indanidine has been researched along with clonidine in 24 studies
Studies (indanidine) | Trials (indanidine) | Recent Studies (post-2010) (indanidine) | Studies (clonidine) | Trials (clonidine) | Recent Studies (post-2010) (clonidine) |
---|---|---|---|---|---|
26 | 0 | 1 | 13,692 | 2,044 | 1,394 |
Protein | Taxonomy | indanidine (IC50) | clonidine (IC50) |
---|---|---|---|
Alpha-2A adrenergic receptor | Homo sapiens (human) | 0.101 | |
Alpha-2B adrenergic receptor | Homo sapiens (human) | 0.0353 | |
Alpha-2C adrenergic receptor | Homo sapiens (human) | 0.0115 | |
5-hydroxytryptamine receptor 1A | Rattus norvegicus (Norway rat) | 5.365 | |
Alpha-2B adrenergic receptor | Rattus norvegicus (Norway rat) | 0.0173 | |
Alpha-2C adrenergic receptor | Rattus norvegicus (Norway rat) | 0.0173 | |
Alpha-2A adrenergic receptor | Rattus norvegicus (Norway rat) | 0.0173 | |
Alpha-1D adrenergic receptor | Homo sapiens (human) | 1.21 | |
5-hydroxytryptamine receptor 1B | Rattus norvegicus (Norway rat) | 5.365 | |
Alpha-2A adrenergic receptor | Bos taurus (cattle) | 0.002 | |
Nischarin | Rattus norvegicus (Norway rat) | 0.3662 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 19 (79.17) | 18.7374 |
1990's | 5 (20.83) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Batink, H; de Jonge, A; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B | 1 |
Esbenshade, TA; Han, C; Hollinger, S; Minneman, KP; Theroux, TL | 1 |
Biguad, M; Julou-Schaeffer, G; Parratt, JR; Stoclet, JC | 1 |
Schott, C; Stoclet, JC; Topouzis, S | 1 |
de Jonge, A; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B | 1 |
McGrath, JC | 2 |
DeMarinis, RM; Hieble, JP; Matthews, WD | 1 |
Bou, J; Massingham, R | 1 |
Chiu, AT; McCall, DE; Thoolen, MJ; Timmermans, PB | 1 |
Contreras-Rodríguez, JL; García-Sáinz, JA | 1 |
Dinovo, EC; Haddox, VG; Menon, MK | 1 |
James, MK; Leighton, HJ | 1 |
de Jonge, A; Mathy, MJ; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B | 2 |
Hong, KW; Jung, HO | 1 |
Coates, J; Jahn, U; Weetman, DF | 1 |
Coates, J; Weetman, DF | 2 |
Chadwick, MA; Coates, J; Ismail, S; Jahn, U; Lawson, K; Thiele, K; Turner, N; Weetman, DF | 1 |
Mathy, MJ; Thoolen, MJ; Timmermans, PB; van Zwieten, PA | 1 |
Lues, I; Schümann, HJ | 1 |
Dong, X; Doughty, MB; Miller, DW; Misse, GA; Tessel, RE | 1 |
Hart, SD; Timmermans, PB; Wong, PC | 1 |
2 review(s) available for indanidine and clonidine
Article | Year |
---|---|
Evidence for and against heterogeneity of alpha 1-adrenoceptors.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Calcium; Calcium Channel Blockers; Clonidine; Dobutamine; Dogs; Humans; In Vitro Techniques; Rabbits; Rats; Receptors, Adrenergic, alpha; Species Specificity; Vasoconstriction | 1986 |
Sgd 101/75: a sympathomimetic that can be used to identify a new subtype of alpha-adrenoceptor, the alpha 1s-adrenoceptor.
Topics: Adrenergic alpha-Agonists; Animals; Clonidine; Electric Stimulation; Hemodynamics; Humans; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Phenoxybenzamine; Receptors, Adrenergic, alpha; Sympathomimetics | 1983 |
22 other study(ies) available for indanidine and clonidine
Article | Year |
---|---|
Quantitative relationships between alpha-adrenergic activity and binding affinity of alpha-adrenoceptor agonists and antagonists.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Blood Pressure; Brain; Cell Membrane; Clonidine; Kinetics; Prazosin; Quinazolines; Rats; Receptors, Adrenergic, alpha; Structure-Activity Relationship; Vasoconstriction | 1984 |
Selectivity of agonists for cloned alpha 1-adrenergic receptor subtypes.
Topics: Adrenergic alpha-1 Receptor Agonists; Animals; Binding, Competitive; Catecholamines; Cattle; Cell Line; Cloning, Molecular; Cricetinae; Humans; Imidazoles; Inositol Phosphates; Phenethylamines; Phenoxybenzamine; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-1; Recombinant Proteins; Tetralones | 1994 |
Endotoxin-induced impairment of vascular smooth muscle contractions elicited by different mechanisms.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic alpha-Agonists; Animals; Aorta, Thoracic; Caffeine; Calcimycin; Calcium; Clonidine; Endothelium, Vascular; Endotoxins; In Vitro Techniques; Inositol 1,4,5-Trisphosphate; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nitrendipine; Phenylephrine; Potassium Chloride; Rats; Rats, Inbred Strains; Sarcoplasmic Reticulum | 1990 |
Participation of endothelium-derived relaxing factor and role of cyclic GMP in inhibitory effects of endothelium on contractile responses elicited by alpha-adrenoceptor agonists in rat aorta.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic alpha-Agonists; Animals; Aorta, Thoracic; Arginine; Azepines; Clonidine; Cyclic GMP; Endothelium, Vascular; Female; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide; Phenylephrine; Rats; Rats, Inbred Strains | 1991 |
Calcium dependency of vasoconstriction mediated by alpha 1- and alpha 2-adrenoceptors.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Azepines; Blood Pressure; Calcium; Calcium Channel Blockers; Clonidine; Imidazoles; Ion Channels; Nifedipine; Rats; Receptors, Adrenergic, alpha; Regional Blood Flow; Structure-Activity Relationship; Vasoconstriction | 1985 |
alpha-Adrenoceptor agonists and the Ca2+-dependence of smooth muscle contraction: evidence for subtypes of receptors or for agonist-dependent differences in the agonist-receptor interaction?
Topics: Adrenergic alpha-Agonists; Animals; Calcium; Clonidine; Ethanolamines; Male; Methoxamine; Muscle Contraction; Muscle, Smooth; Nifedipine; Norepinephrine; Phenylephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Xylazine | 1985 |
Effect of diltiazem upon contractile responses to phenylephrine, cirazoline, Sgd 101/75, St 587 and B-HT 920 in rabbit aorta and dog saphenous vein preparations.
Topics: Adrenergic alpha-Agonists; Animals; Aorta, Thoracic; Azepines; Benzazepines; Clonidine; Diltiazem; Dogs; Drug Interactions; Female; Imidazoles; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Phenylephrine; Rabbits; Saphenous Vein | 1986 |
Ca++ utilization in the constriction of rat aorta to full and partial alpha-1 adrenoceptor agonists.
Topics: Adrenergic alpha-Agonists; Animals; Aorta; Calcium; Clonidine; Dose-Response Relationship, Drug; Ethanolamines; Imidazoles; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Potassium; Rats; Rats, Inbred Strains; Tetrahydronaphthalenes | 1986 |
Possible existence of two mechanisms involved in alpha 1-adrenergic action: effect of Sgd 101/75.
Topics: Adrenalectomy; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Calcium; Clonidine; Cyclic AMP; Epinephrine; Female; Hypothyroidism; In Vitro Techniques; Liver; Propranolol; Rats; Rats, Inbred Strains; Urea | 1986 |
Modification of certain pharmacological effects of ethanol by lipophilic alpha-1 adrenergic agonists.
Topics: Adrenergic alpha-Agonists; Animals; Body Temperature; Clonidine; Drug Interactions; Ethanol; Hypnosis; Imidazoles; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mice, Inbred DBA; Motor Activity; Pentobarbital; Tetrahydronaphthalenes | 1987 |
Analysis of putative alpha-1s adrenoceptor agonism by Sgd 101/75 in the rat anococcygeus muscle.
Topics: Adrenergic alpha-Agonists; Animals; Clonidine; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Muscle Contraction; Norepinephrine; Phenoxybenzamine; Rats; Receptors, Adrenergic, alpha | 1987 |
Effects of the irreversible alpha-adrenoceptor antagonists phenoxybenzamine and benextramine on the effectiveness of nifedipine in inhibiting alpha 1- and alpha 2-adrenoceptor mediated vasoconstriction in pithed rats.
Topics: Animals; Azepines; Clonidine; Cystamine; Decerebrate State; Diastole; Dose-Response Relationship, Drug; Imidazoles; Male; Nifedipine; Phenoxybenzamine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Vasoconstriction | 1985 |
Characterization of inhibition by nifedipine and nitroprusside of the pressor responses to alpha 1-adrenoceptor agonists cirazoline and Sgd 101/75 in pithed rats.
Topics: Animals; Blood Pressure; Clonidine; Ferricyanides; Imidazoles; Male; Nifedipine; Nitroprusside; Rats; Rats, Inbred Strains; Vasoconstriction | 1988 |
The existence of a new subtype of alpha-adrenoceptor on the rat anococcygeus is revealed by SGD 101/75 and phenoxybenzamine.
Topics: Adrenergic alpha-Agonists; Animals; Clonidine; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Norepinephrine; Phenoxybenzamine; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha | 1982 |
Occurrence of alpha 1s-adrenoceptors in the mouse but not in the rabbit isolated anococcygeus preparations.
Topics: Adrenergic alpha-Agonists; Animals; Clonidine; Drug Interactions; Male; Mice; Muscle Contraction; Muscle, Smooth; Norepinephrine; Phenoxybenzamine; Rabbits; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Species Specificity | 1983 |
Demonstration of alpha 1s-adrenoceptors after exposure of the rat anococcygeus to benextramine.
Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Cystamine; In Vitro Techniques; Male; Muscle Contraction; Muscles; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha | 1983 |
Sgd 101/75: cardiovascular effects in various animal preparations; interactions with vascular postjunctional alpha 1- and alpha 2-adrenoceptors.
Topics: Adrenergic alpha-Agonists; Animals; Blood Pressure; Cats; Clonidine; Heart Rate; Hemodynamics; Hypertension; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha | 1984 |
Sgd 101/75 is distinguished from other selective alpha 1-adrenoceptor agonists by the inhibition of its pressor responses by calcium entry blockade and vasodilatation in pithed rats and cats.
Topics: Adrenergic alpha-Agonists; Albuterol; Animals; Blood Pressure; Calcium Channel Blockers; Cats; Clonidine; Decerebrate State; Dose-Response Relationship, Drug; Male; Nifedipine; Rats; Rats, Inbred Strains; Vasoconstriction; Vasodilation | 1983 |
Alpha-adrenoceptor antagonism by apoyohimbine and some observations on the pharmacology of alpha-adrenoceptors in the rat anococcygeus and vas deferens.
Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Cocaine; Electric Stimulation; Ethanolamines; In Vitro Techniques; Male; Muscle, Smooth; Norepinephrine; Rats; Rats, Inbred Strains; Vas Deferens; Xylazine; Yohimbine | 1984 |
Effect of removing the endothelial cells on the reactivity of rat aortic segments to different alpha-adrenoceptor agonists.
Topics: Adrenergic alpha-Agonists; Animals; Aorta, Thoracic; Azepines; Clonidine; Endothelium; Imidazoles; In Vitro Techniques; Male; Methoxamine; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Rats; Rats, Inbred Strains; Xylazine; Yohimbine | 1984 |
Characterization of vascular postsynaptic NPY receptor function and regulation and differential sensitivity of Y1 and Y2 receptor function to changes in extracellular calcium availability and prior in vitro peptide exposure.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic alpha-Agonists; Animals; Calcium; Clonidine; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Neuropeptide Y; Peptide Fragments; Peptides; Rats; Rats, Sprague-Dawley; Receptors, Neuropeptide Y; Synapses; Vasoconstrictor Agents | 1993 |
Effects of nifedipine on phasic and tonic vasoconstrictor responses to Sgd 101/75 in the isolated perfused rabbit ear artery.
Topics: Adrenergic alpha-Agonists; Animals; Arteries; Calcium; Clonidine; Ear; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Rabbits; Vasoconstriction | 1994 |