ici 118551 and carvedilol

ici 118551 has been researched along with carvedilol in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (9.09)18.2507
2000's6 (54.55)29.6817
2010's4 (36.36)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baker, JG1
Abuin, L; Cotecchia, S; Lattion, A; Nenniger-Tosato, M1
Bond, RA; Callaerts-Vegh, Z; Evans, KL; Liu, X1
Bond, RA; Callaerts-Vegh, Z; Cuba, DL; Davies, PJ; Evans, KL; Giles, H; Gurji, HA; Shipley, GL1
Harada, N; Isobe, H; Okajima, K; Uchiba, M1
Christ, T; Kaumann, A; Molenaar, P; Ravens, U1
Abe, H; Anson, BD; Delisle, BP; January, CT; Kawakami, K; Kikuchi, K; Nagatomo, T; Nakashima, Y; Takemasa, H1
Coelho, M; Correia, G; Medeiros, R; Moz, M; Ribeiro, L; Teixeira, A1
Maniak, PJ; O'Grady, SM; Peitzman, ER; Zaidman, NA1
Benovic, JL; Carr, R; Carter, RL; Cheung, JY; Du, Y; Koch, WJ; Schilling, J; Song, J; Tilley, DG; Traynham, CJ; Yoo, SM1
Du, XJ; Hu, HY; Kiriazis, H; Lu, Q; Nguyen, MN; Puthalakath, H; Sadoshima, J; Su, Y; Wang, LN; Zhao, WB; Ziemann, M1

Other Studies

11 other study(ies) available for ici 118551 and carvedilol

ArticleYear
The selectivity of beta-adrenoceptor antagonists at the human beta1, beta2 and beta3 adrenoceptors.
    British journal of pharmacology, 2005, Volume: 144, Issue:3

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Algorithms; Animals; Cell Line; CHO Cells; Cricetinae; Dioxoles; Humans; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3

2005
Constitutively active mutants of the beta1-adrenergic receptor.
    FEBS letters, 1999, Sep-03, Volume: 457, Issue:3

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Amino Acid Substitution; Betaxolol; Carbazoles; Carvedilol; Cell Line; Cyclic AMP; Epinephrine; Humans; Imidazoles; Isoproterenol; Labetalol; Point Mutation; Practolol; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Recombinant Proteins; Timolol

1999
Chronic infusion of beta-adrenoceptor antagonist and inverse agonists decreases elevated protein kinase A activity in transgenic mice with cardiac-specific overexpression of human beta 2-adrenoceptor.
    Journal of cardiovascular pharmacology, 2002, Volume: 40, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Carbazoles; Carvedilol; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Heart Atria; Heart Ventricles; Humans; Infusion Pumps, Implantable; Mice; Mice, Transgenic; Myocardium; Propanolamines; Receptors, Adrenergic, beta-2

2002
Effects of different beta adrenoceptor ligands in mice with permanent occlusion of the left anterior descending coronary artery.
    British journal of pharmacology, 2003, Volume: 138, Issue:8

    Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Carbazoles; Carvedilol; Coronary Disease; Coronary Vessels; Ligands; Male; Mice; Mice, Inbred C57BL; Propanolamines; Receptors, Adrenergic, beta

2003
Activation of capsaicin-sensitive sensory neurons by carvedilol, a nonselective beta-blocker, in spontaneous hypertensive rats.
    The Journal of pharmacology and experimental therapeutics, 2004, Volume: 309, Issue:2

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Bisoprolol; Blood Pressure; Calcitonin Gene-Related Peptide; Capsaicin; Carbazoles; Carvedilol; Cells, Cultured; Drug Interactions; Female; Humans; Hypertension; Kidney; Male; Mice; Neurons, Afferent; Prazosin; Propanolamines; Rats; Rats, Inbred SHR; Rats, Sprague-Dawley; Regional Blood Flow

2004
Carvedilol blocks beta2- more than beta1-adrenoceptors in human heart.
    Cardiovascular research, 2006, Volume: 69, Issue:1

    Topics: Adrenergic beta-Antagonists; Calcium Channels, L-Type; Carbazoles; Carvedilol; Dose-Response Relationship, Drug; Epinephrine; Heart Atria; Heart Failure; Heart Ventricles; Humans; Imidazoles; In Vitro Techniques; Metoprolol; Myocardial Contraction; Myocardium; Norepinephrine; Patch-Clamp Techniques; Propanolamines; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2

2006
Comparison of HERG channel blocking effects of various beta-blockers-- implication for clinical strategy.
    British journal of pharmacology, 2006, Volume: 147, Issue:6

    Topics: Adrenergic beta-Antagonists; Binding Sites; Carbazoles; Cardiovascular Diseases; Carvedilol; Cell Line; Dose-Response Relationship, Drug; Ether-A-Go-Go Potassium Channels; Humans; Long QT Syndrome; Membrane Potentials; Metoprolol; Mutation; Potassium Channel Blockers; Propanolamines; Propranolol; Protein Binding; Transfection

2006
Antiproliferative effects of β-blockers on human colorectal cancer cells.
    Oncology reports, 2015, Volume: 33, Issue:5

    Topics: Adenocarcinoma; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Atenolol; Carbazoles; Carvedilol; Cell Line, Tumor; Cell Proliferation; Colorectal Neoplasms; Epinephrine; HT29 Cells; Humans; Isoproterenol; Norepinephrine; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Signal Transduction

2015
Carvedilol binding to β2-adrenergic receptors inhibits CFTR-dependent anion secretion in airway epithelial cells.
    American journal of physiology. Lung cellular and molecular physiology, 2016, Jan-01, Volume: 310, Issue:1

    Topics: Adrenergic beta-Antagonists; Anions; Arrestins; beta-Arrestins; Carbazoles; Carvedilol; Cells, Cultured; Cyclic AMP; Cystic Fibrosis Transmembrane Conductance Regulator; Epithelial Cells; Humans; Propanolamines; Receptors, Adrenergic, beta-2; Signal Transduction

2016
β-arrestin-biased signaling through the β2-adrenergic receptor promotes cardiomyocyte contraction.
    Proceedings of the National Academy of Sciences of the United States of America, 2016, 07-12, Volume: 113, Issue:28

    Topics: Adrenergic beta-Antagonists; Animals; beta-Arrestins; Carbazoles; Carvedilol; Cell Line, Tumor; Drug Evaluation, Preclinical; Heart Failure; HEK293 Cells; Humans; Lipopeptides; Mice; Myocardial Contraction; Myocytes, Cardiac; Primary Cell Culture; Propanolamines; Protein Conformation

2016
Stimulation of β-adrenoceptors up-regulates cardiac expression of galectin-3 and BIM through the Hippo signalling pathway.
    British journal of pharmacology, 2019, Volume: 176, Issue:14

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bcl-2-Like Protein 11; Cardiovascular Diseases; Carvedilol; Cell Line; Dose-Response Relationship, Drug; Galectin 3; Isoproterenol; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Mice, Transgenic; Propanolamines; Propranolol; Rats; Receptors, Adrenergic, beta-3; Signal Transduction; Up-Regulation

2019