Page last updated: 2024-09-04

ici 147798 and isoproterenol

ici 147798 has been researched along with isoproterenol in 3 studies

Compound Research Comparison

Studies
(ici 147798)
Trials
(ici 147798)
Recent Studies (post-2010)
(ici 147798)
Studies
(isoproterenol)
Trials
(isoproterenol)
Recent Studies (post-2010) (isoproterenol)
70030,7808032,640

Protein Interaction Comparison

ProteinTaxonomyici 147798 (IC50)isoproterenol (IC50)
Beta-2 adrenergic receptorHomo sapiens (human)0.246
Beta-1 adrenergic receptorHomo sapiens (human)0.333
Beta-2 adrenergic receptorRattus norvegicus (Norway rat)0.2125
Polyunsaturated fatty acid lipoxygenase ALOX15Oryctolagus cuniculus (rabbit)1.77
Beta-1 adrenergic receptorRattus norvegicus (Norway rat)0.2125
Beta-3 adrenergic receptorRattus norvegicus (Norway rat)0.2125
Beta-2 adrenergic receptorCanis lupus familiaris (dog)0.6667

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Doggrell, SA; Surman, AJ2
Barnett, CW; Doggrell, SA; Petcu, EB1

Other Studies

3 other study(ies) available for ici 147798 and isoproterenol

ArticleYear
Characterization of the antagonism with metoprolol, ICI 147,798, pindolol, mepindolol and bopindolol on the responses of the rat left atria to isoprenaline.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 346, Issue:6

    Topics: Adrenergic beta-Antagonists; Animals; Heart; Isoproterenol; Male; Metoprolol; Myocardial Contraction; Pindolol; Pyrazines; Rats; Rats, Wistar; Receptors, Adrenergic, beta

1992
Loss of maximum attenuation and receptor reserve for isoprenaline at the beta 2-adrenoceptors of the portal veins of hypertensive rats.
    Journal of hypertension, 1995, Volume: 13, Issue:9

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Hypertension; Hypertrophy; Isoproterenol; Male; Nitroprusside; Portal Vein; Pyrazines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta; Vasodilator Agents; Verapamil

1995
Affinity constants and beta-adrenoceptor reserves for isoprenaline on cardiac tissue from normotensive and hypertensive rats.
    The Journal of pharmacy and pharmacology, 1998, Volume: 50, Issue:2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Female; Heart; Heart Atria; Heart Ventricles; Hypertension; Hypertrophy, Left Ventricular; Isoproterenol; Male; Myocardial Contraction; Myocardium; Papillary Muscles; Pyrazines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta

1998