Page last updated: 2024-08-23

idazoxan and tracizoline

idazoxan has been researched along with tracizoline in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (14.29)18.2507
2000's4 (57.14)29.6817
2010's1 (14.29)24.3611
2020's1 (14.29)2.80

Authors

AuthorsStudies
Baurin, N; Guillaumet, G; Marot, C; Mérour, JY; Morin-Allory, L; Payard, M; Renard, P; Vangrevelinghe, E1
Arrault, A; Guillaumet, G; Mérour, JY; Pfeiffer, B; Renard, P; Rettori, MC; Scalbert, E; Touzeau, F1
Agbaba, D; Azzali, E; Costantino, G; Glisic, S; Laurila, JM; Nikolic, K; Perovic, V; Pieroni, M; Radi, M; Scheinin, M; Srdic-Rajic, T; Tassini, S; Veljkovic, N; Vucicevic, J1
Abás, S; Bagán, A; Brea, J; Brocos-Mosquera, I; Callado, LF; Daelemans, D; de Jonghe, S; Djikic, T; Escolano, C; García-Fuster, MJ; García-Sevilla, JA; Griñán-Ferré, C; Hernández-Hernández, E; Loza, MI; Luque, FJ; Molins, E; Muguruza, C; Naesens, L; Nikolic, K; Pallàs, M; Pérez, B; Pérez-Lozano, P; Radan, M; Rodríguez-Arévalo, S; Vasilopoulou, F1
Bousquet, P; Brasili, L; Carotti, A; Carrieri, A; Cavagna, R; Dontenwill, M; Gentili, F; Giannella, M; Leonetti, F; Piergentili, A; Pigini, M; Quaglia, W1
Gentili, F; Massi, M; Panocka, I; Pigini, M; Polidori, C; Quaglia, W1
Cardinaletti, C; Carrieri, A; Gentili, F; Ghelfi, F; Mattioli, L; Perfumi, M; Pigini, M; Vesprini, C1

Other Studies

7 other study(ies) available for idazoxan and tracizoline

ArticleYear
3D-QSAR CoMFA study on imidazolinergic I(2) ligands: a significant model through a combined exploration of structural diversity and methodology.
    Journal of medicinal chemistry, 2000, Mar-23, Volume: 43, Issue:6

    Topics: Drug Design; Imidazoles; Imidazoline Receptors; Ligands; Models, Molecular; Molecular Structure; Receptors, Drug; Structure-Activity Relationship

2000
Synthesis and biological evaluation of new 2-(4,5-dihydro-1H-imidazol-2-yl)-3,4-dihydro-2H-1,4-benzoxazine derivatives.
    Journal of medicinal chemistry, 2003, May-08, Volume: 46, Issue:10

    Topics: Adrenal Medulla; Animals; Antihypertensive Agents; Binding Sites; Blood Pressure; Cattle; Frontal Lobe; Heart Rate; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Kidney; Oxazines; Rabbits; Radioligand Assay; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Drug; Stereoisomerism; Structure-Activity Relationship

2003
A combined ligand- and structure-based approach for the identification of rilmenidine-derived compounds which synergize the antitumor effects of doxorubicin.
    Bioorganic & medicinal chemistry, 2016, 07-15, Volume: 24, Issue:14

    Topics: Adrenergic alpha-Agonists; Antibiotics, Antineoplastic; Apoptosis; Doxorubicin; Drug Synergism; Humans; K562 Cells; Ligands; Molecular Structure; Oxazoles; Receptors, Adrenergic, alpha-2; Rilmenidine

2016
Bicyclic α-Iminophosphonates as High Affinity Imidazoline I
    Journal of medicinal chemistry, 2020, 04-09, Volume: 63, Issue:7

    Topics: Alzheimer Disease; Animals; Chlorocebus aethiops; Cycloaddition Reaction; Dogs; Female; HeLa Cells; Hippocampus; Humans; Imidazoles; Imidazoline Receptors; Ligands; Madin Darby Canine Kidney Cells; Mice; Molecular Structure; Nootropic Agents; Organophosphonates; Quantitative Structure-Activity Relationship; Vero Cells

2020
Ligand binding to I2 imidazoline receptor: the role of lipophilicity in quantitative structure-activity relationship models.
    Bioorganic & medicinal chemistry, 1998, Volume: 6, Issue:12

    Topics: Animals; Binding, Competitive; Cerebral Cortex; Clonidine; Idazoxan; Imidazoles; Imidazoline Receptors; Kidney; Kinetics; Ligands; Models, Molecular; Molecular Conformation; Molecular Structure; Rabbits; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-2; Receptors, Drug; Regression Analysis; Solubility; Static Electricity; Structure-Activity Relationship

1998
Hyperphagic effect of novel compounds with high affinity for imidazoline I(2) binding sites.
    European journal of pharmacology, 2000, Mar-24, Volume: 392, Issue:1-2

    Topics: Animals; Binding Sites; Dose-Response Relationship, Drug; Drinking; Eating; Idazoxan; Imidazoles; Imidazoline Receptors; Male; Rats; Rats, Wistar; Receptors, Drug

2000
Involvement of I2-imidazoline binding sites in positive and negative morphine analgesia modulatory effects.
    European journal of pharmacology, 2006, Dec-28, Volume: 553, Issue:1-3

    Topics: Adrenergic alpha-Antagonists; Analgesics, Opioid; Animals; Benzofurans; CHO Cells; Cricetinae; Idazoxan; Imidazoles; Imidazoline Receptors; Male; Mice; Models, Molecular; Morphine; Naloxone; Narcotic Antagonists; Pain Measurement; Radioligand Assay; Reaction Time; Receptors, Adrenergic, alpha-2; Receptors, Drug; Receptors, Opioid, mu; Yohimbine

2006