Compounds > indapamide

indapamide and acetazolamide

indapamide has been researched along with acetazolamide in 18 studies

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19903 (16.67)18.7374
1990's1 (5.56)18.2507
2000's4 (22.22)29.6817
2010's10 (55.56)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cecchi, A; Scozzafava, A; Supuran, CT; Temperini, C3
González-Díaz, H; Orallo, F; Quezada, E; Santana, L; Uriarte, E; Viña, D; Yáñez, M1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Čapkauskaitė, E; Gylytė, J; Kišonaitė, M; Matulis, D; Tumkevičius, S; Zubrienė, A1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Čapkauskaitė, E; Gražulis, S; Gylytė, J; Jogaitė, V; Kazokaitė, J; Kišonaitė, M; Manakova, E; Matulis, D; Michailovienė, V; Smirnov, A; Torresan, J; Tumkevičius, S; Zubrienė, A1
Chimirri, A; Damiano, FM; De Luca, L; Ferro, S; Gitto, R; Supuran, CT; Vullo, D1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Čapkauskaitė, E; Gedgaudas, M; Kairys, V; Linkuvienė, V; Matulis, D; Paketurytė, V; Ruibys, V; Zakšauskas, A1
Greenberg, A1
Lettieri, JT; Portelli, ST1
Herbinger, W1
Baican, M; Coltau, M; Domuta, G; Hecht, A; Puscas, I1

Reviews

1 review(s) available for indapamide and acetazolamide

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

17 other study(ies) available for indapamide and acetazolamide

ArticleYear
Carbonic anhydrase inhibitors. Interaction of indapamide and related diuretics with 12 mammalian isozymes and X-ray crystallographic studies for the indapamide-isozyme II adduct.
    Bioorganic & medicinal chemistry letters, 2008, Apr-15, Volume: 18, Issue:8

    Topics: Animals; Carbonic Anhydrase Inhibitors; Carbonic Anhydrases; Computer Simulation; Crystallography, X-Ray; Humans; Indapamide; Isoenzymes; Mice; Models, Molecular; Molecular Structure

2008
Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors.
    Journal of medicinal chemistry, 2008, Nov-13, Volume: 51, Issue:21

    Topics: Computational Biology; Drug Design; Humans; Isoenzymes; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quantitative Structure-Activity Relationship

2008
Carbonic anhydrase inhibitors. Comparison of chlorthalidone and indapamide X-ray crystal structures in adducts with isozyme II: when three water molecules and the keto-enol tautomerism make the difference.
    Journal of medicinal chemistry, 2009, Jan-22, Volume: 52, Issue:2

    Topics: Carbonic Anhydrase Inhibitors; Catalytic Domain; Chlorthalidone; Crystallography, X-Ray; Indapamide; Isoenzymes; Models, Molecular; Stereoisomerism; Water

2009
Carbonic anhydrase inhibitors. Comparison of chlorthalidone, indapamide, trichloromethiazide, and furosemide X-ray crystal structures in adducts with isozyme II, when several water molecules make the difference.
    Bioorganic & medicinal chemistry, 2009, Feb-01, Volume: 17, Issue:3

    Topics: Carbonic Anhydrase II; Carbonic Anhydrase Inhibitors; Chlorthalidone; Crystallography, X-Ray; Furosemide; Indapamide; Isoenzymes; Structure-Activity Relationship; Sulfonamides; Trichlormethiazide; Water

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
Benzenesulfonamides with benzimidazole moieties as inhibitors of carbonic anhydrases I, II, VII, XII and XIII.
    Journal of enzyme inhibition and medicinal chemistry, 2014, Volume: 29, Issue:1

    Topics: Benzenesulfonamides; Carbonic Anhydrase Inhibitors; Magnetic Resonance Spectroscopy; Mass Spectrometry; Spectrophotometry, Infrared; Sulfonamides

2014
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Benzenesulfonamides with pyrimidine moiety as inhibitors of human carbonic anhydrases I, II, VI, VII, XII, and XIII.
    Bioorganic & medicinal chemistry, 2013, Nov-15, Volume: 21, Issue:22

    Topics: Benzenesulfonamides; Binding Sites; Calorimetry; Carbonic Anhydrase Inhibitors; Carbonic Anhydrases; Crystallography, X-Ray; Enzyme Activation; Humans; Isoenzymes; Kinetics; Protein Binding; Protein Structure, Tertiary; Pyrimidines; Recombinant Proteins; Structure-Activity Relationship; Sulfonamides

2013
Structure-based screening for the discovery of new carbonic anhydrase VII inhibitors.
    European journal of medicinal chemistry, 2014, Volume: 71

    Topics: Carbonic Anhydrase Inhibitors; Carbonic Anhydrases; Drug Design; Humans; Molecular Docking Simulation; Structure-Activity Relationship

2014
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
Benzimidazole design, synthesis, and docking to build selective carbonic anhydrase VA inhibitors.
    Bioorganic & medicinal chemistry, 2018, 02-01, Volume: 26, Issue:3

    Topics: Benzimidazoles; Binding Sites; Carbonic Anhydrase Inhibitors; Carbonic Anhydrases; Catalytic Domain; Drug Design; Humans; Isoenzymes; Molecular Docking Simulation; Structure-Activity Relationship

2018
What's new in diuretic therapy.
    American family physician, 1986, Volume: 33, Issue:5

    Topics: Acetazolamide; Acid-Base Imbalance; Biological Transport; Diuretics; Drug Resistance; Ethacrynic Acid; Furosemide; Humans; Hydrochlorothiazide; Hyperkalemia; Hypernatremia; Hypokalemia; Hyponatremia; Indapamide; Kidney Tubules, Distal; Kidney Tubules, Proximal; Loop of Henle; Metolazone; Osmolar Concentration; Spironolactone; Triamterene; Vasopressins

1986
Effects of competitive red blood cell binding and reduced hematocrit on the blood and plasma levels of [14C]Indapamide in the rat.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 224, Issue:2

    Topics: Acetazolamide; Animals; Binding, Competitive; Carbon Radioisotopes; Chlorthalidone; Diuretics; Erythrocytes; Hematocrit; Indapamide; Male; Rats; Rats, Inbred Strains

1983
[Diuretics in the therapy of chronic cardiac insufficiency].
    Wiener medizinische Wochenschrift (1946), 1982, Oct-15, Volume: 132, Issue:19

    Topics: Acetazolamide; Amiloride; Diuretics; Drug Interactions; Ethacrynic Acid; Heart Failure; Humans; Indapamide; Metolazone; Risk; Spironolactone; Sulfonamides; Thiazoles; Ticrynafen; Triamterene

1982
Vasodilatory effect of diuretics is dependent on inhibition of vascular smooth muscle carbonic anhydrase by a direct mechanism of action.
    Drugs under experimental and clinical research, 1999, Volume: 25, Issue:6

    Topics: Acetazolamide; Aged; Amiloride; Animals; Blood Pressure; Carbonic Anhydrase Inhibitors; Carbonic Anhydrases; Diuretics; Erythrocytes; Furosemide; Humans; Hydrochlorothiazide; Hydrogen-Ion Concentration; In Vitro Techniques; Indapamide; Middle Aged; Muscle, Smooth, Vascular; Rabbits; Triamterene; Vasodilation

1999