Compounds > imetit

imetit and clozapine

imetit has been researched along with clozapine in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (71.43)29.6817
2010's2 (28.57)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chang, H; Erlander, MG; Lovenberg, TW; Pyati, J; Wilson, SJ1
Blevitt, J; Carruthers, N; Chai, W; Hofstra, CL; Jiang, X; Li, X; Liu, C; Lovenberg, TW; Ma, X; Pyati, J; Wilson, SJ1
Alston, J; Ames, RS; Bergsma, DJ; Boyce, R; Davenport, CM; Dytko, GM; Fitzgerald, LR; Herrity, NC; Hieble, JP; Li, X; Mannan, IJ; Michalovich, D; Sarau, HM; Tan, KB; Tierney, LA; Vawter, L; Wilson, S; Wu, H; Zhu, Y1
Kuei, C; Liu, C; Lovenberg, TW; Wilson, SJ1
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM1
Berlin, M; Boyce, CW; Ruiz, Mde L1
de Esch, IJ; de Graaf, C; Istyastono, EP; Kooistra, AJ; Leurs, R; Lim, HD; Nijmeijer, S; Roumen, L; van de Stolpe, A; Vischer, HF1

Reviews

1 review(s) available for imetit and clozapine

ArticleYear
Histamine H3 receptor as a drug discovery target.
    Journal of medicinal chemistry, 2011, Jan-13, Volume: 54, Issue:1

    Topics: Animals; Drug Discovery; Drug Industry; Drug Inverse Agonism; Histamine Agonists; Histamine Antagonists; Humans; Ligands; Private Sector; Receptors, Histamine H3

2011

Other Studies

6 other study(ies) available for imetit and clozapine

ArticleYear
Cloning of rat histamine H(3) receptor reveals distinct species pharmacological profiles.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 293, Issue:3

    Topics: Adenylyl Cyclase Inhibitors; Amino Acid Sequence; Animals; Cloning, Molecular; Dose-Response Relationship, Drug; Humans; Methylhistamines; Molecular Sequence Data; Rats; Receptors, Histamine H3; Recombinant Proteins; RNA, Messenger

2000
Cloning and pharmacological characterization of a fourth histamine receptor (H(4)) expressed in bone marrow.
    Molecular pharmacology, 2001, Volume: 59, Issue:3

    Topics: Adenylyl Cyclases; Amino Acid Sequence; Bone Marrow; Cloning, Molecular; Histamine; Humans; Methylhistamines; Molecular Sequence Data; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; RNA, Messenger; Sequence Homology, Amino Acid; Tissue Distribution; Tritium

2001
Cloning, expression, and pharmacological characterization of a novel human histamine receptor.
    Molecular pharmacology, 2001, Volume: 59, Issue:3

    Topics: Amino Acid Sequence; Animals; Calcium; Cloning, Molecular; Dose-Response Relationship, Drug; Gene Expression; Genes, Reporter; Histamine; Humans; Luciferases; Mice; Molecular Sequence Data; Radioligand Assay; Receptors, Histamine; Receptors, Histamine H3; Sequence Homology, Amino Acid; Tissue Distribution; Tritium

2001
Comparison of human, mouse, rat, and guinea pig histamine H4 receptors reveals substantial pharmacological species variation.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 299, Issue:1

    Topics: Amino Acid Sequence; Animals; Calcium; Cell Line; Cloning, Molecular; COS Cells; Cyclic AMP; DNA Fragmentation; Guinea Pigs; Humans; Mice; Molecular Sequence Data; Radioligand Assay; Rats; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Reverse Transcriptase Polymerase Chain Reaction; Species Specificity; Transfection

2001
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:3

    Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4

2005
Molecular determinants of ligand binding modes in the histamine H(4) receptor: linking ligand-based three-dimensional quantitative structure-activity relationship (3D-QSAR) models to in silico guided receptor mutagenesis studies.
    Journal of medicinal chemistry, 2011, Dec-08, Volume: 54, Issue:23

    Topics: Cell Line, Tumor; Histamine Antagonists; Humans; Hydrophobic and Hydrophilic Interactions; Imidazoles; Ligands; Models, Molecular; Molecular Conformation; Molecular Dynamics Simulation; Mutagenesis, Site-Directed; Quantitative Structure-Activity Relationship; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H3; Receptors, Histamine H4; Stereoisomerism; Thiourea

2011