imetit has been researched along with thiourea in 48 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 14 (29.17) | 18.2507 |
| 2000's | 23 (47.92) | 29.6817 |
| 2010's | 11 (22.92) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Arrang, JM; Ganellin, CR; Garbarg, M; Ligneau, X; Rouleau, A; Schwartz, JC; Tuong, MD | 1 |
| Ansay, M; Delaunois, A; Garbarg, M; Gustin, P | 1 |
| Imamura, M; Lander, HM; Levi, R; Seyedi, N | 1 |
| Banks, K; Merali, Z | 1 |
| Buczko, W; Godlewski, G; Malinowska, B; Schlicker, E | 1 |
| Lau, HY; Stenton, GR | 1 |
| Marr, I; Schlicker, E | 1 |
| Bucher, B; Godlewski, G; Malinowska, B; Schlicker, E | 1 |
| Allen, MC | 1 |
| Flood, JF; Morley, JE; Uezu, K | 1 |
| Schlicker, E; Werthwein, S; Zentner, J | 1 |
| Beckers, JF; Bloden, S; Delaunois, A; Gustin, P; Nemmar, A; Sulon, J | 1 |
| Jørgensen, H; Kjaer, A; Knigge, U; Warberg, J; Willems, E | 1 |
| Murakami, Y; Nakamura, K; Okada, S; Wang, M; Yokotani, K | 1 |
| Attarzadeh, M; Farzin, D | 1 |
| Bacciottini, L; Bartolini, L; Blandina, P; Giovannini, MG; Greco, L | 1 |
| Anthes, JC; Bayne, M; Behan, J; Gonsiorek, W; Greene, J; Greenfeder, SA; Gustafson, EL; Hedrick, JA; Hipkin, RW; Laz, TM; Monsma, FJ; Morse, KL; Qiao, X; Shin, N; Umland, S; Wan, Y; Wang, S; West, RE | 1 |
| Alves-Rodrigues, A; Lemstra, S; Leurs, R; Menge, WM; Timmerman, H; Vollinga, RC | 1 |
| Bongers, G; Hashimoto, T; Leurs, R; Lovenberg, TW; Menge, WM; Timmerman, H; Wieland, K; Yamamoto, Y; Yamatodani, A | 1 |
| Blanco, I; Gomez-Ramirez, J; Ortiz, J | 1 |
| Levi, R; Lovenberg, TW; Poonwasi, KS; Seyedi, N; Silver, RB; Wilson, SJ | 1 |
| Debilly, G; Gigout, S; Lin, JS; Vanni-Mercier, G | 1 |
| Cassuto, J; Räntfors, J | 1 |
| Brzozowski, T; Konturek, SJ; Obuchowicz, R; Pawlik, MW; Pawlik, WW | 1 |
| Arrang, JM; Cochois, V; Héron, A; Pillot, C; Rouleau, A; Schwartz, JC | 1 |
| Biernat, J; Brzozowski, T; Konturek, SJ; Obuchowicz, R; Pawlik, MW; Pawlik, WW; Sendur, R | 1 |
| Blanco, I; Gómez-Ramírez, J; Moreno-Delgado, D; Ortiz, J; Rodríguez-Agudo, D; Rodríguez-Caso, C; Sánchez-Jiménez, F; Torrent, A | 1 |
| Blanks, AM; Lee, K; Renaud, LP; Spanswick, D; Whyment, AD | 1 |
| Chen, AS; Chen, HY; Ishihara, A; Kanatani, A; Kotani, H; Macneil, DJ; Miyamoto, Y; Shimamura, K; Takahashi, K; Tokita, S; Yoshimoto, R | 1 |
| Biedka, I; Bortel, A; Brus, R; Dabrowska, J; Kostrzewa, RM; Nowak, P; Szczerbak, G; Słomian, G | 1 |
| Kanatani, A; Tokita, S; Yoshimoto, R | 1 |
| Kamei, C; Kuyama, S; Ogawa, M; Sugimoto, Y; Yokota, E | 1 |
| Banks, ML; Bauzo, RM; Howell, LL; Manvich, DF | 1 |
| Barrett, P; Ebling, FJ; Enright, RA; Jethwa, PH; Murphy, M; Turnbull, Y; Warner, A | 1 |
| Aluisio, L; Boggs, JD; Bonaventure, P; Fraser, IC; Galici, R; Lord, B; Lovenberg, TW | 1 |
| Kamei, C; Masuoka, T | 1 |
| Baranowska, U; Göthert, M; Kurz, C; Lupiński, S; Malinowska, B; Schlicker, E | 1 |
| Li, P; Liu, W; Sun, G; Xu, X; Yang, X | 1 |
| Li, PH; Liu, W; Pan, LJ; Sun, GM; Xu, XG; Yang, XD | 1 |
| Arrang, JM; Motawaj, M | 1 |
| Hall, FS; Kitanaka, J; Kitanaka, N; Morita, Y; Nishiyama, N; Takemura, M; Tanaka, K; Tatsuta, T; Uhl, GR | 1 |
| Clapp, RH; Luckman, SM | 1 |
| Closon, C; Didone, V; Nyssen, L; Quertemont, E; Quoilin, C; Tirelli, E | 1 |
| Jurič, DM; Mele, T | 1 |
| Akhtar, M; Khanam, R; Najmi, AK; Yadav, CH | 1 |
| Akhtar, M; Hass, C; Khanam, R; Najmi, AK; Panda, BP | 1 |
| An, S; Chen, LY; Guo, XX; Hao, Q; Liu, Y; Ma, L; Pediani, JD; Tang, M; Ward, RJ; Wu, N; Xu, TR; Yang, Y; Zeng, H | 1 |
| Ciosek, J; Drobnik, J; Galdyszynska, M; Kun, T; Olczak, S; Piera, L; Szymanski, J | 1 |
48 other study(ies) available for imetit and thiourea
| Article | Year |
|---|---|
S-[2-(4-imidazolyl)ethyl]isothiourea, a highly specific and potent histamine H3 receptor agonist.
Topics: Animals; Cerebral Cortex; Guinea Pigs; Histamine Agonists; Histamine N-Methyltransferase; Histamine Release; Imidazoles; Methylhistamines; Mice; Rats; Receptors, Histamine; Receptors, Histamine H3; Thiourea; Urea | 1992 |
Modulation of acetylcholine, capsaicin and substance P effects by histamine H3 receptors in isolated perfused rabbit lungs.
Topics: Acetylcholine; Animals; Capillary Permeability; Capsaicin; Dose-Response Relationship, Drug; Drug Interactions; Endothelium; Female; Histamine Agonists; Histamine Antagonists; Imidazoles; In Vitro Techniques; Lung; Male; Nerve Fibers; Piperidines; Pulmonary Edema; Rabbits; Receptors, Histamine H3; Serotonin; Substance P; Thiourea | 1995 |
Functional identification of histamine H3-receptors in the human heart.
Topics: Cell Separation; Electric Stimulation; Exocytosis; Heart; Histamine Agonists; Histamine Antagonists; Humans; Imidazoles; In Vitro Techniques; Indoles; Methylhistamines; Myocardial Ischemia; Myocardium; Norepinephrine; Piperidines; Protein Kinase C; Receptors, Histamine H3; Synaptosomes; Thiourea | 1995 |
Does the histaminergic system mediate bombesin/GRP-induced suppression of food intake?
Topics: Animals; Behavior, Animal; Bombesin; Eating; Gastrin-Releasing Peptide; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Male; Methylhistamines; Motor Activity; Peptides; Piperidines; Rats; Rats, Sprague-Dawley; Satiation; Sincalide; Thiourea | 1994 |
Inhibitory H3 receptors on sympathetic nerves of the pithed rat: activation by endogenous histamine and operation in spontaneously hypertensive rats.
Topics: Adrenergic Fibers; Animals; Blood Pressure; Decerebrate State; Electric Stimulation; Histamine; Histamine Agonists; Histamine Antagonists; Hypertension; Imidazoles; Male; Methylhistamines; Piperidines; Pyrimethamine; Rats; Rats, Wistar; Receptors, Histamine H3; Thiourea; Vagotomy; Vascular Resistance | 1997 |
Effects of histamine agonists and antagonists on rat peritoneal mast cells.
Topics: Animals; Dimaprit; Histamine Agonists; Histamine Antagonists; Histamine Release; Imidazoles; Impromidine; Male; Mast Cells; Peritoneal Cavity; Rats; Rats, Sprague-Dawley; Receptors, Histamine H3; Thiourea | 1997 |
Mutual interactions of the presynaptic histamine H3 and prostaglandin EP3 receptors on the noradrenergic terminals in the mouse brain.
Topics: Animals; Brain; Calcium; Cerebral Cortex; Dinoprostone; Electric Stimulation; Histamine; Histamine Agonists; Imidazoles; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Nerve Endings; Norepinephrine; Radioisotope Dilution Technique; Rats; Receptors, Adrenergic, alpha-2; Receptors, Histamine H3; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP3 Subtype; Thiourea; Tritium | 1997 |
Identification of histamine H3 receptors in the tail artery from normotensive and spontaneously hypertensive rats.
Topics: Adrenergic alpha-2 Receptor Antagonists; Animals; Arteries; Electric Stimulation; Histamine; Histamine Agonists; Imidazoles; Male; Norepinephrine; Piperidines; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Histamine H3; Sympathetic Fibers, Postganglionic; Thiourea; Yohimbine | 1997 |
Agonist and antagonist effects of histamine H3 receptor ligands on 5-HT3 receptor-mediated ion currents in NG108-15 cells.
Topics: Animals; Cells, Cultured; Dose-Response Relationship, Drug; Histamine Agonists; Histamine Antagonists; Hybrid Cells; Imidazoles; Ion Channels; Isothiuronium; Membrane Potentials; Mice; Piperidines; Rats; Receptors, Histamine H3; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Serotonin Receptor Agonists; Thiourea | 1998 |
Effect of histamine H2 and H3 receptor modulation in the septum on post-training memory processing.
Topics: Animals; Cimetidine; Dimaprit; Histamine Agonists; Histamine Antagonists; Imidazoles; Limbic System; Male; Memory; Mice; Piperidines; Thiourea | 1998 |
Histamine H3 receptor-mediated inhibition of noradrenaline release in the human brain.
Topics: Animals; Brain; Cerebral Cortex; Dimethindene; Electric Stimulation; Hippocampus; Histamine; Histamine Agonists; Histamine Antagonists; Humans; Imidazoles; Male; Mice; Mice, Inbred Strains; Norepinephrine; Piperidines; Ranitidine; Receptors, Histamine H3; Thiourea; Tritium | 1999 |
Modulatory effect of imetit, a histamine H3 receptor agonist, on C-fibers, cholinergic fibers and mast cells in rabbit lungs in vitro.
Topics: Animals; Capsaicin; Carbachol; Cholinergic Fibers; Drug Interactions; Female; Histamine Agonists; Histamine Release; Imidazoles; In Vitro Techniques; Lung; Male; Mast Cells; Rabbits; Radioimmunoassay; Receptors, Histamine H3; Substance P; Thiourea | 1999 |
Histaminergic and catecholaminergic interactions in the central regulation of vasopressin and oxytocin secretion.
Topics: Animals; Arginine Vasopressin; Blood Pressure; Cerebral Ventricles; Cimetidine; Epinephrine; Histamine; Histamine Agonists; Hypothalamus; Imidazoles; Infusions, Parenteral; Male; Methylhistamines; Norepinephrine; Oxytocin; Pituitary Gland, Posterior; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H2; Thiazoles; Thiourea | 1999 |
Histamine H(3) receptor-mediated inhibition of endogenous acetylcholine release from the isolated, vascularly perfused rat stomach.
Topics: Acetylcholine; Animals; Atropine; Gastric Mucosa; GTP-Binding Proteins; Histamine; Imidazoles; Male; Methylhistamines; Perfusion; Pertussis Toxin; Piperidines; Rats; Rats, Wistar; Receptors, Histamine H3; Thiourea; Vagus Nerve; Virulence Factors, Bordetella | 2000 |
Influence of different histamine receptor agonists and antagonists on apomorphine-induced licking behavior in rat.
Topics: Animals; Apomorphine; Chlorpheniramine; Dimaprit; Diphenhydramine; Dopamine Agonists; Drug Interactions; Famotidine; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Male; Piperidines; Ranitidine; Rats; Rats, Sprague-Dawley; Stereotyped Behavior; Thiourea; Toluidines | 2000 |
Effects of histamine H3 receptor agonists and antagonists on cognitive performance and scopolamine-induced amnesia.
Topics: Amnesia; Analysis of Variance; Animals; Avoidance Learning; Behavior, Animal; Cognition; Histamine Agonists; Histamine Antagonists; Imidazoles; Injections, Intraperitoneal; Injections, Subcutaneous; Male; Methylhistamines; Pattern Recognition, Visual; Piperidines; Rats; Rats, Wistar; Receptors, Histamine H3; Scopolamine; Thiourea | 1999 |
Cloning and characterization of a novel human histamine receptor.
Topics: Amino Acid Sequence; Cells, Cultured; Cloning, Molecular; Histamine; Histamine Agonists; Humans; Imidazoles; Molecular Sequence Data; Radioligand Assay; Receptors, Histamine; Receptors, Histamine H3; RNA, Messenger; Sequence Homology, Amino Acid; Thiourea; Tissue Distribution; Transfection | 2001 |
Pharmacological analysis of immepip and imetit homologues. Further evidence for histamine H(3) receptor heterogeneity?
Topics: Animals; Cerebral Cortex; Guinea Pigs; Histamine Agonists; Imidazoles; Jejunum; Male; Piperidines; Radioligand Assay; Rats; Receptors, Histamine H3; Structure-Activity Relationship; Thiourea | 2001 |
Constitutive activity of histamine h(3) receptors stably expressed in SK-N-MC cells: display of agonism and inverse agonism by H(3) antagonists.
Topics: Animals; Burimamide; Cyclic AMP; Histamine Antagonists; Humans; Imidazoles; Male; Rats; Rats, Wistar; Receptors, Histamine H3; Recombinant Proteins; Thiourea; Tumor Cells, Cultured | 2001 |
Presynaptic H3 autoreceptors modulate histamine synthesis through cAMP pathway.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Brain; Bucladesine; Colforsin; Cyclic AMP; Drug Interactions; Histamine; Imidazoles; In Vitro Techniques; Male; Piperidines; Potassium; Rats; Rats, Sprague-Dawley; Receptors, Histamine H3; Thionucleotides; Thiourea | 2002 |
Decreased intracellular calcium mediates the histamine H3-receptor-induced attenuation of norepinephrine exocytosis from cardiac sympathetic nerve endings.
Topics: Animals; Calcium; Calcium Channel Blockers; Cell Line; Dose-Response Relationship, Drug; Exocytosis; Guinea Pigs; Histamine Agonists; Humans; Imidazoles; Male; Myocardial Ischemia; Myocardium; Neuroblastoma; Neurons; Norepinephrine; omega-Conotoxins; Potassium; Receptors, Histamine H3; Thiourea; Time Factors; Transfection; Tumor Cells, Cultured | 2002 |
Waking selective neurons in the posterior hypothalamus and their response to histamine H3-receptor ligands: an electrophysiological study in freely moving cats.
Topics: Action Potentials; Animals; Cats; Drug Administration Schedule; Electroencephalography; Electromyography; Electrooculography; Electrophysiology; Female; Geniculate Bodies; Hippocampus; Histamine; Histamine Agonists; Histamine Antagonists; Hypothalamus, Posterior; Imidazoles; Immunohistochemistry; Male; Methylhistamines; Neurons; Thiourea; Time Factors; Wakefulness | 2003 |
Role of histamine receptors in the regulation of edema and circulation postburn.
Topics: Animals; Burns; Clemastine; Edema; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Imidazoles; Male; Piperidines; Ranitidine; Rats; Rats, Sprague-Dawley; Receptors, Histamine; Receptors, Histamine H3; Regional Blood Flow; Skin; Statistics, Nonparametric; Thiourea | 2003 |
Involvement of central and peripheral histamine H(3) receptors in the control of the vascular tone and oxygen uptake in the mesenteric circulation of the rat.
Topics: Animals; Blood Pressure; Drug Evaluation, Preclinical; Drug Therapy, Combination; Female; Imidazoles; Injections, Intra-Arterial; Injections, Intraventricular; Intestinal Mucosa; Intestines; Male; Microcirculation; Muscle, Smooth, Vascular; Oxygen Consumption; Rats; Rats, Wistar; Receptors, Histamine H3; Splanchnic Circulation; Tachycardia; Thiourea; Time Factors; Vasoconstriction | 2004 |
Cloning and expression of the mouse histamine H3 receptor: evidence for multiple isoforms.
Topics: Animals; Blotting, Northern; Brain; Chlorocebus aethiops; Cloning, Molecular; Competitive Bidding; COS Cells; Gene Expression; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; In Situ Hybridization; Iodine Radioisotopes; Isoenzymes; Mice; Piperidines; Radioligand Assay; Rats; Receptors, Histamine H3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiourea; Transfection | 2004 |
Histamine H3 receptors modulate reactive hyperemia in rat gut.
Topics: Animals; Blood Pressure; Female; Histamine Agonists; Histamine Antagonists; Hyperemia; Imidazoles; Infusions, Intra-Arterial; Intestinal Mucosa; Intestines; Male; Mesenteric Arteries; Mesenteric Vascular Occlusion; Rats; Rats, Wistar; Receptors, Histamine H3; Regional Blood Flow; Thiourea | 2004 |
H3 autoreceptors modulate histamine synthesis through calcium/calmodulin- and cAMP-dependent protein kinase pathways.
Topics: Amino Acid Sequence; Animals; Brain; Calcium Channel Blockers; Calcium-Calmodulin-Dependent Protein Kinases; Cyclic AMP-Dependent Protein Kinase Type II; Cyclic AMP-Dependent Protein Kinases; Histamine; Histamine Agonists; Histidine Decarboxylase; Imidazoles; In Vitro Techniques; Male; Molecular Sequence Data; Peptide Fragments; Pertussis Toxin; Phosphorylation; Rats; Rats, Sprague-Dawley; Receptors, Histamine H3; Recombinant Proteins; Thiourea | 2005 |
Histamine excites neonatal rat sympathetic preganglionic neurons in vitro via activation of H1 receptors.
Topics: Action Potentials; Animals; Animals, Newborn; Autonomic Fibers, Preganglionic; Barium; Dimaprit; Female; Ganglia, Sympathetic; Histamine; Histamine Agonists; Histamine H1 Antagonists; Imidazoles; In Vitro Techniques; Male; Membrane Potentials; Neurons; Patch-Clamp Techniques; Potassium; Rats; Rats, Inbred WKY; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiourea; Triprolidine | 2006 |
Therapeutic potential of histamine H3 receptor agonist for the treatment of obesity and diabetes mellitus.
Topics: Animals; Appetite; Body Weight; Diabetes Mellitus; Histamine Agonists; Imidazoles; Insulin; Leptin; Mice; Mice, Knockout; Obesity; Piperidines; Receptors, Histamine H3; Thiourea | 2006 |
Histamine H3 receptor agonist- and antagonist-evoked vacuous chewing movements in 6-OHDA-lesioned rats occurs in an absence of change in microdialysate dopamine levels.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Animals, Newborn; Benzazepines; Catalepsy; Corpus Striatum; Dialysis Solutions; Dopamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Male; Mastication; Microdialysis; Motor Activity; Oxidopamine; Piperidines; Rats; Rats, Wistar; Receptors, Histamine H3; Stereotyped Behavior; Thiourea | 2006 |
Distinctive role of central histamine H3 receptor in various orexigenic pathways.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Appetite; Histamine Agonists; Histamine H3 Antagonists; Hyperphagia; Imidazoles; Male; Mice; Mice, Inbred C57BL; Neuropeptide Y; Nociceptin; Opioid Peptides; Piperidines; Receptors, Histamine H3; Thiourea | 2008 |
Participation of histamine H3 receptors in experimental allergic rhinitis of mice.
Topics: Animals; Anti-Allergic Agents; Cetirizine; Chemotaxis, Leukocyte; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Synergism; Eosinophils; Female; Histamine Agonists; Histamine H1 Antagonists, Non-Sedating; Imidazoles; Mice; Mice, Inbred BALB C; Nasal Mucosa; Ovalbumin; Pruritus; Pyrrolidines; Receptors, Histamine H3; Rhinitis, Allergic, Perennial; Sneezing; Thiourea; Time Factors | 2008 |
Effects of histamine H(3) receptor activation on the behavioral-stimulant effects of methamphetamine and cocaine in mice and squirrel monkeys.
Topics: Animals; Behavior, Animal; Central Nervous System Stimulants; Cocaine; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Interactions; Histamine Agonists; Imidazoles; Male; Methamphetamine; Mice; Motor Activity; Receptors, Histamine H3; Reinforcement Schedule; Saimiri; Thiourea | 2009 |
The role of histamine 3 receptors in the control of food intake in a seasonal model of obesity: the Siberian hamster.
Topics: Animals; Body Temperature; Cell Line, Transformed; Cricetinae; Disease Models, Animal; Eating; Histamine; Imidazoles; Injections, Intraventricular; Motor Activity; Obesity; Phodopus; Photoperiod; Piperidines; Receptors, Histamine H3; Seasons; Thiourea; Transfection | 2009 |
JNJ-10181457, a selective non-imidazole histamine H(3) receptor antagonist, normalizes acetylcholine neurotransmission and has efficacy in translational rat models of cognition.
Topics: Acetylcholine; Animals; Anticonvulsants; Brain; Cholinesterase Inhibitors; Cognition; Conditioning, Operant; Donepezil; Drinking Behavior; Drug Evaluation, Preclinical; Histamine Agonists; Histamine Antagonists; Imidazoles; Indans; Learning; Microdialysis; Morpholines; Muscarinic Antagonists; Nootropic Agents; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Histamine H3; Scopolamine; Synaptic Transmission; Thiourea | 2009 |
The ameliorating effects of NMDA receptor agonists on histamine H1 antagonist-induced memory and hippocampal theta disruptions are prevented by the H3 receptor agonist in rats.
Topics: Animals; Cycloserine; Excitatory Amino Acid Agonists; Hippocampus; Histamine Agonists; Histamine H1 Antagonists; Imidazoles; Male; Maze Learning; Memory; Memory Disorders; Pyrilamine; Random Allocation; Rats; Receptors, N-Methyl-D-Aspartate; Space Perception; Spermidine; Theta Rhythm; Thiourea | 2009 |
Urethane, but not pentobarbitone, attenuates presynaptic receptor function in rats: a contribution to the choice of anaesthetic.
Topics: Adrenergic alpha-2 Receptor Agonists; Anesthetics; Animals; Cardiovascular System; Cerebral Cortex; Cyclohexanols; Decerebrate State; Electric Stimulation; Histamine Agonists; Imidazoles; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Pentobarbital; Radioligand Assay; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptors, Presynaptic; Thiourea; Urethane; Vasoconstrictor Agents | 2009 |
[Effect of H3R agonist, IMETIT on allergic rhinitis in guinea pigs].
Topics: Animals; Female; Guinea Pigs; Imidazoles; Male; Receptors, Histamine H3; Receptors, Neurokinin-1; Rhinitis, Allergic, Perennial; Substance P; Thiourea | 2010 |
[Substance P and its receptors are involved in the effect of histamine H3 receptor agonist, IMETIT on nasal allergic symptoms in guinea pigs].
Topics: Animals; Female; Guinea Pigs; Histamine Agonists; Imidazoles; Loratadine; Male; Nasal Mucosa; Receptors, Neurokinin-1; Rhinitis, Allergic, Perennial; RNA, Messenger; Substance P; Thiourea | 2010 |
Ciproxifan, a histamine H₃-receptor antagonist / inverse agonist, modulates methamphetamine-induced sensitization in mice.
Topics: Animals; Behavior, Animal; Brain; Brain-Derived Neurotrophic Factor; Central Nervous System Stimulants; Histamine Agonists; Histamine H3 Antagonists; Humans; Imidazoles; Male; Methamphetamine; Mice; Motor Activity; Receptors, N-Methyl-D-Aspartate; Schizophrenia; Thiourea | 2011 |
Histamine H3 receptor agonists decrease hypothalamic histamine levels and increase stereotypical biting in mice challenged with methamphetamine.
Topics: Animals; Behavior, Animal; Central Nervous System Stimulants; Histamine; Histamine Agonists; Hypothalamus; Imidazoles; Male; Methamphetamine; Methylhistamines; Mice; Motor Activity; Piperidines; Random Allocation; Stereotyped Behavior; Thiourea | 2011 |
Proxyfan acts as a neutral antagonist of histamine H3 receptors in the feeding-related hypothalamic ventromedial nucleus.
Topics: Animals; Eating; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Male; Mice; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Histamine H3; Thiourea; Ventromedial Hypothalamic Nucleus | 2012 |
Effects of L-histidine and histamine H3 receptor modulators on ethanol-induced sedation in mice.
Topics: Animals; Biphenyl Compounds; Brain; Ethanol; Female; Histidine; Hypnotics and Sedatives; Imidazoles; Mice; Nitriles; Piperidines; Pyrrolidines; Receptors, Histamine H3; Reflex, Righting; Thiourea | 2013 |
Identification and pharmacological characterization of the histamine H3 receptor in cultured rat astrocytes.
Topics: Animals; Animals, Newborn; Astrocytes; Binding, Competitive; Brain; Cells, Cultured; Ciprofloxacin; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Methylhistamines; Piperidines; Rats; Rats, Wistar; Receptors, Histamine H3; RNA, Messenger; Thiourea | 2013 |
Cardioprotective role of H₃R agonist imetit on isoproterenol-induced hemodynamic changes and oxidative stress in rats.
Topics: Adrenergic beta-Agonists; Animals; Antioxidants; Biomarkers; Blood Pressure; Body Height; Body Weight; Carbazoles; Cardiotonic Agents; Carvedilol; Heart Diseases; Heart Rate; Hemodynamics; Histamine Agonists; Humans; Imidazoles; Isoproterenol; Male; Myocardium; Oxidative Stress; Propanolamines; Rats; Rats, Wistar; Thiourea | 2015 |
Histamine H3 Receptor Agonist Imetit Attenuated Isoproterenol Induced Renin Angiotensin System and Sympathetic Nervous System Overactivity in Myocardial Infarction of Rats.
Topics: Angiotensin II; Animals; Antioxidants; Cardiotonic Agents; Histamine Agonists; Histamine H3 Antagonists; Imidazoles; Isoproterenol; Losartan; Male; Myocardial Infarction; Myocardium; Norepinephrine; Piperidines; Rats; Renin-Angiotensin System; Sympathetic Nervous System; Thiourea | 2016 |
Visualization of the activation of the histamine H3 receptor (H3R) using novel fluorescence resonance energy transfer biosensors and their potential application to the study of H3R pharmacology.
Topics: Bacterial Proteins; Biosensing Techniques; Cyclic AMP; Fluorescence Resonance Energy Transfer; Gene Expression; Green Fluorescent Proteins; HEK293 Cells; Histamine; Histamine Agonists; Histamine H3 Antagonists; Humans; Imidazoles; Kinetics; Luminescent Proteins; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Phosphorylation; Plasmids; Receptors, Histamine H3; Thiourea; Transfection; Tritium | 2018 |
Disruption of histamine/H
Topics: Animals; Cells, Cultured; Cicatrix; Collagen; Heart; Histamine; Imidazoles; Male; Mast Cells; Myocardial Infarction; Myofibroblasts; Rats; Rats, Wistar; Receptors, Histamine; Thiourea | 2019 |