Page last updated: 2024-09-03

ici 89406 and propranolol

ici 89406 has been researched along with propranolol in 10 studies

Compound Research Comparison

Studies
(ici 89406)
Trials
(ici 89406)
Recent Studies (post-2010)
(ici 89406)
Studies
(propranolol)
Trials
(propranolol)
Recent Studies (post-2010) (propranolol)
451233,3103,4063,218

Protein Interaction Comparison

ProteinTaxonomyici 89406 (IC50)propranolol (IC50)
Beta-1 adrenergic receptor Cavia porcellus (domestic guinea pig)0.0347
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.0288
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)2.294
Cytochrome P450 1A2Homo sapiens (human)4
Beta-2 adrenergic receptorHomo sapiens (human)0.0114
Beta-1 adrenergic receptorHomo sapiens (human)0.0575
5-hydroxytryptamine receptor 1AHomo sapiens (human)3.9811
Beta-2 adrenergic receptorRattus norvegicus (Norway rat)0.012
Cytochrome P450 2D6Homo sapiens (human)2.9706
Beta-3 adrenergic receptorHomo sapiens (human)0.0493
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.0288
Beta-1 adrenergic receptorRattus norvegicus (Norway rat)0.012
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.0288
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0827
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.0288
Beta-3 adrenergic receptorRattus norvegicus (Norway rat)0.012
5-hydroxytryptamine receptor 2AHomo sapiens (human)1.466
5-hydroxytryptamine receptor 2CHomo sapiens (human)2.294
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.0288
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.243
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.0288
Sodium-dependent serotonin transporterHomo sapiens (human)0.38
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.342
5-hydroxytryptamine receptor 6Homo sapiens (human)3.065
Beta-2 adrenergic receptorCanis lupus familiaris (dog)0.017
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.0288
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)2.828
Sodium channel protein type 5 subunit alphaHomo sapiens (human)2.1
Sodium/bile acid cotransporterHomo sapiens (human)5.5
Beta-2 adrenergic receptorCavia porcellus (domestic guinea pig)0.0288
GABA theta subunitRattus norvegicus (Norway rat)0.0288
Sigma non-opioid intracellular receptor 1Homo sapiens (human)2.87
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.0288

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19903 (30.00)18.7374
1990's5 (50.00)18.2507
2000's2 (20.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baker, JG1
Hartling, O; Svendsen, TL; Trap-Jensen, J1
Fraeyman, N; Van de Velde, E; Van Ermen, A; Vanscheeuwijck, P1
Gousse, A; Latifpour, J; Weiss, RM; Yoshida, M1
Ahmad, S; Chrétien, P; Daniel, EE; Shen, SH1
Felder, CC; Jose, PA; McKelvey, AM; Nakamura, KT; Piccio, MM; Robillard, JE1
Frame, LH; Liang, BT; Molinoff, PB1
Gerber, JG; Hedberg, A; Molinoff, PB; Nies, AS; Wolfe, BB1
Murugaiah, KD; O'Donnell, JM1
Kopka, K; Law, MP; Pike, VW; Schäfers, M; Schober, O; Wagner, S1

Trials

1 trial(s) available for ici 89406 and propranolol

ArticleYear
Effects of pindolol and propranolol on beta adrenergic receptors on human lymphocytes.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:1

    Topics: Animals; Cell Membrane; Double-Blind Method; Heart; Humans; Kinetics; Lung; Lymphocytes; Pindolol; Propanolamines; Propranolol; Rats; Receptors, Adrenergic, beta

1986

Other Studies

9 other study(ies) available for ici 89406 and propranolol

ArticleYear
The selectivity of beta-adrenoceptor antagonists at the human beta1, beta2 and beta3 adrenoceptors.
    British journal of pharmacology, 2005, Volume: 144, Issue:3

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Algorithms; Animals; Cell Line; CHO Cells; Cricetinae; Dioxoles; Humans; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3

2005
Immediate haemodynamic effects of propranolol, practolol, pindolol, atenolol and ICI 89,406 in healthy volunteers.
    European journal of clinical pharmacology, 1979, May-21, Volume: 15, Issue:4

    Topics: Adolescent; Adrenergic beta-Antagonists; Adult; Atenolol; Blood Pressure; Cardiac Output; Heart Rate; Hemodynamics; Humans; Male; Pindolol; Practolol; Propanolamines; Propranolol

1979
Influence of age on the beta 1- and beta 2-adrenergic receptors in rat liver.
    Molecular pharmacology, 1992, Volume: 42, Issue:4

    Topics: Adenylyl Cyclases; Aging; Animals; Binding, Competitive; Cell Membrane; Imidazoles; Liver; Liver Glycogen; Male; Pindolol; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta

1992
Beta adrenergic receptor alterations in diabetic rat prostate: effects of insulin and dietary myoinositol.
    The Prostate, 1991, Volume: 19, Issue:2

    Topics: Adrenergic beta-Antagonists; Animals; Blood Glucose; Body Weight; Diabetes Mellitus, Experimental; Dihydroalprenolol; Dose-Response Relationship, Drug; Drinking; Inositol; Insulin; Isoproterenol; Male; Organ Size; Propanolamines; Propranolol; Prostate; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Streptozocin; Urination

1991
Characterization of beta adrenoceptors on cultured endothelial cells by radioligand binding.
    Life sciences, 1990, Volume: 47, Issue:25

    Topics: Adrenergic alpha-Antagonists; Albuterol; Animals; Binding, Competitive; Cattle; Cells, Cultured; Endothelium, Vascular; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Pindolol; Propanolamines; Propranolol; Pulmonary Artery; Receptors, Adrenergic, beta

1990
Ontogeny of renal beta adrenoceptors in the sheep.
    Pediatric nephrology (Berlin, Germany), 1990, Volume: 4, Issue:6

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aging; Animals; Binding, Competitive; Ethanolamines; Isoproterenol; Kidney; Pindolol; Propanolamines; Propranolol; Radioligand Assay; Receptors, Adrenergic, beta; Sheep; Vasodilation

1990
Beta 2-adrenergic receptors contribute to catecholamine-stimulated shortening of action potential duration in dog atrial muscle.
    Proceedings of the National Academy of Sciences of the United States of America, 1985, Volume: 82, Issue:13

    Topics: Action Potentials; Animals; Atropine; Catecholamines; Dogs; Dose-Response Relationship, Drug; Heart Atria; Isoproterenol; Kinetics; Muscle, Smooth, Vascular; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Reserpine

1985
Facilitation of norepinephrine release from cerebral cortex is mediated by beta 2-adrenergic receptors.
    Life sciences, 1995, Volume: 57, Issue:20

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Cerebral Cortex; Drug Interactions; Electric Stimulation; Norepinephrine; Prenalterol; Propanolamines; Propranolol; Rats; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Tritium

1995
Are [O-methyl-11C]derivatives of ICI 89,406 beta1-adrenoceptor selective radioligands suitable for PET?
    European journal of nuclear medicine and molecular imaging, 2008, Volume: 35, Issue:1

    Topics: Adrenergic beta-Antagonists; Air; Animals; Carbon Dioxide; Carbon Radioisotopes; Exhalation; Ligands; Male; Myocardium; Positron-Emission Tomography; Propanolamines; Propranolol; Radioactivity; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Substrate Specificity; Tissue Distribution

2008