imidazole-4-carboxamide has been researched along with olaparib in 1 studies
Studies (imidazole-4-carboxamide) | Trials (imidazole-4-carboxamide) | Recent Studies (post-2010) (imidazole-4-carboxamide) | Studies (olaparib) | Trials (olaparib) | Recent Studies (post-2010) (olaparib) |
---|---|---|---|---|---|
26 | 1 | 15 | 1,313 | 172 | 1,258 |
Protein | Taxonomy | imidazole-4-carboxamide (IC50) | olaparib (IC50) |
---|---|---|---|
Poly [ADP-ribose] polymerase tankyrase-1 | Homo sapiens (human) | 1.538 | |
Cytochrome P450 1A2 | Homo sapiens (human) | 0.02 | |
Cholinesterase | Homo sapiens (human) | 0.0035 | |
Poly [ADP-ribose] polymerase 1 | Homo sapiens (human) | 0.1741 | |
Cytochrome P450 2D6 | Homo sapiens (human) | 0.02 | |
Protein mono-ADP-ribosyltransferase PARP6 | Homo sapiens (human) | 1.8 | |
Protein mono-ADP-ribosyltransferase PARP15 | Homo sapiens (human) | 7.6216 | |
Protein mono-ADP-ribosyltransferase PARP10 | Homo sapiens (human) | 5.2854 | |
Protein mono-ADP-ribosyltransferase PARP16 | Homo sapiens (human) | 5.1143 | |
Poly [ADP-ribose] polymerase tankyrase-2 | Homo sapiens (human) | 2.3349 | |
Histamine H3 receptor | Cavia porcellus (domestic guinea pig) | 0.001 | |
Poly [ADP-ribose] polymerase 2 | Homo sapiens (human) | 0.1866 | |
Protein mono-ADP-ribosyltransferase PARP4 | Homo sapiens (human) | 0.4087 | |
Protein mono-ADP-ribosyltransferase PARP3 | Homo sapiens (human) | 0.1315 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 1 (100.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Jiang, N; Liu, F; Wang, L; Zheng, Z; Zhou, W; Zhou, X | 1 |
1 other study(ies) available for imidazole-4-carboxamide and olaparib
Article | Year |
---|---|
Design, Synthesis, and Biological Evaluation of Novel PARP-1 Inhibitors Based on a 1H-Thieno[3,4-d] Imidazole-4-Carboxamide Scaffold.
Topics: Aminoimidazole Carboxamide; Cell Line; Cell Proliferation; Humans; Phthalazines; Piperazines; Poly (ADP-Ribose) Polymerase-1; Structure-Activity Relationship | 2016 |