imetit has been researched along with piperidines in 25 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 9 (36.00) | 18.2507 |
2000's | 11 (44.00) | 29.6817 |
2010's | 5 (20.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Ansay, M; Delaunois, A; Garbarg, M; Gustin, P | 1 |
Imamura, M; Lander, HM; Levi, R; Seyedi, N | 1 |
Banks, K; Merali, Z | 1 |
Buczko, W; Godlewski, G; Malinowska, B; Schlicker, E | 1 |
Bucher, B; Godlewski, G; Malinowska, B; Schlicker, E | 1 |
Allen, MC | 1 |
Flood, JF; Morley, JE; Uezu, K | 1 |
Schlicker, E; Werthwein, S; Zentner, J | 1 |
Murakami, Y; Nakamura, K; Okada, S; Wang, M; Yokotani, K | 1 |
Attarzadeh, M; Farzin, D | 1 |
Bacciottini, L; Bartolini, L; Blandina, P; Giovannini, MG; Greco, L | 1 |
Alves-Rodrigues, A; Lemstra, S; Leurs, R; Menge, WM; Timmerman, H; Vollinga, RC | 1 |
Blanco, I; Gomez-Ramirez, J; Ortiz, J | 1 |
Cassuto, J; Räntfors, J | 1 |
Arrang, JM; Cochois, V; Héron, A; Pillot, C; Rouleau, A; Schwartz, JC | 1 |
Chen, AS; Chen, HY; Ishihara, A; Kanatani, A; Kotani, H; Macneil, DJ; Miyamoto, Y; Shimamura, K; Takahashi, K; Tokita, S; Yoshimoto, R | 1 |
Biedka, I; Bortel, A; Brus, R; Dabrowska, J; Kostrzewa, RM; Nowak, P; Szczerbak, G; Słomian, G | 1 |
Kanatani, A; Tokita, S; Yoshimoto, R | 1 |
Barrett, P; Ebling, FJ; Enright, RA; Jethwa, PH; Murphy, M; Turnbull, Y; Warner, A | 1 |
Aluisio, L; Boggs, JD; Bonaventure, P; Fraser, IC; Galici, R; Lord, B; Lovenberg, TW | 1 |
Hall, FS; Kitanaka, J; Kitanaka, N; Morita, Y; Nishiyama, N; Takemura, M; Tanaka, K; Tatsuta, T; Uhl, GR | 1 |
Clapp, RH; Luckman, SM | 1 |
Closon, C; Didone, V; Nyssen, L; Quertemont, E; Quoilin, C; Tirelli, E | 1 |
Jurič, DM; Mele, T | 1 |
Akhtar, M; Hass, C; Khanam, R; Najmi, AK; Panda, BP | 1 |
25 other study(ies) available for imetit and piperidines
Article | Year |
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Modulation of acetylcholine, capsaicin and substance P effects by histamine H3 receptors in isolated perfused rabbit lungs.
Topics: Acetylcholine; Animals; Capillary Permeability; Capsaicin; Dose-Response Relationship, Drug; Drug Interactions; Endothelium; Female; Histamine Agonists; Histamine Antagonists; Imidazoles; In Vitro Techniques; Lung; Male; Nerve Fibers; Piperidines; Pulmonary Edema; Rabbits; Receptors, Histamine H3; Serotonin; Substance P; Thiourea | 1995 |
Functional identification of histamine H3-receptors in the human heart.
Topics: Cell Separation; Electric Stimulation; Exocytosis; Heart; Histamine Agonists; Histamine Antagonists; Humans; Imidazoles; In Vitro Techniques; Indoles; Methylhistamines; Myocardial Ischemia; Myocardium; Norepinephrine; Piperidines; Protein Kinase C; Receptors, Histamine H3; Synaptosomes; Thiourea | 1995 |
Does the histaminergic system mediate bombesin/GRP-induced suppression of food intake?
Topics: Animals; Behavior, Animal; Bombesin; Eating; Gastrin-Releasing Peptide; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Male; Methylhistamines; Motor Activity; Peptides; Piperidines; Rats; Rats, Sprague-Dawley; Satiation; Sincalide; Thiourea | 1994 |
Inhibitory H3 receptors on sympathetic nerves of the pithed rat: activation by endogenous histamine and operation in spontaneously hypertensive rats.
Topics: Adrenergic Fibers; Animals; Blood Pressure; Decerebrate State; Electric Stimulation; Histamine; Histamine Agonists; Histamine Antagonists; Hypertension; Imidazoles; Male; Methylhistamines; Piperidines; Pyrimethamine; Rats; Rats, Wistar; Receptors, Histamine H3; Thiourea; Vagotomy; Vascular Resistance | 1997 |
Identification of histamine H3 receptors in the tail artery from normotensive and spontaneously hypertensive rats.
Topics: Adrenergic alpha-2 Receptor Antagonists; Animals; Arteries; Electric Stimulation; Histamine; Histamine Agonists; Imidazoles; Male; Norepinephrine; Piperidines; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Histamine H3; Sympathetic Fibers, Postganglionic; Thiourea; Yohimbine | 1997 |
Agonist and antagonist effects of histamine H3 receptor ligands on 5-HT3 receptor-mediated ion currents in NG108-15 cells.
Topics: Animals; Cells, Cultured; Dose-Response Relationship, Drug; Histamine Agonists; Histamine Antagonists; Hybrid Cells; Imidazoles; Ion Channels; Isothiuronium; Membrane Potentials; Mice; Piperidines; Rats; Receptors, Histamine H3; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Serotonin Receptor Agonists; Thiourea | 1998 |
Effect of histamine H2 and H3 receptor modulation in the septum on post-training memory processing.
Topics: Animals; Cimetidine; Dimaprit; Histamine Agonists; Histamine Antagonists; Imidazoles; Limbic System; Male; Memory; Mice; Piperidines; Thiourea | 1998 |
Histamine H3 receptor-mediated inhibition of noradrenaline release in the human brain.
Topics: Animals; Brain; Cerebral Cortex; Dimethindene; Electric Stimulation; Hippocampus; Histamine; Histamine Agonists; Histamine Antagonists; Humans; Imidazoles; Male; Mice; Mice, Inbred Strains; Norepinephrine; Piperidines; Ranitidine; Receptors, Histamine H3; Thiourea; Tritium | 1999 |
Histamine H(3) receptor-mediated inhibition of endogenous acetylcholine release from the isolated, vascularly perfused rat stomach.
Topics: Acetylcholine; Animals; Atropine; Gastric Mucosa; GTP-Binding Proteins; Histamine; Imidazoles; Male; Methylhistamines; Perfusion; Pertussis Toxin; Piperidines; Rats; Rats, Wistar; Receptors, Histamine H3; Thiourea; Vagus Nerve; Virulence Factors, Bordetella | 2000 |
Influence of different histamine receptor agonists and antagonists on apomorphine-induced licking behavior in rat.
Topics: Animals; Apomorphine; Chlorpheniramine; Dimaprit; Diphenhydramine; Dopamine Agonists; Drug Interactions; Famotidine; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Male; Piperidines; Ranitidine; Rats; Rats, Sprague-Dawley; Stereotyped Behavior; Thiourea; Toluidines | 2000 |
Effects of histamine H3 receptor agonists and antagonists on cognitive performance and scopolamine-induced amnesia.
Topics: Amnesia; Analysis of Variance; Animals; Avoidance Learning; Behavior, Animal; Cognition; Histamine Agonists; Histamine Antagonists; Imidazoles; Injections, Intraperitoneal; Injections, Subcutaneous; Male; Methylhistamines; Pattern Recognition, Visual; Piperidines; Rats; Rats, Wistar; Receptors, Histamine H3; Scopolamine; Thiourea | 1999 |
Pharmacological analysis of immepip and imetit homologues. Further evidence for histamine H(3) receptor heterogeneity?
Topics: Animals; Cerebral Cortex; Guinea Pigs; Histamine Agonists; Imidazoles; Jejunum; Male; Piperidines; Radioligand Assay; Rats; Receptors, Histamine H3; Structure-Activity Relationship; Thiourea | 2001 |
Presynaptic H3 autoreceptors modulate histamine synthesis through cAMP pathway.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Brain; Bucladesine; Colforsin; Cyclic AMP; Drug Interactions; Histamine; Imidazoles; In Vitro Techniques; Male; Piperidines; Potassium; Rats; Rats, Sprague-Dawley; Receptors, Histamine H3; Thionucleotides; Thiourea | 2002 |
Role of histamine receptors in the regulation of edema and circulation postburn.
Topics: Animals; Burns; Clemastine; Edema; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Imidazoles; Male; Piperidines; Ranitidine; Rats; Rats, Sprague-Dawley; Receptors, Histamine; Receptors, Histamine H3; Regional Blood Flow; Skin; Statistics, Nonparametric; Thiourea | 2003 |
Cloning and expression of the mouse histamine H3 receptor: evidence for multiple isoforms.
Topics: Animals; Blotting, Northern; Brain; Chlorocebus aethiops; Cloning, Molecular; Competitive Bidding; COS Cells; Gene Expression; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; In Situ Hybridization; Iodine Radioisotopes; Isoenzymes; Mice; Piperidines; Radioligand Assay; Rats; Receptors, Histamine H3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiourea; Transfection | 2004 |
Therapeutic potential of histamine H3 receptor agonist for the treatment of obesity and diabetes mellitus.
Topics: Animals; Appetite; Body Weight; Diabetes Mellitus; Histamine Agonists; Imidazoles; Insulin; Leptin; Mice; Mice, Knockout; Obesity; Piperidines; Receptors, Histamine H3; Thiourea | 2006 |
Histamine H3 receptor agonist- and antagonist-evoked vacuous chewing movements in 6-OHDA-lesioned rats occurs in an absence of change in microdialysate dopamine levels.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Animals, Newborn; Benzazepines; Catalepsy; Corpus Striatum; Dialysis Solutions; Dopamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Male; Mastication; Microdialysis; Motor Activity; Oxidopamine; Piperidines; Rats; Rats, Wistar; Receptors, Histamine H3; Stereotyped Behavior; Thiourea | 2006 |
Distinctive role of central histamine H3 receptor in various orexigenic pathways.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Appetite; Histamine Agonists; Histamine H3 Antagonists; Hyperphagia; Imidazoles; Male; Mice; Mice, Inbred C57BL; Neuropeptide Y; Nociceptin; Opioid Peptides; Piperidines; Receptors, Histamine H3; Thiourea | 2008 |
The role of histamine 3 receptors in the control of food intake in a seasonal model of obesity: the Siberian hamster.
Topics: Animals; Body Temperature; Cell Line, Transformed; Cricetinae; Disease Models, Animal; Eating; Histamine; Imidazoles; Injections, Intraventricular; Motor Activity; Obesity; Phodopus; Photoperiod; Piperidines; Receptors, Histamine H3; Seasons; Thiourea; Transfection | 2009 |
JNJ-10181457, a selective non-imidazole histamine H(3) receptor antagonist, normalizes acetylcholine neurotransmission and has efficacy in translational rat models of cognition.
Topics: Acetylcholine; Animals; Anticonvulsants; Brain; Cholinesterase Inhibitors; Cognition; Conditioning, Operant; Donepezil; Drinking Behavior; Drug Evaluation, Preclinical; Histamine Agonists; Histamine Antagonists; Imidazoles; Indans; Learning; Microdialysis; Morpholines; Muscarinic Antagonists; Nootropic Agents; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Histamine H3; Scopolamine; Synaptic Transmission; Thiourea | 2009 |
Histamine H3 receptor agonists decrease hypothalamic histamine levels and increase stereotypical biting in mice challenged with methamphetamine.
Topics: Animals; Behavior, Animal; Central Nervous System Stimulants; Histamine; Histamine Agonists; Hypothalamus; Imidazoles; Male; Methamphetamine; Methylhistamines; Mice; Motor Activity; Piperidines; Random Allocation; Stereotyped Behavior; Thiourea | 2011 |
Proxyfan acts as a neutral antagonist of histamine H3 receptors in the feeding-related hypothalamic ventromedial nucleus.
Topics: Animals; Eating; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Male; Mice; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Histamine H3; Thiourea; Ventromedial Hypothalamic Nucleus | 2012 |
Effects of L-histidine and histamine H3 receptor modulators on ethanol-induced sedation in mice.
Topics: Animals; Biphenyl Compounds; Brain; Ethanol; Female; Histidine; Hypnotics and Sedatives; Imidazoles; Mice; Nitriles; Piperidines; Pyrrolidines; Receptors, Histamine H3; Reflex, Righting; Thiourea | 2013 |
Identification and pharmacological characterization of the histamine H3 receptor in cultured rat astrocytes.
Topics: Animals; Animals, Newborn; Astrocytes; Binding, Competitive; Brain; Cells, Cultured; Ciprofloxacin; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Methylhistamines; Piperidines; Rats; Rats, Wistar; Receptors, Histamine H3; RNA, Messenger; Thiourea | 2013 |
Histamine H3 Receptor Agonist Imetit Attenuated Isoproterenol Induced Renin Angiotensin System and Sympathetic Nervous System Overactivity in Myocardial Infarction of Rats.
Topics: Angiotensin II; Animals; Antioxidants; Cardiotonic Agents; Histamine Agonists; Histamine H3 Antagonists; Imidazoles; Isoproterenol; Losartan; Male; Myocardial Infarction; Myocardium; Norepinephrine; Piperidines; Rats; Renin-Angiotensin System; Sympathetic Nervous System; Thiourea | 2016 |