idazoxan has been researched along with 2-(2-benzofuranyl)-2-imidazoline in 24 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 8 (33.33) | 18.2507 |
2000's | 8 (33.33) | 29.6817 |
2010's | 6 (25.00) | 24.3611 |
2020's | 2 (8.33) | 2.80 |
Authors | Studies |
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Baurin, N; Guillaumet, G; Marot, C; Mérour, JY; Morin-Allory, L; Payard, M; Renard, P; Vangrevelinghe, E | 1 |
Arrault, A; Guillaumet, G; Mérour, JY; Pfeiffer, B; Renard, P; Rettori, MC; Scalbert, E; Touzeau, F | 1 |
Abás, S; Bagán, A; Brea, J; Brocos-Mosquera, I; Callado, LF; Daelemans, D; de Jonghe, S; Djikic, T; Escolano, C; García-Fuster, MJ; García-Sevilla, JA; Griñán-Ferré, C; Hernández-Hernández, E; Loza, MI; Luque, FJ; Molins, E; Muguruza, C; Naesens, L; Nikolic, K; Pallàs, M; Pérez, B; Pérez-Lozano, P; Radan, M; Rodríguez-Arévalo, S; Vasilopoulou, F | 1 |
Bagán, A; Brea, J; Brocos-Mosquera, I; Callado, LF; Daelemans, D; De Jonghe, S; Djikic, T; Escolano, C; García-Fuster, MJ; García-Sevilla, JA; Griñán-Ferré, C; Hernández-Hernández, E; Loza, MI; Martínez, AL; Molins, E; Nikolic, K; Pallàs, M; Pérez, B; Radan, M; Rodriguez-Arévalo, S; Vasilopoulou, F | 1 |
Steinberg, MI; Wiest, SA | 1 |
Alemany, R; García-Sevilla, JA; Olmos, G | 1 |
Hudson, AL; Lione, LA; Nutt, DJ | 1 |
Martín-Ruiz, R; Pineda, J; Ruiz-Ortega, JA; Ugedo, L | 1 |
Alemany, R; Boronat, MA; García-Sevilla, JA; Olmos, G | 1 |
Danbury, TC; Hudson, AL; Kestin, SC; Ruban, B; Waterman-Pearson, AE | 1 |
Chen, K; Pickard, RT; Shih, JC; Steinberg, MI; Wiest, SA | 1 |
Artigas, F; Martín-Ruiz, R; Pineda, J; Ruiz-Ortega, JA; Ugedo, L | 1 |
Ballesteros, J; Callado, LF; Gutiérrez, M; Maeztu, AI; Meana, JJ | 1 |
Hudson, AL; Nutt, DJ; Robinson, ES; Tyacke, RJ | 1 |
Handley, SL; MacInnes, N | 1 |
Anderson, NJ; Hudson, AL; Lupo, PA; Nutt, DJ; Robinson, ES | 1 |
Anderson, NJ; Hudson, AL; Nutt, DJ; Robinson, ES; Seif, I | 1 |
Han, Z; Jin, K; Shao, B; Xiao, MJ; Yang, GY; Zheng, RY | 1 |
Han, Z; Hou, ST; Jiang, SX; Li, XL; Zeng, JQ; Zheng, RY | 1 |
Li, JX; Winter, JC; Zhang, Y | 1 |
Aglawe, MM; Chopde, CT; Kotagale, NR; Taksande, BG; Tripathi, SJ; Umekar, MJ | 1 |
He, X; Li, JX; Qiu, Y; Thorn, DA; Zhang, Y | 1 |
Li, JX; Seaman, RW; Shang, L; Siemian, JN; Zhang, Y; Zhu, Q | 1 |
Aglawe, MM; Chopde, CT; Gujar, S; Khade, SD; Kotagale, NR; Taksande, BG | 1 |
24 other study(ies) available for idazoxan and 2-(2-benzofuranyl)-2-imidazoline
Article | Year |
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3D-QSAR CoMFA study on imidazolinergic I(2) ligands: a significant model through a combined exploration of structural diversity and methodology.
Topics: Drug Design; Imidazoles; Imidazoline Receptors; Ligands; Models, Molecular; Molecular Structure; Receptors, Drug; Structure-Activity Relationship | 2000 |
Synthesis and biological evaluation of new 2-(4,5-dihydro-1H-imidazol-2-yl)-3,4-dihydro-2H-1,4-benzoxazine derivatives.
Topics: Adrenal Medulla; Animals; Antihypertensive Agents; Binding Sites; Blood Pressure; Cattle; Frontal Lobe; Heart Rate; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Kidney; Oxazines; Rabbits; Radioligand Assay; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Drug; Stereoisomerism; Structure-Activity Relationship | 2003 |
Bicyclic α-Iminophosphonates as High Affinity Imidazoline I
Topics: Alzheimer Disease; Animals; Chlorocebus aethiops; Cycloaddition Reaction; Dogs; Female; HeLa Cells; Hippocampus; Humans; Imidazoles; Imidazoline Receptors; Ligands; Madin Darby Canine Kidney Cells; Mice; Molecular Structure; Nootropic Agents; Organophosphonates; Quantitative Structure-Activity Relationship; Vero Cells | 2020 |
Benzofuranyl-2-imidazoles as imidazoline I
Topics: Alzheimer Disease; Animals; Apoptosis; Benzofurans; Cell Line, Tumor; Dose-Response Relationship, Drug; Humans; Imidazoles; Imidazoline Receptors; Ligands; Male; Mice; Molecular Structure; Oxidative Stress; Structure-Activity Relationship | 2021 |
Binding of [3H]2-(2-benzofuranyl)-2-imidazoline (BFI) to human brain: potentiation by tranylcypromine.
Topics: Animals; Benzofurans; Binding, Competitive; Brain; Cerebral Cortex; Humans; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Kinetics; Ligands; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Pargyline; Rats; Receptors, Drug; Reticular Formation; Tranylcypromine | 1997 |
Labelling of I2B-imidazoline receptors by [3H]2-(2-benzofuranyl)-2-imidazoline (2-BFI) in rat brain and liver: characterization, regulation and relation to monoamine oxidase enzymes.
Topics: Adrenergic beta-Antagonists; Affinity Labels; Animals; Benzofurans; Binding, Competitive; Brain; Cerebral Cortex; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Isoenzymes; Ligands; Liver; Male; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Phenelzine; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Drug | 1997 |
Characterisation and localisation of [3H]2-(2-benzofuranyl)-2-imidazoline binding in rat brain: a selective ligand for imidazoline I2 receptors.
Topics: Animals; Autoradiography; Benzofurans; Binding, Competitive; Brain; Idazoxan; Imidazoles; Imidazoline Receptors; Kinetics; Ligands; Male; Membranes; Rats; Rats, Wistar; Receptors, Drug; Tritium | 1998 |
Stimulation of locus coeruleus neurons by non-I1/I2-type imidazoline receptors: an in vivo and in vitro electrophysiological study.
Topics: Adenosine Triphosphate; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Benzofurans; Diazoxide; Electrophysiology; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Ligands; Locus Coeruleus; Male; Neurons; Potassium Channels; Rats; Receptors, Adrenergic, alpha-2; Receptors, Drug; Vasodilator Agents | 1998 |
Pharmacologic and molecular discrimination of I2-imidazoline receptor subtypes.
Topics: Amiloride; Animals; Benzofurans; Cell Membrane; Cerebral Cortex; Guanidine; Idazoxan; Imidazoles; Imidazoline Receptors; Male; Monoamine Oxidase Inhibitors; Rabbits; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Drug; Tritium | 1999 |
Imidazoline (I2) binding sites in chicken brain.
Topics: Agmatine; Amiloride; Animals; Benzofurans; Binding Sites; Binding, Competitive; Brain; Chickens; Clonidine; Idazoxan; Imidazoles; Imidazoline Receptors; Kinetics; Receptors, Drug; Tritium | 1999 |
Binding of the imidazoline ligand 3H-2-benzofuranyl-2-imidazoline (BFI) to human brain and platelets. Potentiation by tranylcypromine and role of MAO isoforms.
Topics: Animals; Benzofurans; Blood Platelets; Brain; Cell Membrane; Cerebral Cortex; Humans; Idazoxan; Imidazoles; Imidazoline Receptors; Isoenzymes; Kinetics; Ligands; Monoamine Oxidase; Rats; Receptors, Drug; Tranylcypromine; Tritium | 1999 |
Imidazoline-induced inhibition of firing rate of 5-HT neurons in rat dorsal raphe by modulation of extracellular 5-HT levels.
Topics: Animals; Benzofurans; Clorgyline; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Neurons; Phenylephrine; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, Drug; Serotonin | 1999 |
Differential [(3)H]idazoxan and [(3)H]2-(2-benzofuranyl)-2-imidazoline (2-BFI) binding to imidazoline I(2) receptors in human postmortem frontal cortex.
Topics: Adrenergic alpha-Antagonists; Autopsy; Benzofurans; Binding, Competitive; Dose-Response Relationship, Drug; Frontal Lobe; Humans; Idazoxan; Imidazoles; Imidazoline Receptors; Membranes; Radioligand Assay; Receptors, Drug; Tritium | 2001 |
Distribution of [(3)H]BU224, a selective imidazoline I(2) binding site ligand, in rat brain.
Topics: Animals; Autoradiography; Benzofurans; Binding Sites; Binding, Competitive; Brain; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Kinetics; Ligands; Male; Radioligand Assay; Rats; Rats, Wistar; Receptors, Drug | 2002 |
Autoradiographic localisation of [3H]2-BFI imidazoline I2 binding sites in mouse brain.
Topics: Animals; Autoradiography; Benzofurans; Binding Sites; Binding, Competitive; Brain; Idazoxan; Imidazoles; Male; Mice; Mice, Inbred C57BL; Midline Thalamic Nuclei; Nucleus Accumbens; Radioligand Assay; Raphe Nuclei; Tritium | 2005 |
Characterisation of imidazoline I2 binding sites in pig brain.
Topics: Animals; Benzofurans; Binding Sites; Binding, Competitive; Brain; Carbolines; Clonidine; Dose-Response Relationship, Drug; Female; Idazoxan; Imidazoles; Imidazoline Receptors; Kinetics; Male; Monoamine Oxidase Inhibitors; Picolinic Acids; Radioligand Assay; Receptors, Drug; Swine; Thiazoles; Tritium | 2005 |
Autoradiographical distribution of imidazoline binding sites in monoamine oxidase A deficient mice.
Topics: Animals; Autoradiography; Benzofurans; Binding Sites; Binding, Competitive; Brain; Cell Membrane; Epithelial Cells; Harmine; Idazoxan; Imidazoles; Imidazoline Receptors; Imidazolines; Iodine Radioisotopes; Kidney; Mice; Mice, Inbred C3H; Mice, Knockout; Monoamine Oxidase; Neurons; Picolinic Acids; Radioligand Assay; Receptors, Drug; Thiazoles | 2006 |
Attenuation of ischemia-induced rat brain injury by 2-(-2-benzofuranyl)-2-imidazoline, a high selectivity ligand for imidazoline I(2) receptors.
Topics: Animals; Benzofurans; Brain Injuries; Brain Ischemia; Caspase 3; Disease Models, Animal; Idazoxan; Imidazoles; Imidazoline Receptors; In Situ Nick-End Labeling; Male; Neurologic Examination; Neuroprotective Agents; Rats; Rats, Sprague-Dawley; Tetrazolium Salts | 2009 |
Reversible inhibition of intracellular calcium influx through NMDA receptors by imidazoline I(2) receptor antagonists.
Topics: Animals; Benzofurans; Calcium; Cerebral Cortex; Glutamic Acid; Idazoxan; Imidazoles; Imidazoline Receptors; Intracellular Space; Mice; Molecular Imaging; Neurons; Neuroprotective Agents; Neurotoxins; Receptors, N-Methyl-D-Aspartate | 2010 |
Morphine-induced antinociception in the rat: supra-additive interactions with imidazoline I₂ receptor ligands.
Topics: Adrenergic alpha-2 Receptor Antagonists; Agmatine; Analgesics; Analgesics, Opioid; Animals; Benzofurans; Disease Models, Animal; Drug Synergism; Idazoxan; Imidazoles; Imidazoline Receptors; Ligands; Male; Morphine; Pain; Rats; Rats, Sprague-Dawley; Saline Solution, Hypertonic; Yohimbine | 2011 |
Evidences for the agmatine involvement in antidepressant like effect of bupropion in mouse forced swim test.
Topics: Agmatine; Animals; Antidepressive Agents; Arginine; Benzofurans; Biguanides; Bupropion; Clonidine; Dose-Response Relationship, Drug; Drug Interactions; Eflornithine; Guanidines; Idazoxan; Imidazoles; Immobility Response, Tonic; Injections, Intraventricular; Male; Mice; Motor Activity | 2013 |
Behavioral effects of the imidazoline I(2) receptor ligand BU99006 in rats.
Topics: Animals; Benzofurans; Body Temperature; Central Nervous System Agents; Discrimination, Psychological; Dose-Response Relationship, Drug; Hypothermia; Idazoxan; Imidazoles; Imidazoline Receptors; Male; Rats; Rats, Sprague-Dawley | 2014 |
Effects of imidazoline I2 receptor agonists on reserpine-induced hyperalgesia and depressive-like behavior in rats.
Topics: Analgesics; Animals; Benzofurans; Depression; Disease Models, Animal; Fibromyalgia; Hyperalgesia; Idazoxan; Imidazoles; Imidazoline Receptors; Imidazolines; Male; Pain; Pain Measurement; Quinazolines; Rats; Rats, Sprague-Dawley; Reserpine | 2019 |
Agmatine Inhibits Behavioral Sensitization to Ethanol Through Imidazoline Receptors.
Topics: Agmatine; Animals; Arginine; Benzofurans; Biguanides; Central Nervous System Sensitization; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; Guanidines; Idazoxan; Imidazoles; Imidazoline Receptors; Infusions, Intraventricular; Male; Mice; Microinjections; Motor Activity | 2019 |