idazoxan has been researched along with phentolamine in 55 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 24 (43.64) | 18.7374 |
1990's | 24 (43.64) | 18.2507 |
2000's | 6 (10.91) | 29.6817 |
2010's | 1 (1.82) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Harsing, LG; Somogyi, GT; Szabo, L; Szantay, C; Toth, I; Vizi, ES | 1 |
Butler, RC; Chapleo, CB; Doxey, JC; Myers, PL; Roach, AG; Smith, CF | 1 |
Agbaba, D; Filipic, S; Nikolic, K | 1 |
Warbrick, EV; Ward, SA | 1 |
Schwietert, R; Van Zwieten, PA; Wilffert, B; Wilhelm, D | 1 |
Leslie, FM; Raymon, HK; Smith, TD | 1 |
Chan, SL; Morgan, NG; Stillings, MR | 1 |
Butcher, SP; Clark, AJ; Winn, P | 1 |
Czerwiec, E; De Backer, JP; De Potter, W; De Vos, H; Vauquelin, G | 1 |
Horváth, E; Jaszlits, L; Rabloczky, G | 1 |
Baldwin, DL; Miller, JM; Nuttall, AL; Ohlsén, KA | 1 |
Carpéné, C; Galitzky, J; Lafontan, M; Langin, D; Larrouy, D | 1 |
Majewski, H; Rump, LC | 1 |
Convents, A; Convents, D; De Backer, JP; De Keyser, J; Vauquelin, G | 1 |
Couture, R; Laneuville, O; Reader, TA | 1 |
Harbison, RD; James, RC; Kerger, BD; Roberts, SM | 1 |
Cattaneo, AG; Doxey, JC; Efendic, S; Ostenson, CG | 1 |
Fischer, MR; Limberger, N; Starke, K; Wichmann, T | 1 |
Bickford-Wimer, PC; Freedman, R; Parfitt, KD | 1 |
Rand, MJ; Standford-Starr, CA; Story, DF | 1 |
Heepe, P; Starke, K | 1 |
Loiacono, RE; Rand, MJ; Story, DF | 1 |
Puurunen, J | 1 |
Dickinson, KE; McKernan, RM; Miles, CM; Sever, PS | 1 |
Coupry, I; Dausse, JP; Parini, A; Podevin, RA | 1 |
Bennett, T; Gardiner, SM | 1 |
Edwall, B; Gazelius, B | 1 |
Bucci, TJ; Gandy, J; Harbison, RD; James, RC; Kerger, BD; Roberts, SM | 1 |
Appleby, GJ; Clark, MG; Colquhoun, EQ; Edwards, SJ; McKinstry, WJ; Rattigan, S; Richter, EA | 1 |
Brown, MJ; Burrin, JM; Struthers, AD | 1 |
Convents, A; De Backer, JP; Vauquelin, G | 1 |
Hamilton, CA; Hannah, JA; Reid, JL | 1 |
North, RA; Yoshimura, M | 1 |
Galzin, AM; Langer, SZ; Moret, C | 1 |
Doak, GJ; Reid, AR; Sawynok, J | 1 |
Cooke, HJ; Wood, JD; Zafirov, DH | 1 |
Fukuda, H; Fukushima, C; Ono, H | 1 |
Amabeoku, G; Chandomba, R | 1 |
Amabeoku, GJ | 1 |
Oriowo, MA | 1 |
Göthert, M; Molderings, GJ | 1 |
Berggren, PO; Efanov, AM; Efanova, IB; Efendić, S; Gold, G; Larsson, O; Ostenson, CG; Zaitsev, SV | 1 |
Dunne, MJ; Hashmi, MN; Kane, C; Shepherd, RM; Squires, PE | 1 |
Coupar, IM; Liu, L | 1 |
Regunathan, S; Reis, DJ; Sastre, M | 1 |
Caramona, MM; Figueiredo, IV; Guimarães, S; Moura, D; Paiva, MQ | 1 |
Hasselblatt, A; Kowalewski, R; Leupolt, L; Rustenbeck, I | 1 |
Hasselblatt, A; Köpp, M; Leupolt, L; Ratzka, P; Rustenbeck, I | 1 |
Cox, SL; Gaiser, EG; Meyer, A; Starke, K; Trendelenburg, AU | 1 |
Elliott, J; Morgan, NG; Mourtada, M; Smith, SA | 1 |
Anderson, M; Burleigh, D | 1 |
Berlan, M; Crampes, F; Daviaud, D; Gesta, S; Hejnova, J; Saulnier-Blache, JS; Stich, V; Valet, P | 1 |
Fagerholm, V; Hein, L; Philipp, M; Scheinin, M | 1 |
Dahms, HU; Jin, T; Qian, PY | 1 |
Côrrea, FM; Crestani, CC; Fabri, DR; Gomes, FV; Hott, SC; Reis, DG; Resstel, LB | 1 |
55 other study(ies) available for idazoxan and phentolamine
Article | Year |
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Berbanes: a new class of selective alpha 2-adrenoceptor antagonists.
Topics: Adrenergic alpha-Antagonists; Alkaloids; Animals; Berberine Alkaloids; Chemical Phenomena; Chemistry; Dioxanes; Guinea Pigs; Idazoxan; Ileum; Male; Muscle Contraction; Phentolamine; Prazosin; Pulmonary Artery; Rabbits; Rats; Receptors, Adrenergic, alpha; Vas Deferens; Yohimbine | 1987 |
alpha-adrenoreceptor reagents. 1. Synthesis of some 1,4-benzodioxans as selective presynaptic alpha 2-adrenoreceptor antagonists and potential antidepressants.
Topics: Adrenergic alpha-Antagonists; Animals; Antidepressive Agents; Dioxins; Dose-Response Relationship, Drug; Idazoxan; Male; Mice; Phenylephrine; Rats; Rats, Inbred Strains; Structure-Activity Relationship; Synapses; Vas Deferens | 1983 |
QSAR study of imidazoline antihypertensive drugs.
Topics: Antihypertensive Agents; Binding Sites; Imidazoline Receptors; Imidazolines; Ligands; Models, Molecular; Molecular Structure; Quantitative Structure-Activity Relationship | 2008 |
The effect of catecholamines and catecholamine antagonists on the third larval moult of Dirofilaria immitis in vitro.
Topics: Animals; Catecholamines; Dioxanes; Dirofilaria immitis; Idazoxan; Isoproterenol; Larva; Norepinephrine; Phentolamine; Propranolol | 1992 |
The effect of some alpha-adrenoceptor antagonists on spontaneous myogenic activity in the rat portal vein and the putative involvement of ATP-sensitive K+ channels.
Topics: Adenosine Triphosphate; Adrenergic alpha-Antagonists; Animals; Dioxanes; Dose-Response Relationship, Drug; Idazoxan; In Vitro Techniques; Male; Phentolamine; Portal Vein; Potassium Channels; Prazosin; Rats; Rats, Inbred Strains; Vasoconstriction; Yohimbine | 1992 |
Further pharmacological characterization of [3H]idazoxan binding sites in rat brain: evidence for predominant labeling of alpha 2-adrenergic receptors.
Topics: Adrenergic alpha-Antagonists; Animals; Brain; Buffers; Dioxanes; Epinephrine; Idazoxan; Male; Phentolamine; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Receptors, Drug; Tritium; Yohimbine | 1992 |
Mechanisms involved in stimulation of insulin secretion by the hypoglycaemic alpha-adrenergic antagonist, DG-5128.
Topics: Adrenergic alpha-Antagonists; Animals; Benzofurans; Diazoxide; Dioxanes; Dose-Response Relationship, Drug; Hypoglycemic Agents; Idazoxan; Imidazoles; In Vitro Techniques; Islets of Langerhans; Kinetics; Male; Phentolamine; Rats; Rats, Inbred Strains | 1991 |
Evidence for functional separation of alpha-1 and alpha-2 noradrenaline receptors by pre-synaptic terminal re-uptake mechanisms.
Topics: Adrenergic alpha-Antagonists; Animals; Chromatography, High Pressure Liquid; Cocaine; Dioxanes; Eating; Hydroxydopamines; Idazoxan; In Vitro Techniques; Male; Microinjections; Nerve Endings; Norepinephrine; Oxidopamine; Paraventricular Hypothalamic Nucleus; Phentolamine; Rats; Receptors, Adrenergic, alpha; Synapses | 1991 |
[3H]rauwolscine behaves as an agonist for the 5-HT1A receptors in human frontal cortex membranes.
Topics: Adrenergic alpha-Antagonists; Aged; Dioxanes; Frontal Lobe; GTP-Binding Proteins; Guanine Nucleotides; Humans; Idazoxan; In Vitro Techniques; Kinetics; Membranes; Middle Aged; Mollusk Venoms; Phentolamine; Receptors, Adrenergic, alpha; Receptors, Serotonin; Yohimbine | 1991 |
GYKI-12743 a new postsynaptic vascular alpha-adrenoceptor antagonist.
Topics: Adrenergic alpha-Antagonists; Animals; Azepines; Blood Pressure; Clonidine; Decerebrate State; Dioxanes; Electric Stimulation; Heart Rate; Idazoxan; Phentolamine; Phenylephrine; Pyridazines; Rats; Rats, Inbred Strains; Yohimbine | 1991 |
Influence of topically applied adrenergic agents on cochlear blood flow.
Topics: Administration, Topical; Albuterol; Animals; Azepines; Cochlea; Dioxanes; Epinephrine; Female; Guinea Pigs; Idazoxan; Isoproterenol; Lasers; Male; Norepinephrine; Phentolamine; Phenylephrine; Prazosin; Propranolol; Round Window, Ear; Sympathomimetics | 1991 |
Non-adrenergic sites for imidazolines are not directly involved in the alpha 2-adrenergic antilipolytic effect of UK 14304 in rat adipocytes.
Topics: Adipose Tissue; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding Sites; Binding, Competitive; Brimonidine Tartrate; Bucladesine; Cell Membrane; Colforsin; Dioxanes; Idazoxan; Kinetics; Lipolysis; Phentolamine; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine | 1990 |
Modulation of norepinephrine release through alpha 1- and alpha 2-adrenoceptors in rat isolated kidney.
Topics: Adrenergic alpha-Agonists; Animals; Clonidine; Dioxanes; Electric Stimulation; Idazoxan; In Vitro Techniques; Kidney; Male; Norepinephrine; Phentolamine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Sympathetic Nervous System | 1987 |
High affinity binding of 3H rauwolscine and 3H RX781094 to alpha 2 adrenergic receptors and non-stereoselective sites in human and rabbit brain cortex membranes.
Topics: Adrenergic alpha-Antagonists; Animals; Binding Sites; Cerebral Cortex; Dioxanes; Dioxins; Epinephrine; Humans; Idazoxan; In Vitro Techniques; Phentolamine; Rabbits; Receptors, Adrenergic, alpha; Receptors, Serotonin; Species Specificity; Stereoisomerism; Tritium; Yohimbine | 1989 |
Intrathecal bradykinin acts presynaptically on spinal noradrenergic terminals to produce antinociception in the rat.
Topics: Adrenergic alpha-Antagonists; Analgesics; Animals; Biogenic Monoamines; Bradykinin; Catecholamines; Catheters, Indwelling; Dioxanes; Endorphins; Hydroxydopamines; Idazoxan; Injections, Spinal; Kallidin; Male; Naloxone; Oxidopamine; Phentolamine; Prazosin; Propranolol; Rats; Rats, Inbred Strains; Reaction Time; Spinal Cord; Yohimbine | 1989 |
Antagonism of bromobenzene-induced hepatotoxicity by the alpha-adrenoreceptor blocking agents phentolamine and idazoxan: role of hypothermia.
Topics: Adrenergic alpha-Antagonists; Animals; Body Temperature; Bromobenzenes; Dioxanes; Dioxins; Idazoxan; Liver; Male; Mice; Mice, Inbred Strains; Phentolamine; Sympathetic Nervous System | 1989 |
Alpha-adrenoceptors and insulin release from pancreatic islets of normal and diabetic rats.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Brimonidine Tartrate; Diabetes Mellitus, Experimental; Dioxanes; Female; Glucose; Idazoxan; Insulin; Islets of Langerhans; Male; Phentolamine; Prazosin; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Streptozocin; Yohimbine | 1989 |
Phentolamine blocks presynaptic serotonin autoreceptors in rabbit and rat brain cortex.
Topics: Adrenergic alpha-Antagonists; Animals; Cerebral Cortex; Dioxanes; Electric Stimulation; Female; Idazoxan; In Vitro Techniques; Male; Norepinephrine; Phentolamine; Quipazine; Rabbits; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Sex Factors | 1989 |
Electrophysiological effects of locally applied noradrenergic agents at cerebellar Purkinje neurons: receptor specificity.
Topics: Action Potentials; Animals; Dioxanes; Dioxins; Idazoxan; Neural Inhibition; Norepinephrine; Phencyclidine; Phentolamine; Purkinje Cells; Rats; Rats, Inbred F344; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Yohimbine | 1988 |
Evidence for the involvement of alpha 1-adrenoceptors in negative feedback regulation of noradrenergic transmitter release in rat atria.
Topics: Adrenergic alpha-Antagonists; Animals; Dioxanes; Electric Stimulation; Feedback; Female; Heart Atria; Idazoxan; Methoxamine; Neuromuscular Junction; Norepinephrine; Phentolamine; Prazosin; Rats; Receptors, Adrenergic, alpha; Synaptic Transmission | 1985 |
Alpha-adrenoceptor antagonists and the release of noradrenaline in rabbit cerebral cortex slices: support for the alpha-autoreceptor hypothesis.
Topics: Adrenergic alpha-Antagonists; Animals; Cerebral Cortex; Cocaine; Dioxanes; Electric Stimulation; Female; Idazoxan; In Vitro Techniques; Male; Norepinephrine; Phentolamine; Rabbits; Secologanin Tryptamine Alkaloids; Tetraethylammonium Compounds | 1985 |
Interaction between the inhibitory action of acetylcholine and the alpha-adrenoceptor autoinhibitory feedback system on release of [3H]-noradrenaline from rat atria and rabbit ear artery.
Topics: Acetylcholine; Adrenergic alpha-Antagonists; Animals; Arteries; Catecholamines; Clonidine; Dioxanes; Ear; Electric Stimulation; Feedback; Female; Heart Atria; Idazoxan; Imidazolines; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Myocardial Contraction; Myocardium; Norepinephrine; Phentolamine; Rabbits; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine | 1985 |
Role of putative neurotransmitters in the central gastric antisecretory effect of prostaglandin E2 in rats.
Topics: 5,6-Dihydroxytryptamine; Adrenergic alpha-Antagonists; Animals; Dinoprostone; Dioxanes; Female; Fenclonine; Gastric Juice; Histamine Antagonists; Hydroxydopamines; Idazoxan; Injections, Intraventricular; Male; Naloxone; Neurotransmitter Agents; Oxidopamine; Phentolamine; Propranolol; Prostaglandins E; Rats; Rats, Inbred Strains; Sulpiride; Theophylline | 1985 |
Heterogeneity between soluble human and rabbit splenic alpha 2-adrenoceptors.
Topics: Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Dioxanes; Epinephrine; Humans; Idazoxan; Lectins; Oxymetazoline; Phentolamine; Prazosin; Quinolizines; Quinoxalines; Rabbits; Receptors, Adrenergic, alpha; Solubility; Spleen; Sulfhydryl Reagents; Yohimbine | 1986 |
Evidence for imidazoline binding sites in basolateral membranes from rabbit kidney.
Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Cell Membrane; Dioxanes; Dioxins; Epithelium; Idazoxan; Imidazoles; Kidney; Phentolamine; Rabbits; Receptors, Adrenergic, alpha; Receptors, Cell Surface; Structure-Activity Relationship; Yohimbine | 1987 |
Involvement of beta 2-adrenoceptor-mediated mechanisms in the cardiovascular responses to alpha 1- and alpha 2-adrenoceptor antagonism in conscious, unrestrained, Long Evans and Brattleboro rats.
Topics: Adrenal Medulla; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Blood Pressure; Captopril; Dioxanes; Heart Rate; Hemodynamics; Idazoxan; Male; Phentolamine; Prazosin; Propanolamines; Rats; Rats, Brattleboro; Receptors, Adrenergic, beta; Restraint, Physical | 1988 |
Effects of the alpha-adrenoceptor antagonists phentolamine, phenoxybenzamine, and idazoxan on sympathetic blood flow control in the periodontal ligament of the cat.
Topics: Adrenergic alpha-Antagonists; Animals; Cats; Dioxanes; Dioxins; Electric Stimulation; Epinephrine; Female; Idazoxan; Male; Norepinephrine; Periodontal Ligament; Phenoxybenzamine; Phentolamine; Regional Blood Flow; Sympathetic Nervous System; Vasomotor System | 1988 |
Antagonism of bromobenzene-induced hepatotoxicity by the alpha-adrenergic blocking agents, phentolamine and idazoxan.
Topics: Adrenergic alpha-Antagonists; Alanine Transaminase; Animals; Bromobenzenes; Chemical and Drug Induced Liver Injury; Dioxanes; Dioxins; Dose-Response Relationship, Drug; Epinephrine; Glutathione; Idazoxan; Liver Diseases; Male; Mice; Necrosis; Norepinephrine; Phentolamine; Time Factors | 1988 |
Alpha-adrenergic receptors in rat skeletal muscle.
Topics: Animals; Binding Sites; Dihydroalprenolol; Dioxanes; Female; Idazoxan; Kinetics; Male; Muscles; Peptidyl-Dipeptidase A; Phentolamine; Phenylephrine; Prazosin; Rats; Receptors, Adrenergic, alpha; Sarcolemma; Yohimbine | 1986 |
Exercise-induced increases in plasma catecholamines and growth hormone are augmented by selective alpha 2-adrenoceptor blockade in man.
Topics: Adult; Blood Pressure; Dioxanes; Dioxins; Growth Hormone; Humans; Idazoxan; Insulin; Nervous System Physiological Phenomena; Norepinephrine; Phentolamine; Physical Exertion; Potassium; Receptors, Adrenergic, alpha | 1986 |
Characterization of alpha 2-adrenergic receptors of calf retina membranes by [3H]-rauwolscine and [3H]-RX 781094 binding.
Topics: Animals; Binding, Competitive; Cattle; Dioxanes; Dioxins; Epinephrine; Guanylyl Imidodiphosphate; Idazoxan; Kinetics; Phentolamine; Receptors, Adrenergic, alpha; Retina; Yohimbine | 1987 |
Peripheral alpha 1- and alpha 2-adrenoreceptor mechanisms in blood pressure control.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding Sites; Blood Pressure; Clonidine; Dioxins; Guanabenz; Idazoxan; Male; Muscle, Smooth, Vascular; Norepinephrine; Phenoxybenzamine; Phentolamine; Prazosin; Pressoreceptors; Rabbits; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Synapses; Vascular Resistance | 1983 |
The actions of noradrenaline on neurones of the rat substantia gelatinosa in vitro.
Topics: Adrenergic alpha-Antagonists; Animals; Dioxanes; Idazoxan; Male; Membrane Potentials; Neurons; Norepinephrine; Phentolamine; Prazosin; Propranolol; Rats; Rats, Inbred Strains; Spinal Cord; Substantia Gelatinosa; Tetrodotoxin; Yohimbine | 1984 |
Evidence that exogenous but not endogenous norepinephrine activates the presynaptic alpha-2 adrenoceptors on serotonergic nerve endings in the rat hypothalamus.
Topics: Animals; Cocaine; Desipramine; Dioxins; Hypothalamus; Idazoxan; In Vitro Techniques; Male; Norepinephrine; Phentolamine; Rabbits; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Serotonin; Serotonin; Yohimbine | 1984 |
Caffeine antinociception in the rat hot-plate and formalin tests and locomotor stimulation: involvement of noradrenergic mechanisms.
Topics: Adrenergic alpha-Antagonists; Animals; Caffeine; Dioxanes; Drug Synergism; Formaldehyde; Hot Temperature; Idazoxan; Male; Motor Activity; Norepinephrine; Pain; Pain Measurement; Phentolamine; Prazosin; Rats; Rats, Sprague-Dawley; Stimulation, Chemical | 1995 |
Elevation of cAMP facilitates noradrenergic transmission in submucous neurons of guinea pig ileum.
Topics: 1-Methyl-3-isobutylxanthine; Adrenergic alpha-Antagonists; Animals; Colforsin; Cyclic AMP; Dioxanes; Electric Stimulation; Ganglia; Guinea Pigs; Idazoxan; Ileum; Membrane Potentials; Microelectrodes; Neurons; Norepinephrine; Phentolamine; Receptors, Purinergic; Synaptic Transmission; Yohimbine | 1993 |
Effect of the centrally acting muscle relaxant tizanidine on spinal reflexes: involvement of descending noradrenergic systems.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Clonidine; Decerebrate State; Dioxanes; Hexamethonium Compounds; Idazoxan; Male; Muscle Relaxants, Central; Norepinephrine; Phentolamine; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Reflex; Reflex, Monosynaptic; Spinal Cord; Sympathetic Nervous System | 1993 |
Strychnine-induced seizures in mice: the role of noradrenaline.
Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Disulfiram; Droxidopa; Idazoxan; Imipramine; Male; Mice; Pargyline; Phentolamine; Prazosin; Propranolol; Receptors, Adrenergic; Reserpine; Seizures; Strychnine | 1994 |
The involvement of noradrenaline, 5-hydroxytryptamine and acetylcholine in imipramine-induced seizures in mice.
Topics: 5-Hydroxytryptophan; Acetylcholine; alpha-Methyltyrosine; Animals; Atropine; Clonidine; Dioxanes; Droxidopa; Drug Synergism; Idazoxan; Imipramine; Male; Methyltyrosines; Mice; Norepinephrine; Pargyline; Phentolamine; Physostigmine; Prazosin; Reserpine; Seizures; Serotonin | 1993 |
The prejunctional inhibitory effect of alpha-methylnoradrenaline in the rat vas deferens is not mediated via alpha 2-adrenoceptors.
Topics: Adrenergic alpha-Antagonists; Animals; Benzazepines; Clonidine; Dioxanes; Electric Stimulation; Idazoxan; Imidazoles; Isometric Contraction; Male; Neuromuscular Junction; Nordefrin; Phenoxybenzamine; Phentolamine; Quinolines; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Adrenergic, alpha-2; Vas Deferens; Vasoconstrictor Agents; Yohimbine | 1995 |
Subtype determination of presynaptic alpha 2-autoreceptors in the rabbit pulmonary artery and human saphenous vein.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Benzazepines; Cattle; Dioxanes; Electric Stimulation; Humans; Idazoxan; Imidazoles; In Vitro Techniques; Oxymetazoline; Phentolamine; Presynaptic Terminals; Pulmonary Artery; Rabbits; Rats; Receptors, Adrenergic, alpha-2; Saphenous Vein; Tritium | 1995 |
Imidazoline compounds stimulate insulin release by inhibition of K(ATP) channels and interaction with the exocytotic machinery.
Topics: Animals; Brimonidine Tartrate; Calcium; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Cytosol; Diazoxide; Exocytosis; Glucose; Idazoxan; Imidazoles; Indoles; Insulin; Insulin Secretion; Islets of Langerhans; Male; Membrane Potentials; Phentolamine; Potassium Channels; Potassium Chloride; Protein Kinase C; Quinoxalines; Rats; Rats, Wistar; Tumor Cells, Cultured | 1996 |
Elevation of cytosolic calcium by imidazolines in mouse islets of Langerhans: implications for stimulus-response coupling of insulin release.
Topics: Adrenergic alpha-Antagonists; Agmatine; Animals; Benzofurans; Calcium; Cytosol; Down-Regulation; Glucose; Idazoxan; Imidazoles; Imidazoline Receptors; Insulin; Islets of Langerhans; Mice; Phentolamine; Receptors, Drug; Signal Transduction | 1996 |
Characterisation of pre- and post-synaptic alpha-adrenoceptors in modulation of the rat ileum longitudinal and circular muscle activities.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding Sites; Brimonidine Tartrate; Clonidine; Electric Stimulation; Idazoxan; Ileum; In Vitro Techniques; Muscle Contraction; Oxymetazoline; Phentolamine; Quinoxalines; Rats; Receptors, Adrenergic, alpha; Receptors, Presynaptic | 1997 |
Uptake of agmatine into rat brain synaptosomes: possible role of cation channels.
Topics: Agmatine; Amino Acids; Animals; Biogenic Monoamines; Brain; Cations; Energy Metabolism; Idazoxan; Ion Channels; Male; Phentolamine; Polyamines; Rats; Rats, Sprague-Dawley; Sodium; Synaptosomes | 1997 |
Prejunctional alpha2A-autoreceptors in the human gastric and ileocolic arteries.
Topics: Adrenergic alpha-Antagonists; Aged; Arteries; Autoreceptors; Colon; Dioxanes; Dopamine Antagonists; Dose-Response Relationship, Drug; Electric Stimulation; Female; Gastric Mucosa; Humans; Idazoxan; Ileum; In Vitro Techniques; Male; Middle Aged; Neuromuscular Junction; Norepinephrine; Phentolamine; Prazosin; Receptors, Adrenergic, alpha-2; Spiro Compounds; Stomach; Tritium; Yohimbine | 1998 |
Heterogeneous characteristics of imidazoline-induced insulin secretion.
Topics: Adrenergic alpha-Antagonists; Animals; Anti-Arrhythmia Agents; Calcium; Clonidine; Drug Interactions; Enzyme Inhibitors; Glucose; Idazoxan; Imidazoles; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Membrane Potentials; Mice; Phentolamine; Potassium Channels; Time Factors | 1999 |
Imidazolines and the pancreatic B-cell. Actions and binding sites.
Topics: Adenosine Triphosphate; Animals; Binding Sites; Calcium; Calcium Channels; Cell Line; Cell Membrane; Cytoplasm; Glucose; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Mice; Patch-Clamp Techniques; Phentolamine; Potassium Channels; Protein Kinase C; Receptors, Drug; Tetradecanoylphorbol Acetate | 1999 |
Noradrenaline release from cultured mouse postganglionic sympathetic neurons: autoreceptor-mediated modulation.
Topics: Adenosine; Adenosine Triphosphate; Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Cells, Cultured; Electric Stimulation; Ganglia, Sympathetic; Humans; Idazoxan; Kinetics; Mice; Mice, Inbred Strains; Neurons; Norepinephrine; Phenethylamines; Phentolamine; Purinergic P1 Receptor Agonists; Quinoxalines; Receptors, Adrenergic, alpha-2; Tritium; Yohimbine | 1999 |
Effects of imidazoline binding site ligands on the growth and viability of clonal pancreatic beta-cells.
Topics: Animals; Antazoline; Apoptosis; Benzofurans; Binding Sites; Cell Division; Cell Survival; Idazoxan; Imidazoles; Imidazoline Receptors; Insulin; Insulin Secretion; Islets of Langerhans; PC12 Cells; Phentolamine; Rats; Receptors, Drug | 2000 |
Imidazolines inhibit secretory responses of rat colonic mucosa to calcium-dependent but not cyclic AMP-dependent secretagogues.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Calcium; Clonidine; Colon; Cyclic AMP; Idazoxan; Imidazoles; In Vitro Techniques; Intestinal Mucosa; Male; Phentolamine; Rats; Rats, Wistar | 2001 |
In vitro and in vivo impairment of alpha2-adrenergic receptor-dependent antilipolysis by fatty acids in human adipose tissue.
Topics: Adipocytes; Adipose Tissue; Adrenergic Agents; Adult; Biopsy, Needle; Dietary Fats; Dose-Response Relationship, Drug; Epinephrine; Exercise; Fatty Acids; Female; Gene Expression; Glycerol; GTP-Binding Proteins; Humans; Idazoxan; Isoproterenol; Lipolysis; Middle Aged; Palmitates; Phentolamine; Receptors, Adrenergic, alpha-2 | 2001 |
[Ethyl-3H]RS-79948-197 alpha2-adrenoceptor autoradiography validation in alpha2-adrenoceptor knockout mice.
Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Animals; Autoradiography; Binding Sites; Binding, Competitive; Cerebral Cortex; Idazoxan; In Vitro Techniques; Isoquinolines; Ligands; Mice; Mice, Knockout; Naphthyridines; Oxymetazoline; Phentolamine; Prazosin; Putamen; Radioligand Assay; Receptors, Adrenergic, alpha-2; Tritium; Yohimbine | 2004 |
Adrenoceptor compounds prevent the settlement of marine invertebrate larvae: Balanus amphitrite (Cirripedia), Bugula neritina (Bryozoa) and Hydroides elegans (Polychaeta).
Topics: Adrenergic alpha-Antagonists; Animals; Bryozoa; Idazoxan; Larva; Mortality; Paint; Pest Control; Phentolamine; Polychaeta; Seawater; Thoracica | 2004 |
Both α1- and β1-adrenoceptors in the bed nucleus of the stria terminalis are involved in the expression of conditioned contextual fear.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Conditioning, Psychological; Dioxanes; Electroshock; Fear; Idazoxan; Imidazoles; Male; Phentolamine; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-1; Septal Nuclei | 2012 |