Page last updated: 2024-09-05

iclaprim and linezolid

iclaprim has been researched along with linezolid in 6 studies

Compound Research Comparison

Studies
(iclaprim)
Trials
(iclaprim)
Recent Studies (post-2010)
(iclaprim)
Studies
(linezolid)
Trials
(linezolid)
Recent Studies (post-2010) (linezolid)
457163,9162222,188

Protein Interaction Comparison

ProteinTaxonomyiclaprim (IC50)linezolid (IC50)
Prostaglandin G/H synthase 1Homo sapiens (human)8.19
Amine oxidase [flavin-containing] BHomo sapiens (human)2.1
Succinate dehydrogenase [ubiquinone] flavoprotein subunit, mitochondrialHomo sapiens (human)8.19

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (66.67)29.6817
2010's2 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hawser, S; Islam, K; Schneider, P1
Fritsche, TR; Jones, RN; Sader, HS1
Hawser, S; Islam, K; Laue, H; Lociuro, S; Seguin, A; Valensise, T1
Barrow, EW; Barrow, WW; Berlin, KD; Bourne, CR; Bourne, PC; Bunce, RA1
Corey, GR; Stryjewski, ME1
Cattoir, V; Daurel, C1

Reviews

2 review(s) available for iclaprim and linezolid

ArticleYear
New treatments for methicillin-resistant Staphylococcus aureus.
    Current opinion in critical care, 2009, Volume: 15, Issue:5

    Topics: Acetamides; Anti-Bacterial Agents; Cephalosporins; Clinical Trials as Topic; Daptomycin; Evidence-Based Medicine; Glycopeptides; Humans; Linezolid; Methicillin-Resistant Staphylococcus aureus; Minocycline; Oxazolidinones; Pyrimidines; Streptococcal Infections; Tigecycline

2009
[Update on antimicrobial chemotherapy].
    Medecine et maladies infectieuses, 2010, Volume: 40, Issue:3

    Topics: Acetamides; Aminoglycosides; Anti-Infective Agents; beta-Lactams; Carbapenems; Cephalosporins; Daptomycin; Doripenem; Drug Resistance, Bacterial; Ertapenem; Fluoroquinolones; France; Humans; Linezolid; Lipoglycopeptides; Minocycline; Oxazolidinones; Penicillins; Pyrimidines; Teicoplanin; Tigecycline

2010

Other Studies

4 other study(ies) available for iclaprim and linezolid

ArticleYear
Iclaprim, a novel diaminopyrimidine with potent activity on trimethoprim sensitive and resistant bacteria.
    Bioorganic & medicinal chemistry letters, 2003, Dec-01, Volume: 13, Issue:23

    Topics: Animals; Drug Resistance, Bacterial; Folic Acid Antagonists; Lung; Methicillin Resistance; Mice; Microbial Sensitivity Tests; Pyrimidines; Sepsis; Staphylococcus aureus; Structure-Activity Relationship; Tetrahydrofolate Dehydrogenase; Trimethoprim Resistance; Vancomycin

2003
Potency and bactericidal activity of iclaprim against recent clinical gram-positive isolates.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:5

    Topics: Anti-Bacterial Agents; Enterococcus faecalis; Europe; Gram-Positive Bacterial Infections; Gram-Positive Cocci; Hospitalization; Humans; Methicillin; Methicillin-Resistant Staphylococcus aureus; Microbial Sensitivity Tests; Pyrimidines; Staphylococcus aureus; Streptococcus; United States

2009
In vitro bactericidal activity of iclaprim in human plasma.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:10

    Topics: Anti-Bacterial Agents; Humans; Methicillin-Resistant Staphylococcus aureus; Microbial Sensitivity Tests; Plasma; Pyrimidines; Staphylococcus aureus

2009
Inhibition of antibiotic-resistant Staphylococcus aureus by the broad-spectrum dihydrofolate reductase inhibitor RAB1.
    Antimicrobial agents and chemotherapy, 2010, Volume: 54, Issue:9

    Topics: Anti-Bacterial Agents; Enzyme Inhibitors; Inhibitory Concentration 50; Microbial Sensitivity Tests; Protein Structure, Secondary; Protein Structure, Tertiary; Staphylococcus aureus; Tetrahydrofolate Dehydrogenase

2010
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