Page last updated: 2024-08-23

idazoxan and agmatine

idazoxan has been researched along with agmatine in 43 studies

Research

Studies (43)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's13 (30.23)18.2507
2000's20 (46.51)29.6817
2010's9 (20.93)24.3611
2020's1 (2.33)2.80

Authors

AuthorsStudies
Arrault, A; Guillaumet, G; Mérour, JY; Pfeiffer, B; Renard, P; Rettori, MC; Scalbert, E; Touzeau, F1
Hussain, JF; Kendall, DA; Pinthong, D; Wilson, VG1
Li, G; Regunathan, S; Reis, DJ; Wang, H; Youngson, C1
Dunne, MJ; Hashmi, MN; Kane, C; Shepherd, RM; Squires, PE1
Bramwell, S; McGowan, D; Regunathan, S; Reis, DJ; Wang, H1
Regunathan, S; Reis, DJ1
Regunathan, S; Reis, DJ; Sastre, M1
Danbury, TC; Hudson, AL; Kestin, SC; Ruban, B; Waterman-Pearson, AE1
Feinstein, DL; Regunathan, S; Reis, DJ1
Li, J; Li, X; Pei, G; Qin, BY2
Assumpció Boronat, M; DeGregorio-Rocasolano, N; García-Sevilla, JA; Gasull, T; Lerma, J; Olmos, G; Paz Regalado, M; Trullas, R; Villarroel, A1
Gacar, MN; Ulak, G; Utkan, T; Yardimoglu, M; Yildiran, HG1
Duan, HR; He, RR; Li, XT; Liu, LL; Liu, S; Zhang, WL; Zhao, H1
Fan, ZZ; He, RR; Li, XT1
He, RR; Li, XT1
Duan, HR; He, RR; Li, XT1
He, RR; Qin, XM1
Li, J; Li, X; Qin, BY; Su, RB1
Dominiak, P; Häuser, W; Jungbluth, B; Raasch, W; Schäfer, U2
Hou, SW; Qi, JS; Qiao, JT; Zhang, Y1
Garcez-do-Carmo, L; Jurkiewicz, A; Piçarro, I; Santos, WC; Smaili, SS1
Li, J; Lu, G; Qin, BY; Su, RB1
Aricioglu, F; Dulger, G; Ercil, E1
Shen, FM; Su, DF; Wang, WZ; Yang, J1
Berntsson, K; Dahlström, M; Elwing, H; Jonsson, PR; Lindgren, F; Mårtensson, LG; Sjögren, M1
Rawls, SM; Tallarida, RJ; Zisk, J1
Amin, M; Rawls, SM; Zisk, J1
Ferguson, TB; Johnson, FK; Johnson, RA; Joshi, MS; Lancaster, JR; Parthasarathy, S1
Li, J; Lu, XQ; Su, RB; Wei, XL; Wu, N; Zheng, JQ1
Chen, HX; Jiang, XZ; Li, J; Li, YF; Wang, NP; Zhang, YZ1
Aggarwal, S; Kim, E; Rawls, SM; Shavalian, B1
Chopde, CT; Gahane, AY; Kotagale, NR; Taksande, BG; Ugale, RR1
Bi, GH; Dong, HJ; Li, J; Lu, W; Su, RB; Yang, Z; Zhao, YQ1
Dong, HJ; Gong, ZH; Li, J; Lu, W; Su, RB1
Bhalla, S; Gulati, A; Rapolaviciute, V1
Li, JX; Winter, JC; Zhang, Y1
Andurkar, SV; Bhalla, S; Gulati, A1
Aglawe, MM; Chopde, CT; Kotagale, NR; Taksande, BG; Tripathi, SJ; Umekar, MJ1
Bernard, R; Bernstein, HG; Laube, G; Veh, RW; Weiss, T1
Aglawe, MM; Chopde, CT; Gujar, S; Khade, SD; Kotagale, NR; Taksande, BG1
Manole, OM; Moraru, C; Nechita, P; Rusu-Zota, G; Şorodoc, V1

Other Studies

43 other study(ies) available for idazoxan and agmatine

ArticleYear
Synthesis and biological evaluation of new 2-(4,5-dihydro-1H-imidazol-2-yl)-3,4-dihydro-2H-1,4-benzoxazine derivatives.
    Journal of medicinal chemistry, 2003, May-08, Volume: 46, Issue:10

    Topics: Adrenal Medulla; Animals; Antihypertensive Agents; Binding Sites; Blood Pressure; Cattle; Frontal Lobe; Heart Rate; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Kidney; Oxazines; Rabbits; Radioligand Assay; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Drug; Stereoisomerism; Structure-Activity Relationship

2003
Comparison of the interaction of agmatine and crude methanolic extracts of bovine lung and brain with alpha 2-adrenoceptor binding sites.
    British journal of pharmacology, 1995, Volume: 115, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Agmatine; Animals; Binding, Competitive; Brimonidine Tartrate; Cattle; Cerebral Cortex; Clonidine; Dioxanes; Idazoxan; Imidazoles; Lung; Methanol; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-2; Yohimbine

1995
Coexpression of imidazoline receptors and agmatine in rat carotid body.
    Annals of the New York Academy of Sciences, 1995, Jul-12, Volume: 763

    Topics: Agmatine; Animals; Binding Sites; Carotid Body; Cells, Cultured; Dioxanes; Idazoxan; Imidazoles; Imidazoline Receptors; Immunohistochemistry; Rats; Rats, Wistar; Receptors, Drug

1995
Elevation of cytosolic calcium by imidazolines in mouse islets of Langerhans: implications for stimulus-response coupling of insulin release.
    British journal of pharmacology, 1996, Volume: 119, Issue:5

    Topics: Adrenergic alpha-Antagonists; Agmatine; Animals; Benzofurans; Calcium; Cytosol; Down-Regulation; Glucose; Idazoxan; Imidazoles; Imidazoline Receptors; Insulin; Islets of Langerhans; Mice; Phentolamine; Receptors, Drug; Signal Transduction

1996
An antiserum to idazoxan recognizes an immunoreactive substance in human serum and cerebral spinal fluid which is not agmatine.
    Neurochemistry international, 1997, Volume: 30, Issue:1

    Topics: Agmatine; Animals; Antibody Specificity; Antigens; Cattle; Clonidine; Humans; Idazoxan; Imidazoline Receptors; Immune Sera; Radioimmunoassay; Rats; Receptors, Drug; Serum Albumin, Bovine

1997
Stimulation of imidazoline receptors inhibits proliferation of human coronary artery vascular smooth muscle cells.
    Hypertension (Dallas, Tex. : 1979), 1997, Volume: 30, Issue:2 Pt 1

    Topics: Adrenergic alpha-Antagonists; Agmatine; Animals; Arteries; Carrier Proteins; Cell Division; Cells, Cultured; Coronary Vessels; GTP-Binding Proteins; Humans; Idazoxan; Imidazoline Receptors; Muscle, Smooth, Vascular; Rats; Receptors, Drug

1997
Uptake of agmatine into rat brain synaptosomes: possible role of cation channels.
    Journal of neurochemistry, 1997, Volume: 69, Issue:6

    Topics: Agmatine; Amino Acids; Animals; Biogenic Monoamines; Brain; Cations; Energy Metabolism; Idazoxan; Ion Channels; Male; Phentolamine; Polyamines; Rats; Rats, Sprague-Dawley; Sodium; Synaptosomes

1997
Imidazoline (I2) binding sites in chicken brain.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Agmatine; Amiloride; Animals; Benzofurans; Binding Sites; Binding, Competitive; Brain; Chickens; Clonidine; Idazoxan; Imidazoles; Imidazoline Receptors; Kinetics; Receptors, Drug; Tritium

1999
Anti-proliferative and anti-inflammatory actions of imidazoline agents. Are imidazoline receptors involved?
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Agmatine; Animals; Animals, Newborn; Astrocytes; Cell Division; Cell Line; Cells, Cultured; Cerebral Cortex; Enzyme Induction; Gene Expression Regulation; Idazoxan; Imidazoles; Imidazoline Receptors; Inflammation; Macrophages; Mice; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Rats; Rats, Sprague-Dawley; Receptors, Drug

1999
Effects of agmatine on tolerance to and substance dependence on morphine in mice.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1999, Volume: 20, Issue:3

    Topics: Adrenergic alpha-Antagonists; Agmatine; Analgesics, Opioid; Animals; Drug Tolerance; Female; Idazoxan; Male; Mice; Morphine; Morphine Dependence; Substance Withdrawal Syndrome

1999
Protection by imidazol(ine) drugs and agmatine of glutamate-induced neurotoxicity in cultured cerebellar granule cells through blockade of NMDA receptor.
    British journal of pharmacology, 1999, Volume: 127, Issue:6

    Topics: Agmatine; Animals; Antazoline; Benzofurans; Cell Line; Cells, Cultured; Cerebellum; Dioxanes; Dizocilpine Maleate; Dose-Response Relationship, Drug; Electrophysiology; Glutamic Acid; Humans; Idazoxan; Imidazoles; Neuroprotective Agents; Patch-Clamp Techniques; Potassium; Radioligand Assay; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Styrenes

1999
Influence of agmatine in adaptation of cAMP signal transduction system of opiate receptors.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1999, Volume: 20, Issue:7

    Topics: Adaptation, Physiological; Adrenergic alpha-Antagonists; Agmatine; Analgesics; Animals; Cyclic AMP; Enkephalin, D-Penicillamine (2,5)-; Glioma; Guanosine 5'-O-(3-Thiotriphosphate); Hybrid Cells; Idazoxan; Imidazoline Receptors; Mice; Morphine; Neuroblastoma; Rats; Receptors, Drug; Signal Transduction; Tumor Cells, Cultured

1999
Investigation on the mechanism involved in the effects of agmatine on ethanol-induced gastric mucosal injury in rats.
    Life sciences, 2000, Mar-24, Volume: 66, Issue:18

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Agmatine; Animals; Central Nervous System Depressants; Ethanol; Female; Gastrointestinal Hemorrhage; Idazoxan; Imidazoline Receptors; Intestinal Mucosa; Male; Nitric Oxide; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, Drug; Stomach Ulcer; Yohimbine

2000
Electrophysiological effects of agmatine on human atrial fibers.
    Life sciences, 2000, May-05, Volume: 66, Issue:24

    Topics: Action Potentials; Adolescent; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Agmatine; Atrial Appendage; Child; Child, Preschool; Electrophysiology; Heart Defects, Congenital; Humans; Idazoxan; Imidazoline Receptors; In Vitro Techniques; Infant; Myocardial Contraction; NG-Nitroarginine Methyl Ester; Receptors, Drug

2000
Electrophysiologic effects of agmatine on pacemaker cells in sinoatrial node of rabbits.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1999, Volume: 20, Issue:10

    Topics: Action Potentials; Adrenergic alpha-Antagonists; Agmatine; Animals; Calcium Channels; Cromakalim; Dose-Response Relationship, Drug; Electrophysiology; Female; Idazoxan; Imidazoline Receptors; Male; Potassium Channels; Rabbits; Receptors, Drug; Sinoatrial Node

1999
[Hemodynamic effects of agmatine and its cellular mechanism in anesthetized rats].
    Sheng li xue bao : [Acta physiologica Sinica], 1999, Volume: 51, Issue:2

    Topics: Adrenergic alpha-Antagonists; Agmatine; Animals; Antihypertensive Agents; Hemodynamics; Idazoxan; Imidazoline Receptors; Injections, Intravenous; Male; Rats; Rats, Sprague-Dawley; Receptors, Drug

1999
Inhibition by agmatine on spontaneous activity of rabbit atrioventricular node cells.
    Acta pharmacologica Sinica, 2000, Volume: 21, Issue:10

    Topics: Action Potentials; Adrenergic alpha-Antagonists; Agmatine; Animals; Atrioventricular Node; Biological Transport, Active; Calcium; Calcium Channels; Female; Idazoxan; Male; Potassium; Rabbits

2000
Agmatine inhibits carotid sinus baroreflex in anesthetized rats.
    Acta pharmacologica Sinica, 2001, Volume: 22, Issue:3

    Topics: Adrenergic alpha-Antagonists; Agmatine; Animals; Baroreflex; Blood Pressure; Carotid Sinus; Idazoxan; Imidazoline Receptors; In Vitro Techniques; Male; Rats; Rats, Sprague-Dawley; Receptors, Drug

2001
Down-regulation of MAO-B activity and imidazoline receptors in rat brain following chronic treatment of morphine.
    Acta pharmacologica Sinica, 2001, Volume: 22, Issue:7

    Topics: Agmatine; Animals; Brain; Chromatography, High Pressure Liquid; Down-Regulation; Idazoxan; Imidazoline Receptors; Male; Monoamine Oxidase; Morphine; Morphine Dependence; Rats; Rats, Wistar; Receptors, Drug

2001
Modification of noradrenaline release in pithed spontaneously hypertensive rats by I1-binding sites in addition to alpha2-adrenoceptors.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 304, Issue:3

    Topics: Adrenergic alpha-Antagonists; Agmatine; Animals; Antihypertensive Agents; Benzofurans; Binding Sites; Blood Pressure; Disease Models, Animal; Heart Rate; Idazoxan; Imidazoles; Male; Norepinephrine; Phenoxybenzamine; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha-2

2003
Spinal antinociceptive effect of agmatine and tentative analysis of involved receptors: study in an electrophysiological model of rats.
    Brain research, 2003, Apr-11, Volume: 968, Issue:2

    Topics: Action Potentials; Adrenergic alpha-Antagonists; Agmatine; Analgesics; Animals; Dose-Response Relationship, Drug; Electrophysiology; Female; Idazoxan; Injections, Spinal; Intralaminar Thalamic Nuclei; Male; Neural Pathways; Neurons; Physical Stimulation; Rats; Rats, Wistar; Spinal Cord; Tail; Yohimbine

2003
Dual effect of agmatine in the bisected rat vas deferens.
    The Journal of pharmacy and pharmacology, 2003, Volume: 55, Issue:3

    Topics: Adenosine Triphosphate; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Agmatine; Animals; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Epididymis; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Male; Muscle Contraction; Norepinephrine; Phenoxybenzamine; Potassium Chloride; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, Drug; Sympathetic Nervous System; Synaptic Transmission; Vas Deferens; Yohimbine

2003
Modulation by alpha-difluoromethyl-ornithine and aminoguanidine of pain threshold, morphine analgesia and tolerance.
    European journal of pharmacology, 2003, Oct-08, Volume: 478, Issue:2-3

    Topics: Acetic Acid; Adrenergic alpha-Antagonists; Agmatine; Analgesics, Opioid; Animals; Behavior, Animal; Drug Tolerance; Eflornithine; Female; Guanidines; Hot Temperature; Idazoxan; Injections, Intraventricular; Injections, Subcutaneous; Male; Mice; Morphine; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Pain Measurement; Pain Threshold

2003
Agmatine inhibits naloxone-induced contractions in morphine-dependent Guinea pig ileum.
    Annals of the New York Academy of Sciences, 2003, Volume: 1009

    Topics: Adrenergic alpha-Antagonists; Agmatine; Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Guinea Pigs; Idazoxan; Ileum; Male; Morphine; Morphine Dependence; Muscle Contraction; Naloxone; Narcotic Antagonists; Substance Withdrawal Syndrome; Yohimbine

2003
Norepinephrine release is reduced by I(1)-receptors in addition to alpha(2)-adrenoceptors.
    Annals of the New York Academy of Sciences, 2003, Volume: 1009

    Topics: Adrenergic alpha-Antagonists; Agmatine; Animals; Benzofurans; Blood Pressure; Bridged Bicyclo Compounds; Electric Stimulation; Heptanes; Hypertension; Idazoxan; Imidazoles; Imidazoline Receptors; Male; Norepinephrine; Phenoxybenzamine; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha-2; Receptors, Drug; Spinal Cord

2003
Cardiovascular effects of agmatine within the rostral ventrolateral medulla are similar to those of clonidine in anesthetized rats.
    Experimental brain research, 2005, Volume: 160, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Agmatine; Anesthesia; Animals; Baroreflex; Blood Pressure; Cardiovascular Physiological Phenomena; Clonidine; Efferent Pathways; Glutamic Acid; Heart Rate; Idazoxan; Imidazoline Receptors; Male; Medulla Oblongata; Rats; Rats, Sprague-Dawley; Receptors, Drug; Sympathetic Nervous System

2005
Evidence for different pharmacological targets for imidazoline compounds inhibiting settlement of the barnacle Balanus improvisus.
    Journal of experimental zoology. Part A, Comparative experimental biology, 2005, Jul-01, Volume: 303, Issue:7

    Topics: Adrenergic Agonists; Adrenergic alpha-Antagonists; Agmatine; Analysis of Variance; Animals; Dose-Response Relationship, Drug; Idazoxan; Imidazoles; Imidazolines; Metamorphosis, Biological; Movement; Thoracica

2005
Agmatine and a cannabinoid agonist, WIN 55212-2, interact to produce a hypothermic synergy.
    European journal of pharmacology, 2006, Dec-28, Volume: 553, Issue:1-3

    Topics: Adrenergic alpha-Antagonists; Agmatine; Animals; Benzoxazines; Body Temperature; Cannabinoid Receptor Agonists; Cannabinoids; Dose-Response Relationship, Drug; Drug Synergism; Hypothermia; Idazoxan; Imidazoline Receptors; Injections, Intraventricular; Male; Morpholines; Naphthalenes; Rats; Rats, Sprague-Dawley; Receptors, Drug; Yohimbine

2006
Agmatine blocks morphine-evoked hyperthermia in rats.
    Brain research, 2007, May-25, Volume: 1147

    Topics: Agmatine; Analgesics, Non-Narcotic; Analysis of Variance; Animals; Biogenic Amines; Body Temperature Regulation; Dose-Response Relationship, Drug; Drug Interactions; Fever; Idazoxan; Imidazoline Receptors; Male; Morphine; Rats; Rats, Sprague-Dawley; Receptors, Drug; Receptors, Opioid, mu; Yohimbine

2007
Receptor-mediated activation of nitric oxide synthesis by arginine in endothelial cells.
    Proceedings of the National Academy of Sciences of the United States of America, 2007, Jun-12, Volume: 104, Issue:24

    Topics: Adrenergic alpha-Antagonists; Agmatine; Aniline Compounds; Arginine; Calcium; Calcium Channel Blockers; Cell Culture Techniques; Cells, Cultured; Culture Media, Serum-Free; Dexmedetomidine; Dose-Response Relationship, Drug; Endothelial Cells; Endothelium, Vascular; Enzyme Activation; Estrenes; Fluorescent Dyes; Humans; Idazoxan; Imidazolines; Lipopolysaccharides; Molecular Structure; NG-Nitroarginine Methyl Ester; Nifedipine; Nitrates; Nitric Oxide; Nitric Oxide Synthase Type III; Nitrites; Pyrrolidinones; Receptors, Adrenergic, alpha-2; Second Messenger Systems; Type C Phospholipases; Umbilical Veins; Virulence Factors, Bordetella; Xanthenes; Yohimbine

2007
Agmatine inhibits morphine-induced locomotion sensitization and morphine-induced changes in striatal dopamine and metabolites in rats.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2007, Volume: 17, Issue:12

    Topics: 3,4-Dihydroxyphenylacetic Acid; Adrenergic alpha-Antagonists; Agmatine; Analysis of Variance; Animals; Behavior, Animal; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Dynorphins; Gene Expression Regulation; Homovanillic Acid; Idazoxan; Locomotion; Male; Morphine; Narcotics; Rats; Rats, Wistar; Time Factors

2007
[5-HT1A/1B receptors, alpha2-adrenoceptors and the post-receptor adenylate cyclase activation in the mice brain are involved in the antidepressant-like action of agmatine].
    Yao xue xue bao = Acta pharmaceutica Sinica, 2008, Volume: 43, Issue:5

    Topics: Adenylyl Cyclases; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Agmatine; Animals; Antidepressive Agents; Behavior, Animal; Depression; Dose-Response Relationship, Drug; Fenclonine; Idazoxan; Male; Mice; Pindolol; Random Allocation; Rats; Rats, Wistar; Receptors, Biogenic Amine; Serotonin 5-HT1 Receptor Antagonists; Swimming; Synapses; Yohimbine

2008
Agmatine enhances cannabinoid action in the hot-plate assay of thermal nociception.
    Pharmacology, biochemistry, and behavior, 2009, Volume: 93, Issue:4

    Topics: Adrenergic alpha-Antagonists; Agmatine; Animals; Benzoxazines; Cannabinoids; Dose-Response Relationship, Drug; Drug Synergism; Hot Temperature; Idazoxan; Imidazoline Receptors; Male; Morpholines; Naphthalenes; Pain Measurement; Rats; Rats, Sprague-Dawley; Reaction Time; Receptor, Cannabinoid, CB1; Receptors, Adrenergic, alpha-2; Yohimbine

2009
Repeated agmatine treatment attenuates nicotine sensitization in mice: modulation by alpha2-adrenoceptors.
    Behavioural brain research, 2010, Dec-01, Volume: 213, Issue:2

    Topics: Agmatine; Animals; Arginine; Biguanides; Clonidine; Dose-Response Relationship, Drug; Drug Interactions; Eflornithine; Enzyme Inhibitors; Guanidines; Idazoxan; Male; Mice; Motor Activity; Nicotine; Receptors, Adrenergic, alpha-2; Yohimbine

2010
Effect of agmatine on long-term potentiation in morphine-treated rats.
    Pharmacology, biochemistry, and behavior, 2010, Volume: 96, Issue:2

    Topics: Agmatine; Animals; Dentate Gyrus; Drug Interactions; Hippocampus; Idazoxan; Imidazoline Receptors; Long-Term Potentiation; Male; Morphine; Rats; Rats, Wistar

2010
Agmatine inhibits morphine-induced memory impairment in the mouse step-down inhibitory avoidance task.
    Pharmacology, biochemistry, and behavior, 2010, Volume: 97, Issue:2

    Topics: Adrenergic alpha-Antagonists; Agmatine; Analgesics, Opioid; Animals; Avoidance Learning; Dose-Response Relationship, Drug; Idazoxan; Imidazoline Receptors; Male; Memory Disorders; Mental Recall; Mice; Morphine

2010
Determination of α(2)-adrenoceptor and imidazoline receptor involvement in augmentation of morphine and oxycodone analgesia by agmatine and BMS182874.
    European journal of pharmacology, 2011, Jan-25, Volume: 651, Issue:1-3

    Topics: Agmatine; Analgesics; Animals; Dansyl Compounds; Drug Synergism; Idazoxan; Imidazoline Receptors; Male; Mice; Morphine; Naloxone; Oxycodone; Receptors, Adrenergic, alpha-2; Receptors, Endothelin; Yohimbine

2011
Morphine-induced antinociception in the rat: supra-additive interactions with imidazoline I₂ receptor ligands.
    European journal of pharmacology, 2011, Nov-01, Volume: 669, Issue:1-3

    Topics: Adrenergic alpha-2 Receptor Antagonists; Agmatine; Analgesics; Analgesics, Opioid; Animals; Benzofurans; Disease Models, Animal; Drug Synergism; Idazoxan; Imidazoles; Imidazoline Receptors; Ligands; Male; Morphine; Pain; Rats; Rats, Sprague-Dawley; Saline Solution, Hypertonic; Yohimbine

2011
Involvement of α₂-adrenoceptors, imidazoline, and endothelin-A receptors in the effect of agmatine on morphine and oxycodone-induced hypothermia in mice.
    Fundamental & clinical pharmacology, 2013, Volume: 27, Issue:5

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Agmatine; Animals; Body Temperature Regulation; Dansyl Compounds; Dose-Response Relationship, Drug; Endothelin A Receptor Antagonists; Hypothermia; Idazoxan; Imidazoline Receptors; Male; Mice; Morphine; Oxycodone; Receptor, Endothelin A; Receptors, Adrenergic, alpha-2; Yohimbine

2013
Evidences for the agmatine involvement in antidepressant like effect of bupropion in mouse forced swim test.
    Pharmacology, biochemistry, and behavior, 2013, Volume: 107

    Topics: Agmatine; Animals; Antidepressive Agents; Arginine; Benzofurans; Biguanides; Bupropion; Clonidine; Dose-Response Relationship, Drug; Drug Interactions; Eflornithine; Guanidines; Idazoxan; Imidazoles; Immobility Response, Tonic; Injections, Intraventricular; Male; Mice; Motor Activity

2013
Agmatine modulates spontaneous activity in neurons of the rat medial habenular complex-a relevant mechanism in the pathophysiology and treatment of depression?
    Translational psychiatry, 2018, 09-24, Volume: 8, Issue:1

    Topics: Action Potentials; Agmatine; Animals; Benzofurans; Depression; Female; Habenula; Humans; Idazoxan; Imidazoles; Imidazoline Receptors; Male; Middle Aged; Neurons; Rats, Wistar; Ureohydrolases

2018
Agmatine Inhibits Behavioral Sensitization to Ethanol Through Imidazoline Receptors.
    Alcoholism, clinical and experimental research, 2019, Volume: 43, Issue:4

    Topics: Agmatine; Animals; Arginine; Benzofurans; Biguanides; Central Nervous System Sensitization; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; Guanidines; Idazoxan; Imidazoles; Imidazoline Receptors; Infusions, Intraventricular; Male; Mice; Microinjections; Motor Activity

2019
Effects of imidazoline agents in a rat conditioned place preference model of addiction.
    Naunyn-Schmiedeberg's archives of pharmacology, 2022, Volume: 395, Issue:3

    Topics: Agmatine; Analgesics, Opioid; Animals; Benzofurans; Conditioning, Psychological; Drug Interactions; Idazoxan; Imidazoles; Imidazoline Receptors; Male; Rats; Rats, Wistar; Time Factors; Tramadol

2022