Page last updated: 2024-09-03

indatraline and gsk1210151a

indatraline has been researched along with gsk1210151a in 2 studies

Compound Research Comparison

Studies
(indatraline)
Trials
(indatraline)
Recent Studies (post-2010)
(indatraline)
Studies
(gsk1210151a)
Trials
(gsk1210151a)
Recent Studies (post-2010) (gsk1210151a)
460241091106

Protein Interaction Comparison

ProteinTaxonomyindatraline (IC50)gsk1210151a (IC50)
Chain A, BROMODOMAIN-CONTAINING PROTEIN 2Homo sapiens (human)0.5
Chain A, BROMODOMAIN-CONTAINING PROTEIN 2Homo sapiens (human)0.5
Bromodomain-containing protein 4Homo sapiens (human)0.3054
Cytochrome P450 3A4Homo sapiens (human)9.7
Cytochrome P450 2C9 Homo sapiens (human)7.4875
Bromodomain-containing protein 2Homo sapiens (human)0.3127
cAMP-specific 3',5'-cyclic phosphodiesterase 4BHomo sapiens (human)3.9811
Bromodomain-containing protein 3Homo sapiens (human)0.1531
Bromodomain testis-specific proteinHomo sapiens (human)0.5801

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (50.00)24.3611
2020's1 (50.00)2.80

Authors

AuthorsStudies
Kabir, M; Kerns, E; Nguyen, K; Shah, P; Sun, H; Wang, Y; Xu, X; Yu, KR1
Kabir, M; Kerns, E; Neyra, J; Nguyen, K; Nguyễn, ÐT; Shah, P; Siramshetty, VB; Southall, N; Williams, J; Xu, X; Yu, KR1

Other Studies

2 other study(ies) available for indatraline and gsk1210151a

ArticleYear
Predictive models of aqueous solubility of organic compounds built on A large dataset of high integrity.
    Bioorganic & medicinal chemistry, 2019, 07-15, Volume: 27, Issue:14

    Topics: Drug Discovery; Organic Chemicals; Pharmaceutical Preparations; Solubility

2019
Retrospective assessment of rat liver microsomal stability at NCATS: data and QSAR models.
    Scientific reports, 2020, 11-26, Volume: 10, Issue:1

    Topics: Animals; Computer Simulation; Databases, Factual; Drug Discovery; High-Throughput Screening Assays; Liver; Machine Learning; Male; Microsomes, Liver; National Center for Advancing Translational Sciences (U.S.); Pharmaceutical Preparations; Quantitative Structure-Activity Relationship; Rats; Rats, Sprague-Dawley; Retrospective Studies; United States

2020