Page last updated: 2024-09-03

ilomastat and pepstatin

ilomastat has been researched along with pepstatin in 2 studies

Compound Research Comparison

Studies
(ilomastat)
Trials
(ilomastat)
Recent Studies (post-2010)
(ilomastat)
Studies
(pepstatin)
Trials
(pepstatin)
Recent Studies (post-2010) (pepstatin)
1030456960125

Protein Interaction Comparison

ProteinTaxonomyilomastat (IC50)pepstatin (IC50)
Pepsin ASus scrofa (pig)0.011
ReninHomo sapiens (human)1.9333
Cathepsin DHomo sapiens (human)0.3597
Procathepsin LHomo sapiens (human)0.8
Cathepsin BHomo sapiens (human)4.26
Candidapepsin-2Candida albicans0.09
Pepsin A-5Homo sapiens (human)0.059
Cathepsin EHomo sapiens (human)0.5558
Plasmepsin-1Plasmodium falciparum (malaria parasite P. falciparum)0.0009
Plasmepsin-2Plasmodium falciparum (malaria parasite P. falciparum)0.0005
Cathepsin D Bos taurus (cattle)0.0235
Disintegrin and metalloproteinase domain-containing protein 9Homo sapiens (human)0.0563
Plasmepsin 4 Plasmodium falciparum (malaria parasite P. falciparum)0.0003
Cysteine proteaseLeishmania donovani0.16
Protease Human immunodeficiency virus 10.947

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's1 (50.00)2.80

Authors

AuthorsStudies
Eksioglu, EA; Kwan, JC; Liu, C; Luesch, H; Paul, VJ1
Dranchak, PK; Huang, R; Inglese, J; Lamy, L; Oliphant, E; Queme, B; Tao, D; Wang, Y; Xia, M1

Other Studies

2 other study(ies) available for ilomastat and pepstatin

ArticleYear
Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation.
    Journal of medicinal chemistry, 2009, Sep-24, Volume: 52, Issue:18

    Topics: Amino Acids; Animals; Antigen Presentation; Cathepsin E; Cell Line, Tumor; Cyanobacteria; Dendritic Cells; Humans; Inhibitory Concentration 50; Magnetic Resonance Spectroscopy; Models, Molecular; Molecular Conformation; Oceans and Seas; Oligopeptides; Protease Inhibitors; Spectrometry, Mass, Electrospray Ionization; Substrate Specificity

2009
In vivo quantitative high-throughput screening for drug discovery and comparative toxicology.
    Disease models & mechanisms, 2023, 03-01, Volume: 16, Issue:3

    Topics: Animals; Caenorhabditis elegans; Drug Discovery; High-Throughput Screening Assays; Humans; Proteomics; Small Molecule Libraries

2023