Page last updated: 2024-08-26

ici 164384 and afimoxifene

ici 164384 has been researched along with afimoxifene in 58 studies

Research

Studies (58)

Timeframe	Studies, this research(%)	All Research%
pre-1990	4 (6.90)	18.7374
1990's	50 (86.21)	18.2507
2000's	3 (5.17)	29.6817
2010's	1 (1.72)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Cotnoir-White, D; Gleason, JL; Jutras, I; Kulpa, J; Mader, S; Mendoza-Sanchez, R; Moitessier, N; Pottel, J	1
Chang, C; Jiang, SY; Jordan, VC; Wolf, DM; Yingling, JM	1
Beug, H; Boehmelt, G; Enrietto, PJ; Kabrun, N; Mellitzer, G; Walker, A; Zenke, M	1
Albaladejo, V; Andre, J; Joly-Pharaboz, MO; Nicolas, B; Zhou-Li, F	1
Ballejo, G; Gong, Y; Murphy, LC; Murphy, LJ	1
Emmas, CE; Fawell, SE; Hoare, SA; Parker, MG	1
Abbondanza, C; Armetta, I; Medici, N; Minucci, S; Molinari, AM; Moncharmont, B; Nigro, V; Puca, GA	1
Croxtall, JD; Jamil, A; White, JO	1
Giambiagi, N; Pasqualini, JR	1
Chetrite, G; Pasqualini, JR	1
Berry, M; Chambon, P; Metzger, D	1
Baxter, JD; Greene, GL; Hort, E; Kushner, PJ; Shine, J	1
Jordan, VC; Murphy, CS; Pink, JJ	1
Dickson, RB; Katz, D; Lippman, ME; Shima, TB; Thompson, EW; Wakeling, AE	1
Dufour, JM; Labrie, F; Levesque, C; Merand, Y; Poirier, D; Poulin, R	1
Wakeling, AE	1
Chambon, P; Green, S; Jin, JR; Webster, NJ	1
Chambon, P; Endoh, H; Gotoh, Y; Kato, S; Kawashima, H; Kitamoto, T; Masuhiro, Y; Masushige, S; Metzger, D; Nishida, E; Sasaki, H; Uchiyama, S	1
Dekker, A; Dorssers, LC; Foekens, JA; van Agthoven, T; van Agthoven, TL	1
Chambon, P; Chiba, H; Clifford, J; Metzger, D	1
Aliau, S; Borgna, JL; Groblewski, T	1
Dickson, RB; Johnson, GR; Martínez-Lacaci, I; Normanno, N; Plowman, GD; Saceda, M; Salomon, DS	1
Dauvois, S; Mahfoudi, A; Parker, MG; Roulet, E; Wahli, W	1
Fritsch, M; Jiang, SY; Jordan, VC; Pink, JJ	1
Halliwell, B; Wiseman, H	1
King, RJ; Lewis, DF; Parker, MG	1
Clairmont, A; Drewes, T; Klein-Hitpass, L; Ryffel, GU	1
Cavaillès, V; Danielian, PS; Dauvois, S; Parker, MG	1
Badia, E; Duchesne, MJ; Fournier-Bidoz, S; Nicolas, JC; Pons, M; Simar-Blanchet, AE; Terouanne, B	1
Musgrove, EA; Sutherland, RL; Sweeney, KJ; Warlters, A; Watts, CK	1
Miksicek, RJ	1
Aronica, SM; Katzenellenbogen, BS; Kraus, WL	1
Dauvois, S; Parker, MG; White, R	1
Bicknell, R; Harris, AL; Toi, M	1
Brünner, N; Clarke, R; Coopman, P; Derocq, D; Garcia, M; Rochefort, H	1
Chalbos, D; Philips, A; Rochefort, H	1
Conneely, OM; O'Malley, BW; Smith, CL	1
Chalbos, D; Galtier, F; Philips, A; Rochefort, H	1
Chetrite, G; Pasqualini, JR; Urabe, M	1
Santen, RJ; Santner, SJ	1
Sager, R; Webster, L; Zajchowski, DA	1
Ali, S; Bornert, JM; Chambon, P; Metzger, D	1
Adlercreutz, H; Garey, J; Gurpide, E; Markiewicz, L	1
Clerico, L; de Cupis, A; Favoni, RE; Ferrera, A; Noonan, D; Pirani, P	1
Clemm, DL; Goldman, ME; Hermann, T; McDonnell, DP; Pike, JW	1
Ekena, K; Katzenellenbogen, BS; Keller, AL; Krueger, KD; Montano, MM	1
Fournier, B; Häring, S; Kaye, AM; Sömjen, D	1
Flouriot, G; Pakdel, F; Valotaire, Y	1
Gurpide, E; Markiewicz, L	1
Eng, FC; Ferrara, J; Lee, HS; White, JH; Willson, TM	1
Bonnet, S; Brouillet, JP; Derocq, D; Garcia, M; Platet, N; Rochefort, H; Touitou, I	1
Bartholdi, M; Humm, R; Simmons, SJ; Webster, L; White, FA; Zajchowski, DA	1
Anghel, SI; Barsalou, A; Carrière, J; Gao, W; Mader, S	1
Jeannin, E; Liu, JW; Picard, D	1
Löwik, CW; Papapoulos, SE; van Bezooijen, RL; Van der Bent, C	1
Cenni, B; Delafontaine, P; Picard, D; Scheidegger, KJ	1
Katzenellenbogen, BS; van der Burg, B; van der Saag, PT; Wissink, S	1
Flouriot, G; Métivier, R; Pakdel, F; Penot, G	1

Other Studies

58 other study(ies) available for ici 164384 and afimoxifene

Article	Year
Design, synthesis and evaluation of antiestrogen and histone deacetylase inhibitor molecular hybrids. Bioorganic & medicinal chemistry, 2015, Dec-15, Volume: 23, Issue:24 Topics: Antineoplastic Agents; Benzamides; Breast; Breast Neoplasms; Cell Line, Tumor; Estradiol; Estrogen Receptor Modulators; Female; Histone Deacetylase Inhibitors; Histone Deacetylases; Humans; Molecular Docking Simulation; Polyunsaturated Alkamides; Pyridines	2015
An estrogen receptor positive MCF-7 clone that is resistant to antiestrogens and estradiol. Molecular and cellular endocrinology, 1992, Volume: 90, Issue:1 Topics: Breast Neoplasms; Cell Division; Clone Cells; DNA, Neoplasm; Drug Resistance; ErbB Receptors; Estradiol; Estrogen Antagonists; Estrogens; Female; Gene Expression Regulation, Neoplastic; Humans; Neoplasm Proteins; Neoplasms, Hormone-Dependent; Polymerase Chain Reaction; Polyunsaturated Alkamides; Progesterone; Receptors, Estrogen; Recombinant Fusion Proteins; Signal Transduction; Tamoxifen; Transfection; Transforming Growth Factor alpha; Tumor Cells, Cultured	1992
Hormone-regulated v-rel estrogen receptor fusion protein: reversible induction of cell transformation and cellular gene expression. The EMBO journal, 1992, Volume: 11, Issue:12 Topics: Animals; Bone Marrow; Bone Marrow Cells; Cell Transformation, Neoplastic; Cells, Cultured; Chickens; Culture Techniques; DNA, Single-Stranded; Estradiol; Estrogen Antagonists; Estrogens; Gene Expression Regulation; Humans; Molecular Sequence Data; NF-kappa B; Oncogene Proteins v-rel; Polyunsaturated Alkamides; Protein-Tyrosine Kinases; Receptors, Estrogen; Recombinant Fusion Proteins; Retroviridae Proteins, Oncogenic; RNA, Messenger; Tamoxifen; Transcription, Genetic	1992
Antiestrogens prevent the stimulatory effects of L-triiodothyronine on cell proliferation. Endocrinology, 1992, Volume: 130, Issue:3 Topics: Breast Neoplasms; Cell Division; DNA, Neoplasm; Estradiol; Estrogen Antagonists; Female; Humans; Insulin-Like Growth Factor I; Pituitary Neoplasms; Polyunsaturated Alkamides; Receptors, Estrogen; Receptors, Thyroid Hormone; RNA, Messenger; Tamoxifen; Transcription, Genetic; Triiodothyronine; Tumor Cells, Cultured	1992
Differential effects of estrogen and antiestrogen on transforming growth factor gene expression in endometrial adenocarcinoma cells. Cancer research, 1992, Apr-01, Volume: 52, Issue:7 Topics: Adenocarcinoma; Analysis of Variance; Cell Division; Cell Line; Dose-Response Relationship, Drug; Endometrial Neoplasms; ErbB Receptors; Estradiol; Estrogen Antagonists; Female; Gene Expression; Humans; Kinetics; Polyunsaturated Alkamides; Pyrrolidines; RNA, Messenger; Tamoxifen; Thiophenes; Transforming Growth Factor alpha; Tumor Cells, Cultured	1992
Effect of ligand binding and DNA binding on the structure of the mouse oestrogen receptor. The Journal of steroid biochemistry and molecular biology, 1992, Volume: 41, Issue:3-8 Topics: Animals; Baculoviridae; Base Sequence; Binding Sites; Binding, Competitive; Cell Line; DNA-Binding Proteins; Endopeptidases; Estradiol; Estrogen Antagonists; Kinetics; Ligands; Mice; Molecular Sequence Data; Peptide Mapping; Polyunsaturated Alkamides; Receptors, Estrogen; Recombinant Proteins; Regulatory Sequences, Nucleic Acid; Tamoxifen; Transfection	1992
Proteolytic activity of the purified hormone-binding subunit in the estrogen receptor. Proceedings of the National Academy of Sciences of the United States of America, 1991, May-15, Volume: 88, Issue:10 Topics: Amino Acid Sequence; Animals; Aprotinin; Cattle; Chromogenic Compounds; Electrophoresis, Polyacrylamide Gel; Endopeptidases; Estradiol; Estrogen Antagonists; Female; Hydrolysis; Isoflurophate; Molecular Sequence Data; Polyunsaturated Alkamides; Receptors, Estrogen; Tamoxifen; Uterus	1991
The effect of anti-oestrogens on cell growth and progesterone receptor concentration in human endometrial cancer cells (Ishikawa). Journal of molecular endocrinology, 1991, Volume: 6, Issue:3 Topics: Cell Division; Estradiol; Estrogen Antagonists; Female; Humans; Polyunsaturated Alkamides; Receptors, Progesterone; Tamoxifen; Tumor Cells, Cultured; Uterine Neoplasms	1991
Studies on the activation of the oestrogen receptor bound to the anti-oestrogens 4-hydroxytamoxifen and ICI 164,384 by using three monoclonal antibodies. Journal of molecular endocrinology, 1991, Volume: 7, Issue:1 Topics: Animals; Antibodies, Monoclonal; Binding Sites; DNA; Estradiol; Estrogen Antagonists; Female; Guinea Pigs; Polyunsaturated Alkamides; Receptors, Estrogen; Structure-Activity Relationship; Tamoxifen; Temperature; Uterus	1991
Biological responses of ICI 164,384 and other anti-estrogens in vaginal and uterine cells of fetal guinea pig in culture. Acta endocrinologica, 1991, Volume: 125, Issue:4 Topics: Animals; Cell Division; Cell Separation; Cells, Cultured; DNA; Estradiol; Estrogen Antagonists; Female; Fetus; Guinea Pigs; Polyunsaturated Alkamides; Receptors, Progesterone; Tamoxifen; Uterus; Vagina	1991
Role of the two activating domains of the oestrogen receptor in the cell-type and promoter-context dependent agonistic activity of the anti-oestrogen 4-hydroxytamoxifen. The EMBO journal, 1990, Volume: 9, Issue:9 Topics: Animals; beta-Galactosidase; Chick Embryo; Chloramphenicol O-Acetyltransferase; Estradiol; Estrogen Antagonists; Fibroblasts; HeLa Cells; Humans; Polyunsaturated Alkamides; Promoter Regions, Genetic; Receptors, Estrogen; Saccharomyces cerevisiae; Tamoxifen; Transcription, Genetic; Transfection	1990
Construction of cell lines that express high levels of the human estrogen receptor and are killed by estrogens. Molecular endocrinology (Baltimore, Md.), 1990, Volume: 4, Issue:10 Topics: Animals; Cadmium; Cell Line; Cell Survival; Cricetinae; Drug Resistance; Enhancer Elements, Genetic; Estradiol; Estrogens; Female; Gene Amplification; Gene Expression; Metallothionein; Ovary; Polyunsaturated Alkamides; Promoter Regions, Genetic; Receptors, Estrogen; Simian virus 40; Tamoxifen; Transfection	1990
Characterization of a receptor-negative, hormone-nonresponsive clone derived from a T47D human breast cancer cell line kept under estrogen-free conditions. Cancer research, 1990, Nov-15, Volume: 50, Issue:22 Topics: Blotting, Northern; Breast Neoplasms; Cell Division; Clone Cells; Cytidine; DNA Fingerprinting; DNA, Neoplasm; ErbB Receptors; Estradiol; Gene Expression; Humans; In Vitro Techniques; Polyunsaturated Alkamides; Receptors, Estrogen; Receptors, Progesterone; RNA, Messenger; Tamoxifen; Transforming Growth Factor alpha; Transforming Growth Factor beta; Tumor Cells, Cultured	1990
ICI 164,384, a pure antagonist of estrogen-stimulated MCF-7 cell proliferation and invasiveness. Cancer research, 1989, Dec-15, Volume: 49, Issue:24 Pt 1 Topics: Basement Membrane; Binding, Competitive; Breast Neoplasms; Cell Cycle; Estradiol; Estrogen Antagonists; Humans; Neoplasm Invasiveness; Polyunsaturated Alkamides; Pyrrolidines; Receptors, Estrogen; Stimulation, Chemical; Tamoxifen; Thiophenes; Tumor Cells, Cultured	1989
Antiestrogenic properties of keoxifene, trans-4-hydroxytamoxifen, and ICI 164384, a new steroidal antiestrogen, in ZR-75-1 human breast cancer cells. Breast cancer research and treatment, 1989, Volume: 14, Issue:1 Topics: Binding, Competitive; Breast Neoplasms; Cell Division; Dexamethasone; Dihydrotestosterone; Dose-Response Relationship, Drug; Drug Interactions; Estradiol; Estrogen Antagonists; Humans; Piperidines; Polyunsaturated Alkamides; Raloxifene Hydrochloride; Receptors, Estrogen; Tamoxifen; Time Factors; Tumor Cells, Cultured	1989
Comparative studies on the effects of steroidal and nonsteroidal oestrogen antagonists on the proliferation of human breast cancer cells. Journal of steroid biochemistry, 1989, Volume: 34, Issue:1-6 Topics: Breast Neoplasms; Cell Division; Cell Line; Estradiol; Estrogen Antagonists; Female; Humans; Insulin; Kinetics; Polyunsaturated Alkamides; Structure-Activity Relationship; Tamoxifen; Tumor Cells, Cultured	1989
The hormone-binding domains of the estrogen and glucocorticoid receptors contain an inducible transcription activation function. Cell, 1988, Jul-15, Volume: 54, Issue:2 Topics: DNA; Estradiol; Estrenes; Estrogen Antagonists; Estrogens; Glucocorticoids; HeLa Cells; Hormones; Humans; Mifepristone; Polyunsaturated Alkamides; Receptors, Estrogen; Receptors, Glucocorticoid; Tamoxifen; Transcription Factors; Transcription, Genetic; Transfection	1988
Activation of the estrogen receptor through phosphorylation by mitogen-activated protein kinase. Science (New York, N.Y.), 1995, Dec-01, Volume: 270, Issue:5241 Topics: Amino Acid Sequence; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Enzyme Activation; Epidermal Growth Factor; Estradiol; Estrogen Antagonists; Humans; Mitogen-Activated Protein Kinase Kinases; Molecular Sequence Data; Mutation; Phosphorylation; Polyunsaturated Alkamides; Protein Kinases; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-raf; Proto-Oncogene Proteins p21(ras); Receptors, Estrogen; Recombinant Fusion Proteins; Serine; Somatomedins; Tamoxifen; Transcriptional Activation; Transfection	1995
Induction of estrogen independence of ZR-75-1 human breast cancer cells by epigenetic alterations. Molecular endocrinology (Baltimore, Md.), 1994, Volume: 8, Issue:11 Topics: Azacitidine; Breast Neoplasms; Down-Regulation; ErbB Receptors; Estradiol; Estrogen Antagonists; Estrogens; Female; Gene Expression Regulation, Neoplastic; Humans; Keratins; Neoplasm Proteins; Neoplasms, Hormone-Dependent; Polyunsaturated Alkamides; Proteins; Receptor, ErbB-2; Receptors, Estradiol; Receptors, Progesterone; Tamoxifen; Trefoil Factor-1; Tumor Cells, Cultured; Tumor Suppressor Proteins	1994
Conditional site-specific recombination in mammalian cells using a ligand-dependent chimeric Cre recombinase. Proceedings of the National Academy of Sciences of the United States of America, 1995, Jul-18, Volume: 92, Issue:15 Topics: DNA Nucleotidyltransferases; Enzyme Induction; Estradiol; Estrogen Antagonists; Gene Targeting; Genetic Vectors; Integrases; Mutagenesis, Site-Directed; Polyunsaturated Alkamides; Receptors, Estrogen; Receptors, Retinoic Acid; Recombinant Fusion Proteins; Recombination, Genetic; Repetitive Sequences, Nucleic Acid; Tamoxifen; Tumor Cells, Cultured; Viral Proteins	1995
The effect of free DNA on the interactions of the estrogen receptor bound to hormone, partial antagonist or pure antagonist with target DNA. European journal of biochemistry, 1995, Jul-01, Volume: 231, Issue:1 Topics: Animals; Bacterial Proteins; Base Sequence; DNA; Estradiol; Estrogen Antagonists; Estrogens; Female; Molecular Sequence Data; Polyunsaturated Alkamides; Receptors, Estrogen; Sheep; Streptavidin; Tamoxifen	1995
Estrogen and phorbol esters regulate amphiregulin expression by two separate mechanisms in human breast cancer cell lines. Endocrinology, 1995, Volume: 136, Issue:9 Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amphiregulin; Antineoplastic Agents; Blotting, Western; Breast Neoplasms; Bryostatins; Culture Media, Conditioned; Cycloheximide; Dose-Response Relationship, Drug; EGF Family of Proteins; Estradiol; Estrogen Antagonists; Estrogens; Gene Expression Regulation, Neoplastic; Glycoproteins; Growth Substances; Humans; Intercellular Signaling Peptides and Proteins; Isoquinolines; Lactones; Macrolides; Piperazines; Polyunsaturated Alkamides; Protein Kinase C; Receptors, Estrogen; RNA, Messenger; Tamoxifen; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured	1995
Specific mutations in the estrogen receptor change the properties of antiestrogens to full agonists. Proceedings of the National Academy of Sciences of the United States of America, 1995, May-09, Volume: 92, Issue:10 Topics: Amino Acid Sequence; Animals; Binding Sites; Cell Line; Chickens; Conserved Sequence; DNA-Binding Proteins; Estradiol; Estrogen Antagonists; Gene Expression; HeLa Cells; Humans; Mice; Molecular Sequence Data; Mutagenesis, Site-Directed; Oncorhynchus mykiss; Point Mutation; Polyunsaturated Alkamides; Protein Structure, Secondary; Rats; Receptors, Estrogen; Recombinant Proteins; Sequence Homology, Amino Acid; Tamoxifen; Transcription, Genetic; Transfection; Xenopus	1995
An estrogen-independent MCF-7 breast cancer cell line which contains a novel 80-kilodalton estrogen receptor-related protein. Cancer research, 1995, Jun-15, Volume: 55, Issue:12 Topics: Blotting, Western; Breast Neoplasms; Cell Division; Clone Cells; Electrophoresis, Polyacrylamide Gel; Estradiol; Estrogen Antagonists; Female; Humans; Kinetics; Luciferases; Molecular Weight; Polyunsaturated Alkamides; Protein Biosynthesis; Proteins; Receptors, Estrogen; Receptors, Progesterone; Recombinant Proteins; Tamoxifen; Time Factors; Transfection; Tumor Cells, Cultured; Up-Regulation	1995
Tamoxifen and related compounds protect against lipid peroxidation in isolated nuclei: relevance to the potential anticarcinogenic benefits of breast cancer prevention and therapy with tamoxifen? Free radical biology & medicine, 1994, Volume: 17, Issue:5 Topics: Animals; Anticarcinogenic Agents; Breast Neoplasms; Cell Nucleus; Estradiol; Estrogen Antagonists; Female; Humans; Lipid Peroxidation; Liver; Male; Nafoxidine; Polyunsaturated Alkamides; Rats; Rats, Wistar; Structure-Activity Relationship; Tamoxifen	1994
Molecular modelling of the human estrogen receptor and ligand interactions based on site-directed mutagenesis and amino acid sequence homology. The Journal of steroid biochemistry and molecular biology, 1995, Volume: 52, Issue:1 Topics: Computer Simulation; Estradiol; Estrogen Antagonists; Humans; Ligands; Models, Molecular; Mutagenesis, Site-Directed; Polyunsaturated Alkamides; Protein Conformation; Receptors, Estrogen; Tamoxifen	1995
Estrogen-inducible derivatives of hepatocyte nuclear factor-4, hepatocyte nuclear factor-3 and liver factor B1 are differently affected by pure and partial antiestrogens. European journal of biochemistry, 1994, Oct-01, Volume: 225, Issue:1 Topics: Animals; Base Sequence; Cell Line; Diethylstilbestrol; DNA Primers; DNA-Binding Proteins; Estradiol; Estrogen Antagonists; Estrogens; Gene Expression; Hepatocyte Nuclear Factor 1; Hepatocyte Nuclear Factor 1-alpha; Hepatocyte Nuclear Factor 1-beta; Hepatocyte Nuclear Factor 3-alpha; Hepatocyte Nuclear Factor 3-beta; Hepatocyte Nuclear Factor 3-gamma; Hepatocyte Nuclear Factor 4; Kinetics; Liver; Liver Neoplasms, Experimental; Molecular Sequence Data; Nuclear Proteins; Phosphoproteins; Polymerase Chain Reaction; Polyunsaturated Alkamides; Rats; Receptors, Estrogen; Substrate Specificity; Tamoxifen; Transcription Factors; Transcriptional Activation; Transfection; Tumor Cells, Cultured	1994
Interaction of proteins with transcriptionally active estrogen receptors. Proceedings of the National Academy of Sciences of the United States of America, 1994, Oct-11, Volume: 91, Issue:21 Topics: Animals; Base Sequence; Blotting, Western; Cell Line; Cell Nucleus; Cell-Free System; Chlorocebus aethiops; DNA Primers; DNA-Binding Proteins; Estradiol; Estrogen Antagonists; Fulvestrant; Glutathione Transferase; HeLa Cells; Humans; Kidney; Molecular Sequence Data; Nuclear Proteins; Polyunsaturated Alkamides; Receptors, Estrogen; Recombinant Fusion Proteins; Tamoxifen; Transcription, Genetic	1994
Hydroxytamoxifen induces a rapid and irreversible inactivation of an estrogenic response in an MCF-7-derived cell line. Cancer research, 1994, Nov-15, Volume: 54, Issue:22 Topics: Base Sequence; Breast Neoplasms; Cell Division; Cell Line; Enzyme Induction; Estradiol; Estrogen Antagonists; Gene Expression Regulation, Enzymologic; Humans; Luciferases; Molecular Sequence Data; Plasmids; Polyunsaturated Alkamides; Receptors, Estrogen; RNA, Messenger; Tamoxifen; Transfection; Tumor Cells, Cultured	1994
Antiestrogen regulation of cell cycle progression and cyclin D1 gene expression in MCF-7 human breast cancer cells. Breast cancer research and treatment, 1994, Volume: 31, Issue:1 Topics: Animals; Breast Neoplasms; Cell Cycle; Cell Division; Cell Line; Culture Media, Serum-Free; Cyclin D1; Cyclins; Dose-Response Relationship, Drug; Estradiol; Estrogen Antagonists; Female; Gene Expression Regulation, Neoplastic; Humans; Kinetics; Mice; Mice, Nude; Oncogene Proteins; Polyunsaturated Alkamides; Tamoxifen; Time Factors; Transplantation, Heterologous; Tumor Cells, Cultured	1994
Interaction of naturally occurring nonsteroidal estrogens with expressed recombinant human estrogen receptor. The Journal of steroid biochemistry and molecular biology, 1994, Volume: 49, Issue:2-3 Topics: Binding, Competitive; Estradiol; Estrogens, Non-Steroidal; Fungi; HeLa Cells; Humans; Plants; Polyunsaturated Alkamides; Receptors, Estrogen; Recombinant Proteins; Tamoxifen; Transcription, Genetic; Transfection	1994
Estrogen action via the cAMP signaling pathway: stimulation of adenylate cyclase and cAMP-regulated gene transcription. Proceedings of the National Academy of Sciences of the United States of America, 1994, Aug-30, Volume: 91, Issue:18 Topics: Adenylyl Cyclases; Animals; Base Sequence; Breast Neoplasms; Cells, Cultured; Cyclic AMP; Estradiol; Female; Gene Expression Regulation; Humans; In Vitro Techniques; Molecular Sequence Data; Oligodeoxyribonucleotides; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Signal Transduction; Tamoxifen; Transcription, Genetic; Tumor Cells, Cultured; Uterus	1994
The antiestrogen ICI 182780 disrupts estrogen receptor nucleocytoplasmic shuttling. Journal of cell science, 1993, Volume: 106 ( Pt 4) Topics: Amino Acid Sequence; Animals; Biological Transport; Cell Compartmentation; Cell Nucleus; Cells, Cultured; Chlorocebus aethiops; Cytoplasm; Estradiol; Estrogen Antagonists; Fulvestrant; Hybrid Cells; Mice; Molecular Sequence Data; Oligomycins; Polyunsaturated Alkamides; Receptors, Estrogen; Recombinant Proteins; Sequence Homology, Amino Acid; Tamoxifen; Transfection	1993
cDNA transfection followed by the isolation of a MCF-7 breast cell line resistant to tamoxifen in vitro and in vivo. British journal of cancer, 1993, Volume: 68, Issue:6 Topics: Animals; Breast Neoplasms; Cloning, Molecular; Culture Media, Conditioned; DNA, Complementary; DNA, Neoplasm; DNA, Recombinant; Drug Resistance; Estradiol; Estrogen Antagonists; Estrogens; Female; Growth Substances; Humans; Mice; Mice, Inbred BALB C; Mice, Nude; Neoplasm Transplantation; Polyunsaturated Alkamides; Receptors, Estrogen; Tamoxifen; Transfection; Tumor Cells, Cultured; Tumor Stem Cell Assay	1993
Anti-proliferative and anti-estrogenic effects of ICI 164,384 and ICI 182,780 in 4-OH-tamoxifen-resistant human breast-cancer cells. International journal of cancer, 1994, Jan-15, Volume: 56, Issue:2 Topics: Antineoplastic Agents; Breast Neoplasms; Cathepsin D; Cell Division; Drug Resistance; Estradiol; Estrogen Antagonists; Estrogens; Fulvestrant; Gene Expression Regulation, Neoplastic; Humans; Neoplasm Proteins; Neoplasms, Hormone-Dependent; Polyunsaturated Alkamides; Proteins; Receptors, Estrogen; Tamoxifen; Trefoil Factor-1; Tumor Cells, Cultured; Tumor Suppressor Proteins	1994
Estradiol increases and anti-estrogens antagonize the growth factor-induced activator protein-1 activity in MCF7 breast cancer cells without affecting c-fos and c-jun synthesis. The Journal of biological chemistry, 1993, Jul-05, Volume: 268, Issue:19 Topics: Breast Neoplasms; Chloramphenicol O-Acetyltransferase; Epidermal Growth Factor; Estradiol; Estrogen Antagonists; Female; Genes, fos; Genes, jun; Humans; Insulin-Like Growth Factor I; Kinetics; Polyunsaturated Alkamides; Proto-Oncogene Proteins c-fos; Proto-Oncogene Proteins c-jun; Receptors, Estrogen; Recombinant Fusion Proteins; RNA, Messenger; Tamoxifen; Thymidine Kinase; Time Factors; Transfection; Tumor Cells, Cultured	1993
Modulation of the ligand-independent activation of the human estrogen receptor by hormone and antihormone. Proceedings of the National Academy of Sciences of the United States of America, 1993, Jul-01, Volume: 90, Issue:13 Topics: Chloramphenicol O-Acetyltransferase; Dopamine; Estradiol; Estrogen Antagonists; Estrogens; HeLa Cells; Humans; Ligands; Polyunsaturated Alkamides; Receptors, Dopamine; Receptors, Estrogen; Tamoxifen	1993
Synthetic antiestrogens modulate induction of pS2 and cathepsin-D messenger ribonucleic acid by growth factors and adenosine 3',5'-monophosphate in MCF7 cells. Endocrinology, 1993, Volume: 133, Issue:2 Topics: 8-Bromo Cyclic Adenosine Monophosphate; Breast Neoplasms; Cathepsin D; Epidermal Growth Factor; Estradiol; Estrogen Antagonists; Growth Substances; Humans; Insulin-Like Growth Factor I; Neoplasm Proteins; Polyunsaturated Alkamides; Proteins; RNA, Messenger; Tamoxifen; Tetradecanoylphorbol Acetate; Transcription, Genetic; Trefoil Factor-1; Tumor Cells, Cultured; Tumor Suppressor Proteins	1993
Transformation of estrone, estradiol, and estrone sulfate in uterine and vaginal isolated cells of fetal guinea pig. Effect of various antiestrogens in the conversion of estrone sulfate to estradiol. Steroids, 1993, Volume: 58, Issue:5 Topics: Animals; Cells, Cultured; Culture Media; DNA; Estradiol; Estrogen Antagonists; Estrone; Female; Guinea Pigs; Polyunsaturated Alkamides; Pregnancy; Tamoxifen; Uterus; Vagina	1993
Inhibition of estrone sulfatase and 17 beta-hydroxysteroid dehydrogenase by antiestrogens. The Journal of steroid biochemistry and molecular biology, 1993, Volume: 45, Issue:5 Topics: 17-Hydroxysteroid Dehydrogenases; Animals; Binding, Competitive; Dehydroepiandrosterone; Dehydroepiandrosterone Sulfate; Estradiol; Female; Kinetics; Mammary Neoplasms, Experimental; Polyunsaturated Alkamides; Pregnenolone; Rats; Rats, Sprague-Dawley; Sulfatases; Tamoxifen	1993
Estrogen inhibits the growth of estrogen receptor-negative, but not estrogen receptor-positive, human mammary epithelial cells expressing a recombinant estrogen receptor. Cancer research, 1993, Oct-15, Volume: 53, Issue:20 Topics: Animals; Breast; Breast Neoplasms; Cell Cycle; Cell Division; Cell Line; Dose-Response Relationship, Drug; Epithelial Cells; Epithelium; Estradiol; Estrogen Antagonists; Female; Humans; Kinetics; Mice; Mice, Nude; Polyunsaturated Alkamides; Receptors, Estrogen; Recombinant Proteins; Tamoxifen; Transfection; Transplantation, Heterologous; Tumor Cells, Cultured	1993
Modulation of transcriptional activation by ligand-dependent phosphorylation of the human oestrogen receptor A/B region. The EMBO journal, 1993, Volume: 12, Issue:3 Topics: Amino Acid Sequence; Animals; Cell Line; Chloramphenicol O-Acetyltransferase; Estradiol; Estrogen Antagonists; Humans; Ligands; Molecular Sequence Data; Mutagenesis, Site-Directed; Phosphorylation; Point Mutation; Polyunsaturated Alkamides; Receptors, Estrogen; Sequence Deletion; Serine; Tamoxifen; Transcription, Genetic	1993
In vitro bioassays of non-steroidal phytoestrogens. The Journal of steroid biochemistry and molecular biology, 1993, Volume: 45, Issue:5 Topics: Adenocarcinoma; Alkaline Phosphatase; Biological Assay; Chromans; Coumestrol; Dinoprost; Endometrial Neoplasms; Endometrium; Equol; Estradiol; Female; Genistein; Humans; Isoflavones; Polyunsaturated Alkamides; Tamoxifen; Tumor Cells, Cultured	1993
Comparison between novel steroid-like and conventional nonsteroidal antioestrogens in inhibiting oestradiol- and IGF-I-induced proliferation of human breast cancer-derived cells. British journal of pharmacology, 1995, Volume: 116, Issue:5 Topics: Base Sequence; Blotting, Western; Breast Neoplasms; Cell Division; Culture Media, Conditioned; DNA; Estradiol; Estrogen Antagonists; Fulvestrant; Humans; Insulin-Like Growth Factor I; Molecular Sequence Data; Polyunsaturated Alkamides; RNA, Messenger; Steroids; Tamoxifen; Tumor Cells, Cultured	1995
Analysis of estrogen receptor function in vitro reveals three distinct classes of antiestrogens. Molecular endocrinology (Baltimore, Md.), 1995, Volume: 9, Issue:6 Topics: Animals; Cell Line; Chlorocebus aethiops; DNA; Estradiol; Estrogen Antagonists; Gene Expression Regulation; Kidney; Molecular Structure; Piperidines; Polyunsaturated Alkamides; Protein Binding; Protein Conformation; Raloxifene Hydrochloride; Receptors, Estrogen; Recombinant Proteins; Structure-Activity Relationship; Tamoxifen; Transfection	1995
Human estrogen receptor ligand activity inversion mutants: receptors that interpret antiestrogens as estrogens and estrogens as antiestrogens and discriminate among different antiestrogens. Molecular endocrinology (Baltimore, Md.), 1996, Volume: 10, Issue:3 Topics: 3T3 Cells; Animals; Breast Neoplasms; CHO Cells; Cricetinae; Cricetulus; Estradiol; Estrogen Antagonists; Estrogens; Female; Humans; Ligands; Mice; Neoplasms, Hormone-Dependent; Point Mutation; Polyunsaturated Alkamides; Promoter Regions, Genetic; Protein Binding; Receptors, Estrogen; Recombinant Fusion Proteins; Structure-Activity Relationship; Substrate Specificity; Tamoxifen; Transcription, Genetic; Tumor Cells, Cultured	1996
Stimulation of creatine kinase specific activity in human osteoblast and endometrial cells by estrogens and anti-estrogens and its modulation by calciotropic hormones. The Journal of endocrinology, 1996, Volume: 150, Issue:2 Topics: Calcitriol; Creatine Kinase; Endometrium; Estradiol; Estrogen Antagonists; Female; Humans; Osteoblasts; Piperidines; Plasmids; Polyunsaturated Alkamides; Raloxifene Hydrochloride; Recombinant Proteins; Stimulation, Chemical; Tamoxifen; Teriparatide; Tumor Cells, Cultured	1996
Transcriptional and post-transcriptional regulation of rainbow trout estrogen receptor and vitellogenin gene expression. Molecular and cellular endocrinology, 1996, Nov-29, Volume: 124, Issue:1-2 Topics: Animals; Cells, Cultured; Cycloheximide; Estradiol; Estrogen Antagonists; Gene Expression Regulation; Liver; Male; Oncorhynchus mykiss; Polyunsaturated Alkamides; Protein Synthesis Inhibitors; Receptors, Estrogen; RNA Processing, Post-Transcriptional; RNA, Messenger; Tamoxifen; Transcription, Genetic; Vitellogenins	1996
Estrogenic and progestagenic activities of physiologic and synthetic androgens, as measured by in vitro bioassays. Methods and findings in experimental and clinical pharmacology, 1997, Volume: 19, Issue:4 Topics: Adenocarcinoma; Alkaline Phosphatase; Androgen Antagonists; Androgens; Breast Neoplasms; Cyproterone Acetate; Endometrial Neoplasms; Estradiol; Estrogen Antagonists; Female; Flutamide; Gonanes; Humans; Mifepristone; Polyunsaturated Alkamides; Progestins; Tamoxifen; Testosterone; Testosterone Congeners; Tumor Cells, Cultured	1997
Probing the structure and function of the estrogen receptor ligand binding domain by analysis of mutants with altered transactivation characteristics. Molecular and cellular biology, 1997, Volume: 17, Issue:8 Topics: Amino Acid Sequence; Animals; Cloning, Molecular; COS Cells; Estradiol; Estrogen Antagonists; Estrone; HSP90 Heat-Shock Proteins; Hydroxyestrones; Ligands; Molecular Sequence Data; Mutation; Nuclear Proteins; Polyunsaturated Alkamides; Receptors, Estrogen; Saccharomyces cerevisiae; Sequence Alignment; Tamoxifen; Transcriptional Activation	1997
Both estradiol and tamoxifen decrease proliferation and invasiveness of cancer cells transfected with a mutated estrogen receptor. The Journal of steroid biochemistry and molecular biology, 1997, Volume: 61, Issue:1-2 Topics: Animals; Cell Division; Estradiol; Estrogen Antagonists; Mice; Mice, Inbred BALB C; Mice, Nude; Mutation; Neoplasm Invasiveness; Neoplasms, Experimental; Polyunsaturated Alkamides; Rats; Receptors, Estrogen; Tamoxifen; Transfection	1997
Different estrogen receptor structural domains are required for estrogen- and tamoxifen-dependent anti-proliferative activity in human mammary epithelial cells expressing an exogenous estrogen receptor. The Journal of steroid biochemistry and molecular biology, 1997, Volume: 62, Issue:5-6 Topics: Base Sequence; Binding Sites; Breast; Cell Division; Cell Line; DNA; DNA Primers; Epithelial Cells; Estradiol; Estrogen Antagonists; Female; Gene Expression; Humans; Mutation; Polymerase Chain Reaction; Polyunsaturated Alkamides; Receptors, Estrogen; Tamoxifen; Transfection	1997
Estrogen response elements can mediate agonist activity of anti-estrogens in human endometrial Ishikawa cells. The Journal of biological chemistry, 1998, Jul-03, Volume: 273, Issue:27 Topics: Animals; Base Sequence; Cell Line; COS Cells; Electrophoresis, Polyacrylamide Gel; Endometrium; Estradiol; Estrogen Antagonists; Estrogens; Female; Gene Expression Regulation; Humans; Polyunsaturated Alkamides; Promoter Regions, Genetic; Receptors, Progesterone; Tamoxifen; Transcription, Genetic; Tumor Cells, Cultured	1998
The anti-estrogen hydroxytamoxifen is a potent antagonist in a novel yeast system. Biological chemistry, 1999, Volume: 380, Issue:11 Topics: Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Estradiol; Estrogen Antagonists; Estrogen Receptor alpha; Humans; Indoles; Nafoxidine; Piperidines; Polyunsaturated Alkamides; Receptors, Estrogen; Saccharomyces cerevisiae; Sulfones; Tamoxifen; Two-Hybrid System Techniques	1999
Oestrogenic compounds modulate cytokine-induced nitric oxide production in mouse osteoblast-like cells. The Journal of pharmacy and pharmacology, 1999, Volume: 51, Issue:12 Topics: Animals; Cells, Cultured; Cytokines; Estradiol; Estrogen Antagonists; Estrogens; Interferon-gamma; Interleukin-1; Lipopolysaccharides; Mice; Nitric Oxide; Osteoblasts; Polyunsaturated Alkamides; Tamoxifen; Tumor Necrosis Factor-alpha	1999
Estradiol decreases IGF-1 and IGF-1 receptor expression in rat aortic smooth muscle cells. Mechanisms for its atheroprotective effects. The Journal of biological chemistry, 2000, Dec-08, Volume: 275, Issue:49 Topics: Animals; Aorta; Cells, Cultured; Estradiol; Estrogen Antagonists; Estrogen Receptor alpha; Estrogen Receptor beta; Gene Expression Regulation; HeLa Cells; Humans; Muscle, Smooth, Vascular; Polyunsaturated Alkamides; Promoter Regions, Genetic; Rats; Receptor, IGF Type 1; Receptor, IGF Type 2; Receptors, Estrogen; Recombinant Proteins; Tamoxifen; Transfection	2000
Synergistic activation of the serotonin-1A receptor by nuclear factor-kappa B and estrogen. Molecular endocrinology (Baltimore, Md.), 2001, Volume: 15, Issue:4 Topics: Animals; Cells, Cultured; Estradiol; Estrogen Antagonists; Estrogen Receptor alpha; Estrogen Receptor beta; Estrogens; Humans; NF-kappa B; Polyunsaturated Alkamides; Promoter Regions, Genetic; Protein Structure, Tertiary; Receptors, Estrogen; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Tamoxifen; Transcriptional Activation	2001
Synergism between ERalpha transactivation function 1 (AF-1) and AF-2 mediated by steroid receptor coactivator protein-1: requirement for the AF-1 alpha-helical core and for a direct interaction between the N- and C-terminal domains. Molecular endocrinology (Baltimore, Md.), 2001, Volume: 15, Issue:11 Topics: Amino Acid Sequence; Animals; Cells, Cultured; Coenzyme A; Cricetinae; DEAD-box RNA Helicases; Estradiol; Estrogen Antagonists; Estrogen Receptor alpha; Histone Acetyltransferases; Humans; Ligands; Molecular Sequence Data; Mutation; Nuclear Receptor Coactivator 1; Phosphorylation; Polyunsaturated Alkamides; Protein Conformation; Protein Kinases; Protein Structure, Tertiary; Rabbits; Receptors, Estrogen; RNA Helicases; Tamoxifen; Trans-Activators; Transcription Factors	2001