imetit and piperidines

imetit has been researched along with piperidines in 25 studies

Research

Studies (25)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's9 (36.00)18.2507
2000's11 (44.00)29.6817
2010's5 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ansay, M; Delaunois, A; Garbarg, M; Gustin, P1
Imamura, M; Lander, HM; Levi, R; Seyedi, N1
Banks, K; Merali, Z1
Buczko, W; Godlewski, G; Malinowska, B; Schlicker, E1
Bucher, B; Godlewski, G; Malinowska, B; Schlicker, E1
Allen, MC1
Flood, JF; Morley, JE; Uezu, K1
Schlicker, E; Werthwein, S; Zentner, J1
Murakami, Y; Nakamura, K; Okada, S; Wang, M; Yokotani, K1
Attarzadeh, M; Farzin, D1
Bacciottini, L; Bartolini, L; Blandina, P; Giovannini, MG; Greco, L1
Alves-Rodrigues, A; Lemstra, S; Leurs, R; Menge, WM; Timmerman, H; Vollinga, RC1
Blanco, I; Gomez-Ramirez, J; Ortiz, J1
Cassuto, J; Räntfors, J1
Arrang, JM; Cochois, V; Héron, A; Pillot, C; Rouleau, A; Schwartz, JC1
Chen, AS; Chen, HY; Ishihara, A; Kanatani, A; Kotani, H; Macneil, DJ; Miyamoto, Y; Shimamura, K; Takahashi, K; Tokita, S; Yoshimoto, R1
Biedka, I; Bortel, A; Brus, R; Dabrowska, J; Kostrzewa, RM; Nowak, P; Szczerbak, G; Słomian, G1
Kanatani, A; Tokita, S; Yoshimoto, R1
Barrett, P; Ebling, FJ; Enright, RA; Jethwa, PH; Murphy, M; Turnbull, Y; Warner, A1
Aluisio, L; Boggs, JD; Bonaventure, P; Fraser, IC; Galici, R; Lord, B; Lovenberg, TW1
Hall, FS; Kitanaka, J; Kitanaka, N; Morita, Y; Nishiyama, N; Takemura, M; Tanaka, K; Tatsuta, T; Uhl, GR1
Clapp, RH; Luckman, SM1
Closon, C; Didone, V; Nyssen, L; Quertemont, E; Quoilin, C; Tirelli, E1
Jurič, DM; Mele, T1
Akhtar, M; Hass, C; Khanam, R; Najmi, AK; Panda, BP1

Other Studies

25 other study(ies) available for imetit and piperidines

ArticleYear
Modulation of acetylcholine, capsaicin and substance P effects by histamine H3 receptors in isolated perfused rabbit lungs.
    European journal of pharmacology, 1995, Apr-24, Volume: 277, Issue:2-3

    Topics: Acetylcholine; Animals; Capillary Permeability; Capsaicin; Dose-Response Relationship, Drug; Drug Interactions; Endothelium; Female; Histamine Agonists; Histamine Antagonists; Imidazoles; In Vitro Techniques; Lung; Male; Nerve Fibers; Piperidines; Pulmonary Edema; Rabbits; Receptors, Histamine H3; Serotonin; Substance P; Thiourea

1995
Functional identification of histamine H3-receptors in the human heart.
    Circulation research, 1995, Volume: 77, Issue:1

    Topics: Cell Separation; Electric Stimulation; Exocytosis; Heart; Histamine Agonists; Histamine Antagonists; Humans; Imidazoles; In Vitro Techniques; Indoles; Methylhistamines; Myocardial Ischemia; Myocardium; Norepinephrine; Piperidines; Protein Kinase C; Receptors, Histamine H3; Synaptosomes; Thiourea

1995
Does the histaminergic system mediate bombesin/GRP-induced suppression of food intake?
    The American journal of physiology, 1994, Volume: 267, Issue:6 Pt 2

    Topics: Animals; Behavior, Animal; Bombesin; Eating; Gastrin-Releasing Peptide; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Male; Methylhistamines; Motor Activity; Peptides; Piperidines; Rats; Rats, Sprague-Dawley; Satiation; Sincalide; Thiourea

1994
Inhibitory H3 receptors on sympathetic nerves of the pithed rat: activation by endogenous histamine and operation in spontaneously hypertensive rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 355, Issue:2

    Topics: Adrenergic Fibers; Animals; Blood Pressure; Decerebrate State; Electric Stimulation; Histamine; Histamine Agonists; Histamine Antagonists; Hypertension; Imidazoles; Male; Methylhistamines; Piperidines; Pyrimethamine; Rats; Rats, Wistar; Receptors, Histamine H3; Thiourea; Vagotomy; Vascular Resistance

1997
Identification of histamine H3 receptors in the tail artery from normotensive and spontaneously hypertensive rats.
    Journal of cardiovascular pharmacology, 1997, Volume: 29, Issue:6

    Topics: Adrenergic alpha-2 Receptor Antagonists; Animals; Arteries; Electric Stimulation; Histamine; Histamine Agonists; Imidazoles; Male; Norepinephrine; Piperidines; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Histamine H3; Sympathetic Fibers, Postganglionic; Thiourea; Yohimbine

1997
Agonist and antagonist effects of histamine H3 receptor ligands on 5-HT3 receptor-mediated ion currents in NG108-15 cells.
    European journal of pharmacology, 1998, Nov-20, Volume: 361, Issue:2-3

    Topics: Animals; Cells, Cultured; Dose-Response Relationship, Drug; Histamine Agonists; Histamine Antagonists; Hybrid Cells; Imidazoles; Ion Channels; Isothiuronium; Membrane Potentials; Mice; Piperidines; Rats; Receptors, Histamine H3; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Serotonin Receptor Agonists; Thiourea

1998
Effect of histamine H2 and H3 receptor modulation in the septum on post-training memory processing.
    Psychopharmacology, 1998, Volume: 140, Issue:3

    Topics: Animals; Cimetidine; Dimaprit; Histamine Agonists; Histamine Antagonists; Imidazoles; Limbic System; Male; Memory; Mice; Piperidines; Thiourea

1998
Histamine H3 receptor-mediated inhibition of noradrenaline release in the human brain.
    Fundamental & clinical pharmacology, 1999, Volume: 13, Issue:1

    Topics: Animals; Brain; Cerebral Cortex; Dimethindene; Electric Stimulation; Hippocampus; Histamine; Histamine Agonists; Histamine Antagonists; Humans; Imidazoles; Male; Mice; Mice, Inbred Strains; Norepinephrine; Piperidines; Ranitidine; Receptors, Histamine H3; Thiourea; Tritium

1999
Histamine H(3) receptor-mediated inhibition of endogenous acetylcholine release from the isolated, vascularly perfused rat stomach.
    European journal of pharmacology, 2000, Mar-24, Volume: 392, Issue:1-2

    Topics: Acetylcholine; Animals; Atropine; Gastric Mucosa; GTP-Binding Proteins; Histamine; Imidazoles; Male; Methylhistamines; Perfusion; Pertussis Toxin; Piperidines; Rats; Rats, Wistar; Receptors, Histamine H3; Thiourea; Vagus Nerve; Virulence Factors, Bordetella

2000
Influence of different histamine receptor agonists and antagonists on apomorphine-induced licking behavior in rat.
    European journal of pharmacology, 2000, Sep-15, Volume: 404, Issue:1-2

    Topics: Animals; Apomorphine; Chlorpheniramine; Dimaprit; Diphenhydramine; Dopamine Agonists; Drug Interactions; Famotidine; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Male; Piperidines; Ranitidine; Rats; Rats, Sprague-Dawley; Stereotyped Behavior; Thiourea; Toluidines

2000
Effects of histamine H3 receptor agonists and antagonists on cognitive performance and scopolamine-induced amnesia.
    Behavioural brain research, 1999, Volume: 104, Issue:1-2

    Topics: Amnesia; Analysis of Variance; Animals; Avoidance Learning; Behavior, Animal; Cognition; Histamine Agonists; Histamine Antagonists; Imidazoles; Injections, Intraperitoneal; Injections, Subcutaneous; Male; Methylhistamines; Pattern Recognition, Visual; Piperidines; Rats; Rats, Wistar; Receptors, Histamine H3; Scopolamine; Thiourea

1999
Pharmacological analysis of immepip and imetit homologues. Further evidence for histamine H(3) receptor heterogeneity?
    Behavioural brain research, 2001, Oct-15, Volume: 124, Issue:2

    Topics: Animals; Cerebral Cortex; Guinea Pigs; Histamine Agonists; Imidazoles; Jejunum; Male; Piperidines; Radioligand Assay; Rats; Receptors, Histamine H3; Structure-Activity Relationship; Thiourea

2001
Presynaptic H3 autoreceptors modulate histamine synthesis through cAMP pathway.
    Molecular pharmacology, 2002, Volume: 61, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Brain; Bucladesine; Colforsin; Cyclic AMP; Drug Interactions; Histamine; Imidazoles; In Vitro Techniques; Male; Piperidines; Potassium; Rats; Rats, Sprague-Dawley; Receptors, Histamine H3; Thionucleotides; Thiourea

2002
Role of histamine receptors in the regulation of edema and circulation postburn.
    Burns : journal of the International Society for Burn Injuries, 2003, Volume: 29, Issue:8

    Topics: Animals; Burns; Clemastine; Edema; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Imidazoles; Male; Piperidines; Ranitidine; Rats; Rats, Sprague-Dawley; Receptors, Histamine; Receptors, Histamine H3; Regional Blood Flow; Skin; Statistics, Nonparametric; Thiourea

2003
Cloning and expression of the mouse histamine H3 receptor: evidence for multiple isoforms.
    Journal of neurochemistry, 2004, Volume: 90, Issue:6

    Topics: Animals; Blotting, Northern; Brain; Chlorocebus aethiops; Cloning, Molecular; Competitive Bidding; COS Cells; Gene Expression; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; In Situ Hybridization; Iodine Radioisotopes; Isoenzymes; Mice; Piperidines; Radioligand Assay; Rats; Receptors, Histamine H3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiourea; Transfection

2004
Therapeutic potential of histamine H3 receptor agonist for the treatment of obesity and diabetes mellitus.
    Proceedings of the National Academy of Sciences of the United States of America, 2006, Sep-12, Volume: 103, Issue:37

    Topics: Animals; Appetite; Body Weight; Diabetes Mellitus; Histamine Agonists; Imidazoles; Insulin; Leptin; Mice; Mice, Knockout; Obesity; Piperidines; Receptors, Histamine H3; Thiourea

2006
Histamine H3 receptor agonist- and antagonist-evoked vacuous chewing movements in 6-OHDA-lesioned rats occurs in an absence of change in microdialysate dopamine levels.
    European journal of pharmacology, 2006, Dec-15, Volume: 552, Issue:1-3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Animals, Newborn; Benzazepines; Catalepsy; Corpus Striatum; Dialysis Solutions; Dopamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Male; Mastication; Microdialysis; Motor Activity; Oxidopamine; Piperidines; Rats; Rats, Wistar; Receptors, Histamine H3; Stereotyped Behavior; Thiourea

2006
Distinctive role of central histamine H3 receptor in various orexigenic pathways.
    European journal of pharmacology, 2008, Jan-28, Volume: 579, Issue:1-3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Appetite; Histamine Agonists; Histamine H3 Antagonists; Hyperphagia; Imidazoles; Male; Mice; Mice, Inbred C57BL; Neuropeptide Y; Nociceptin; Opioid Peptides; Piperidines; Receptors, Histamine H3; Thiourea

2008
The role of histamine 3 receptors in the control of food intake in a seasonal model of obesity: the Siberian hamster.
    Behavioural pharmacology, 2009, Volume: 20, Issue:2

    Topics: Animals; Body Temperature; Cell Line, Transformed; Cricetinae; Disease Models, Animal; Eating; Histamine; Imidazoles; Injections, Intraventricular; Motor Activity; Obesity; Phodopus; Photoperiod; Piperidines; Receptors, Histamine H3; Seasons; Thiourea; Transfection

2009
JNJ-10181457, a selective non-imidazole histamine H(3) receptor antagonist, normalizes acetylcholine neurotransmission and has efficacy in translational rat models of cognition.
    Neuropharmacology, 2009, Volume: 56, Issue:8

    Topics: Acetylcholine; Animals; Anticonvulsants; Brain; Cholinesterase Inhibitors; Cognition; Conditioning, Operant; Donepezil; Drinking Behavior; Drug Evaluation, Preclinical; Histamine Agonists; Histamine Antagonists; Imidazoles; Indans; Learning; Microdialysis; Morpholines; Muscarinic Antagonists; Nootropic Agents; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Histamine H3; Scopolamine; Synaptic Transmission; Thiourea

2009
Histamine H3 receptor agonists decrease hypothalamic histamine levels and increase stereotypical biting in mice challenged with methamphetamine.
    Neurochemical research, 2011, Volume: 36, Issue:10

    Topics: Animals; Behavior, Animal; Central Nervous System Stimulants; Histamine; Histamine Agonists; Hypothalamus; Imidazoles; Male; Methamphetamine; Methylhistamines; Mice; Motor Activity; Piperidines; Random Allocation; Stereotyped Behavior; Thiourea

2011
Proxyfan acts as a neutral antagonist of histamine H3 receptors in the feeding-related hypothalamic ventromedial nucleus.
    British journal of pharmacology, 2012, Volume: 167, Issue:5

    Topics: Animals; Eating; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Male; Mice; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Histamine H3; Thiourea; Ventromedial Hypothalamic Nucleus

2012
Effects of L-histidine and histamine H3 receptor modulators on ethanol-induced sedation in mice.
    Behavioural brain research, 2013, Feb-01, Volume: 238

    Topics: Animals; Biphenyl Compounds; Brain; Ethanol; Female; Histidine; Hypnotics and Sedatives; Imidazoles; Mice; Nitriles; Piperidines; Pyrrolidines; Receptors, Histamine H3; Reflex, Righting; Thiourea

2013
Identification and pharmacological characterization of the histamine H3 receptor in cultured rat astrocytes.
    European journal of pharmacology, 2013, Nov-15, Volume: 720, Issue:1-3

    Topics: Animals; Animals, Newborn; Astrocytes; Binding, Competitive; Brain; Cells, Cultured; Ciprofloxacin; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Methylhistamines; Piperidines; Rats; Rats, Wistar; Receptors, Histamine H3; RNA, Messenger; Thiourea

2013
Histamine H3 Receptor Agonist Imetit Attenuated Isoproterenol Induced Renin Angiotensin System and Sympathetic Nervous System Overactivity in Myocardial Infarction of Rats.
    Drug research, 2016, Volume: 66, Issue:6

    Topics: Angiotensin II; Animals; Antioxidants; Cardiotonic Agents; Histamine Agonists; Histamine H3 Antagonists; Imidazoles; Isoproterenol; Losartan; Male; Myocardial Infarction; Myocardium; Norepinephrine; Piperidines; Rats; Renin-Angiotensin System; Sympathetic Nervous System; Thiourea

2016