Pathologic; Protein Kinase Inhibitors; Receptor Protein-Tyrosine Kinases; Structure-Activity Relationship; Thiourea

2017
Pyrimido[1,2-b]indazole derivatives: Selective inhibitors of human monoamine oxidase B with neuroprotective activity.
    European journal of medicinal chemistry, 2021, Jan-01, Volume: 209

    Topics: Antiparkinson Agents; Bromides; Coordination Complexes; Humans; Indazoles; Metals; Molecular Docking Simulation; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Neuroblastoma; Neuroprotective Agents; Protein Binding; Small Molecule Libraries; Structure-Activity Relationship; Tyramine

2021