Page last updated: 2024-09-03

imatinib mesylate and kw 2449

imatinib mesylate has been researched along with kw 2449 in 1 studies

Compound Research Comparison

Studies
(imatinib mesylate)
Trials
(imatinib mesylate)
Recent Studies (post-2010)
(imatinib mesylate)
Studies
(kw 2449)
Trials
(kw 2449)
Recent Studies (post-2010) (kw 2449)
11,4779605,77323020

Protein Interaction Comparison

ProteinTaxonomyimatinib mesylate (IC50)kw 2449 (IC50)
Replicase polyprotein 1abBetacoronavirus England 13.6
Tyrosine-protein kinase ABL1Homo sapiens (human)0.009
Receptor-type tyrosine-protein kinase FLT3Homo sapiens (human)0.0066

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Attkisson, E; Dai, Y; Grant, S; Jordan, N; Kolluri, N; Kramer, L; Muschen, M; Nguyen, N; Nguyen, T1

Other Studies

1 other study(ies) available for imatinib mesylate and kw 2449

ArticleYear
HDAC inhibitors potentiate the activity of the BCR/ABL kinase inhibitor KW-2449 in imatinib-sensitive or -resistant BCR/ABL+ leukemia cells in vitro and in vivo.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 2011, May-15, Volume: 17, Issue:10

    Topics: Adult; Animals; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Cell Line, Tumor; Drug Resistance, Neoplasm; Drug Synergism; Fusion Proteins, bcr-abl; Histone Deacetylase Inhibitors; Humans; Imatinib Mesylate; Indazoles; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Mice; Mice, Inbred BALB C; Mice, SCID; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Xenograft Model Antitumor Assays

2011