ici 118551 has been researched along with prazosin in 44 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 11 (25.00) | 18.7374 |
1990's | 17 (38.64) | 18.2507 |
2000's | 10 (22.73) | 29.6817 |
2010's | 6 (13.64) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET | 1 |
Bartoccini, F; Carminati, P; Castorina, M; Di Cesare, MA; Di Serio, S; Gallo, G; Ghirardi, O; Giorgi, F; Giorgi, L; Minetti, P; Piersanti, G; Tarzia, G; Tinti, MO | 1 |
Altenbach, RJ; Brioni, JD; Carr, TL; Chandran, P; Cowart, MD; Esbenshade, TA; Honore, P; Hsieh, GC; Lewis, LG; Liu, H; Manelli, AM; Marsh, KC; Milicic, I; Miller, TR; Strakhova, MI; Vortherms, TA; Wakefield, BD; Wetter, JM; Witte, DG | 1 |
Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K | 1 |
Colau, D; Dolusić, E; Frédérick, R; Larrieu, P; Masereel, B; Moineaux, L; Pilotte, L; Pochet, L; Stroobant, V; Van den Eynde, B; Wouters, J | 1 |
Anzini, M; Brogi, S; Butini, S; Campiani, G; Cappelli, A; Caselli, G; Castriconi, F; Gemma, S; Giordani, A; Giorgi, G; Giuliani, G; Lanza, M; Letari, O; Makovec, F; Manini, M; Mennuni, L; Valenti, S | 1 |
Belyakov, S; Dambrova, M; Kazoka, H; Kuznecovs, J; Lebedev, A; Liepinsh, E; Mishnev, A; Orlova, N; Ponomaryov, Y; Vavers, E; Veinberg, G; Vikainis, S; Vilskersts, R; Vorona, M; Zvejniece, L | 1 |
Bednarski, M; Gunia-Krzyżak, A; Marona, H; Nitek, W; Pękala, E; Powroźnik, B; Słoczyńska, K; Walczak, M; Waszkielewicz, AM; Żesławska, E | 1 |
Filipek, B; Gunia-Krzyżak, A; Marona, H; Nitek, W; Pańczyk, K; Pękala, E; Rapacz, A; Słoczyńska, K; Waszkielewicz, AM; Żelaszczyk, D; Żesławska, E | 1 |
Goldberg, SR; Schindler, CW; Tella, SR | 1 |
Garcia-Barrado, MJ; Moratinos, J; Reverte, M | 1 |
Amstislavskaja, TG; Naumenko, EV; Osadchuk, AV | 1 |
Birkeland, S; Grong, K; Kvitting, P; Lekven, J; Westby, J | 1 |
Hyman, AL; Kadowitz, PJ; Lippton, HL | 1 |
Hyman, AL; Kadowitz, PJ | 2 |
Costall, B; Naylor, RJ; Tan, CC | 1 |
Bennett, T; Gardiner, SM | 2 |
Haynes, J; Pennefather, JN | 1 |
Forler, C; Fozard, JR; Middlemiss, DN; Tricklebank, MD | 1 |
Knudtzon, J | 1 |
De Jonge, A; Thoolen, MJ; Timmermans, PB; Van Zwieten, PA; Wilffert, B | 1 |
McWilliam, JR; Meldrum, BS | 1 |
Chojnacka-Wójcik, E; Filip, M; Przegaliński, E; Tatarczyńska, E | 1 |
Abe, K; Hidaka, S; Okina, A; Tashiro, M | 1 |
De Ridder, WJ; Higashino, M; Kinoshita, H; Meulemans, AL; Schuurkes, JA; Tokuhara, T | 1 |
Bültmann, R; Driessen, B; Gonçalves, J; Starke, K | 1 |
Burrello, N; Calogero, AE; D'Agata, R; Ossino, AM; Weber, RF | 1 |
Goepel, M; Michel, MC; Rübben, H; Wittmann, A | 1 |
Bearham, MC; Heal, DJ; Hutchins, LJ; Jackson, HC; Mazurkiewicz, SE; Needham, AM | 1 |
Carón, RW; Deis, RP; Salicioni, AM | 1 |
Butterworth, RF; Buu, PN; Michalak, A; Rose, C | 1 |
Dang, H; Gruber, DD; Scofield, MA; Shimozono, M; Wangemann, P | 1 |
Badino, P; Bergamasco, L; Borgarelli, M; Girardi, C; Odore, R; Re, G; Tarducci, A; Zanatta, R | 1 |
Colucci, WS; Communal, C; Sawyer, DB; Singh, K | 1 |
Cheng, H; Koch, WJ; Lakatta, EG; Lefkowitz, RJ; Spurgoen, H; Wang, DJ; Xiao, RP; Zhang, SJ; Zhou, YY; Zhu, W; Ziman, B | 1 |
Lee, TJ; Sarwinski, S; Zhang, W | 1 |
Harada, N; Isobe, H; Okajima, K; Uchiba, M | 1 |
Brahmadevara, N; MacDonald, A; Shaw, AM | 1 |
Chakir, K; Crow, MT; Jo, SH; Lakatta, EG; Leblais, V; Maltsev, V; Wang, W; Xiao, RP; Zheng, M | 1 |
Chartier, D; Ehrlich, JR; Hébert, TE; Nattel, S; Qi, X; Yeh, YH | 1 |
Chen, P; Liu, Z; Ma, K; Yang, H; Zhang, Y; Zhou, C | 1 |
Berger, SP; Bernardi, RE; Lattal, KM; Ryabinin, AE | 1 |
44 other study(ies) available for ici 118551 and prazosin
Article | Year |
---|---|
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium | 1985 |
2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A2A adenosine receptor antagonists. Design, synthesis, and pharmacological characterization.
Topics: Adenine; Adenosine A2 Receptor Antagonists; Animals; Cell Line; Cricetinae; Cricetulus; Drug Design; Humans; Imidazoles; Male; Models, Molecular; Motor Activity; Purines; Radioligand Assay; Rats; Rats, Inbred F344; Structure-Activity Relationship; Triazoles | 2005 |
cis-4-(Piperazin-1-yl)-5,6,7a,8,9,10,11,11a-octahydrobenzofuro[2,3-h]quinazolin-2-amine (A-987306), a new histamine H4R antagonist that blocks pain responses against carrageenan-induced hyperalgesia.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzofurans; Carrageenan; Disease Models, Animal; Drug Design; Drug Evaluation, Preclinical; Humans; Hyperalgesia; Ligands; Mice; Molecular Structure; Pain; Peritonitis; Quinazolines; Rats; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Stereoisomerism; Structure-Activity Relationship | 2008 |
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship | 2010 |
Tryptophan 2,3-dioxygenase (TDO) inhibitors. 3-(2-(pyridyl)ethenyl)indoles as potential anticancer immunomodulators.
Topics: Animals; Antineoplastic Agents; Biological Availability; Cell Line; Drug Design; Enzyme Inhibitors; Humans; Immunologic Factors; Indoles; Kinetics; Mice; Neoplasms; Structure-Activity Relationship; Tryptophan Oxygenase | 2011 |
Synthesis and structure-activity relationship studies in serotonin 5-HT(1A) receptor agonists based on fused pyrrolidone scaffolds.
Topics: Animals; Area Under Curve; Humans; Intestinal Absorption; Ligands; Male; Metabolic Clearance Rate; Models, Chemical; Models, Molecular; Molecular Structure; Protein Binding; Protein Structure, Tertiary; Pyrrolidinones; Radioligand Assay; Receptor, Serotonin, 5-HT1A; Receptors, Serotonin, 5-HT3; Serotonin 5-HT1 Receptor Agonists; Structure-Activity Relationship | 2013 |
Synthesis and biological evaluation of 2-(5-methyl-4-phenyl-2-oxopyrrolidin-1-yl)-acetamide stereoisomers as novel positive allosteric modulators of sigma-1 receptor.
Topics: Acetamides; Allosteric Regulation; Animals; Rats; Rats, Wistar; Receptors, sigma; Sigma-1 Receptor; Stereoisomerism; Structure-Activity Relationship | 2013 |
Design, physico-chemical properties and biological evaluation of some new N-[(phenoxy)alkyl]- and N-{2-[2-(phenoxy)ethoxy]ethyl}aminoalkanols as anticonvulsant agents.
Topics: Amino Alcohols; Animals; Anticonvulsants; Chemistry, Physical; Dose-Response Relationship, Drug; Drug Design; Epilepsy; Male; Mice; Microsomes, Liver; Molecular Structure; Pilocarpine | 2016 |
Structure-anticonvulsant activity studies in the group of (E)-N-cinnamoyl aminoalkanols derivatives monosubstituted in phenyl ring with 4-Cl, 4-CH
Topics: Amino Alcohols; Animals; Anticonvulsants; Crystallography, X-Ray; Disease Models, Animal; Dose-Response Relationship, Drug; Electroshock; Mice; Models, Molecular; Molecular Structure; Rats; Seizures; Structure-Activity Relationship | 2017 |
Adrenoceptor mechanisms in the cardiovascular effects of cocaine in conscious squirrel monkeys.
Topics: Adrenergic beta-Antagonists; Animals; Atenolol; Blood Pressure; Cocaine; Heart Rate; Labetalol; Male; Phentolamine; Prazosin; Propanolamines; Propranolol; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Saimiri; Yohimbine | 1992 |
Changes in plasma glucose and lactate evoked by alpha and beta 2-adrenoceptor stimulation in conscious fasted rabbits.
Topics: Albuterol; Analysis of Variance; Animals; Blood Glucose; Clonidine; Dioxanes; Epinephrine; Fasting; Idazoxan; Lactates; Male; Picolinic Acids; Prazosin; Propanolamines; Rabbits; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Spectrophotometry | 1991 |
The role of the adrenoceptors in the activation of the hypothalamic-pituitary-testicular complex of mice induced by the presence of a female.
Topics: Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Female; Hypothalamo-Hypophyseal System; Male; Metoprolol; Mice; Mice, Inbred CBA; Phentolamine; Prazosin; Propanolamines; Propranolol; Radioimmunoassay; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Sexual Behavior, Animal; Testis; Testosterone; Yohimbine | 1991 |
Regional perfusion in hearts with acute coronary artery occlusion and subsequent beta 2- and alpha 1-adrenergic blockade.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Cats; Coronary Circulation; Coronary Disease; Doxazosin; Drug Interactions; Hemodynamics; Male; Myocardium; Oxygen Consumption; Prazosin; Propanolamines; Renal Circulation; Renin | 1990 |
Analysis of pulmonary vascular responses in cats to sympathetic nerve stimulation under elevated tone conditions. Evidence that neuronally released norepinephrine acts on alpha 1-, alpha 2-, and beta 2-adrenoceptors.
Topics: Adrenergic beta-Antagonists; Animals; Blood Pressure; Cats; Electric Stimulation; Female; Lung; Male; Norepinephrine; Prazosin; Propanolamines; Propranolol; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Sympathetic Nervous System; Yohimbine | 1990 |
Analysis of responses to sympathetic nerve stimulation in the feline pulmonary vascular bed.
Topics: Adrenergic beta-Antagonists; Animals; Cats; Electric Stimulation; Lung; Norepinephrine; Prazosin; Propanolamines; Propranolol; Pulmonary Circulation; Sympathetic Nervous System; Tyramine; Vascular Resistance; Yohimbine | 1989 |
Mechanism of action of apomorphine on rat gastric secretion.
Topics: Adrenergic beta-Antagonists; Animals; Antipsychotic Agents; Apomorphine; Atenolol; Drug Interactions; Gastric Acid; Gastric Mucosa; Male; Prazosin; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Time Factors; Yohimbine | 1985 |
Enhancement of alpha- and beta-adrenoceptor responses by elevations in vascular tone in pulmonary circulation.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-Antagonists; Animals; Brimonidine Tartrate; Cats; Female; Male; Muscle Tonus; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Prazosin; Propanolamines; Pulmonary Circulation; Quinoxalines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Yohimbine | 1986 |
Involvement of beta 2-adrenoceptor-mediated mechanisms in the cardiovascular responses to alpha 1- and alpha 2-adrenoceptor antagonism in conscious, unrestrained, Long Evans and Brattleboro rats.
Topics: Adrenal Medulla; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Blood Pressure; Captopril; Dioxanes; Heart Rate; Hemodynamics; Idazoxan; Male; Phentolamine; Prazosin; Propanolamines; Rats; Rats, Brattleboro; Receptors, Adrenergic, beta; Restraint, Physical | 1988 |
Regional hemodynamic responses to adrenoceptor antagonism in conscious rats.
Topics: Adrenergic alpha-Antagonists; Animals; Aorta, Abdominal; Blood Pressure; Captopril; Deamino Arginine Vasopressin; Dioxanes; Idazoxan; Male; Mesenteric Arteries; Prazosin; Propanolamines; Propranolol; Rats; Rats, Brattleboro; Reference Values; Species Specificity; Ultrasonics; Vascular Resistance | 1988 |
Alpha 1-and alpha 2-adrenoceptors of the circular myometrium from the dioestrous guinea-pig.
Topics: Adrenergic beta-Antagonists; Animals; Diestrus; Estrus; Female; Fluoxetine; Guinea Pigs; Myometrium; Norepinephrine; Phenylephrine; Prazosin; Propanolamines; Receptors, Adrenergic, alpha; Uterine Contraction | 1988 |
Subtypes of the 5-HT receptor mediating the behavioural responses to 5-methoxy-N,N-dimethyltryptamine in the rat.
Topics: Animals; Apomorphine; Behavior, Animal; Betaxolol; Haloperidol; Ketanserin; Male; Pindolol; Piperidines; Prazosin; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reserpine; Spiperone | 1985 |
Adrenergic effects on plasma levels of glucagon, insulin, glucose and free fatty acids in rabbits--influences of selective blocking drugs.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Blood Glucose; Epinephrine; Fatty Acids, Nonesterified; Female; Glucagon; Insulin; Isoproterenol; Metoprolol; Prazosin; Propanolamines; Rabbits; Yohimbine | 1984 |
Heterogeneity of the interaction between alpha 1- and alpha 2-adrenoceptor agonists with their respective receptors in the vascular system of the pithed rat.
Topics: Adrenergic alpha-Agonists; Animals; Azepines; Blood Pressure; Cocaine; Dopamine; Electric Stimulation; Emetics; Ethanolamines; Hemodynamics; Male; Naphthols; Prazosin; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tetrahydronaphthalenes; Yohimbine | 1984 |
Noradrenergic regulation of growth hormone secretion in the baboon.
Topics: Albuterol; Animals; Brimonidine Tartrate; Dose-Response Relationship, Drug; Female; Growth Hormone; Male; Papio; Practolol; Prazosin; Propanolamines; Propranolol; Quinoxalines; Receptors, Adrenergic | 1983 |
The role of 5-hydroxytryptamine1A (5-HT1A) receptors in the anticonflict activity of beta-adrenoceptor antagonists.
Topics: Adrenergic beta-Antagonists; Animals; Anxiety; Betaxolol; Conflict, Psychological; Disease Models, Animal; Drug Interactions; Male; p-Chloroamphetamine; Pindolol; Piperazines; Prazosin; Propanolamines; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists | 1994 |
The effects of tyramine on salivary flow rate and protein secretion by rat submandibular glands.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Isoelectric Focusing; Male; Metoprolol; Phenoxybenzamine; Prazosin; Propanolamines; Propranolol; Protease Inhibitors; Rats; Rats, Sprague-Dawley; Saliva; Salivary Proteins and Peptides; Salivation; Secretory Rate; Serine Endopeptidases; Stimulation, Chemical; Submandibular Gland; Tyramine; Yohimbine | 1993 |
Effect of adrenoceptor agonists on striated muscle strips of the canine oesophagus.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dogs; Esophagus; Female; In Vitro Techniques; Isometric Contraction; Isoproterenol; Male; Muscle, Smooth; Norepinephrine; Phenylephrine; Prazosin; Propanolamines; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Ritodrine | 1993 |
Opposite modulation of noradrenaline and ATP release in guinea-pig vas deferens through prejunctional beta-adrenoceptors: evidence for the beta 2 subtype.
Topics: Adenosine Triphosphate; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Imidazoles; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Neuromuscular Junction; Norepinephrine; Prazosin; Propanolamines; Receptors, Adrenergic, beta-2; Suramin; Terbutaline; Vas Deferens | 1996 |
Interaction between prolactin and catecholamines on hypothalamic GnRH release in vitro.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Atenolol; Corticotropin-Releasing Hormone; Depression, Chemical; Dose-Response Relationship, Drug; Gonadotropin-Releasing Hormone; Hypothalamus; Male; Organ Culture Techniques; Phentolamine; Prazosin; Prolactin; Propanolamines; Propranolol; Rats; Rats, Sprague-Dawley; Yohimbine | 1996 |
Comparison of adrenoceptor subtype expression in porcine and human bladder and prostate.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Female; Humans; Imidazoles; Isoquinolines; Male; Oxymetazoline; Piperazines; Prazosin; Propanolamines; Prostate; Radioligand Assay; Receptors, Adrenergic; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta; Swine; Urinary Bladder; Yohimbine | 1997 |
Investigation of the mechanisms underlying the hypophagic effects of the 5-HT and noradrenaline reuptake inhibitor, sibutramine, in the rat.
Topics: Adrenergic Uptake Inhibitors; Animals; Cyclobutanes; Eating; Idazoxan; Male; Metoprolol; Prazosin; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors | 1997 |
Participation of both adrenergic and opioidergic systems in the negative feedback of adrenal progesterone on LH secretion.
Topics: Adrenal Glands; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Estradiol; Feedback; Female; Hormone Antagonists; Idazoxan; Luteinizing Hormone; Metoprolol; Mifepristone; Naloxone; Ovariectomy; Prazosin; Progesterone; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic; Receptors, Opioid | 1997 |
Evidence for altered central noradrenergic function in experimental acute liver failure in the rat.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Autoradiography; Cerebral Cortex; Chromatography, High Pressure Liquid; Coma; Dopamine; Frontal Lobe; Hippocampus; Hypothalamus; Idazoxan; Liver Failure, Acute; Microdialysis; Norepinephrine; Pindolol; Prazosin; Propanolamines; Putamen; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic; Serotonin; Thalamus | 1998 |
Alpha1A-adrenergic receptors mediate vasoconstriction of the isolated spiral modiolar artery in vitro.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Arteries; Cochlea; Dose-Response Relationship, Drug; Enzyme Inhibitors; Gerbillinae; Nitric Oxide Synthase; Nitroarginine; Norepinephrine; Piperazines; Polymerase Chain Reaction; Prazosin; Propanolamines; Receptors, Adrenergic, alpha-1; RNA; Vasoconstriction; Yohimbine | 1998 |
Canine dilated cardiomyopathy: lymphocyte and cardiac alpha(1)- and beta-adrenoceptor concentrations in normal and affected great danes.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Cardiomyopathy, Dilated; Catecholamines; Dog Diseases; Dogs; Electrocardiography; Female; Heart Failure; Lymphocyte Count; Lymphocytes; Male; Myocardium; Prazosin; Propanolamines; Receptors, Adrenergic; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2 | 1999 |
Opposing effects of beta(1)- and beta(2)-adrenergic receptors on cardiac myocyte apoptosis : role of a pertussis toxin-sensitive G protein.
Topics: Adenylate Cyclase Toxin; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Apoptosis; Carbachol; Cardiotonic Agents; Cyclic AMP; GTP-Binding Protein alpha Subunits, Gi-Go; Heart; Imidazoles; Isoproterenol; Male; Muscarinic Agonists; Myocardium; Pertussis Toxin; Prazosin; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Second Messenger Systems; Virulence Factors, Bordetella | 1999 |
Inhibition of spontaneous beta 2-adrenergic activation rescues beta 1-adrenergic contractile response in cardiomyocytes overexpressing beta 2-adrenoceptor.
Topics: Adrenergic beta-Agonists; Animals; beta-Adrenergic Receptor Kinases; Carbachol; Cells, Cultured; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; G-Protein-Coupled Receptor Kinase 2; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Heart; Heart Ventricles; Humans; Mice; Myocardial Contraction; Myocardium; Norepinephrine; Pertussis Toxin; Prazosin; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Recombinant Proteins; Transfection; Virulence Factors, Bordetella | 2000 |
Presynaptic beta(2)-adrenoceptors mediate nicotine-induced NOergic neurogenic dilation in porcine basilar arteries.
Topics: Adrenergic beta-Antagonists; Animals; Basilar Artery; Butoxamine; Endothelium, Vascular; Female; In Vitro Techniques; Male; Models, Cardiovascular; Muscle, Smooth, Vascular; Nicotine; Nitric Oxide; Prazosin; Propanolamines; Receptors, Adrenergic, beta-2; Swine; Vasodilation; Yohimbine | 2000 |
Activation of capsaicin-sensitive sensory neurons by carvedilol, a nonselective beta-blocker, in spontaneous hypertensive rats.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Bisoprolol; Blood Pressure; Calcitonin Gene-Related Peptide; Capsaicin; Carbazoles; Carvedilol; Cells, Cultured; Drug Interactions; Female; Humans; Hypertension; Kidney; Male; Mice; Neurons, Afferent; Prazosin; Propanolamines; Rats; Rats, Inbred SHR; Rats, Sprague-Dawley; Regional Blood Flow | 2004 |
ALpha1-adrenoceptor antagonist properties of CGP 12177A and other beta-adrenoceptor ligands: evidence against beta(3)- or atypical beta-adrenoceptors in rat aorta.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-1 Receptor Antagonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Aorta, Thoracic; Binding Sites; Bupranolol; Cell Membrane; Cerebral Cortex; Dose-Response Relationship, Drug; Ethanolamines; Imidazoles; Male; Muscle, Smooth, Vascular; Phenylephrine; Pindolol; Prazosin; Propanolamines; Propranolol; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-3; Tritium; United Kingdom; Vasoconstriction | 2004 |
Phosphatidylinositol 3-kinase offsets cAMP-mediated positive inotropic effect via inhibiting Ca2+ influx in cardiomyocytes.
Topics: Androstadienes; Animals; Calcium; Calcium Channels, L-Type; Calcium Signaling; Cells, Cultured; Chromones; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein beta Subunits; GTP-Binding Protein gamma Subunits; Insulin-Like Growth Factor I; Ion Transport; Isoproterenol; Morpholines; Myocardial Contraction; Myocytes, Cardiac; Norepinephrine; Patch-Clamp Techniques; Peptide Fragments; Pertussis Toxin; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Prazosin; Propanolamines; Protein Processing, Post-Translational; Rats; Receptors, Adrenergic, beta-1; Recombinant Proteins; Second Messenger Systems; Signal Transduction; Wortmannin | 2004 |
Adrenergic control of a constitutively active acetylcholine-regulated potassium current in canine atrial cardiomyocytes.
Topics: Acetylcholine; Action Potentials; Adrenergic Agents; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Bee Venoms; Clonidine; Cyclic AMP-Dependent Protein Kinases; Dihydropyridines; Dogs; Dose-Response Relationship, Drug; Estrenes; Heart Atria; Imidazoles; Indoles; Isoproterenol; Isoquinolines; Maleimides; Myocytes, Cardiac; Patch-Clamp Techniques; Phenylephrine; Phorbol 12,13-Dibutyrate; Piperazines; Potassium Channels; Prazosin; Propanolamines; Propranolol; Protein Kinase C; Pyrrolidinones; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-1; Sulfonamides; Type C Phospholipases | 2007 |
Mouse embryonic stem cell-derived cardiomyocytes express functional adrenoceptors.
Topics: Animals; Cell Differentiation; Cell Line; Embryonic Stem Cells; Extracellular Signal-Regulated MAP Kinases; Gene Expression; Imidazoles; Isoproterenol; Mice; Myocytes, Cardiac; Phenylephrine; Prazosin; Propanolamines; Propranolol; Receptor, Muscarinic M2; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta; Tyrosine 3-Monooxygenase | 2008 |
Post-retrieval disruption of a cocaine conditioned place preference by systemic and intrabasolateral amygdala beta2- and alpha1-adrenergic antagonists.
Topics: Adrenergic alpha-Antagonists; Adrenergic Antagonists; Adrenergic beta-Antagonists; Amygdala; Analysis of Variance; Animals; Cocaine; Conditioning, Operant; Dopamine Uptake Inhibitors; Drug Administration Routes; Mental Recall; Microinjections; Oncogene Proteins v-fos; Prazosin; Propanolamines; Rats; Rats, Sprague-Dawley | 2009 |