Page last updated: 2024-08-23

idazoxan and oxymetazoline

idazoxan has been researched along with oxymetazoline in 24 studies

Research

Studies (24)

TimeframeStudies, this research(%)All Research%
pre-19906 (25.00)18.7374
1990's13 (54.17)18.2507
2000's5 (20.83)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Agbaba, D; Filipic, S; Nikolic, K1
De Backer, JP; De Keyser, J; De Vos, H; Van Liefde, I; Vauquelin, G1
Briand, R; de Champlain, J; Gagne, J; Nadeau, R; Yamaguchi, N1
Angel, I; Langer, SZ; Niddam, R1
Berlan, M; Galitzky, J; Lafontan, M; Montastruc, JL; Senard, JM; Stillings, M1
Brandon, S; Cragoe, EJ; Guyer, CA; Horstman, DA; Limbird, LE; Wilson, AL1
Lacroix, JS; Lundberg, JM1
Dickinson, KE; McKernan, RM; Miles, CM; Sever, PS1
Diop, L; Kolta, A; Reader, TA1
de Champlain, J; Foucart, S; Nadeau, R2
Curet, O; de Montigny, C1
Etgen, AM; Karkanias, GB1
Ala-Uotila, S; Kurose, H; Marjamäki, A; Oker-Blom, C; Pohjanoksa, K; Scheinin, M; Sizmann, D1
Göthert, M; Molderings, GJ1
Blandizzi, C; Carignani, D; Colucci, R; Crema, F; Del Tacca, M; Lazzeri, G; Natale, G1
Bylund, DB; Cerutis, DR; Deupree, JD; Hinton, KA1
Flügge, G1
Coupar, IM; Liu, L1
Bobirnac, I; Gazi, L; Loetscher, E; Parsley, S; Schoeffter, P1
Cockcroft, V; Frang, H; Marjamäki, A; Pihlavisto, M; Scheinin, M1
Colpaert, FC; Pauwels, PJ1
Fagerholm, V; Hein, L; Philipp, M; Scheinin, M1
Díez-Alarcia, R; Fernández-López, A; Meana, JJ; Paniagua, MA; Pilar-Cuéllar, F1

Other Studies

24 other study(ies) available for idazoxan and oxymetazoline

ArticleYear
QSAR study of imidazoline antihypertensive drugs.
    Bioorganic & medicinal chemistry, 2008, Aug-01, Volume: 16, Issue:15

    Topics: Antihypertensive Agents; Binding Sites; Imidazoline Receptors; Imidazolines; Ligands; Models, Molecular; Molecular Structure; Quantitative Structure-Activity Relationship

2008
Regional distribution of alpha 2A- and alpha 2B-adrenoceptor subtypes in postmortem human brain.
    Journal of neurochemistry, 1992, Volume: 58, Issue:4

    Topics: Adrenergic alpha-Antagonists; Aged; Binding, Competitive; Brain; Cadaver; Dioxanes; Humans; Idazoxan; Middle Aged; Oxymetazoline; Prazosin; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Tissue Distribution

1992
Alpha 2-adrenoceptor modulation of catecholamine and neuropeptide Y responses during haemorrhagic hypotension in anaesthetized dogs.
    Journal of the autonomic nervous system, 1990, Volume: 30, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Cardiovascular System; Catecholamines; Dioxanes; Dogs; Hemorrhage; Hypotension; Idazoxan; Neuropeptide Y; Oxymetazoline; Receptors, Adrenergic, alpha

1990
Involvement of alpha-2 adrenergic receptor subtypes in hyperglycemia.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 254, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Glucose; Brimonidine Tartrate; Dioxanes; Dioxins; Drug Interactions; Hyperglycemia; Idazoxan; Imidazoles; Insulin; Male; Mice; Oxymetazoline; Quinoxalines; Receptors, Adrenergic, alpha

1990
Identification of human platelet alpha 2-adrenoceptors with a new antagonist [3H]-RX821002, a 2-methoxy derivative of idazoxan.
    British journal of pharmacology, 1990, Volume: 100, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adult; Blood Platelets; Brimonidine Tartrate; Dioxanes; Epinephrine; Humans; Idazoxan; In Vitro Techniques; Kinetics; Male; Membranes; Oxymetazoline; Prazosin; Quinoxalines; Radioligand Assay; Receptors, Adrenergic, alpha; Yohimbine

1990
An aspartate conserved among G-protein receptors confers allosteric regulation of alpha 2-adrenergic receptors by sodium.
    The Journal of biological chemistry, 1990, Dec-15, Volume: 265, Issue:35

    Topics: Affinity Labels; Allosteric Regulation; Amino Acid Sequence; Animals; Aspartic Acid; Brimonidine Tartrate; Dioxanes; DNA Mutational Analysis; Epinephrine; Idazoxan; In Vitro Techniques; Molecular Sequence Data; Oxymetazoline; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha; Sodium; Structure-Activity Relationship; Swine; Transfection; Yohimbine

1990
Sympathetic vascular control of the pig nasal mucosa: adrenoceptor mechanisms in blood flow and volume control.
    British journal of pharmacology, 1989, Volume: 97, Issue:4

    Topics: Animals; Antihypertensive Agents; Brimonidine Tartrate; Desipramine; Dioxanes; Electric Stimulation; Female; Idazoxan; Male; Nasal Mucosa; Norepinephrine; Oxymetazoline; Phenylephrine; Prazosin; Quinoxalines; Receptors, Adrenergic; Regional Blood Flow; Rheology; Swine; Sympathetic Nervous System

1989
Heterogeneity between soluble human and rabbit splenic alpha 2-adrenoceptors.
    Biochemical pharmacology, 1986, Oct-15, Volume: 35, Issue:20

    Topics: Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Dioxanes; Epinephrine; Humans; Idazoxan; Lectins; Oxymetazoline; Phentolamine; Prazosin; Quinolizines; Quinoxalines; Rabbits; Receptors, Adrenergic, alpha; Solubility; Spleen; Sulfhydryl Reagents; Yohimbine

1986
Noradrenergic effects on rat visual cortex: single-cell microiontophoretic studies of alpha-2 adrenergic receptors.
    Life sciences, 1987, Jul-20, Volume: 41, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Antagonists; Animals; Clonidine; Dioxanes; Idazoxan; Male; Neurons; Norepinephrine; Oxymetazoline; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Visual Cortex

1987
In vivo modulation by alpha 2-adrenoceptors of adrenal catecholamine release in the anaesthetized dog.
    Canadian journal of physiology and pharmacology, 1988, Volume: 66, Issue:4

    Topics: Adrenal Glands; Adrenergic alpha-Antagonists; Anesthesia; Animals; Catecholamines; Dioxanes; Dogs; Electric Stimulation; Female; Idazoxan; Male; Oxymetazoline; Receptors, Adrenergic, alpha; Splanchnic Nerves

1988
Electrophysiological characterization of adrenoceptors in the rat dorsal hippocampus. I. Receptors mediating the effect of microiontophoretically applied norepinephrine.
    Brain research, 1988, Dec-13, Volume: 475, Issue:1

    Topics: Action Potentials; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Dioxanes; Hippocampus; Idazoxan; Iontophoresis; Male; Norepinephrine; Oxymetazoline; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha

1988
The release of catecholamines from the adrenal medulla and its modulation by alpha 2-adrenoceptors in the anaesthetized dog.
    Canadian journal of physiology and pharmacology, 1987, Volume: 65, Issue:4

    Topics: Adrenal Medulla; Animals; Catecholamines; Clonidine; Dioxanes; Dogs; Dopamine; Electric Stimulation; Epinephrine; Female; Idazoxan; Male; Norepinephrine; Oxymetazoline; Receptors, Adrenergic, alpha; Splanchnic Nerves; Yohimbine

1987
A thermodynamic analysis of estrogen regulation of alpha 2-adrenoceptor binding.
    Brain research, 1995, Mar-13, Volume: 674, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Binding Sites; Binding, Competitive; Dioxanes; Estradiol; Female; Guanylyl Imidodiphosphate; Hypothalamus; Idazoxan; Ligands; Ovariectomy; Oxymetazoline; Preoptic Area; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Temperature; Thermodynamics

1995
Similar ligand binding in recombinant human alpha 2 C2-adrenoceptors produced in mammalian, insect and yeast cells.
    European journal of pharmacology, 1994, Mar-15, Volume: 267, Issue:1

    Topics: Adrenergic alpha-Antagonists; Amino Acid Sequence; Animals; Cells, Cultured; Chlorpromazine; Dioxanes; Humans; Idazoxan; Immunoblotting; Mammary Neoplasms, Experimental; Mice; Molecular Sequence Data; Moths; Oxymetazoline; Prazosin; Receptors, Adrenergic, alpha; Recombinant Proteins; Saccharomyces cerevisiae; Transfection; Tumor Cells, Cultured; Yohimbine

1994
Subtype determination of presynaptic alpha 2-autoreceptors in the rabbit pulmonary artery and human saphenous vein.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Benzazepines; Cattle; Dioxanes; Electric Stimulation; Humans; Idazoxan; Imidazoles; In Vitro Techniques; Oxymetazoline; Phentolamine; Presynaptic Terminals; Pulmonary Artery; Rabbits; Rats; Receptors, Adrenergic, alpha-2; Saphenous Vein; Tritium

1995
Determination on functional basis of presynaptic alpha 2-adrenoceptor subtypes in guinea-pig duodenum.
    Neuroscience letters, 1996, May-24, Volume: 210, Issue:1

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Cholinergic Fibers; Duodenum; Electric Stimulation; Gastrointestinal Motility; Guinea Pigs; Idazoxan; Imidazoles; Indoles; Isoindoles; Isoquinolines; Male; Medetomidine; Muscle Contraction; Nordefrin; Norepinephrine; Oxymetazoline; Piperazines; Prazosin; Receptors, Adrenergic, alpha-2; Synaptic Membranes; Vasoconstrictor Agents; Xylazine; Yohimbine

1996
Buffers differentially alter the binding of [3H]rauwolscine and [3H]RX821002 to the alpha-2 adrenergic receptor subtypes.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 278, Issue:3

    Topics: Animals; Buffers; CHO Cells; Cricetinae; Humans; Idazoxan; Kinetics; Opossums; Oxymetazoline; Prazosin; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-2; Recombinant Proteins; Species Specificity; Yohimbine

1996
Alterations in the central nervous alpha 2-adrenoceptor system under chronic psychosocial stress.
    Neuroscience, 1996, Volume: 75, Issue:1

    Topics: Adrenergic alpha-2 Receptor Agonists; Animals; Brimonidine Tartrate; Chronic Disease; Down-Regulation; Hydrocortisone; Idazoxan; Locus Coeruleus; Male; Nerve Tissue Proteins; Norepinephrine; Oxymetazoline; Pituitary-Adrenal System; Prefrontal Cortex; Quinoxalines; Receptors, Adrenergic, alpha-2; Social Dominance; Solitary Nucleus; Stress, Psychological; Tupaiidae; Up-Regulation; Vagus Nerve

1996
Characterisation of pre- and post-synaptic alpha-adrenoceptors in modulation of the rat ileum longitudinal and circular muscle activities.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding Sites; Brimonidine Tartrate; Clonidine; Electric Stimulation; Idazoxan; Ileum; In Vitro Techniques; Muscle Contraction; Oxymetazoline; Phentolamine; Quinoxalines; Rats; Receptors, Adrenergic, alpha; Receptors, Presynaptic

1997
Functional alpha2C-adrenoceptors in human neuroblastoma SH-SY5Y cells.
    European journal of pharmacology, 1999, May-07, Volume: 372, Issue:1

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Brimonidine Tartrate; Clonidine; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Guanfacine; Humans; Idazoxan; Isoquinolines; Neuroblastoma; Oxymetazoline; Piperazines; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tumor Cells, Cultured; Yohimbine

1999
Ligand recognition of serine-cysteine amino acid exchanges in transmembrane domain 5 of alpha2-adrenergic receptors by UK 14,304.
    Journal of neurochemistry, 2000, Volume: 74, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding Sites; Binding, Competitive; Brimonidine Tartrate; Chlorpromazine; CHO Cells; Cricetinae; Cysteine; Dopamine Antagonists; Humans; Idazoxan; Ligands; Mice; Models, Molecular; Molecular Sequence Data; Oxymetazoline; Protein Structure, Tertiary; Quinoxalines; Radioligand Assay; Receptors, Adrenergic, alpha-2; Sequence Homology, Amino Acid; Serine; Transfection; Tritium; Yohimbine

2000
Partial to complete antagonism by putative antagonists at the wild-type alpha(2C)-adrenoceptor based on kinetic analyses of agonist:antagonist interactions.
    British journal of pharmacology, 2000, Volume: 131, Issue:7

    Topics: Adrenergic Agonists; Adrenergic Antagonists; Animals; Azepines; Brimonidine Tartrate; Calcium; CHO Cells; Clonidine; Cricetinae; DNA, Recombinant; Dose-Response Relationship, Drug; Drug Interactions; Epinephrine; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gq-G11; Heterotrimeric GTP-Binding Proteins; Idazoxan; Kinetics; Medetomidine; Mice; Oxymetazoline; Quinoxalines; Rats; Receptors, Adrenergic, alpha-2; Recombinant Fusion Proteins; Transfection

2000
[Ethyl-3H]RS-79948-197 alpha2-adrenoceptor autoradiography validation in alpha2-adrenoceptor knockout mice.
    European journal of pharmacology, 2004, Aug-30, Volume: 497, Issue:3

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Animals; Autoradiography; Binding Sites; Binding, Competitive; Cerebral Cortex; Idazoxan; In Vitro Techniques; Isoquinolines; Ligands; Mice; Mice, Knockout; Naphthyridines; Oxymetazoline; Phentolamine; Prazosin; Putamen; Radioligand Assay; Receptors, Adrenergic, alpha-2; Tritium; Yohimbine

2004
Pharmacological characterization and autoradiographic distribution of alpha2-adrenoceptor antagonist [3H]RX 821002 binding sites in the chicken brain.
    Neuroscience, 2006, Aug-11, Volume: 141, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Brain; Chickens; Dose-Response Relationship, Drug; Drug Interactions; Idazoxan; In Vitro Techniques; Male; Oxymetazoline; Radioligand Assay; Rats; Rats, Sprague-Dawley; Serotonin; Tritium

2006