Page last updated: 2024-09-02

idarubicinol and idarubicin

idarubicinol has been researched along with idarubicin in 47 studies

Compound Research Comparison

Studies
(idarubicinol)
Trials
(idarubicinol)
Recent Studies (post-2010)
(idarubicinol)
Studies
(idarubicin)
Trials
(idarubicin)
Recent Studies (post-2010) (idarubicin)
541001,795454487

Research

Studies (47)

TimeframeStudies, this research(%)All Research%
pre-19904 (8.51)18.7374
1990's30 (63.83)18.2507
2000's13 (27.66)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ames, MM; Spreafico, F1
Ames, MM; Kuffel, MJ; Reid, JM1
Camaggi, CM; Carisi, P; Pannuti, F; Strocchi, E1
Camaggi, CM; Carisi, P; Efthymiopoulos, C; Guaraldi, M; Martoni, A; Pannuti, F; Strocchi, E; Strolin-Benedetti, M; Tononi, A1
Huet, S; Hurteloup, P; Pris, J; Rigal-Huguet, F; Robert, J1
Ames, MM; Hammond, GD; Krailo, MD; Pendergrass, TW; Reid, JM1
Barbui, T; Biondi, A; Catapano, C; D'Incalci, M; Giudici, G; Limonta, M; Masera, G; Specchia, G1
D'Incalci, M; Erranti, D; Freshi, A; Tirelli, U; Zanette, L; Zucchetti, M1
Bastholt, L; Dalmark, M; Ebbehøj, E; Elbaek, K; Jakobsen, A; Juul, P; Rasmussen, SN; Steiness, E1
Eksborg, S; Nilsson, B1
de Graaf, SS; Evans, WE; Riley-Stewart, CA1
Harousseau, JL; Huet, S; Hurteloup, P; Pris, J; Reiffers, J; Rigal-Huguet, F; Robert, J; Tamassia, V1
Cornblatt, B; Doyle, LA; Ross, DD; Tong, Y; Yang, W1
Ames, MM; Kuffel, MJ1
Fukushima, T; Kawai, Y; Nakamura, T; Ueda, T; Urasaki, Y; Yoshida, A1
Biersack, H; Brieden, T; Gieseler, F; Manderscheid, J; Nüssler, V1
Boezeman, J; de Witte, T; Haanen, C; Linssen, P; Minderman, H; van der Lely, N; Wessels, J1
Paul, C; Sundman-Engberg, B; Tidefelt, U1
Braess, J; Hiddemann, W; Kaufmann, CC; Kern, W; Kühn, S; Rührs, H; Schleyer, E; Sträubel, G; Unterhalt, M2
Boiocchi, M; Corona, G; De Angeli, S; Gigante, M; Simone, F; Toffoli, G1
Paul, C; Prenkert, M; Tidefelt, U1
Abbadessa, V; Cajozzo, A; Gancitano, RA; Musso, M; Perricone, R; Porretto, F; Tolomeo, M1
Baltes-Engler, S; Dederichs, B; Diehl, V; Engelhard, M; Engert, A; Küpper, F; Lathan, B; Reiser, M; Scheulen, ME; Schnell, R; Tesch, H; Wilhelm, M; Winterhalter, B; Wörmann, B1
Linke, R; Looby, M; Weiss, M1
Björkholm, M; Eksborg, S; Fagerlund, E; Hast, R1
Blaschke, G; Boos, J; Haberland, S; Hempel, G; Möhling, N; Schulze-Westhoff, P1
Brieden, T; Gieseler, F; Kunze, J; Nüssler, V; Valsamas, S1
Fiallo, M; Gallois, L; Garnier-Suillerot, A1
Bondi, F; Crescimanno, A; Mariani, G; Musso, M; Polizzi, V; Porretto, F; Scalone, R; Tolomeo, M1
Fukushima, T; Imamura, S; Inai, K; Inoue, H; Kishi, S; Nakamura, T; Nakayama, T; Takemura, H; Ueda, T; Urasaki, Y; Yamauchi, T1
Fukushima, T; Imamura, S; Misaki, H; Ueda, T; Urasaki, Y; Yamashita, T; Yamauchi, T; Yoshio, N1
Hofmann, S; Kuhlmann, O; Weiss, M1
Barbui, T; Bassan, R; Chiodini, B1
Kasimir-Bauer, S; Scheulen, ME; Schröder, JK; Seeber, S1
Clark, M; Gieseler, F; Puschmann, M; Stiebeling, K; Valsamas, S1
Aita, P; Bearz, A; Boiocchi, M; Colussi, AM; Corona, G; Crivellari, D; Robieux, I; Sorio, R; Stocco, F; Toffoli, G1
de Witte, T; Linssen, P; Masereeuw, R; Muus, P; Raymakers, R; Smeets, M; Vierwinden, G1
Fukushima, T; Goto, N; Kuraishi, Y; Ogawa, M; Ohno, R; Okabe, KI; Ueda, T; Urabe, A; Yamashita, T1
Kang, W; Weiss, M2
Bargoni, A; Cavalli, R; Fundarò, A; Gasco, MR; Vighetto, D; Zara, GP1
Bengala, C; Biadi, O; Conte, PF; Danesi, R; Del Tacca, M; Donati, S; Favre, C; Fogli, S; Guarneri, V; Innocenti, F; Mariani, M; Pazzagli, I1
Aita, P; Basso, B; Boiocchi, M; Corona, G; Ruolo, G; Rupolo, M; Sorio, R; Toffoli, G1
Giessler, C; Kang, W; Weiss, M1
Barbara, C; Bocci, G; Danesi, R; Del Tacca, M; Di Paolo, A; Fioravanti, A; Orlandi, P1
Corona, G; Crivellari, D; Lestuzzi, C; Lombardi, D; Lucenti, A; Magri, MD; Massacesi, C; Sorio, R; Talamini, R; Toffoli, G; Veronesi, A1

Reviews

1 review(s) available for idarubicinol and idarubicin

ArticleYear
Selected pharmacologic characteristics of idarubicin and idarubicinol.
    Leukemia, 1992, Volume: 6 Suppl 1

    Topics: Animals; Daunorubicin; Humans; Idarubicin

1992

Trials

9 trial(s) available for idarubicinol and idarubicin

ArticleYear
Idarubicin metabolism and pharmacokinetics after intravenous and oral administration in cancer patients: a crossover study.
    Cancer chemotherapy and pharmacology, 1992, Volume: 30, Issue:4

    Topics: Administration, Oral; Biological Availability; Daunorubicin; Glycosylation; Humans; Idarubicin; Infusions, Intravenous; Kidney; Kidney Diseases; Liver Neoplasms; Neoplasms

1992
Pharmacokinetics of idarubicin after oral administration in elderly leukemic patients.
    Leukemia, 1990, Volume: 4, Issue:3

    Topics: Administration, Oral; Aged; Biological Availability; Daunorubicin; Drug Evaluation; Female; Humans; Idarubicin; Leukemia, Myeloid, Acute; Male; Multicenter Studies as Topic

1990
Plasma pharmacokinetics and cerebrospinal fluid concentrations of idarubicin and idarubicinol in pediatric leukemia patients: a Childrens Cancer Study Group report.
    Cancer research, 1990, Oct-15, Volume: 50, Issue:20

    Topics: Adolescent; Adult; Child; Child, Preschool; Daunorubicin; Drug Evaluation; Humans; Idarubicin; Infant; Leukemia

1990
Oral idarubicin pharmacokinetics--correlation of trough level with idarubicin area under curve.
    Leukemia, 1996, Volume: 10, Issue:4

    Topics: Acute Disease; Administration, Oral; Adult; Antibiotics, Antineoplastic; Antineoplastic Combined Chemotherapy Protocols; Chromatography, High Pressure Liquid; Cytarabine; Daunorubicin; Drug Administration Schedule; Humans; Idarubicin; Leukemia, Myeloid; Lymphoma, Non-Hodgkin; Metabolic Clearance Rate; Middle Aged

1996
A phase-II study with idarubicin, ifosfamide and VP-16 (IIVP-16) in patients with refractory or relapsed aggressive and high grade non-Hodgkin's lymphoma.
    Leukemia & lymphoma, 1997, Volume: 24, Issue:5-6

    Topics: Adult; Aged; Antineoplastic Combined Chemotherapy Protocols; Daunorubicin; Etoposide; Female; Humans; Idarubicin; Ifosfamide; Individuality; Lymphoma, Non-Hodgkin; Male; Middle Aged

1997
Plasma pharmacokinetics of idarubicin and its 13-dihydro metabolite--a comparison of bolus versus 2 h infusion during a 3 day course.
    Anti-cancer drugs, 1997, Volume: 8, Issue:1

    Topics: Aged; Aged, 80 and over; Antibiotics, Antineoplastic; Area Under Curve; Chromatography, Liquid; Cross-Over Studies; Daunorubicin; Female; Humans; Idarubicin; Infusions, Intravenous; Injections, Intravenous; Leukemia, Myeloid, Acute; Male; Middle Aged; Spectrometry, Fluorescence

1997
Dose-finding and pharmacologic study of chronic oral idarubicin therapy in metastatic breast cancer patients.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 2000, Volume: 6, Issue:6

    Topics: Administration, Oral; Adult; Aged; Antibiotics, Antineoplastic; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Area Under Curve; Breast Neoplasms; Cyclophosphamide; Daunorubicin; Docetaxel; Dose-Response Relationship, Drug; Doxorubicin; Epirubicin; Female; Fluorouracil; Humans; Idarubicin; Maximum Tolerated Dose; Methotrexate; Middle Aged; Neoplasm Metastasis; Paclitaxel; Taxoids; Time Factors

2000
A pharmacokinetic study of idarubicin in Japanese patients with malignant lymphoma: relationship with leukocytopenia and neutropenia.
    International journal of hematology, 2001, Volume: 74, Issue:3

    Topics: Aged; Antibiotics, Antineoplastic; Area Under Curve; Biotransformation; Daunorubicin; Dose-Response Relationship, Drug; Female; Half-Life; Humans; Idarubicin; Japan; Leukocyte Count; Leukopenia; Lymphoma; Male; Middle Aged; Neutropenia

2001
Innovative schedule of oral idarubicin in elderly patients with metastatic breast cancer: comprehensive results of a phase II multi-institutional study with pharmacokinetic drug monitoring.
    Annals of oncology : official journal of the European Society for Medical Oncology, 2006, Volume: 17, Issue:5

    Topics: Administration, Oral; Aged; Aged, 80 and over; Antibiotics, Antineoplastic; Bone Neoplasms; Breast Neoplasms; Chromatography, High Pressure Liquid; Daunorubicin; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Monitoring; Female; Humans; Idarubicin; Liver Neoplasms; Lung Neoplasms; Soft Tissue Neoplasms

2006

Other Studies

37 other study(ies) available for idarubicinol and idarubicin

ArticleYear
Anthracyclines and their C-13 alcohol metabolites: growth inhibition and DNA damage following incubation with human tumor cells in culture.
    Cancer chemotherapy and pharmacology, 1992, Volume: 30, Issue:1

    Topics: Antibiotics, Antineoplastic; Cell Division; Daunorubicin; DNA Damage; DNA, Neoplasm; Doxorubicin; Epirubicin; Glioma; Humans; Idarubicin; Leukemia, Myeloid; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Tumor Cells, Cultured

1992
High-performance liquid chromatographic analysis of idarubicin and fluorescent metabolites in biological fluids.
    Cancer chemotherapy and pharmacology, 1992, Volume: 30, Issue:4

    Topics: Calibration; Chromatography, High Pressure Liquid; Daunorubicin; Fluorescence; Humans; Idarubicin; Reference Standards

1992
Cytotoxicity and DNA damage caused by 4-demethoxydaunorubicin and its metabolite 4-demethoxy-13-hydroxydaunorubicin in human acute myeloid leukemia cells.
    Cancer chemotherapy and pharmacology, 1990, Volume: 26, Issue:5

    Topics: Adult; Antineoplastic Agents; Cell Division; Daunorubicin; DNA Damage; DNA, Neoplasm; Humans; Idarubicin; Leukemia, Myeloid, Acute; Tumor Cells, Cultured; Tumor Stem Cell Assay

1990
Pharmacokinetics of 4-demethoxydaunorubicin in cancer patients.
    Cancer chemotherapy and pharmacology, 1990, Volume: 25, Issue:6

    Topics: Administration, Oral; Adult; Aged; Aged, 80 and over; Biological Availability; Daunorubicin; Female; Half-Life; Humans; Idarubicin; Injections, Intravenous; Male; Middle Aged; Neoplasms

1990
Pharmacokinetics of oral idarubicin in breast cancer patients with reference to antitumor activity and side effects.
    Clinical pharmacology and therapeutics, 1989, Volume: 45, Issue:6

    Topics: Administration, Oral; Aged; Biological Availability; Breast Neoplasms; Daunorubicin; Half-Life; Humans; Idarubicin; Male; Middle Aged

1989
Reversed-phase liquid chromatographic determination of idarubicin and its 13-hydroxy metabolite in human plasma.
    Journal of chromatography, 1989, Mar-24, Volume: 488, Issue:2

    Topics: Chemical Phenomena; Chemistry; Chromatography, High Pressure Liquid; Daunorubicin; Humans; Hydrogen-Ion Concentration; Idarubicin; Spectrometry, Fluorescence

1989
Improved high-performance liquid chromatographic method using loop-column extraction for analysis of idarubicin and idarubicinol in plasma.
    Journal of chromatography, 1989, Jul-21, Volume: 491, Issue:2

    Topics: Chromatography, High Pressure Liquid; Daunorubicin; Humans; Idarubicin; Time Factors

1989
Pharmacokinetics of idarubicin after daily intravenous administration in leukemic patients.
    Leukemia research, 1987, Volume: 11, Issue:11

    Topics: Antibiotics, Antineoplastic; Biotransformation; Daunorubicin; Humans; Idarubicin; Injections, Intravenous; Kinetics; Leukemia, Myeloid, Acute

1987
Susceptibility of idarubicin, daunorubicin, and their C-13 alcohol metabolites to transport-mediated multidrug resistance.
    Biochemical pharmacology, 1995, Nov-09, Volume: 50, Issue:10

    Topics: Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Breast Neoplasms; Cell Survival; Culture Media; Cyclosporine; Daunorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Stability; HL-60 Cells; Humans; Idarubicin; Intracellular Fluid; Tumor Cells, Cultured

1995
Comparative resistance of idarubicin, doxorubicin and their C-13 alcohol metabolites in human MDR1 transfected NIH-3T3 cells.
    Cancer chemotherapy and pharmacology, 1995, Volume: 36, Issue:3

    Topics: 3T3 Cells; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cell Line; Daunorubicin; Doxorubicin; Drug Resistance, Multiple; Humans; Idarubicin; Mice; Transfection

1995
Influence of idarubicinol on the antileukemic effect of idarubicin.
    Leukemia research, 1994, Volume: 18, Issue:12

    Topics: Daunorubicin; DNA; DNA Damage; Humans; Idarubicin; In Vitro Techniques; Leukemia, Myeloid; Nucleic Acid Synthesis Inhibitors; Tumor Cells, Cultured

1994
Cytotoxicity of anthracyclines: correlation with cellular uptake, intracellular distribution and DNA binding.
    Annals of hematology, 1994, Volume: 69 Suppl 1

    Topics: Antibiotics, Antineoplastic; Antineoplastic Agents; Cell Nucleus; Cell Survival; Daunorubicin; DNA; Humans; Idarubicin; Lethal Dose 50; Lymphocytes; Tumor Cells, Cultured

1994
Toxicity of idarubicin and doxorubicin towards normal and leukemic human bone marrow progenitors in relation to their proliferative state.
    Leukemia, 1994, Volume: 8, Issue:3

    Topics: Acute Disease; Antineoplastic Agents; Cell Division; Daunorubicin; Doxorubicin; Granulocytes; Hematopoietic Stem Cells; Humans; Idarubicin; Leukemia, Myeloid; Macrophages; Tumor Stem Cell Assay

1994
Comparison of the intracellular pharmacokinetics of daunorubicin and idarubicin in patients with acute leukemia.
    Leukemia research, 1994, Volume: 18, Issue:4

    Topics: Acute Disease; Aged; Daunorubicin; Female; Humans; Idarubicin; Leukemia, Myeloid, Acute; Male; Middle Aged

1994
Cellular pharmacology of idarubicinol in multidrug-resistant LoVo cell lines.
    International journal of cancer, 1996, Jul-03, Volume: 67, Issue:1

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Daunorubicin; Drug Resistance, Multiple; Humans; Idarubicin; Tumor Cells, Cultured

1996
Comparison of idarubicin and daunorubicin and their main metabolites regarding intracellular uptake and effect on sensitive and multidrug-resistant HL60 cells.
    Cancer chemotherapy and pharmacology, 1996, Volume: 38, Issue:5

    Topics: Antibiotics, Antineoplastic; Antineoplastic Agents; Cell Division; Daunorubicin; Dose-Response Relationship, Drug; Drug Resistance, Multiple; HL-60 Cells; Humans; Idarubicin

1996
Comparative activity of idarubicin and idarubicinol in combination with cyclosporin A in multidrug-resistant leukemia cells.
    Cancer chemotherapy and pharmacology, 1996, Volume: 39, Issue:1-2

    Topics: Antibiotics, Antineoplastic; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Cyclosporine; Daunorubicin; Drug Resistance, Multiple; Flow Cytometry; Idarubicin; Immunosuppressive Agents; Tumor Cells, Cultured

1996
Pharmacokinetics and tissue distribution of idarubicin and its active metabolite idarubicinol in the rabbit.
    Cancer chemotherapy and pharmacology, 1997, Volume: 39, Issue:6

    Topics: Animals; Antibiotics, Antineoplastic; Chromatography, High Pressure Liquid; Daunorubicin; Idarubicin; Rabbits; Tissue Distribution

1997
Determination of idarubicin and idarubicinol in plasma by capillary electrophoresis.
    Journal of chromatography. B, Biomedical sciences and applications, 1997, Sep-26, Volume: 698, Issue:1-2

    Topics: Antibiotics, Antineoplastic; Child; Daunorubicin; Electrophoresis, Capillary; Humans; Idarubicin; Reference Standards

1997
Oral idarubicin pharmacokinetics--correlation of trough level with idarubicin area under curve.
    Leukemia, 1997, Volume: 11 Suppl 5

    Topics: Administration, Oral; Adult; Antibiotics, Antineoplastic; Antineoplastic Agents; Chromatography, High Pressure Liquid; Daunorubicin; Half-Life; Humans; Idarubicin; Leukemia, Myeloid, Acute; Lymphoma, Non-Hodgkin; Metabolic Clearance Rate; Middle Aged; Regression Analysis

1997
Intracellular pharmacokinetics of anthracyclines in human leukemia cells: correlation of DNA-binding with apoptotic cell death.
    International journal of clinical pharmacology and therapeutics, 1998, Volume: 36, Issue:1

    Topics: Antibiotics, Antineoplastic; Antineoplastic Agents; Apoptosis; Cell Nucleus; Daunorubicin; DNA Damage; DNA, Neoplasm; Drug Resistance, Neoplasm; HL-60 Cells; Humans; Idarubicin; Leukemia

1998
Comparison of the interaction of doxorubicin, daunorubicin, idarubicin and idarubicinol with large unilamellar vesicles. Circular dichroism study.
    Biochimica et biophysica acta, 1998, Mar-06, Volume: 1370, Issue:1

    Topics: Anthracyclines; Circular Dichroism; Daunorubicin; Dimerization; Doxorubicin; Idarubicin; Lipid Bilayers; Liposomes; Membranes, Artificial; Models, Molecular; Solvents

1998
Only association of low concentrations of idarubicin plus idarubicinol induced apoptosis on leukaemic cells.
    Leukemia research, 1998, Volume: 22, Issue:6

    Topics: Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Daunorubicin; HL-60 Cells; Humans; Idarubicin

1998
Idarubicin and idarubicinol are less affected by topoisomerase II-related multidrug resistance than is daunorubicin.
    Leukemia research, 1998, Volume: 22, Issue:7

    Topics: Antineoplastic Agents; Cell Division; Cell Extracts; Cell Survival; Cytotoxins; Daunorubicin; DNA Topoisomerases, Type II; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Humans; Idarubicin; Trypan Blue; Tumor Cells, Cultured

1998
Effect of PSC 833 on the cytotoxicity of idarubicin and idarubicinol in multidrug-resistant K562 cells.
    Leukemia research, 1999, Volume: 23, Issue:1

    Topics: Antibiotics, Antineoplastic; Antineoplastic Combined Chemotherapy Protocols; Cyclosporins; Daunorubicin; Drug Resistance, Multiple; Humans; Idarubicin; K562 Cells

1999
Determination of idarubicin and idarubicinol in rat plasma using reversed-phase high-performance liquid chromatography and fluorescence detection.
    Journal of chromatography. B, Biomedical sciences and applications, 1999, May-28, Volume: 728, Issue:2

    Topics: Animals; Antibiotics, Antineoplastic; Chromatography, High Pressure Liquid; Daunorubicin; Idarubicin; Male; Rats; Rats, Wistar; Reproducibility of Results; Sensitivity and Specificity; Spectrometry, Fluorescence

1999
Apoptosis by anthracyclines at therapeutic concentrations in MDR1+ human leukemic cells.
    Advances in experimental medicine and biology, 1999, Volume: 457

    Topics: Annexin A5; Antibiotics, Antineoplastic; Apoptosis; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Membrane; Daunorubicin; Drug Resistance, Multiple; Flow Cytometry; Genes, MDR; Humans; Idarubicin; Leukemia-Lymphoma, Adult T-Cell; Membrane Lipids; Necrosis; Phosphatidylserines; Tumor Cells, Cultured

1999
In vitro effect of multidrug resistance modifiers on idarubicinol efflux in blasts of acute myeloid leukemia.
    Journal of cancer research and clinical oncology, 2000, Volume: 126, Issue:2

    Topics: Antineoplastic Agents; Blast Crisis; Calcium Channel Blockers; Daunorubicin; Dihydropyridines; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Idarubicin; Leukemia, Myeloid, Acute; Tumor Cells, Cultured; Verapamil

2000
Induction of apoptosis by idarubicin: how important is the plasma peak?
    International journal of clinical pharmacology and therapeutics, 2000, Volume: 38, Issue:4

    Topics: Antibiotics, Antineoplastic; Antineoplastic Agents; Apoptosis; Area Under Curve; Daunorubicin; DNA, Neoplasm; HL-60 Cells; Humans; Idarubicin; Leukemia, Promyelocytic, Acute

2000
Cyclosporin increases cellular idarubicin and idarubicinol concentrations in relapsed or refractory AML mainly due to reduced systemic clearance.
    Leukemia, 2001, Volume: 15, Issue:1

    Topics: Acute Disease; Adolescent; Adult; Aged; Antineoplastic Combined Chemotherapy Protocols; Cyclosporine; Daunorubicin; Female; Humans; Idarubicin; Immunosuppressive Agents; Leukemia, Myeloid; Male; Middle Aged; Pilot Projects; Prospective Studies; Recurrence

2001
Influence of P-glycoprotein modulators on cardiac uptake, metabolism, and effects of idarubicin.
    Pharmaceutical research, 2001, Volume: 18, Issue:11

    Topics: Algorithms; Animals; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cyclosporins; Daunorubicin; Heart; Idarubicin; In Vitro Techniques; Male; Myocardium; Rats; Rats, Sprague-Dawley; Stroke Volume; Verapamil

2001
Pharmacokinetics and tissue distribution of idarubicin-loaded solid lipid nanoparticles after duodenal administration to rats.
    Journal of pharmaceutical sciences, 2002, Volume: 91, Issue:5

    Topics: Animals; Antibiotics, Antineoplastic; Daunorubicin; Drug Administration Routes; Drug Carriers; Duodenum; Idarubicin; Nanotechnology; Rats; Rats, Wistar; Solutions; Tissue Distribution

2002
High-dose consolidation chemotherapy with Idarubicin and alkylating agents following induction with gemcitabine-epirubicin-paclitaxel in metastatic breast cancer: a dose finding study.
    Bone marrow transplantation, 2003, Volume: 31, Issue:4

    Topics: Adult; Antineoplastic Agents, Alkylating; Antineoplastic Combined Chemotherapy Protocols; Breast Neoplasms; Daunorubicin; Deoxycytidine; Disease Progression; Disease-Free Survival; Dose-Response Relationship, Drug; Epirubicin; Female; Humans; Idarubicin; Melphalan; Middle Aged; Neoplasm Metastasis; Paclitaxel; Remission Induction; Taxoids; Thiotepa; Time Factors; Transplantation Conditioning; Treatment Outcome

2003
Modeling the metabolism of idarubicin to idarubicinol in rat heart: effect of rutin and phenobarbital.
    Drug metabolism and disposition: the biological fate of chemicals, 2003, Volume: 31, Issue:4

    Topics: Amiodarone; Animals; Antineoplastic Agents; Daunorubicin; Drug Design; Excitatory Amino Acid Antagonists; Heart; Idarubicin; Kinetics; Male; Phenobarbital; Rats; Rats, Sprague-Dawley; Rutin; Time Factors; Vasodilator Agents; Verapamil

2003
Pharmacokinetic comparison of 120-hour infusion versus hyperfractionated oral administration of idarubicin.
    Journal of chemotherapy (Florence, Italy), 2004, Volume: 16, Issue:2

    Topics: Administration, Oral; Adult; Aged; Aged, 80 and over; Antibiotics, Antineoplastic; Area Under Curve; Daunorubicin; Female; Humans; Idarubicin; Infusions, Intravenous; Lymphoma, Non-Hodgkin; Male; Middle Aged

2004
Effects of idarubicin and idarubicinol on rat coronary resistance and vasoconstrictor responsiveness of isolated aorta and mesentery.
    Anti-cancer drugs, 2006, Volume: 17, Issue:1

    Topics: Animals; Antibiotics, Antineoplastic; Aorta, Thoracic; Coronary Circulation; Daunorubicin; Dose-Response Relationship, Drug; Heart; Idarubicin; In Vitro Techniques; Inhibitory Concentration 50; Male; Mesenteric Arteries; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Potassium Chloride; Rats; Rats, Wistar; Vascular Resistance; Vasoconstriction; Vasoconstrictor Agents

2006
Idarubicin and idarubicinol effects on breast cancer multicellular spheroids.
    Journal of chemotherapy (Florence, Italy), 2005, Volume: 17, Issue:6

    Topics: Antibiotics, Antineoplastic; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; Cell Survival; Daunorubicin; Dose-Response Relationship, Drug; Female; Humans; Idarubicin; Inhibitory Concentration 50; Spheroids, Cellular; Time Factors

2005