Page last updated: 2024-08-26

hydroxyflutamide and dihydrotestosterone

hydroxyflutamide has been researched along with dihydrotestosterone in 98 studies

Research

Studies (98)

Timeframe	Studies, this research(%)	All Research%
pre-1990	10 (10.20)	18.7374
1990's	48 (48.98)	18.2507
2000's	27 (27.55)	29.6817
2010's	12 (12.24)	24.3611
2020's	1 (1.02)	2.80

Authors

Authors	Studies
Ackerman, JH; Bell, MR; Christiansen, RG; D'Ambra, TE; Herrmann, JL; Kullnig, RK; Mallamo, JP; Opalka, CJ; Snyder, BW; Winneker, RC	1
Breton, R; Labrie, F; Martel, C; Poirier, D; Roy, J	1
Bydal, P; Labrie, F; Luu-The, V; Poirier, D	1
Bellavance, E; Luu-The, V; Poirier, D	1
Badalassi, F; Bertozzi, F; Bradley, SR; Fejzic, A; Gardell, LR; Lewinsky, R; Lund, BW; Olsson, R; Pawlas, J; Piu, F; Schlienger, N; Tabatabaei, A; Thygesen, MB	1
Arias, DA; Barbieri, LR; Berrodin, TJ; Bigelis, R; Chang, LP; Luckman, SW; McDonald, LA; Roll, DM; Singh, MP; Yudt, MR	1
Fournier, MA; Maltais, R; Poirier, D	1
Wang, S; Xiang, W	1
Connors, K; Geller, J; Hoffman, RM; Sionit, LR	1
Huber, GK; Kirschenbaum, A; Levine, AC; Ren, M	1
Chalmers, D; Kirk, D; Leake, RE; Lloyd, SN	1
Beato, M; Bock, K; Filmer, A; Hackenberg, R; Hawighorst, T; Schulz, KD; Slater, EP	1
Bernasconi, D; Cassulo, S; Fazzuoli, L; Giordano, G; Marugo, M; Miglietta, L; Ravera, F	1
de Launoit, Y; Dufour, M; Labrie, F; Simard, J; Veilleux, R	1
Korpacheva, T; Reznikov, A	1
Arbusow, V; Bojar, H; Fittler, F; Klobeck, HG; Schulz, P; Wolf, D	1
Olea, N; Sakabe, K; Sonnenschein, C; Soto, AM	1
Dauvois, S; Haagensen, DE; Labrie, F; Lévesque, C; Mérand, Y; Simard, J	1
Begin, DJ; Labrie, F; Luthy, IA	1
Baylink, DJ; Farley, JR; Kasperk, CH; Linkhart, TA; Turner, RT; Wergedal, JE	1
Hammond, JM; Spicer, LJ	1
Dias, JA; Swift, TA	1
Duleba, AJ; Ho Yuen, B; Kim, KS; Moon, YS	1
Baker, D; Labrie, F; Poulin, R	1
Mauvais-Jarvis, P; Mowszowicz, I; Portois, MC; Santen, RJ	1
Hillier, SG; Purohit, A; Reichert, LE	1
Azzolin, GC; Saiduddin, S	1
King, RJ; Yates, J	1
Boccuzzi, G; Brignardello, E; Di Monaco, M; Gatto, V; Leonardi, L	1
Baird, A; Connors, KM; Geller, J; Hoffman, RM; Kohls, M; Sionit, LR	1
Calabrò, M; Carruba, G; Castagnetta, LA; Farruggio, R; Miceli, MD; Oliveri, G; Pfeffer, U; Sorci, CM	1
Bravo, AI; Calandra, RS; Capurro, MI; Donaldson, M; Luthy, IA; Mordoh, J; Morvillo, V; Quintans, C	1
Carruba, G; Castagnetta, LA; Comito, L; D'Amico, D; Farruggio, R; Miceli, D; Montesanti, A; Polito, L	1
Charreau, EH; Dran, G; Lanari, C; Luthy, IA; Molinolo, AA; Montecchia, F; Pasqualini, CD	1
Kelce, WR; Sar, M; Wilson, EM; Wong, C	1
Gorczynska, E; Handelsman, DJ	1
Bentel, JM; Birrell, SN; Hickey, TE; Horsfall, DJ; Ricciardelli, C; Tilley, WD; Weger, MA	1
Biordi, L; Bologna, M; Festuccia, C; Muzi, P; Vicentini, C	1
Kelley, DB; Robertson, JC; Watson, JT	1
Boccuzzi, G; Brignardello, E; Di Monaco, M; Gallo, M; Gatto, V; Leonardi, L; Pizzini, A	1
Dell'Acqua, G; Fattorossi, A; Iacopino, F; Marchetti, P; Pavone-Macaluso, M; Sica, G; van der Kwast, TH	1
Govindan, MV; Koutsilieris, M; Pagé, N; Warriar, N	2
Fanger, GR; Henderson, LP; Maue, RA; Tabb, JS; Wilson, EM	1
Couture, P; Labrie, F; Simard, J; Thériault, C	1
Chang, C; Yeh, S	1
Beck, S; Hackenberg, R; Hannig, K; Schmidt-Rhode, P; Scholz, A; Schulz, KD	1
Batchelor, KW; Grant, ES; Habib, FK	1
Jimenez, J; Luizzi, MF; Sonnenschein, C; Soto, AM; Szelei, J	1
Chen, Y; Elbrecht, A; Rutledge, SJ; Schmidt, A; Toney, JH	1
Galosy, S; Gudmundsson, GO; Newcomer, B; Sridaran, R; Talamantes, F; Thordarson, G	1
Barañao, JL; Bley, MA; Saragüeta, PE	1
Boschelli, F; Caplan, AJ; Fang, Y; Fliss, AE	1
Belsham, DD; Brown, TJ; Duc, VL; Evangelou, A; Roy, D	1
Danielpour, D; Lucia, MS; Roberts, AB; Sporn, MB; Stewart, LV	1
Gaido, KW; Maness, SC; McDonnell, DP	1
Hicok, KC; Hofbauer, LC; Khosla, S	1
Balk, SP; Bubley, GJ; Fenton, MA; Fertig, AM; Kolvenbag, G; Shuster, TD; Taplin, ME	1
Cavazzini, P; degli Uberti, EC; del Senno, L; Fallo, F; Rossi, R; Valentini, A; Zatelli, MC	1
Fournier, A; Labrie, C; Lapointe, J; Richard, V	1
Judd, J; Kremer, M; Oursler, MJ; Pascoe, D; Pederson, L; Riggs, BL; Spelsberg, TC	1
Budman, DR; Kreis, W; Liu, XM; Wang, LG	1
Hackenberg, R; Loos, S; Schulz, KD	1
Hofbauer, LC; Khosla, S; Ten, RM	1
Fan, Z; Mendelsohn, J; Ye, D	1
Celermajer, DS; Death, AK; Handelsman, DJ; Jessup, W; McCrohon, JA; Nakhla, S; Stanley, KK	1
Brown, TJ; Evangelou, A; Jindal, SK; Letarte, M	1
Jones, GR; Lyng, FM; Rommerts, FF	1
Damien, E; Lanyon, LE; Price, JS	1
Bentel, JM; Buchanan, G; Greenberg, NM; Han, G; Harris, JM; Horsfall, DJ; Marshall, VR; Matusik, RJ; Moore, N; Nahm, HS; Tilley, WD; Yang, M	1
Appa Rao, KB; Gui, Y; Lessey, BA; Lovely, LP	1
Chen, Q; Chihara, K; Kaji, H; Sugimoto, T	1
Goto, K; Morinaga, H; Nawata, H; Nomura, M; Okabe, T; Takayanagi, R; Tomura, A; Yanase, T	1
Bobseine, KL; Britt, BH; Cardon, MC; Gray, LE; Hartig, PC; Lambright, CR; Wilson, VS	1
Furutani, T; Hashimoto, T; Kato, S; Koutoku, H; Kudoh, M; Shikama, H; Shimizu, Y; Tanimoto, K; Watanabe, T	1
Bongers, G; Buttini, M; LeFevour, A; Mucke, L; Raber, J	1
Bonmassar, E; Faraoni, I; Missale, C; Rizzetti, MC; Sigala, S; Spano, P; Tognazzi, N	1
Aozasa, K; Chang, C; Chang, HC; Harada, Y; Kang, HY; Miyamoto, H; Nishimura, K; Nonomura, N; Okuyama, A; Shin, M; Ting, HJ; Tokizane, T; Yeh, S	1
Armstrong, DT; Gilchrist, RB; Hickey, TE; Marrocco, DL; Norman, RJ	1
Lou, YR; Nazarova, N; Talonpoika, R; Tuohimaa, P	1
Amato, F; Armstrong, DT; Gilchrist, RB; Hickey, TE; Marrocco, DL; Norman, RJ; Ritter, LJ	1
Hajszan, T; Johansen, JA; Jordan, CL; Leranth, C; MacLusky, NJ	1
Chang, CY; Elbi, C; Hager, GL; Hendarwanto, A; Klokk, TI; Kurys, P; Nagaich, AK; Saatcioglu, F; Slagsvold, T	1
De Rosier, T; Eliason, HC; Ervin, KM; Gowda, K; Kupcho, KR; Marks, BD; Ozers, MS; Qadir, N; Riddle, SM; Shekhani, MS	1
Fuse, H; Hiyama, T; Ito, T; Kato, S; Kimura, K; Korenaga, S; Sakari, M	1
Akahoshi, T; Ariga, H; Hayashi, H; Itoh, Y; Miyazawa, K; Okamoto, T; Onozaki, K; Otsuka, T; Takii, T; Waguri-Nagaya, Y; Xu, J	1
Hara, S; Isaacs, JT; Ishioka, J; Kageyama, Y; Nishikawa, K; Tomura, A	1
Dubbink, HJ; Hersmus, R; Jenster, G; Lusher, SJ; Molier, M; Trapman, J; van de Wijngaart, DJ	1
Chippari, S; Crabtree, JS; Harris, HA; Kenney, T; Kilbourne, EJ; McNally, C; Nagpal, S; Peano, BJ; Thompson, CC; Wang, W; Winneker, RC	1
Walker, WH	1
Anonuevo, A; Bingham, B; Gray, M; Innala, L; Myung, C; Viau, V	1
Andrieu, T; Baker, ME; Bertolini, R; Frey, BM; Frey, FJ; Nichols, SE; Setoud, R	1
Chang, C; Hsu, JW; Izumi, K; Miyamoto, H; Zheng, Y	1
Imasaka, T; Li, X; Miyake, R; Uchimura, T	1
Makita, M; Miyano, T	1
Hara, N; Ishizaki, F; Nishiyama, T; Takeda, K; Tasaki, M; Tomita, Y	1
El-Shishtawy, KA; Ide, H; Kashiwagi, E; Kawahara, T; Li, Y; Miyamoto, H; Reis, LO; Zheng, Y	1
Azhagiya Singam, ER; Durkin, KA; La Merrill, MA; Smith, MT; Tachachartvanich, P	1

Reviews

1 review(s) available for hydroxyflutamide and dihydrotestosterone

Article	Year
Therapeutic Strategies to Target the Androgen Receptor. Journal of medicinal chemistry, 2022, 07-14, Volume: 65, Issue:13 Topics: Androgen Antagonists; Androgen Receptor Antagonists; Humans; Male; Prostatic Neoplasms, Castration-Resistant; Receptors, Androgen	2022

Other Studies

97 other study(ies) available for hydroxyflutamide and dihydrotestosterone

Article	Year
Antiandrogenic steroidal sulfonylpyrazoles. Journal of medicinal chemistry, 1990, Volume: 33, Issue:8 Topics: Androgen Antagonists; Animals; Male; Molecular Structure; Orchiectomy; Organ Size; Pregnanes; Prostate; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, Androgen; Structure-Activity Relationship; Testosterone; X-Ray Diffraction	1990
Chemical synthesis and biological activities of 16alpha-derivatives of 5alpha-androstane-3alpha,17beta-diol as antiandrogens. Bioorganic & medicinal chemistry, 2007, Apr-15, Volume: 15, Issue:8 Topics: Androgen Antagonists; Androstane-3,17-diol; Antineoplastic Agents, Hormonal; Cell Line, Tumor; Cell Proliferation; Humans; Indicators and Reagents; Magnetic Resonance Spectroscopy; Models, Molecular; Receptors, Androgen; Spectrophotometry, Infrared; Structure-Activity Relationship	2007
Steroidal lactones as inhibitors of 17beta-hydroxysteroid dehydrogenase type 5: chemical synthesis, enzyme inhibitory activity, and assessment of estrogenic and androgenic activities. European journal of medicinal chemistry, 2009, Volume: 44, Issue:2 Topics: 17-Hydroxysteroid Dehydrogenases; Cell Line; Cell Proliferation; Enzyme Inhibitors; Humans; Lactones; Male; Prostatic Diseases; Receptors, Androgen; Receptors, Estrogen; Receptors, Glucocorticoid; Receptors, Progesterone; Steroids; Structure-Activity Relationship	2009
Potent and selective steroidal inhibitors of 17beta-hydroxysteroid dehydrogenase type 7, an enzyme that catalyzes the reduction of the key hormones estrone and dihydrotestosterone. Journal of medicinal chemistry, 2009, Dec-10, Volume: 52, Issue:23 Topics: 17-Hydroxysteroid Dehydrogenases; Androstane-3,17-diol; Androstanes; Biocatalysis; Cell Line; Dihydrotestosterone; Enzyme Inhibitors; Estradiol; Estrone; Humans; Inhibitory Concentration 50; Oxidation-Reduction; Substrate Specificity	2009
Synthesis, structure-activity relationships, and characterization of novel nonsteroidal and selective androgen receptor modulators. Journal of medicinal chemistry, 2009, Nov-26, Volume: 52, Issue:22 Topics: Administration, Oral; Androgen Receptor Antagonists; Androgens; Animals; Azabicyclo Compounds; Dogs; Drug Design; Humans; Ligands; Male; Mice; Microsomes, Liver; Mutation; NIH 3T3 Cells; Orchiectomy; Prostatic Neoplasms; Rats; Receptors, Androgen; Structure-Activity Relationship; Substrate Specificity; Testosterone Propionate	2009
The lecanindoles, nonsteroidal progestins from the terrestrial fungus Verticillium lecanii 6144. Journal of natural products, 2009, Volume: 72, Issue:11 Topics: Animals; Chlorocebus aethiops; Female; Humans; Hypocreales; Indoles; Luciferases; Molecular Structure; Nuclear Magnetic Resonance, Biomolecular; Progestins; Receptors, Progesterone; Sesquiterpenes	2009
Development of 3-substituted-androsterone derivatives as potent inhibitors of 17β-hydroxysteroid dehydrogenase type 3. Bioorganic & medicinal chemistry, 2011, Aug-01, Volume: 19, Issue:15 Topics: 17-Hydroxysteroid Dehydrogenases; Androsterone; Enzyme Inhibitors; HEK293 Cells; Humans; Inhibitory Concentration 50; Male; Prostatic Neoplasms; Structure-Activity Relationship	2011
Measurement of androgen sensitivity in the human prostate in in vitro three-dimensional histoculture. The Prostate, 1992, Volume: 21, Issue:4 Topics: Androgen Antagonists; Androgen Receptor Antagonists; Dihydrotestosterone; Flutamide; Histological Techniques; Humans; Male; Prostate; Prostatic Hyperplasia; Receptors, Androgen; Thymidine	1992
The effect of androgen, estrogen, and growth factors on the proliferation of cultured fibroblasts derived from human fetal and adult prostates. Endocrinology, 1992, Volume: 130, Issue:4 Topics: Cell Division; Cells, Cultured; Dihydrotestosterone; Epidermal Growth Factor; Estradiol; Female; Fetus; Fibroblasts; Flutamide; Genes, fos; Growth Substances; Humans; Immunohistochemistry; Male; Pregnancy; Prostate; Prostatic Hyperplasia; RNA, Messenger	1992
Local hyperthermia for prostatic disease: in vitro studies on human prostatic cancer cell lines. British journal of urology, 1992, Volume: 70, Issue:5 Topics: Cell Division; Cell Survival; Dihydrotestosterone; DNA, Neoplasm; Flutamide; Humans; Hyperthermia, Induced; Male; Prostatic Neoplasms; Tumor Cells, Cultured	1992
Regulation of androgen receptor mRNA and protein level by steroid hormones in human mammary cancer cells. The Journal of steroid biochemistry and molecular biology, 1992, Volume: 43, Issue:7 Topics: Blotting, Northern; Breast Neoplasms; Cyproterone; Dihydrotestosterone; Estradiol; Flutamide; Gene Expression Regulation, Neoplastic; Hormones; Humans; Immunohistochemistry; Progesterone Congeners; Radioligand Assay; Receptors, Androgen; RNA, Messenger; Steroids; Tumor Cells, Cultured	1992
Effects of dihydrotestosterone and hydroxyflutamide on androgen receptors in cultured human breast cancer cells (EVSA-T). The Journal of steroid biochemistry and molecular biology, 1992, Volume: 42, Issue:5 Topics: Androgen Antagonists; Breast Neoplasms; Cell Division; Dihydrotestosterone; Flutamide; Humans; Receptors, Androgen; Tumor Cells, Cultured	1992
Characteristics of the biphasic action of androgens and of the potent antiproliferative effects of the new pure antiestrogen EM-139 on cell cycle kinetic parameters in LNCaP human prostatic cancer cells. Cancer research, 1991, Oct-01, Volume: 51, Issue:19 Topics: Androgens; Androstane-3,17-diol; Binding, Competitive; Cell Cycle; Dihydrotestosterone; Dose-Response Relationship, Drug; Drug Antagonism; Estradiol; Estrogen Antagonists; Estrone; Flow Cytometry; Flutamide; Humans; In Vitro Techniques; Male; Metribolone; Piperidines; Prostatic Neoplasms; Raloxifene Hydrochloride; Tamoxifen; Testosterone; Time Factors; Tumor Cells, Cultured	1991
Nonsteroid antiandrogen inhibiting effect on testosterone metabolism in rat prostate and liver. Endocrinologia experimentalis, 1990, Volume: 24, Issue:4 Topics: 3-Oxo-5-alpha-Steroid 4-Dehydrogenase; Animals; Dihydrotestosterone; Flutamide; Liver; Male; Orchiectomy; Prostate; Rats; Rats, Inbred Strains; Testosterone	1990
The synthetic androgen mibolerone induces transient suppression of the transformed phenotype in an androgen responsive human prostatic carcinoma cell line. Andrologia, 1990, Volume: 22 Suppl 1 Topics: Androgen Antagonists; Androgens; Cell Division; Cell Transformation, Neoplastic; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; Flutamide; Humans; Male; Nandrolone; Prostatic Neoplasms; Receptors, Androgen; RNA, Messenger; Tumor Cells, Cultured	1990
The proliferative effect of "anti-androgens" on the androgen-sensitive human prostate tumor cell line LNCaP. Endocrinology, 1990, Volume: 126, Issue:3 Topics: Androgens; Antibodies; Cell Division; Dihydrotestosterone; Estradiol; Flutamide; Humans; Male; Nandrolone; Prostatic Neoplasms; Receptors, Androgen; Testosterone Congeners; Tumor Cells, Cultured	1990
Regulation of progesterone-binding breast cyst protein GCDFP-24 secretion by estrogens and androgens in human breast cancer cells: a new marker of steroid action in breast cancer. Endocrinology, 1990, Volume: 126, Issue:6 Topics: Androgens; Apolipoproteins; Apolipoproteins D; Binding, Competitive; Biomarkers, Tumor; Breast Neoplasms; Carrier Proteins; Cell Division; Dihydrotestosterone; Estradiol; Estrogen Antagonists; Estrogens; Female; Flutamide; Glycoproteins; Humans; Kinetics; Membrane Transport Proteins; Neoplasm Proteins; Progesterone; Tumor Cells, Cultured	1990
Androgenic activity of synthetic progestins and spironolactone in androgen-sensitive mouse mammary carcinoma (Shionogi) cells in culture. Journal of steroid biochemistry, 1988, Volume: 31, Issue:5 Topics: Androgens; Animals; Cell Division; Chlormadinone Acetate; Dihydrotestosterone; Flutamide; Male; Mammary Neoplasms, Experimental; Medroxyprogesterone; Medroxyprogesterone Acetate; Megestrol; Mice; Progestins; Spironolactone; Tumor Cells, Cultured	1988
Androgens directly stimulate proliferation of bone cells in vitro. Endocrinology, 1989, Volume: 124, Issue:3 Topics: Alkaline Phosphatase; Androgens; Animals; Binding, Competitive; Cell Count; Cell Differentiation; Cell Division; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; DNA; Dose-Response Relationship, Drug; Fluoxymesterone; Flutamide; Humans; Methenolone; Mice; Osteoblasts; Testosterone; Tumor Cells, Cultured	1989
Comparative effects of androgens and catecholestrogens on progesterone production by porcine granulosa cells. Molecular and cellular endocrinology, 1988, Volume: 56, Issue:3 Topics: 2-Methoxyestradiol; Androstenedione; Animals; Cell Count; Cells, Cultured; Dihydrotestosterone; Dose-Response Relationship, Drug; Estradiol; Estrogens, Catechol; Female; Flutamide; Follicle Stimulating Hormone; Granulosa Cells; Ovum; Progesterone; Swine; Testosterone	1988
Testosterone suppression of ornithine decarboxylase activity in rat Sertoli cells. Endocrinology, 1988, Volume: 123, Issue:2 Topics: Animals; Bucladesine; Cells, Cultured; Cyclic AMP; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; Enzyme Induction; Estradiol; Flutamide; Follicle Stimulating Hormone; Male; Ornithine Decarboxylase; Rats; Rats, Inbred Strains; Sertoli Cells; Testosterone	1988
Inhibition of 20 alpha-hydroxysteroid dehydrogenase activity by follicle-stimulating hormone and androgens in cultured rat granulosa cells: a search for the mechanism of action. Biology of reproduction, 1985, Volume: 33, Issue:2 Topics: 20-alpha-Hydroxysteroid Dehydrogenase; 20-Hydroxysteroid Dehydrogenases; Androgens; Androstenedione; Animals; Bucladesine; Cells, Cultured; Cholera Toxin; Dihydrotestosterone; Estradiol; Estrone; Female; Flutamide; Follicle Stimulating Hormone; Granulosa Cells; Progesterone; Rats; Rats, Inbred Strains; Testosterone	1985
Androgens inhibit basal and estrogen-induced cell proliferation in the ZR-75-1 human breast cancer cell line. Breast cancer research and treatment, 1988, Volume: 12, Issue:2 Topics: Androgen Antagonists; Androstenedione; Breast Neoplasms; Cell Division; Cell Line; Dihydrotestosterone; Dose-Response Relationship, Drug; Estradiol; Estrogen Antagonists; Flutamide; Humans; Piperidines; Raloxifene Hydrochloride; Receptors, Androgen; Receptors, Estrogen; Testosterone	1988
Androgen dependence of the Dunning R3327G cell line in monolayer culture. The Prostate, 1987, Volume: 11, Issue:4 Topics: Androgen Antagonists; Androgens; Animals; Cell Division; Cell Line; Dihydrotestosterone; Flutamide; Male; Neoplasms, Hormone-Dependent; Orchiectomy; Prostatic Neoplasms; Rats; Tumor Cells, Cultured	1987
Control of granulosa cell lactate production by follicle-stimulating hormone and androgen. Endocrinology, 1985, Volume: 116, Issue:3 Topics: Androgens; Animals; Dihydrotestosterone; Dose-Response Relationship, Drug; Drug Synergism; Female; Flutamide; Follicle Stimulating Hormone; Granulosa Cells; Lactates; Osmolar Concentration; Progesterone; Rats; Rats, Inbred Strains; Testosterone; Time Factors	1985
Effect of androgens on the ovarian morphology of the hypophysectomized rat. Proceedings of the Society for Experimental Biology and Medicine. Society for Experimental Biology and Medicine (New York, N.Y.), 1983, Volume: 172, Issue:1 Topics: Animals; Diethylstilbestrol; Dihydrotestosterone; Female; Flutamide; Hypophysectomy; Ovarian Follicle; Rats; Testosterone	1983
Antiandrogen effects on androgen-responsive mammary tumour cells in culture. Journal of steroid biochemistry, 1981, Volume: 14, Issue:9 Topics: Anilides; Animals; Cell Division; Cells, Cultured; Cyproterone; Dihydrotestosterone; Dose-Response Relationship, Drug; Flutamide; Mammary Neoplasms, Experimental; Mice; Receptors, Androgen; Testosterone	1981
Inhibitory effect of hydroxyflutamide plus tamoxifen on oestradiol-induced growth of MCF-7 breast cancer cells. Journal of cancer research and clinical oncology, 1995, Volume: 121, Issue:12 Topics: Antineoplastic Combined Chemotherapy Protocols; Breast Neoplasms; Cell Division; Dihydrotestosterone; Drug Synergism; Estradiol; Estrogen Antagonists; Flutamide; Humans; Neoplasms, Hormone-Dependent; Tamoxifen; Tumor Cells, Cultured	1995
In vivo and in vitro effects of androgen on fibroblast growth factor-2 concentrations in the human prostate. The Prostate, 1994, Volume: 25, Issue:4 Topics: Androgen Antagonists; Cell Division; Culture Techniques; Dihydrotestosterone; Fibroblast Growth Factor 2; Flutamide; Humans; Male; Megestrol; Megestrol Acetate; Orchiectomy; Prostate; Prostatic Hyperplasia; Radioimmunoassay	1994
Growth of LNCaP human prostate cancer cells is stimulated by estradiol via its own receptor. Endocrinology, 1995, Volume: 136, Issue:5 Topics: Androgen Antagonists; Base Sequence; Breast Neoplasms; Cell Division; Cell Line; Cell Nucleus; Cytosol; Dihydrotestosterone; DNA Primers; DNA, Neoplasm; Estradiol; Female; Flutamide; Gene Expression; Humans; Kinetics; Male; Molecular Sequence Data; Polymerase Chain Reaction; Prostate-Specific Antigen; Prostatic Neoplasms; Radioligand Assay; Receptors, Estradiol; Transcription, Genetic; Tumor Cells, Cultured	1995
Atypical androgen receptor in the human melanoma cell line IIB-MEL-J. Pigment cell research, 1995, Volume: 8, Issue:3 Topics: Androgen Antagonists; Animals; Antibodies, Monoclonal; Antineoplastic Agents, Hormonal; Binding, Competitive; Cell Division; Dihydrotestosterone; Estradiol; Flutamide; Humans; Hydrocortisone; Immunohistochemistry; Male; Melanoma; Metribolone; Mice; Mice, Nude; Progesterone; Receptors, Androgen; Testosterone; Tumor Cells, Cultured	1995
Sex steroids up-regulate E-cadherin expression in hormone-responsive LNCaP human prostate cancer cells. Biochemical and biophysical research communications, 1995, Jul-17, Volume: 212, Issue:2 Topics: Androgen Antagonists; Cadherins; Dihydrotestosterone; Estradiol; Estrogen Antagonists; Flutamide; Fulvestrant; Gonadal Steroid Hormones; Humans; Immunoblotting; Immunohistochemistry; Male; Prostatic Neoplasms	1995
Effect of medroxyprogesterone acetate (MPA) and serum factors on cell proliferation in primary cultures of an MPA-induced mammary adenocarcinoma. Breast cancer research and treatment, 1995, Volume: 35, Issue:2 Topics: Adenocarcinoma; Androgen Antagonists; Animals; Blood Physiological Phenomena; Cell Division; Dexamethasone; Dihydrotestosterone; Estradiol; Female; Flutamide; Mammary Neoplasms, Experimental; Medroxyprogesterone Acetate; Mice; Mice, Inbred BALB C; Mifepristone; Ovariectomy; Progesterone; Tumor Cells, Cultured	1995
Androgen receptor antagonist versus agonist activities of the fungicide vinclozolin relative to hydroxyflutamide. The Journal of biological chemistry, 1995, Aug-25, Volume: 270, Issue:34 Topics: Androgen Receptor Antagonists; Androgens; Animals; Binding, Competitive; Cell Line; Dihydrotestosterone; DNA; Flutamide; Fungicides, Industrial; Humans; Kinetics; Male; Oxazoles; Receptors, Androgen; Recombinant Proteins; Reproduction; Transcription, Genetic; Transfection; Tumor Cells, Cultured	1995
Androgens rapidly increase the cytosolic calcium concentration in Sertoli cells. Endocrinology, 1995, Volume: 136, Issue:5 Topics: Androgen Antagonists; Androgens; Animals; Calcium; Cells, Cultured; Cyclic AMP; Cytosol; Dihydrotestosterone; Drug Synergism; Finasteride; Flutamide; Follicle Stimulating Hormone; Kinetics; Male; Progesterone; Rats; Rats, Wistar; Sertoli Cells; Spermatogenesis; Testosterone; Time Factors	1995
Androgens induce divergent proliferative responses in human breast cancer cell lines. The Journal of steroid biochemistry and molecular biology, 1995, Volume: 52, Issue:5 Topics: Androgen Receptor Antagonists; Androgens; Breast Neoplasms; Cell Division; Dihydrotestosterone; Flutamide; Humans; Imidazoles; Imidazolidines; Nandrolone; Oligonucleotides, Antisense; Receptors, Androgen; Tumor Cells, Cultured	1995
Finasteride dose-dependently reduces the proliferation rate of the LnCap human prostatic cancer cell line in vitro. Urology, 1995, Volume: 45, Issue:2 Topics: Androgen Antagonists; Cell Division; Cyproterone Acetate; Dihydrotestosterone; Dose-Response Relationship, Drug; Finasteride; Flutamide; Humans; Linear Models; Male; Prostatic Neoplasms; Testosterone; Tumor Cells, Cultured	1995
Androgen directs sexual differentiation of laryngeal innervation in developing Xenopus laevis. Journal of neurobiology, 1994, Volume: 25, Issue:12 Topics: Animals; Axons; Dihydrotestosterone; Female; Flutamide; Laryngeal Muscles; Laryngeal Nerves; Male; Microscopy, Electron; Muscle Development; Sex Differentiation; Testosterone; Xenopus laevis	1994
5-En-androstene-3 beta,17 beta-diol inhibits the growth of MCF-7 breast cancer cells when oestrogen receptors are blocked by oestradiol. British journal of cancer, 1994, Volume: 70, Issue:6 Topics: Androstenediol; Breast Neoplasms; Cell Division; Diethylstilbestrol; Dihydrotestosterone; Estradiol; Flutamide; Humans; Receptors, Estrogen; Tamoxifen; Tumor Cells, Cultured	1994
Androgen receptors and hormone sensitivity of a human prostatic cancer cell line (PC-3) are modulated by natural beta-interferon. Urological research, 1994, Volume: 22, Issue:1 Topics: Androgen Antagonists; Androgens; Cell Cycle; Cell Division; Dihydrotestosterone; Drug Resistance; Flutamide; Humans; Immunohistochemistry; Interferon-beta; Male; Prostatic Neoplasms; Receptors, Androgen; Tumor Cells, Cultured	1994
Antiandrogens inhibit human androgen receptor-dependent gene transcription activation in the human prostate cancer cells LNCaP. The Prostate, 1994, Volume: 24, Issue:4 Topics: Amino Acid Sequence; Androgen Antagonists; Binding, Competitive; Blotting, Western; Chloramphenicol O-Acetyltransferase; Cyproterone Acetate; Dihydrotestosterone; Dose-Response Relationship, Drug; Flutamide; Gene Expression Regulation, Viral; Humans; Imidazoles; Imidazolidines; Male; Mammary Tumor Virus, Mouse; Molecular Sequence Data; Promoter Regions, Genetic; Prostatic Neoplasms; Receptors, Androgen; Transcription, Genetic; Transfection; Tumor Cells, Cultured	1994
Interaction of antiandrogen-androgen receptor complexes with DNA and transcription activation. The Journal of steroid biochemistry and molecular biology, 1993, Volume: 46, Issue:6 Topics: Androgen Antagonists; Animals; Binding, Competitive; Blotting, Western; Cell Line; Chloramphenicol O-Acetyltransferase; Chlorocebus aethiops; Cyproterone Acetate; Dihydrotestosterone; DNA; Flutamide; Gene Expression Regulation; Humans; Imidazoles; Imidazolidines; Kidney; Kinetics; Mammary Tumor Virus, Mouse; Metribolone; Receptors, Androgen; Recombinant Proteins; Transcription Factors; Transcription, Genetic; Transcriptional Activation; Transfection	1993
Suppression of sodium channel function in differentiating C2 muscle cells stably overexpressing rat androgen receptors. The Journal of neuroscience : the official journal of the Society for Neuroscience, 1994, Volume: 14, Issue:2 Topics: Acetylcholine; Androgen Antagonists; Animals; Bungarotoxins; Cell Differentiation; Cell Line; Dihydrotestosterone; Flutamide; Gene Expression; Metribolone; Mice; Muscles; Rats; Receptors, Androgen; Receptors, Cholinergic; Sodium Channels; Transfection	1994
Androgen receptor-mediated stimulation of 17 beta-hydroxysteroid dehydrogenase activity by dihydrotestosterone and medroxyprogesterone acetate in ZR-75-1 human breast cancer cells. Endocrinology, 1993, Volume: 132, Issue:1 Topics: 17-Hydroxysteroid Dehydrogenases; Breast Neoplasms; Dexamethasone; Dihydrotestosterone; Estradiol; Estrone; Flutamide; Humans; Kinetics; Medroxyprogesterone Acetate; Receptors, Androgen; Tumor Cells, Cultured	1993
Cloning and characterization of a specific coactivator, ARA70, for the androgen receptor in human prostate cells. Proceedings of the National Academy of Sciences of the United States of America, 1996, May-28, Volume: 93, Issue:11 Topics: Amino Acid Sequence; Base Sequence; Blotting, Northern; Cell Line; Chloramphenicol O-Acetyltransferase; Cloning, Molecular; Dihydrotestosterone; DNA-Binding Proteins; Flutamide; Humans; Male; Molecular Sequence Data; Nuclear Receptor Coactivators; Oncogene Proteins; Prostate; Prostatic Neoplasms; Receptors, Androgen; Receptors, Steroid; Recombinant Proteins; RNA, Messenger; Testosterone; Trans-Activators; Transcription Factors; Transcription, Genetic; Transfection; Tumor Cells, Cultured	1996
Androgen-like and anti-androgen-like effects of antiprogestins in human mammary cancer cells. European journal of cancer (Oxford, England : 1990), 1996, Volume: 32A, Issue:4 Topics: Androgen Antagonists; Antineoplastic Agents; Binding, Competitive; Breast Neoplasms; Cell Division; Dihydrotestosterone; Estrenes; Flutamide; Gonanes; Humans; Mifepristone; Models, Biological; Progestins; Receptors, Androgen; Transfection; Tumor Cells, Cultured	1996
Androgen independence of primary epithelial cultures of the prostate is associated with a down-regulation of androgen receptor gene expression. The Prostate, 1996, Volume: 29, Issue:6 Topics: Androgen Antagonists; Androgens; Base Sequence; Blotting, Northern; Cell Division; Dihydrotestosterone; DNA, Neoplasm; Dose-Response Relationship, Drug; Down-Regulation; Epithelium; Flutamide; Gene Expression Regulation, Neoplastic; Humans; Male; Molecular Sequence Data; Polymerase Chain Reaction; Prostatic Neoplasms; Receptors, Androgen; RNA, Messenger; Transfection; Tumor Cells, Cultured	1996
Androgen-induced inhibition of proliferation in human breast cancer MCF7 cells transfected with androgen receptor. Endocrinology, 1997, Volume: 138, Issue:4 Topics: Androgen Antagonists; Androgens; Anilides; Blotting, Western; Breast Neoplasms; Cell Cycle; Cell Division; Dihydrotestosterone; Dose-Response Relationship, Drug; Female; Flutamide; Humans; In Vitro Techniques; Metribolone; Nandrolone; Nitriles; Receptors, Androgen; Testosterone; Testosterone Congeners; Tosyl Compounds; Transfection; Tumor Cells, Cultured	1997
Non-steroidal L-245,976 acts as a classical antiandrogen in vitro. The Journal of steroid biochemistry and molecular biology, 1997, Volume: 60, Issue:1-2 Topics: Amides; Androgen Antagonists; Androgen-Binding Protein; Androgens; Aniline Compounds; Animals; Cell Division; Cell Line; CHO Cells; Colorimetry; Cricetinae; Dihydrotestosterone; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Flutamide; Formazans; Humans; Male; Receptors, Androgen; Recombinant Proteins; Testosterone; Tetrazolium Salts; Thiazoles; Transcriptional Activation; Transfection; Vas Deferens	1997
Interaction of mouse placental lactogens and androgens in regulating progesterone release in cultured mouse luteal cells. Endocrinology, 1997, Volume: 138, Issue:8 Topics: Androgen Receptor Antagonists; Androgens; Androstenedione; Animals; Aromatase Inhibitors; Cattle; Cells, Cultured; Cycloheximide; Dihydrotestosterone; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Estradiol; Estrogen Antagonists; Fadrozole; Female; Flutamide; Luteal Cells; Mice; Placental Lactogen; Pregnancy; Progesterone; Prolactin; Protein Synthesis Inhibitors; Rabbits; Testosterone	1997
Concerted stimulation of rat granulosa cell deoxyribonucleic acid synthesis by sex steroids and follicle-stimulating hormone. The Journal of steroid biochemistry and molecular biology, 1997, Volume: 62, Issue:1 Topics: Androgen Antagonists; Androgens; Androstenedione; Androsterone; Animals; Bucladesine; Cells, Cultured; Diethylstilbestrol; Dihydrotestosterone; DNA; Estradiol; Female; Flutamide; Follicle Stimulating Hormone; Granulosa Cells; Insulin; Insulin-Like Growth Factor I; Kinetics; Medroxyprogesterone; Ovary; Progesterone; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Testosterone; Thymidine	1997
Differential in vivo regulation of steroid hormone receptor activation by Cdc37p. Molecular biology of the cell, 1997, Volume: 8, Issue:12 Topics: Amino Acid Sequence; Androgen Antagonists; Cell Cycle Proteins; Chaperonins; Desoxycorticosterone; Dihydrotestosterone; Drosophila Proteins; Flutamide; Genes, Reporter; Humans; Ligands; Molecular Chaperones; Molecular Sequence Data; Mutation; Protein Structure, Tertiary; Receptors, Androgen; Receptors, Glucocorticoid; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Temperature; Thermodynamics; Transcriptional Activation	1997
Regulation of gonadotropin-releasing hormone (GnRH) gene expression by 5alpha-dihydrotestosterone in GnRH-secreting GT1-7 hypothalamic neurons. Endocrinology, 1998, Volume: 139, Issue:3 Topics: Animals; Cells, Cultured; Dihydrotestosterone; Flutamide; Gene Expression Regulation; Gonadotropin-Releasing Hormone; Humans; Hypothalamus; Mice; Neurons; Receptors, Androgen; RNA, Messenger	1998
The role of transforming growth factor-beta1, -beta2, and -beta3 in androgen-responsive growth of NRP-152 rat prostatic epithelial cells. Journal of cellular physiology, 1998, Volume: 175, Issue:2 Topics: Androgen Antagonists; Androgens; Animals; Antibodies; Cell Division; Cell Line; Dihydrotestosterone; Down-Regulation; Finasteride; Flutamide; Male; Prostate; Rats; Testosterone; Transforming Growth Factor beta	1998
Inhibition of androgen receptor-dependent transcriptional activity by DDT isomers and methoxychlor in HepG2 human hepatoma cells. Toxicology and applied pharmacology, 1998, Volume: 151, Issue:1 Topics: Androgen Antagonists; Androgen Receptor Antagonists; Androgens; Antineoplastic Agents, Hormonal; Carcinoma, Hepatocellular; DDT; Dihydrotestosterone; Estradiol; Flutamide; Humans; Insecticides; Isomerism; Methoxychlor; Progesterone; Receptors, Androgen; Testosterone; Transcription, Genetic; Tumor Cells, Cultured	1998
Effects of gonadal and adrenal androgens in a novel androgen-responsive human osteoblastic cell line. Journal of cellular biochemistry, 1998, Oct-01, Volume: 71, Issue:1 Topics: Adrenal Glands; Aged; Alkaline Phosphatase; Androgen Antagonists; Androgens; Cell Division; Cell Line; Collagen; Dehydroepiandrosterone; Dihydrotestosterone; DNA-Binding Proteins; Early Growth Response Transcription Factors; Flutamide; Gene Expression Regulation; Humans; Kruppel-Like Transcription Factors; Male; Osteoblasts; Osteocalcin; Testosterone; Transcription Factors; Transforming Growth Factor beta	1998
Functional characterization of mutant androgen receptors from androgen-independent prostate cancer. Clinical cancer research : an official journal of the American Association for Cancer Research, 1997, Volume: 3, Issue:8 Topics: Amino Acid Substitution; Androgen Antagonists; Androgens; Androstenedione; Animals; beta-Galactosidase; Cell Line; Dihydrotestosterone; Estradiol; Flutamide; Genes, Reporter; Imidazoles; Imidazolidines; Luciferases; Male; Point Mutation; Progesterone; Prostatic Neoplasms; Receptors, Androgen; Recombinant Fusion Proteins; Transfection	1997
Evidence for androgen receptor gene expression and growth inhibitory effect of dihydrotestosterone on human adrenocortical cells. The Journal of endocrinology, 1998, Volume: 159, Issue:3 Topics: Adrenal Cortex; Androgen Antagonists; Cell Division; Cells, Cultured; Cyproterone Acetate; Dihydrotestosterone; Female; Flutamide; Gene Expression; Humans; Immunohistochemistry; Male; Receptors, Androgen; Reverse Transcriptase Polymerase Chain Reaction; Tumor Cells, Cultured	1998
Androgens down-regulate bcl-2 protooncogene expression in ZR-75-1 human breast cancer cells. Endocrinology, 1999, Volume: 140, Issue:1 Topics: Androgen Antagonists; Androgens; Breast Neoplasms; Caspase 3; Caspases; Dihydrotestosterone; Down-Regulation; Estradiol; Estrogens; Female; Flutamide; Humans; Immunohistochemistry; Proto-Oncogene Proteins c-bcl-2; Tumor Cells, Cultured	1999
Androgens regulate bone resorption activity of isolated osteoclasts in vitro. Proceedings of the National Academy of Sciences of the United States of America, 1999, Jan-19, Volume: 96, Issue:2 Topics: Acid Phosphatase; Androgen Antagonists; Androgens; Animals; Bone Resorption; Cathepsin B; Chickens; Dihydrotestosterone; Flutamide; Genes, Reporter; Humans; Isoenzymes; Metribolone; Mice; Osteoclasts; Receptors, Androgen; Regulatory Sequences, Nucleic Acid; Tartrate-Resistant Acid Phosphatase; Transfection; Transforming Growth Factor beta	1999
Phosphorylation/dephosphorylation of androgen receptor as a determinant of androgen agonistic or antagonistic activity. Biochemical and biophysical research communications, 1999, May-27, Volume: 259, Issue:1 Topics: Androgen Antagonists; Androgens; Anilides; Animals; Base Sequence; Dihydrotestosterone; Estradiol; Estramustine; Flutamide; Humans; Ligands; Male; Molecular Sequence Data; Nitriles; Phosphorylation; Prostate-Specific Antigen; Prostatic Neoplasms; Receptors, Androgen; RNA, Messenger; Tosyl Compounds; Tumor Cells, Cultured	1999
Regulation of GCDFP-15 expression in human mammary cancer cells. International journal of molecular medicine, 1999, Volume: 4, Issue:2 Topics: Androgen Antagonists; Anilides; Apolipoproteins; Apolipoproteins D; Breast Neoplasms; Carrier Proteins; Cell Division; Dihydrotestosterone; Flutamide; Gene Expression Regulation, Neoplastic; Glycoproteins; Humans; Membrane Transport Proteins; Nitriles; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tosyl Compounds; Tumor Cells, Cultured	1999
The anti-androgen hydroxyflutamide and androgens inhibit interleukin-6 production by an androgen-responsive human osteoblastic cell line. Journal of bone and mineral research : the official journal of the American Society for Bone and Mineral Research, 1999, Volume: 14, Issue:8 Topics: Analysis of Variance; Androgen Antagonists; Androgens; Cell Line; Dihydrotestosterone; Flutamide; Humans; Interleukin-1; Interleukin-6; NF-kappa B; Osteoblasts; Paracrine Communication; Protein Binding; RNA, Messenger; Stimulation, Chemical; Tumor Necrosis Factor-alpha	1999
Androgen and epidermal growth factor down-regulate cyclin-dependent kinase inhibitor p27Kip1 and costimulate proliferation of MDA PCa 2a and MDA PCa 2b prostate cancer cells. Clinical cancer research : an official journal of the American Association for Cancer Research, 1999, Volume: 5, Issue:8 Topics: Androgen Antagonists; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Cell Cycle Proteins; Cell Division; Cyclin-Dependent Kinase Inhibitor p27; Cyclin-Dependent Kinases; Cycloheximide; Dihydrotestosterone; Down-Regulation; Drug Synergism; Enzyme Inhibitors; Epidermal Growth Factor; ErbB Receptors; Flutamide; Humans; Male; Metribolone; Microtubule-Associated Proteins; Prostatic Neoplasms; Protein Synthesis Inhibitors; Receptors, Androgen; Testosterone Congeners; Trastuzumab; Tumor Cells, Cultured; Tumor Suppressor Proteins	1999
Androgen receptor expression is greater in macrophages from male than from female donors. A sex difference with implications for atherogenesis. Circulation, 2000, Jan-25, Volume: 101, Issue:3 Topics: Adult; Aged; Arteriosclerosis; Cholesterol Esters; Dihydrotestosterone; Female; Flutamide; Humans; Macrophages; Male; Middle Aged; Receptors, Androgen; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sex Factors	2000
Down-regulation of transforming growth factor beta receptors by androgen in ovarian cancer cells. Cancer research, 2000, Feb-15, Volume: 60, Issue:4 Topics: Dihydrotestosterone; Down-Regulation; Female; Flutamide; Gene Expression Regulation; Humans; Ovarian Neoplasms; Receptors, Androgen; Receptors, Transforming Growth Factor beta; RNA, Messenger; Transforming Growth Factor beta; Tumor Cells, Cultured	2000
Rapid androgen actions on calcium signaling in rat sertoli cells and two human prostatic cell lines: similar biphasic responses between 1 picomolar and 100 nanomolar concentrations. Biology of reproduction, 2000, Volume: 63, Issue:3 Topics: Androgen Antagonists; Androgens; Animals; Calcium Signaling; Cell Line; Cyproterone Acetate; Dihydrotestosterone; Dose-Response Relationship, Drug; Flutamide; Gap Junctions; Humans; Kinetics; Male; Metribolone; Prostate; Prostatic Neoplasms; Rats; Rats, Wistar; Sertoli Cells; Testosterone; Tumor Cells, Cultured	2000
Mechanical strain stimulates osteoblast proliferation through the estrogen receptor in males as well as females. Journal of bone and mineral research : the official journal of the American Society for Bone and Mineral Research, 2000, Volume: 15, Issue:11 Topics: Androgen Antagonists; Androstenedione; Animals; Antibodies; Aromatase Inhibitors; Cells, Cultured; Dihydrotestosterone; Enzyme Inhibitors; Estradiol; Estrogen Antagonists; Estrogens; Flutamide; Fulvestrant; Insulin-Like Growth Factor I; Insulin-Like Growth Factor II; Male; Osteoblasts; Rats; Rats, Sprague-Dawley; Receptors, Estrogen; Stress, Mechanical; Tamoxifen; Testosterone; Thymidine	2000
Mutations at the boundary of the hinge and ligand binding domain of the androgen receptor confer increased transactivation function. Molecular endocrinology (Baltimore, Md.), 2001, Volume: 15, Issue:1 Topics: Adenocarcinoma; Androgen Antagonists; Androgens; Animals; Binding Sites; Cell Line; COS Cells; Dihydrotestosterone; DNA; Estradiol; Flutamide; Humans; Male; Mice; Mice, Transgenic; Models, Molecular; Mutagenesis; Mutation; Progesterone; Prostatic Neoplasms; Protein Structure, Secondary; Receptors, Androgen; Structure-Activity Relationship; Transcriptional Activation; Transfection	2001
Characterization of androgen receptors in a well-differentiated endometrial adenocarcinoma cell line (Ishikawa). The Journal of steroid biochemistry and molecular biology, 2000, Nov-15, Volume: 74, Issue:4 Topics: Adenocarcinoma; Alkaline Phosphatase; Androgens; Cell Differentiation; Cell Nucleus; Diethylstilbestrol; Dihydrotestosterone; Endometrial Neoplasms; Endometrium; Estradiol; Estrogen Receptor Modulators; Estrogens; Female; Flutamide; Fulvestrant; Humans; Metribolone; Progesterone; Receptors, Androgen; Reverse Transcriptase Polymerase Chain Reaction; Tumor Cells, Cultured	2000
Testosterone inhibits osteoclast formation stimulated by parathyroid hormone through androgen receptor. FEBS letters, 2001, Feb-23, Volume: 491, Issue:1-2 Topics: Androgen Antagonists; Androstenedione; Animals; Aromatase Inhibitors; Cell Division; Cells, Cultured; Dihydrotestosterone; Enzyme Inhibitors; Estradiol; Estrogen Antagonists; Flutamide; Fulvestrant; Glucuronates; Mice; Mice, Inbred ICR; Osteoclasts; Parathyroid Hormone; Receptors, Androgen; Teriparatide; Testosterone	2001
The subnuclear three-dimensional image analysis of androgen receptor fused to green fluorescence protein. The Journal of biological chemistry, 2001, Jul-27, Volume: 276, Issue:30 Topics: Active Transport, Cell Nucleus; Androgen Antagonists; Animals; Cell Nucleus; COS Cells; Dihydrotestosterone; Euchromatin; Flutamide; Green Fluorescent Proteins; Heterochromatin; Humans; Ligands; Luminescent Proteins; Microscopy, Confocal; Plasmids; Point Mutation; Progesterone; Protein Binding; Receptors, Androgen; Receptors, Progesterone; Recombinant Fusion Proteins; Transcription, Genetic; Transcriptional Activation	2001
Development of two androgen receptor assays using adenoviral transduction of MMTV-luc reporter and/or hAR for endocrine screening. Toxicological sciences : an official journal of the Society of Toxicology, 2002, Volume: 66, Issue:1 Topics: Adenoviridae; Androgen Antagonists; Androgen Receptor Antagonists; Androgens; Animals; Cell Line; Dexamethasone; Dihydrotestosterone; Flutamide; Gene Expression; Glucocorticoids; Humans; Luciferases; Mammary Tumor Virus, Mouse; Pesticides; Progesterone; Promoter Regions, Genetic; Receptors, Androgen; Receptors, Estrogen; Receptors, Glucocorticoid; Receptors, Progesterone; Recombinant Fusion Proteins; Transduction, Genetic; Transfection; Tumor Cells, Cultured	2002
Stabilization of androgen receptor protein is induced by agonist, not by antagonists. Biochemical and biophysical research communications, 2002, Jun-21, Volume: 294, Issue:4 Topics: Androgen Receptor Antagonists; Androgens; Anilides; Animals; Blotting, Northern; Blotting, Western; CHO Cells; Cricetinae; Dihydrotestosterone; Dose-Response Relationship, Drug; Flutamide; Humans; Ligands; Luciferases; Nitriles; Plasmids; Receptors, Androgen; RNA Processing, Post-Transcriptional; Time Factors; Tosyl Compounds; Transcriptional Activation; Transfection; Tumor Cells, Cultured	2002
Androgens protect against apolipoprotein E4-induced cognitive deficits. The Journal of neuroscience : the official journal of the Society for Neuroscience, 2002, Jun-15, Volume: 22, Issue:12 Topics: Androgen Antagonists; Androgens; Animals; Apolipoprotein E3; Apolipoprotein E4; Apolipoproteins E; Brain; Cognition; Cognition Disorders; Dihydrotestosterone; Female; Flutamide; Male; Maze Learning; Memory; Mice; Mice, Inbred C57BL; Mice, Knockout; Neuroprotective Agents; Receptors, Androgen; Recognition, Psychology; Sex Factors; Testosterone	2002
Nerve growth factor induces the re-expression of functional androgen receptors and p75(NGFR) in the androgen-insensitive prostate cancer cell line DU145. European journal of endocrinology, 2002, Volume: 147, Issue:3 Topics: Androgen Antagonists; Androgens; Apoptosis; Cell Division; Cyproterone Acetate; Dihydrotestosterone; Flutamide; Gene Expression; Humans; Male; Nerve Growth Factor; Prostatic Neoplasms; Receptor, Nerve Growth Factor; Receptors, Androgen; RNA, Messenger; Telomerase; Tumor Cells, Cultured	2002
Modulation of androgen receptor transactivation by gelsolin: a newly identified androgen receptor coregulator. Cancer research, 2003, Aug-15, Volume: 63, Issue:16 Topics: Animals; Cloning, Molecular; COS Cells; Dihydrotestosterone; Flutamide; Gelsolin; Humans; Male; Mice; Prostatic Neoplasms; Receptors, Androgen; Transcriptional Activation	2003
Interactions between androgen and growth factors in granulosa cell subtypes of porcine antral follicles. Biology of reproduction, 2004, Volume: 71, Issue:1 Topics: Androgen Antagonists; Androgens; Animals; Cell Division; Dihydrotestosterone; DNA; Drug Combinations; Female; Flutamide; Follicle Stimulating Hormone; Granulosa Cells; Growth Substances; Insulin-Like Growth Factor I; Progesterone; Swine; Time Factors	2004
5alpha-dihydrotestosterone inhibits 1alpha,25-dihydroxyvitamin D3-induced expression of CYP24 in human prostate cancer cells. The Prostate, 2005, May-15, Volume: 63, Issue:3 Topics: Androgen Receptor Antagonists; Androgens; Anilides; Calcitriol; Cycloheximide; Cytochrome P-450 Enzyme System; Dihydrotestosterone; Drug Interactions; Flutamide; Gene Expression Regulation, Enzymologic; Humans; Male; Nitriles; Prostatic Neoplasms; Protein Synthesis Inhibitors; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; Steroid Hydroxylases; Tosyl Compounds; Tumor Cells, Cultured; Vitamin D3 24-Hydroxylase	2005
Androgens augment the mitogenic effects of oocyte-secreted factors and growth differentiation factor 9 on porcine granulosa cells. Biology of reproduction, 2005, Volume: 73, Issue:4 Topics: Androgen Antagonists; Androgens; Animals; Bone Morphogenetic Protein 15; Cell Proliferation; Cells, Cultured; Coculture Techniques; Dihydrotestosterone; Dose-Response Relationship, Drug; Female; Flutamide; Follicle Stimulating Hormone; Granulosa Cells; Growth Differentiation Factor 9; Insulin-Like Growth Factor I; Intercellular Signaling Peptides and Proteins; Mice; Mitogens; Oocytes; Progesterone; Recombinant Proteins; Swine; Testosterone	2005
Androgen effects on hippocampal CA1 spine synapse numbers are retained in Tfm male rats with defective androgen receptors. Endocrinology, 2006, Volume: 147, Issue:5 Topics: Androgens; Animals; Dendrites; Dendritic Cells; Dihydrotestosterone; Estradiol; Flutamide; Genotype; Hippocampus; Male; Microscopy, Electron; Models, Statistical; Mutation; Neurons; Orchiectomy; Rats; Receptors, Androgen; Sesame Oil; Synapses; Time Factors	2006
Ligand-specific dynamics of the androgen receptor at its response element in living cells. Molecular and cellular biology, 2007, Volume: 27, Issue:5 Topics: Adenocarcinoma; Androgen Antagonists; Androgens; Anilides; Animals; Cell Line, Tumor; Chromatin Assembly and Disassembly; Cyproterone Acetate; Dihydrotestosterone; Female; Fluorescence Recovery After Photobleaching; Flutamide; Genes, Reporter; Green Fluorescent Proteins; In Situ Hybridization, Fluorescence; Ligands; Luciferases; Mammary Neoplasms, Animal; Mammary Tumor Virus, Mouse; Metribolone; Mice; Microscopy, Video; Mifepristone; Models, Biological; Nitriles; Plasmids; Promoter Regions, Genetic; Receptors, Androgen; Response Elements; Testosterone; Tosyl Compounds; Transcription, Genetic	2007
The androgen receptor T877A mutant recruits LXXLL and FXXLF peptides differently than wild-type androgen receptor in a time-resolved fluorescence resonance energy transfer assay. Biochemistry, 2007, Jan-23, Volume: 46, Issue:3 Topics: Amino Acid Sequence; Amino Acid Substitution; Androgen Antagonists; Anilides; Animals; Cyproterone Acetate; Dihydrotestosterone; Fluoresceins; Fluorescence Resonance Energy Transfer; Flutamide; Ligands; Mifepristone; Nitriles; Oligopeptides; Rats; Receptors, Androgen; Tosyl Compounds	2007
Non-steroidal antiandrogens act as AF-1 agonists under conditions of high androgen-receptor expression. The Prostate, 2007, May-01, Volume: 67, Issue:6 Topics: Androgens; Anilides; Dihydrotestosterone; Dose-Response Relationship, Drug; Drug Resistance, Neoplasm; Female; Flutamide; HeLa Cells; Humans; Male; Nitriles; Prostatic Neoplasms; Receptors, Androgen; Receptors, Interferon; Tosyl Compounds; Transcriptional Activation	2007
Dihydrotestosterone inhibits tumor necrosis factor alpha induced interleukin-1alpha mRNA expression in rheumatoid fibroblast-like synovial cells. Biological & pharmaceutical bulletin, 2007, Volume: 30, Issue:6 Topics: Androgen Receptor Antagonists; Arthritis, Rheumatoid; Cell Culture Techniques; Cell Line, Transformed; Cells, Cultured; Dihydrotestosterone; Flutamide; Genes, Reporter; Humans; Interleukin-1alpha; Luciferases; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Synovial Membrane; Time Factors; Transfection; Tumor Necrosis Factor-alpha	2007
Suppression of mutant androgen receptors by flutamide. International journal of urology : official journal of the Japanese Urological Association, 2009, Volume: 16, Issue:5 Topics: Androgen Antagonists; Androgens; Binding, Competitive; Cell Line, Tumor; Dihydrotestosterone; Flutamide; Humans; Luciferases; Male; Promoter Regions, Genetic; Prostatic Neoplasms; Receptors, Androgen; Transcriptional Activation	2009
Systematic structure-function analysis of androgen receptor Leu701 mutants explains the properties of the prostate cancer mutant L701H. The Journal of biological chemistry, 2010, Feb-12, Volume: 285, Issue:7 Topics: Androgen Antagonists; Anilides; Blotting, Western; Cell Line, Tumor; Cyproterone Acetate; Dihydrotestosterone; Flutamide; Humans; Hydrocortisone; Hydrophobic and Hydrophilic Interactions; Male; Mutation; Nitriles; Progesterone; Prostatic Neoplasms; Protein Structure, Secondary; Receptors, Androgen; Steroids; Structure-Activity Relationship; Tosyl Compounds	2010
A mouse model of androgenetic alopecia. Endocrinology, 2010, Volume: 151, Issue:5 Topics: Alopecia; Androgen Antagonists; Androgens; Animals; beta Catenin; Blotting, Western; Cell Line; Cell Line, Tumor; Dihydrotestosterone; Disease Models, Animal; Female; Flutamide; Hair; Humans; Keratin-5; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Promoter Regions, Genetic; Protein Binding; Receptors, Androgen; Transfection	2010
Is the "comb over" dying? A mouse model for male pattern baldness (androgenic alopecia). Endocrinology, 2010, Volume: 151, Issue:5 Topics: Alopecia; Androgen Antagonists; Androgens; Animals; beta Catenin; Dihydrotestosterone; Disease Models, Animal; Flutamide; Hair Follicle; Humans; Mice; Mice, Transgenic; Models, Biological; Protein Binding; Receptors, Androgen; Testosterone	2010
Androgen receptors in the posterior bed nucleus of the stria terminalis increase neuropeptide expression and the stress-induced activation of the paraventricular nucleus of the hypothalamus. Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2011, Volume: 36, Issue:7 Topics: Analysis of Variance; Androgen Antagonists; Androgens; Animals; Arginine Vasopressin; Castration; Corticosterone; Dihydrotestosterone; Flutamide; Functional Laterality; Gene Expression Regulation; Glutamate Decarboxylase; Male; Neuropeptides; Paraventricular Hypothalamic Nucleus; Rats; Rats, Sprague-Dawley; Receptors, Androgen; RNA, Messenger; Septal Nuclei; Stress, Psychological	2011
A novel steroidal antiandrogen targeting wild type and mutant androgen receptors. Biochemical pharmacology, 2011, Dec-01, Volume: 82, Issue:11 Topics: Androgen Antagonists; Animals; Binding, Competitive; Carbamates; Cell Line, Tumor; Cell Proliferation; Chlorocebus aethiops; Dihydrotestosterone; Drug Screening Assays, Antitumor; Flutamide; Humans; Male; Models, Molecular; Mutation; Prostate-Specific Antigen; Prostatic Neoplasms; Protein Transport; Receptors, Androgen; Structure-Activity Relationship; Transcriptional Activation	2011
Androgen receptor signals regulate UDP-glucuronosyltransferases in the urinary bladder: a potential mechanism of androgen-induced bladder carcinogenesis. Molecular carcinogenesis, 2013, Volume: 52, Issue:2 Topics: Aged; Aged, 80 and over; Androgen Antagonists; Animals; Cell Line; Cystectomy; Dihydrotestosterone; Down-Regulation; Female; Flutamide; Follow-Up Studies; Gene Expression Regulation, Enzymologic; Glucuronosyltransferase; Humans; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Middle Aged; Orchiectomy; Receptors, Androgen; Reference Values; Signal Transduction; UDP-Glucuronosyltransferase 1A9; Urinary Bladder; Urinary Bladder Neoplasms	2013
Fluorescence lifetime imaging microscopy for the monitoring of green fluorescent protein-tagged androgen receptors in living cells. Chemical & pharmaceutical bulletin, 2013, Volume: 61, Issue:1 Topics: Animals; Cell Survival; Chlorocebus aethiops; COS Cells; Dihydrotestosterone; Flutamide; Green Fluorescent Proteins; Microscopy, Fluorescence; Receptors, Androgen	2013
Androgens promote the acquisition of maturation competence in bovine oocytes. The Journal of reproduction and development, 2015, Volume: 61, Issue:3 Topics: Androgen Receptor Antagonists; Androgens; Animals; Cattle; Cell Nucleus; Dihydrotestosterone; Estradiol; Female; Flutamide; Granulosa Cells; Metaphase; Microscopy, Fluorescence; Oocytes; Receptors, Androgen	2015
Corepressive function of nuclear receptor coactivator 2 in androgen receptor of prostate cancer cells treated with antiandrogen. BMC cancer, 2016, 05-25, Volume: 16 Topics: Androgen Antagonists; Anilides; Cell Line, Tumor; Cell Proliferation; Dihydrotestosterone; Flutamide; Gene Expression Regulation, Neoplastic; Humans; Male; Mutation; Nitriles; Nuclear Receptor Coactivators; Prostatic Neoplasms; Receptors, Androgen; Tosyl Compounds	2016
Enzalutamide inhibits androgen receptor-positive bladder cancer cell growth. Urologic oncology, 2016, Volume: 34, Issue:10 Topics: Androgen Antagonists; Anilides; Animals; Antineoplastic Agents; Apoptosis; Benzamides; Cell Line, Tumor; Cell Movement; Cell Proliferation; Cell Survival; Dihydrotestosterone; Down-Regulation; Flutamide; Humans; Interleukin-6; Male; Matrix Metalloproteinase 2; Mice; Mice, Inbred NOD; Mice, SCID; Neoplasm Transplantation; Nitriles; Phenylthiohydantoin; Receptors, Androgen; RNA; Tosyl Compounds; Transcription, Genetic; Urinary Bladder Neoplasms	2016
Structural Dynamics of Agonist and Antagonist Binding to the Androgen Receptor. The journal of physical chemistry. B, 2019, 09-12, Volume: 123, Issue:36 Topics: Androgen Receptor Antagonists; Androgens; Anilides; Binding Sites; Dihydrotestosterone; Flutamide; Humans; Molecular Dynamics Simulation; Nitriles; Receptors, Androgen; Testosterone; Tosyl Compounds	2019