histamine and thiourea

histamine has been researched along with thiourea in 365 studies

Research

Studies (365)

TimeframeStudies, this research(%)All Research%
pre-1990268 (73.42)18.7374
1990's42 (11.51)18.2507
2000's38 (10.41)29.6817
2010's15 (4.11)24.3611
2020's2 (0.55)2.80

Authors

AuthorsStudies
Code, CF2
Schofield, B; Tepperman, BL; Tepperman, FS1
Durant, GJ; Emmett, JC; Ganellin, CR1
Brimblecombe, RW; Duncan, WA; Owen, DA; Parsons, ME1
Ledda, F; Mantelli, L; Mugelli, A1
Bunce, KT; Parsons, ME3
Jellinek, M; Kaminski, DL; Ruwart, MJ1
Burks, TF1
Reinhardt, D; Schümann, HJ; Wiemann, HM1
Olbe, L; Ryberg, B; Sjöstrand, SE1
Haith, LR; Reynolds, ES; Szabo, S1
Morrissey, SM; Tymvios, MC1
Buck, SH; Gilman, DJ; Jones, DF; Wardleworth, JM; Yellin, TO1
Adamik, R; Baxter, JH1
Lundell, L2
Magee, DF1
Advenier, C; Mallard, B; Ruff, F; Santais, MC1
Bertaccini, G; Coruzzi, G; Plazzi, V1
Becker, M; Malchow, H; Painz, B; Rack, M; Ruoff, HJ; Sewing, KF1
Drazen, JM; Schneider, MW; Venugopalan, CS1
Bertaccini, G; Bocchi, P; Melotti, G; Zappia, L1
Kreutner, W; Yen, SS1
Ferrario, E; Lebrecht, U; Nowak, JZ1
Beaven, MA; Shaff, RE1
Aksulu, HE; Ercan, ZS; Türker, RK1
Michel, IM; Weinryb, I1
Kostopoulos, GK; Odutola, A; Phillis, JW1
Berglindh, T1
Anderson, R; Glover, A; Rabson, AR1
Allouche, G; Foussard, C; Parrot, JL; Ruff, F; Santais, MC1
Cherry, KJ; Ritchie, WP1
Edvinsson, L; Owman, C1
Bailey, BA; Fordtran, JS; Richardson, CT; Walsh, JH1
Buck, SH; Sperow, JW; Yellin, TO1
Bareicha, I; Silva, MR1
Code, CF; Preiss, DU1
Fuchs, W; Mitznegg, P; Schubert, E1
Albinus, M; Blair, EL; Hirst, BH; Reed, JD; Schally, AV; Shaw, B1
Boĭko, NS; Fokina, AA; Klimov, PK1
Bolton, JP; Cohen, MM1
Berti, F; Folco, GC; Nicosia, S; Omini, C; Pasargiklian, R1
Jacobson, ED; Miller, TA; Pawlik, W; Tague, LL; Tepperman, BL1
Chiavarini, M; Impicciatore, M; Razzetti, R; Vitali, T1
Szelenyi, I; Thiemer, K1
Bertaccini, G; Coruzzi, G; Musso, E1
Bertaccini, G; Impicciatore, M; Morini, G1
Barkla, DH; Tutton, PJ1
Huszti, Z1
Carter, DC; Grossman, MI; Impicciatore, M1
Banks, RO; Fondacaro, JD; Jacobson, ED; Schwaiger, MM1
Grossman, MI; Petersen, H1
Bajaj, SC; Hirschowitz, BI1
Doyle, TF; Kobrine, AI; Rizzoli, HV1
Giles, RW; Heise, G; Wilcken, DE1
Durant, GJ; Ganellin, CR; Parsons, ME1
Biegańaki, T; Fogel, WA; Maśliński, C1
Kwong, F; Orzechowski, RF1
Dormann, P; Hamelmann, H; Lorenz, W; Schingale, F; Schmal, A; Thermann, M1
Chakrin, LW; Krell, RD1
Chiba, S1
Johnston, BM; Owen, DA1
Holstein, B2
Feldman, EJ; Isenberg, JI1
Francis, D; Greaves, MW; Yamamoto, S1
Ruoff, HJ; Sewing, KF1
Lin, TM; Warrick, MW1
Lippe, C; Schettino, T1
Bank, S; Barbezat, GO; Grant, B; Vinik, A1
Bowen, JC; Jacobson, ED; Kuo, YJ; Pawlik, W; Shanbour, LL; Williams, D1
Hood, AJ; Smy, JR; Weetman, DF1
Debbas, G; Goodman, FR; Weiss, GB1
Shumaker, JB1
Buschauer, A; Höer, A; Schwaner, I; Seifert, R1
Donné-Op den Kelder, GM; Haaksma, EE; Timmerman, H; Vernooijs, P1
Barker, LA; Petropoulos, AC; Winbery, SL1
Brink, C; Gorenne, I; Labat, C; Norel, X; Ortiz, JL; Verley, J1
Maeyama, K; Ohkawara, Y; Ohrui, T; Sasaki, H; Sasaki, M; Sekizawa, K; Takemura, M; Wada, H; Watanabe, T; Yamauchi, K1
Bast, A; Brozius, MM; Leurs, R; Smit, MJ; Timmerman, H1
Donné- op den Kelder, GM; Haaksma, EE; Timmerman, H; Weinstein, H1
Hannibal, T; Jørgensen, H; Knigge, U; Matzen, S; Warberg, J1
Nowak, JZ; Sek, B1
Krielaart, MJ; van Buuren, KJ; Veenstra, DM1
Benedito, S; Nyborg, NC; Prieto, D1
Giri, SN; Hollinger, MA; Rice, SA2
Benedito, S; Nielsen, PJ; Nyborg, NC; Prieto, D1
Bermejo, E; Egozcue, J; Gimeno, M; Lazzari, MA; Maugeri, N; Serpente, N1
Matsumoto, M; Nishio, A; Obi, T1
Chediak, AD; Csete, ME; Elsasser, S; Gazeroglu, H; Wanner, A1
Mutafova-Yambolieva, V; Staneva-Stoytcheva, D; Todorov, S; Vassilev, P1
Dy, M; Piquet-Pellorce, C; Schneider, E2
Chiba, S; Tsukada, M1
Campillo, M; Giraldo, J; Martín, M; Pardo, L1
Dolata, J; Lindberg, S; Mercke, U1
Amerini, S; Cerbai, E; Mugelli, A1
Gerges, E; Gertner, SB1
Almeida, L; Figueiredo, A; Gonçalo, M; Poiares-Baptista, A; Ribeiro, CA; Teixeira, F1
Cooke, HJ; Wang, YZ1
Młynarska, MS1
Matsuki, T; Ohhashi, T1
Asea, A; Hellstrand, K; Hermodsson, S1
Clark, MA; Egan, RW; Shih, NY; Siegel, MI; West, RE; Zweig, A1
Borchard, U; Hafner, D; Hirth, C1
Borchard, U; Hafner, D1
Donné-Op den Kelder, GM; Haaksma, EE; Ravenek, W; Timmerman, H; Vernooijs, P1
Hashimoto, K; Motomura, S1
Bugajski, J; Gadek-Michalska, A1
Cortijo, J; Esplugues, J; Morcillo, EJ; Orón, JD; Ortiz, JL; Perpiñá, M; Sanz, C1
Bueno, L; Fargeas, MJ; Fioramonti, J1
Abboud, HE; Sedor, JR1
Gannon, MN; Hough, LB1
Girard, A; Marche, P1
Batzri, S; Thompson, WF; Toles, R1
Bertaccini, G; Coruzzi, G; Poli, E1
Mieda, M; Sakuma, H; Shiratsuchi, K; Tarutani, M1
Rising, TJ; Steward, A1
Sterk, GJ; Timmerman, H; van der Goot, H1
Hutchison, VH; Spriestersbach, KK1
Knigge, U; Matzen, S; Warberg, J2
Coruzzi, G; Noci, MT1
Boucher, M; Duchene-Marullaz, P; Li, JH1
Blandina, P; Brunelleschi, S; Fantozzi, R; Giannella, E; Mannaioni, PF; Masini, E1
Bertaccini, G; Coruzzi, G1
Salonen, RO; Webber, SE; Widdicombe, JG1
Akahori, H; Kamei, C; Kitazumi, K; Tasaka, K1
Ledgard, SE; Nieves, AL; Woodward, DF1
Beaudoin, J; Beaulieu, L; Hébert, J; Jobin, M1
Barker, LA; Winbery, SL1
Donaldson, J; Hill, SJ1
Bordi, F; Chiavarini, M; Impicciatore, M; Morini, G; Plazzi, PV; Vitali, F2
Adami, M; Bertaccini, G; Coruzzi, G1
Fan, HX; Wen, R1
Kim, LE; Oudart, N; Sercombe, R; Teste, JF1
Gertner, SB; Poulakos, JJ1
Granata, AR; Reis, DJ1
Hayashi, S; Miichi, H; Tanaka, H; Umemoto, M1
Jouvet, M; Lin, JS; Sakai, K1
Chiba, S; Nakane, T1
Nishiwaki, H; Okabe, S; Okada, M; Takeuchi, K1
Knigge, U; Matzen, S; Sleimann, I; Warberg, J1
Fromm, D; Furukawa, T; Olender, EJ; Woods, DJ1
Ekblad, EB; Licko, V2
Altman, CB; Bassett, AL; Cameron, JS; Cuevas, J; Gaide, MS; Goad, PL; Myerburg, RJ1
Faanes, R; French, S; Susskind, B; Walker, M1
Leff, P; Trist, DG1
Dimlich, RV1
Black, JW; Hesselbo, T; Wyllie, JH2
Gillespie, E; Henney, CS; Lichtenstein, LM; Plaut, M1
Gillespie, E; Lichtenstein, LM1
Türker, RK1
Ambache, N; Killick, SW; Zar, MA1
Bovaird, L; Kobayashi, Y; Maudsley, DV; Williamson, E1
Henney, CS; Lichtenstein, LM; Plaut, M1
Burns, LR; Hackney, V; Jenkins, BC; Sachs, G; Spenney, JG; Sung, CP; Wiebelhaus, VD1
Code, CF; Dousa, TP1
Taylor, KM1
Assem, ES; Schild, HO; Wan, BY2
McNeill, JH; Verma, SC2
Eyre, P1
Black, JW; Duncan, WA; Emmett, JC; Ganellin, CR; Hesselbo, T; Parsons, ME; Wyllie, JH1
Barth, H; Lorenz, W; Niemeyer, I2
Fantozzi, R; Mannaioni, PF; Moroni, F2
Schayer, RW1
Black, JW; Durant, GJ; Emmett, JC; Ganellin, CR1
Grossman, MI; Konturek, SJ1
Buckner, E; Sachs, G; Shoemaker, RL; Spenney, JG1
Harris, D; Reed, JD; Smy, JR; Venables, CW1
Dembiński, A; Demitrescu, T; Konturek, S; Mitis, M; Radecki, T1
Albinus, M; Sewing, KF3
Gibson, R; Hirschowitz, BI; Hutchison, G1
Dick, WC; Gilbertson, E; Grennan, DM; Rooney, PJ1
Hirschowitz, BI1
Csongrady, A; Kobinger, W1
Main, IH; Whittle, BJ1
Fantozzi, R; Ledda, F; Mannaioni, PF; Moroni, F; Mugelli, A2
Brimblecombe, RW; Owen, DA; Parsons, ME1
Bökesoy, TA; Türker, RK1
Mathé, AA; Puri, SK; Volicer, L1
carroll, PR; Glover, WE; Latt, N1
Demitrescu, T; Konturek, SJ; Radecki, T1
Okpako, DT1
Owen, DA; Parsons, ME1
Reinhardt, D; Schümann, HJ; Wagner, J1
Albinus, M; Sewing, KR1
Kolodej, A; Kowalewski, K1
Bogatyrev, GP; Chirkov, IuIu; Goncharenko, EN; Kudriashov, IuB1
Cronin, SR; Giri, SN1
Karppanen, HO; Westermann, E1
Brimble, MJ; Wallis, DI1
Black, JW; Duncan, WA; Durant, CJ; Ganellin, CR; Parsons, EM1
Guthrie, PD; Johnson, LR1
Bovaird, L; Kobayashi, Y; Maudsley, DV; Zeidel, M1
McNeil, JH; Verma, SC1
Biernat, J; Konturek, SJ; Oleksy, J1
Curwain, BP; Holton, P; Spencer, J1
Blyth, DI1
Spencer, J1
Bank, S; Barbezat, GO; Daniel, M; Grant, B; Vinik, A1
Suzuki, T1
Cotton, WR; Leonard, EP1
Davis, EM; Simons, HA1
Hirshfeld, A; Mechoulam, R1
Batzri, S1
Kume, S; Ohashi, T; Ozaki, Y1
Gerber, JG; Nies, AS2
Gristwood, RW; Lincoln, JC; Owen, DA1
Daniel, D; Owen, DA; Poy, E; Woodward, DF1
Askenase, PW; Gershon, RK; Schwartz, A1
Cho, CH; Pfeiffer, CJ1
Fondacaro, JD; Jacobson, ED; Walus, KM1
Eyre, P; Norris, AA1
Colboc, O; Costentin, J; Protais, P1
Oriowo, MA1
Ooi, YM1
Clineschmidt, BV; Cook, PG; Hanson, CA; Pendleton, RG; Torchiana, ML1
Birkett, DH; La Morte, WW; Schoetz, DJ; Williams, LF; Wise, WE1
Fletcher, MP; Gallin, JI; Seligmann, BE1
Heldsinger, AA; Skoglund, ML; Vinik, AI1
Donoso, AO; Zárate, MB1
Guldvog, I; Linnestad, P; Schrumpf, E1
Nemeth, PR; Ort, CA; Wood, JD1
Tsai, BS; Yellin, TO1
Burtin, C; Lebel, B; Soubrane, C1
Bielkiewicz, B; Kordecka, A; Lebrecht, U; Maslinski, C; Nowak, JZ1
Rothschild, AM1
Johnson, CL; Kalinyak, K; Sawutz, DG; Whitsett, JA1
Birkett, DH; Gaca, JM; LaMorte, WW; Schoetz, DJ; Williams, LF; Wise, WE1
Christiansen, VJ; Horst, MA; Robinson, CP1
Eyre, P; Mirbahar, KB1
Ganellin, CR; Martin, D; Milliner, K; Vickers, MR1
Sykes, KJ; Vickers, MR1
Horowitz, GP; Isaacson, RL; O'Callaghan, M1
Badger, AM; Poste, G; Young, J1
Bertaccini, G; Bezzi, E; Potenzoni, D; Zappia, L1
Salvati, P; Whittle, BJ1
Bugajski, J; Gadek, A1
Bugajski, J; Janusz, Z1
Brooks, HL; Christensen, CW; Gross, GJ; Hardman, HF; Warltier, DC1
Owen, DA; Pipkin, MA; Woodward, DF1
Clark, KE; Harrington, DJ; Mills, EG1
Jespersen, LT; Mikkelsen, E; Sakr, AM1
Cooke, HJ; Nemeth, PR; Wood, JD1
Christiansen, VJ; Horst, MA; Robinson, C1
Dale, MM; Ladd, R1
Horst, MA; Robinson, CP1
Cheret, AM; Lewin, MJ; Mangeat, P; Marchis-Mouren, G1
Brown, EM1
Baumann, G; Blömer, H; Erhardt, WD; Felix, SB; Heidecke, CD; Loher, U; Ludwig, L; Riess, G; Schrader, J; Sebening, F1
Nishibori, M1
Daly, MJ; Humphray, JM; Stables, R1
Batzri, S; Harmon, JW; Thompson, WF1
Eckel, L; Gristwood, RW; Nawrath, H; Owen, DA; Satter, P1
Bonnet, M; Burtin, C; Lespinats, G1
Del Soldato, P1
Konturek, SJ; Siebers, R1
Hughes, MJ1
Birkett, DH; Gaca, JM; LaMorte, WW; Williams, LF; Wise, WE1
Anderson, C; Busse, WW; Cooper, W1
Eriksson, L; Tuomisto, L1
Davies, MG; Greaves, MW1
Gertner, SB; Klein, MC1
Hingston, SJ; La Morte, WW; Wise, WE1
Harvey, CA; Owen, DA; Quinn, EH1
Philippu, A; Wiedemann, K2
Pang, PK; Tenner, TE; Yang, MC1
Bielkiewicz, B; Nowak, JZ1
Tenner, TE1
Di Donato, M; Mantovani, P; Santicioli, P1
Nunoki, K; Shimizu, T; Taira, N1
Gross, PM; Harper, AM; Teasdale, GM1
Baker, AP; Chakrin, LW; Holden, DA; Smith, WJ; Sung, CP1
Brink, C; Douglas, JS; Duncan, PG1
Bertaccini, G; Coruzzi, G; Scarpignato, C1
Bedate, H; Esplugues, J; Moragues, A; Morcillo, E1
Beck, H; Engler, H; Szelenyi, I1
Chambers, MM; Russell, JC1
Wikel, SK1
Banks, K; Merali, Z1
Buczko, W; Godlewski, G; Malinowska, B; Schlicker, E1
Banchelli, G; Conforti, L; Pirisino, R; Raimondi, L; Sgromo, L1
Marr, I; Schlicker, E1
Bucher, B; Godlewski, G; Malinowska, B; Schlicker, E1
Hemedah, M; Mitchelson, F1
Kou, YR; Lai, CJ1
Bacciottini, L; Blandina, P; Cecchi, M; Giorgetti, M; Giovannini, MG1
Aarden, LA; Alewijnse, AE; Boeije, LC; de Groot, ER; Leurs, R; Snijders, A; van der Pouw Kraan, TC1
Schlicker, E; Werthwein, S; Zentner, J1
Jørgensen, H; Kjaer, A; Knigge, U; Warberg, J; Willems, E1
Murakami, Y; Nakamura, K; Okada, S; Wang, M; Yokotani, K1
de Wildt, DJ; Hendriksen, CF; van de Kuil, A; van den Hout, JW; Vleeming, W1
Chen, Z; Fujii, Y; Ishizawa, K; Kamei, C; Okuma, C; Sugimoto, Y1
Attarzadeh, M; Farzin, D1
Anthes, JC; Bayne, M; Behan, J; Gonsiorek, W; Greene, J; Greenfeder, SA; Gustafson, EL; Hedrick, JA; Hipkin, RW; Laz, TM; Monsma, FJ; Morse, KL; Qiao, X; Shin, N; Umland, S; Wan, Y; Wang, S; West, RE1
Aceves, J; Arias-Montaño, JA; Floran, B; Garcia, M; Young, JM1
Chen, Z1
Barnes, W; Boyd, D; Hough, L1
Blanco, I; Gomez-Ramirez, J; Ortiz, J1
Chen, J; Liu, C; Lovenberg, TW1
Chen, Z; Hu, WW; Huang, YW; Wei, EQ; Yanai, K; Zhang, LS1
Debilly, G; Gigout, S; Lin, JS; Vanni-Mercier, G1
Buckland, KF; Conroy, DM; Williams, TJ1
Fujii, Y; Hossen, MA; Kamei, C; Kayasuga, R; Sugimoto, Y1
GIUSTI, G; TESI, A1
Chen, Z; Hu, WW; Jin, CL; Shen, HQ; Zhang, LS; Zhao, MH1
Arrang, JM; Cochois, V; Héron, A; Pillot, C; Rouleau, A; Schwartz, JC1
Blanco, I; Gómez-Ramírez, J; Moreno-Delgado, D; Ortiz, J; Rodríguez-Agudo, D; Rodríguez-Caso, C; Sánchez-Jiménez, F; Torrent, A1
Fu, YL; He, SH; Xie, H1
Espinosa-Tanguma, R1
Djahanguiri, B; Khalilzadeh, A; Zarrindast, MR1
Blanks, AM; Lee, K; Renaud, LP; Spanswick, D; Whyment, AD1
Eckman, JR; Wagner, MC; Wick, TM1
Holopainen, IE; Kukko-Lukjanov, TK; Michelsen, KA; Panula, P; Soini, S; Taira, T1
Carr, TL; Cassar, S; Esbenshade, TA; Faghih, R; Hancock, AA; Krueger, KM; Miller, TR; Sharma, R; Surber, BW; Witte, DG; Yao, BB1
Blanco, I; de Esch, I; Gómez-Ramírez, J; Moreno-Delgado, D; Ortiz, J; Torrent, A1
Arias-Montaño, JA; Garduño-Torres, B; Gutiérrez, R; Treviño, M1
Hirota, S; Janssen, LJ; Pertens, E1
Chen, Z; Dai, HB; Fu, QL; Shen, Y1
Algara-Suárez, P; Chrones, T; Espinosa-Tanguma, R; Meza, U; Romero-Méndez, C; Sánchez-Armass, S; Sims, SM1
Alvarez, J; Hernández-Sanmiguel, E; Lobatón, CD; Montero, M; Moreno, A; Santo-Domingo, J; Vay, L1
Chazot, P; Dijkstra, D; Gutzmer, R; Leurs, R; Shenton, FC; Stark, H; Werfel, T1
Brzozowski, T; Gaca, P; Hahn, EG; Konturek, PC; Konturek, SJ; Pawlik, M; Raithel, M1
Bergoc, R; Crescenti, E; Cricco, G; Croci, M; Martin, G; Massari, N; Medina, V; Mohamad, N; Nuñez, M; Rivera, E; Sanchez-Jiménez, F1
Hatano, K; Ishizuka, T; Murotani, T; Yamatodani, A1
Kamei, C; Kuyama, S; Ogawa, M; Yokota, E1
Bäumer, W; Chazot, P; Dijkstra, D; Gutzmer, R; Kietzmann, M; Stark, H; Wendorff, S; Werfel, T1
Barrett, P; Ebling, FJ; Enright, RA; Jethwa, PH; Murphy, M; Turnbull, Y; Warner, A1
Khodarahmi, P; Oryan, S; Rezayof, A; Zarrindast, MR1
Bäumer, W; Kietzmann, M; Leurs, R; Rossbach, K; Sander, K; Stark, H1
Antigny, F; Frieden, M; Girardin, NC1
Khanam, R; Manocha, A; Uma Devi, P; Vohora, D1
Bertron, AF; Dy, M; Schneider, E1
Hall, FS; Kitanaka, J; Kitanaka, N; Morita, Y; Nishiyama, N; Takemura, M; Tanaka, K; Tatsuta, T; Uhl, GR1
Bergoc, RM; Cricco, GP; Croci, M; Martinel Lamas, DJ; Massari, NA; Medina, VA; Rivera, ES; Sambuco, L1
Clapp, RH; Luckman, SM1
Jurič, DM; Mele, T1
Ciz, M; Jancinova, V; Lojek, A; Nosal, R; Vasicek, O1
Akhtar, M; Goswami, D; Jahan, K; Mahmood, D1
Durante, M; Galeotti, N; Ghelardini, C; Lucarini, L; Masini, E; Sanna, MD1
Bachelerie, F; Chauveau, L; Cutolo, P; Davidson, S; Durroux, T; Dutrieux, J; Dy, M; Herbeuval, JP; Manoury, B; McCort-Tranchepain, I; Münch, J; Nisole, S; Pietrancosta, N; Schwartz, O; Scott-Algara, D; Smith, N; Wack, A; Zirafi, O1
Fernandes, CEM; Gianlorenco, ACL; Mattioli, R; Serafim, KR1
An, S; Chen, LY; Guo, XX; Hao, Q; Liu, Y; Ma, L; Pediani, JD; Tang, M; Ward, RJ; Wu, N; Xu, TR; Yang, Y; Zeng, H1
Ciosek, J; Drobnik, J; Galdyszynska, M; Kun, T; Olczak, S; Piera, L; Szymanski, J1
Borgonetti, V; Galeotti, N; Masini, E; Sanna, MD1
Bryukhovetskiy, I; Buzoianu, AD; Castellani, RJ; Lafuente, JV; Manzhulo, I; Menon, PK; Muresanu, DF; Nozari, A; Patnaik, R; Sahib, S; Sharma, A; Sharma, HS; Skaper, SD; Tian, ZR; Wiklund, L1

Reviews

3 review(s) available for histamine and thiourea

ArticleYear
[Burimamid and metiamid, a new pharmacological principle].
    Der Internist, 1974, Volume: 15, Issue:3

    Topics: Animals; Cats; Dose-Response Relationship, Drug; Female; Gastric Mucosa; Gastrointestinal Motility; Guinea Pigs; Heart Atria; Histamine; Histamine H1 Antagonists; Humans; Ileum; Imidazoles; In Vitro Techniques; Methylation; Molecular Conformation; Pentagastrin; Rats; Receptors, Drug; Sulfides; Swine; Thiourea; Uterus

1974
Modulation of hematopoiesis through histamine receptor signaling.
    Frontiers in bioscience (Scholar edition), 2011, 01-01, Volume: 3, Issue:2

    Topics: Animals; Cell Cycle; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclin-Dependent Kinase Inhibitor p21; Hematopoiesis; Hematopoietic Stem Cells; Histamine; Humans; Imidazoles; Mice; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Signal Transduction; Thiourea

2011
Histamine H3 and H4 receptors modulate Parkinson's disease induced brain pathology. Neuroprotective effects of nanowired BF-2649 and clobenpropit with anti-histamine-antibody therapy.
    Progress in brain research, 2021, Volume: 266

    Topics: Corpus Striatum; Histamine; Humans; Imidazoles; Neuroprotective Agents; Parkinson Disease; Receptors, Histamine H4; Thiourea

2021

Trials

4 trial(s) available for histamine and thiourea

ArticleYear
Human gastric mucosal adenylate cyclase: activation by histamine-H2-receptor stimulation and inhibition by cimetidine in vitro and in peptic ulcer patients.
    European journal of clinical pharmacology, 1979, Apr-17, Volume: 15, Issue:3

    Topics: Adenylyl Cyclases; Cimetidine; Clinical Trials as Topic; Enzyme Activation; Female; Gastric Mucosa; Guanidines; Histamine; Humans; Male; Middle Aged; Peptic Ulcer; Phenethylamines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H2; Thiourea

1979
The effect of an H2-receptor antagonist on food-stimulated acid secretion, serum gastrin, and gastric emptying in patients with duodenal ulcers. Comparison with an anticholinergic drug.
    The Journal of clinical investigation, 1975, Volume: 55, Issue:3

    Topics: Adult; Clinical Trials as Topic; Drug Therapy, Combination; Duodenal Ulcer; Female; Food; Gastric Juice; Gastrins; Gastrointestinal Motility; Histamine; Humans; Imidazoles; Male; Middle Aged; Placebos; Quaternary Ammonium Compounds; Receptors, Drug; Stomach; Sulfides; Thiourea

1975
The effect of histamine H2-receptor blockade with metiamide on serum gastrin levels in man.
    Gut, 1975, Volume: 16, Issue:3

    Topics: Adolescent; Adult; Drinking; Gastrins; Histamine; Humans; Meat; Metiamide; Radioimmunoassay; Receptors, Drug; Thiourea

1975
Sensory responses of human skin to synthetic histamine analogues and histamine.
    British journal of clinical pharmacology, 1980, Volume: 9, Issue:5

    Topics: Adult; Chlorpheniramine; Dimaprit; Female; Histamine; Humans; Male; Methylhistamines; Pruritus; Receptors, Histamine H1; Receptors, Histamine H2; Skin; Thiourea

1980

Other Studies

358 other study(ies) available for histamine and thiourea

ArticleYear
Proceedings: Suppression of histamine leucocytosis by metiamide.
    The Journal of physiology, 1976, Volume: 254, Issue:1

    Topics: Animals; Dogs; Histamine; Histamine H1 Antagonists; Leukocytosis; Metiamide; Neutrophils; Thiourea

1976
Effect of metiamide on acid secretion from isolated kitten fundic mucosa.
    Canadian journal of physiology and pharmacology, 1975, Volume: 53, Issue:6

    Topics: Acetylcholine; Animals; Cats; Female; Gastric Juice; Gastric Mucosa; Histamine; Histamine H1 Antagonists; In Vitro Techniques; Male; Metiamide; Pentagastrin; Stimulation, Chemical; Thiourea; Time Factors

1975
Some chemical aspects of histamine H2-receptor antagonists.
    Federation proceedings, 1976, Volume: 35, Issue:8

    Topics: Burimamide; Histamine; Histamine H1 Antagonists; Isoelectric Point; Metiamide; Molecular Conformation; Receptors, Drug; Structure-Activity Relationship; Thiourea

1976
The pharmacology of burimamide and metiamide, two histamine H2-receptor antagonists.
    Federation proceedings, 1976, Volume: 35, Issue:8

    Topics: Animals; Anti-Inflammatory Agents; Burimamide; Catecholamines; Dogs; Female; Gastric Mucosa; Guinea Pigs; Histamine; Histamine H1 Antagonists; Metiamide; Muscle Contraction; Myocardial Contraction; Rats; Receptors, Drug; Thiourea; Uterus

1976
Blockade by burimamide of the restorative effect of histamine in tetrodotoxin-treated heart preparations.
    British journal of pharmacology, 1976, Volume: 57, Issue:2

    Topics: Action Potentials; Animals; Burimamide; Edetic Acid; Gallopamil; Guinea Pigs; Heart; Histamine; Histamine H1 Antagonists; In Vitro Techniques; Tetrodotoxin; Thiourea

1976
A quantitative study of metiamide, a histamine H2-antagonist, on the isolated whole rat stomach.
    The Journal of physiology, 1976, Volume: 258, Issue:2

    Topics: Animals; Dose-Response Relationship, Drug; Female; Gastric Juice; Gastric Mucosa; Histamine; Histamine H1 Antagonists; In Vitro Techniques; Male; Metiamide; Rats; Stomach; Thiourea

1976
Effect of the histamine (H2) inhibitor metiamide on histamine-stimulated bile flow in dogs.
    The American journal of physiology, 1976, Volume: 231, Issue:2

    Topics: Animals; Bile; Binding, Competitive; Dogs; Dose-Response Relationship, Drug; Duodenum; Gastric Juice; Histamine; Histamine H1 Antagonists; Hydrogen-Ion Concentration; Metiamide; Thiourea

1976
Antiadrenergic actions of metiamide in cat thermoregulatory mechanisms.
    Proceedings of the Western Pharmacology Society, 1976, Volume: 19

    Topics: Animals; Body Temperature Regulation; Cats; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Metiamide; Morphine; Norepinephrine; Prostaglandins E; Sympatholytics; Thiourea

1976
Effects of the H1-antagonist promethazine and the H2-antagonist burimamide on chronotropic, inotropic and coronary vascular responses to histamine in isolated perfused guinea-pig hearts.
    Agents and actions, 1976, Volume: 6, Issue:6

    Topics: Animals; Burimamide; Coronary Circulation; Drug Interactions; Guinea Pigs; Heart Rate; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Myocardial Contraction; Promethazine; Stimulation, Chemical; Thiourea

1976
Analysis of the actions of cimetidine and metiamide on gastric acid secretion in the isolated guinea pig gastric mucosa.
    Naunyn-Schmiedeberg's archives of pharmacology, 1977, Volume: 296, Issue:2

    Topics: Animals; Female; Gastric Juice; Gastric Mucosa; Guanidines; Guinea Pigs; Histamine; Histamine H2 Antagonists; Imidazoles; In Vitro Techniques; Metiamide; Models, Biological; Receptors, Drug; Thiourea

1977
Investigation of the role of histamine H1-receptors in the control of gastric acid secretion in the rat.
    The Journal of pharmacy and pharmacology, 1978, Volume: 30, Issue:4

    Topics: Animals; Dose-Response Relationship, Drug; Ethylamines; Female; Gastric Juice; Histamine; Pyrilamine; Rats; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1978
Pathogenesis of duodenal ulceration produced by cysteamine or propionitrile: influence of vagotomy, sympathectomy, histamine depletion, H-2 receptor antagonists and hormones.
    Digestive diseases and sciences, 1979, Volume: 24, Issue:6

    Topics: Adrenalectomy; Animals; Castration; Cimetidine; Cysteamine; Disease Models, Animal; Duodenal Ulcer; Gastric Juice; Guanidines; Histamine; Histamine H2 Antagonists; Hypophysectomy; Metiamide; Nitriles; Rats; Sympathectomy; Thiourea; Thyroidectomy; Vagotomy

1979
The effect of histamine, metiamide and cystic fibrosis factor on the electrophysiological properties of the frog's gastric mucosa [proceedings].
    The Journal of physiology, 1979, Volume: 291

    Topics: Animals; Anura; Biological Transport, Active; Chlorides; Cystic Fibrosis; Gastric Mucosa; Histamine; Humans; Hydrogen-Ion Concentration; In Vitro Techniques; Membrane Potentials; Metiamide; Thiourea

1979
ICI 125,211: a new gastric antisecretory agent acting on histamine H2-receptors.
    Life sciences, 1979, Dec-03, Volume: 25, Issue:23

    Topics: Animals; Cimetidine; Dogs; Female; Gastric Mucosa; Guanidines; Guinea Pigs; Heart; Heart Rate; Histamine; Histamine H2 Antagonists; Myocardial Contraction; Thiazoles; Thiourea; Time Factors

1979
Control of histamine release: effects of various conditions on rate of release and rate of cell desensitization.
    Journal of immunology (Baltimore, Md. : 1950), 1975, Volume: 114, Issue:3

    Topics: Desensitization, Immunologic; Dextrans; Histamine; Histamine Release; Immune Sera; Immunization; Immunodiffusion; Indomethacin; Mast Cells; Ovalbumin; Passive Cutaneous Anaphylaxis; Pertussis Vaccine; Phenoxybenzamine; Phosphatidylserines; Promethazine; Temperature; Thiourea

1975
Elicidation by a H-2-receptor antagonist of the significance of mucosal histamine mobilization in exciting acid secretion.
    The Journal of physiology, 1975, Volume: 244, Issue:2

    Topics: Animals; Cholecystokinin; Deoxyglucose; Eating; Female; Gastric Juice; Gastric Mucosa; Histamine; Histamine Release; Methacholine Compounds; Metiamide; Pentagastrin; Peptides; Rats; Receptors, Drug; Secretory Rate; Thiourea; Time Factors

1975
Metiamide: an antagonist of histamine-stimulated gastric acid secretion.
    Annals of surgery, 1975, Volume: 182, Issue:5

    Topics: Animals; Deoxyglucose; Dogs; Eating; Gastric Juice; Histamine; Histamine H1 Antagonists; Histamine Release; Metiamide; Pentagastrin; Pepsin A; Pilocarpine; Secretin; Stomach; Thiourea

1975
The effects of metiamide and H1 receptor blocking agents on anaphylactic response in guinea-pigs.
    Agents and actions, 1979, Volume: 9, Issue:5-6

    Topics: Airway Resistance; Anaphylaxis; Animals; Blood Pressure; Bronchial Spasm; Guinea Pigs; Heart Rate; Histamine; Histamine H1 Antagonists; Histamine Release; Lung; Male; Metiamide; Thiourea

1979
[Action of some H2 receptor agonists on the cardiac atria of the guinea pig].
    Bollettino della Societa italiana di biologia sperimentale, 1978, May-30, Volume: 54, Issue:10

    Topics: Animals; Guinea Pigs; Heart Atria; Heart Rate; Histamine; Receptors, Histamine; Receptors, Histamine H2; Thiourea

1978
Bronchodilator activity of dimaprit in the guinea pig in vitro and in vivo.
    European journal of pharmacology, 1979, May-01, Volume: 55, Issue:3

    Topics: Airway Resistance; Animals; Bronchodilator Agents; Guinea Pigs; Histamine; In Vitro Techniques; Lung Compliance; Male; Phenethylamines; Receptors, Histamine; Receptors, Histamine H2; Thiourea; Trachea

1979
[Histamine receptors in the human saphenous vein].
    Bollettino della Societa italiana di biologia sperimentale, 1978, Oct-15, Volume: 54, Issue:19

    Topics: Cimetidine; Histamine; Humans; Pheniramine; Receptors, Histamine; Receptors, Histamine H1; Saphenous Vein; Thiourea

1978
Histamine H2-receptors in guinea pig peripheral airway smooth muscle.
    Life sciences, 1979, Aug-06, Volume: 25, Issue:6

    Topics: Animals; Chlorpheniramine; Drug Synergism; Guinea Pigs; Histamine; Lung; Male; Metiamide; Muscle Contraction; Muscle, Smooth; Propranolol; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1979
Dimaprit-induced hypothermia in normal rats: its attenuation by cimetidine and by tricyclic antidepressant drugs.
    Neuropharmacology, 1979, Volume: 18, Issue:10

    Topics: Animals; Antidepressive Agents, Tricyclic; Body Temperature; Cimetidine; Female; Fenclonine; Guanidines; Histamine; Metergoline; Methylhistamines; Rats; Receptors, Histamine; Receptors, Histamine H2; Thiourea; Time Factors

1979
Inhibition of histamine methylation in vivo by the dimaprit analog, SKF Compound 91488.
    Agents and actions, 1979, Volume: 9, Issue:5-6

    Topics: Amine Oxidase (Copper-Containing); Animals; Brain; Dimaprit; Guanidines; Histamine; Histamine N-Methyltransferase; Kidney; Male; Methylation; Methyltransferases; Mice; Rats; Thiourea

1979
A comparative study with impromidine (SKF 92676), a potent agonist for histamine H2-receptors.
    Agents and actions, 1979, Volume: 9, Issue:5-6

    Topics: Airway Resistance; Animals; Blood Pressure; Cats; Dimaprit; Diuresis; Drug Interactions; Female; Guanidines; Guinea Pigs; Histamine; Imidazoles; Impromidine; In Vitro Techniques; Kidney; Lung; Male; Metiamide; Rabbits; Receptors, Histamine; Receptors, Histamine H2; Tachyphylaxis; Thiourea; Trachea

1979
Comparison of the effects of histamine and tolazoline on adenylate cyclase activity from guinea pig heart.
    Journal of medicinal chemistry, 1975, Volume: 18, Issue:1

    Topics: Adenosine Triphosphatases; Adenylyl Cyclases; Animals; Benzyl Compounds; Cyclic AMP; Dose-Response Relationship, Drug; Drug Synergism; Ethylenediamines; Guinea Pigs; Heart; Histamine; Imidazoles; In Vitro Techniques; Isoproterenol; Myocardium; Phosphoric Diester Hydrolases; Pyridines; Receptors, Drug; Stimulation, Chemical; Thiourea; Tolazoline

1975
On the specificity of histamine H2-receptor antagonists in the rat cerebral cortex.
    Canadian journal of physiology and pharmacology, 1975, Volume: 53, Issue:6

    Topics: Acetylcholine; Animals; Biogenic Amines; Burimamide; Cerebral Cortex; Cyclic AMP; Histamine; In Vitro Techniques; Male; Metiamide; Neurons; Rats; Receptors, Drug; Thiourea

1975
Effects of common inhibitors of gastric acid secretion on secretagogue-induced respiration and aminopyrine accumulation in isolated gastric glands.
    Biochimica et biophysica acta, 1977, Jan-04, Volume: 464, Issue:1

    Topics: Aminopyrine; Animals; Atropine; Biological Transport; Bucladesine; Burimamide; Gastric Juice; Gastric Mucosa; Histamine; In Vitro Techniques; Kinetics; Oxygen Consumption; Rabbits; Thiocyanates; Thiourea

1977
The in vitro effects of histamine and metiamide on neutrophil motility and their relationship to intracellular cyclic nucleotide levels.
    Journal of immunology (Baltimore, Md. : 1950), 1977, Volume: 118, Issue:5

    Topics: Cell Movement; Chemotaxis, Leukocyte; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Histamine; Levamisole; Metiamide; Neutrophils; Receptors, Histamine; Thiourea

1977
Role of H2-receptor antagonists in the feedback of histamine [proceedings].
    Agents and actions, 1977, Volume: 7, Issue:1

    Topics: Amine Oxidase (Copper-Containing); Anaphylaxis; Animals; Burimamide; Cyclic AMP; Feedback; Guinea Pigs; Histamine; Lung; Metiamide; Pyridines; Pyrilamine; Thiourea

1977
Influence of metiamide on "alkaline tide".
    Surgical forum, 1978, Volume: 29

    Topics: Animals; Bicarbonates; Dogs; Gastric Mucosa; Histamine; Metiamide; Protons; Thiourea

1978
A pharmacologic comparison of histamine receptors in isolated extracranial and intracranial arteries in vitro.
    Neurology, 1975, Volume: 25, Issue:3

    Topics: Animals; Arteries; Benzyl Compounds; Binding, Competitive; Cats; Cerebrovascular Circulation; Chlorpheniramine; Dilatation; Ethylenediamines; Female; Histamine; Histamine H1 Antagonists; In Vitro Techniques; Male; Pyridines; Receptors, Adrenergic; Serotonin; Thiourea; Vasomotor System

1975
Antagonism of tolazoline by histamine H2-receptor blockers.
    Nature, 1975, Feb-13, Volume: 253, Issue:5492

    Topics: Animals; Dogs; Dose-Response Relationship, Drug; Gastric Juice; Gastric Mucosa; Guinea Pigs; Heart Rate; Histamine; Hydrogen-Ion Concentration; Imidazoles; Kinetics; Male; Receptors, Drug; Stimulation, Chemical; Sulfides; Thiourea; Tolazoline

1975
Occurrence of H2-receptors for histamine in the guinea-pig intestine.
    Biochemical pharmacology, 1975, Jun-15, Volume: 24, Issue:11-12

    Topics: Amine Oxidase (Copper-Containing); Animals; Binding Sites; Burimamide; Dose-Response Relationship, Drug; Drug Synergism; Duodenum; Guanidines; Guinea Pigs; Histamine; Histamine H1 Antagonists; Ileum; In Vitro Techniques; Intestinal Mucosa; Mathematics; Thiourea

1975
Effect of the H2-receptor antagonists (burimamide and metiamide) on gastric secretion stimulated by histamine and its methyl derivatives.
    The Journal of pharmacology and experimental therapeutics, 1975, Volume: 193, Issue:2

    Topics: Animals; Burimamide; Dogs; Female; Gastric Juice; Gastric Mucosa; Histamine; Histamine H1 Antagonists; Metiamide; Stimulation, Chemical; Stomach; Thiourea; Time Factors; Vagus Nerve

1975
Relations between the effects of histamine, pheniramin and metiamide on spontaneous motility and the formation of cyclic AMP in the isolated rat uterus.
    Naunyn-Schmiedeberg's archives of pharmacology, 1975, Volume: 287, Issue:3

    Topics: Animals; Cyclic AMP; Female; Histamine; Histamine H1 Antagonists; In Vitro Techniques; Metiamide; Pheniramine; Rats; Receptors, Drug; Thiourea; Uterine Contraction; Uterus

1975
The effects of somatostatin and metiamide on tachyphylaxis of pentagastrin stimulated gastric acid and pepsin secretion in the conscious cat.
    The Journal of physiology, 1977, Volume: 266, Issue:3

    Topics: Animals; Cats; Depression, Chemical; Gastric Juice; Gastric Mucosa; Histamine; Metiamide; Pentagastrin; Pepsin A; Receptors, Histamine H2; Somatostatin; Tachyphylaxis; Thiourea

1977
[Analysis of regulation of gastric secretion].
    Fiziologicheskii zhurnal SSSR imeni I. M. Sechenova, 1977, Volume: 63, Issue:5

    Topics: Animals; Burimamide; Dogs; Drug Interactions; Gastric Juice; Gastric Mucosa; Gastrins; Histamine; Male; Pepsin A; Reaction Time; Receptors, Drug; Serotonin; Thiourea

1977
The effect of prostaglandin E2, 15-methyl prostaglandin E2, and metiamide on established canine gastric mucosal barrier damage.
    Surgery, 1979, Volume: 85, Issue:3

    Topics: Administration, Topical; Animals; Aspirin; Cell Membrane Permeability; Disease Models, Animal; Dogs; Female; Gastric Juice; Gastric Mucosa; Histamine; Injections, Intravenous; Metiamide; Prostaglandins E, Synthetic; Regression Analysis; Secretory Rate; Stimulation, Chemical; Stomach Ulcer; Thiourea

1979
The role of histamine H1- and H2-receptors in the generation of thromboxane A2 in perfused guinea-pig lungs.
    British journal of pharmacology, 1979, Volume: 65, Issue:4

    Topics: Adenosine Triphosphate; Animals; Guinea Pigs; Histamine; In Vitro Techniques; Lung; Male; Methylhistamines; Prostaglandins; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea; Thromboxane A2; Thromboxanes

1979
Characteristics of H2-receptor blockade in the canine mesenteric circulation.
    The Journal of surgical research, 1979, Volume: 27, Issue:2

    Topics: Animals; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Female; Histamine; Male; Mesenteric Arteries; Metiamide; Receptors, Histamine; Regional Blood Flow; Thiourea; Vasodilation

1979
Effects of alkyl analogs of histamine and metiamide on gastric acid secretion.
    European journal of pharmacology, 1979, Jul-15, Volume: 57, Issue:1

    Topics: Animals; Cats; Female; Gastric Juice; Histamine; Male; Methylhistamines; Metiamide; Thiourea

1979
Influence of metiamide and atropine on pepsinogen secretion in the conscious rat.
    Experientia, 1977, Dec-15, Volume: 33, Issue:12

    Topics: Animals; Atropine; Carbachol; Gastric Acidity Determination; Gastric Fistula; Histamine; Male; Metiamide; Pentagastrin; Pepsinogens; Rats; Thiourea

1977
[Histamine receptors in the guinea pig papillary muscle].
    Bollettino della Societa italiana di biologia sperimentale, 1977, Dec-15, Volume: 53, Issue:23

    Topics: Animals; Cimetidine; Epinephrine; Female; Guinea Pigs; Histamine; Male; Papillary Muscles; Pyrilamine; Receptors, Histamine; Thiazoles; Thiourea

1977
The effects of stimulants and inhibitors of histamine receptors on acid secretion from guinea pig gastric fundus.
    European journal of pharmacology, 1978, Apr-01, Volume: 48, Issue:3

    Topics: Animals; Cimetidine; Female; Gastric Mucosa; Guinea Pigs; Histamine; In Vitro Techniques; Male; Methylhistamines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea; Time Factors

1978
Stimulation of cell proliferation by histamine H2 receptors in dimethylhdrazine-induced adenocarcinomata.
    Cell biology international reports, 1978, Volume: 2, Issue:2

    Topics: Adenocarcinoma; Animals; Cell Division; Cimetidine; Colon; Colonic Neoplasms; Dimethylhydrazines; Histamine; Intestinal Mucosa; Male; Metiamide; Pyrilamine; Rats; Receptors, Histamine; Receptors, Histamine H2; Stimulation, Chemical; Thiourea

1978
Regulation of histamine synthesis: metiamide-induced synthesis of histamine in the rat stomach and the effect of histidine decarboxylase inhibitors on the elevated 14C-histamine level and histidine decarboxylase activity [proceedings].
    Agents and actions, 1978, Volume: 8, Issue:4

    Topics: Animals; Carboxy-Lyases; Gastric Mucosa; Histamine; Histidine Decarboxylase; Male; Metiamide; Rats; Stomach; Thiourea

1978
Effect of dimaprit on gastric acid secretion in conscious cats.
    Agents and actions, 1978, Volume: 8, Issue:5

    Topics: Animals; Cats; Cimetidine; Gastric Juice; Histamine; Methylhistamines; Pentagastrin; Pyrilamine; Receptors, Histamine H2; Thiourea; Time Factors

1978
Renal histamine H1 and H2 receptors: characterization and functional significance.
    The American journal of physiology, 1978, Volume: 235, Issue:6

    Topics: Animals; Cimetidine; Dogs; Ethylamines; Female; Histamine; Kidney; Male; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Regional Blood Flow; Thiourea; Tripelennamine; Vasodilation

1978
Stimulation of gastric acid secretion by dimaprit in unanesthetized rats.
    Agents and actions, 1978, Volume: 8, Issue:6

    Topics: Animals; Dose-Response Relationship, Drug; Gastric Juice; Histamine; Male; Pentagastrin; Rats; Receptors, Histamine; Receptors, Histamine H2; Thiourea

1978
Inhibition by metiamide of secretagogue-induced gastric acid secretion in the conscious Heidenhain pouch rat.
    The Journal of physiology, 1978, Volume: 285

    Topics: Animals; Bethanechol Compounds; Female; Gastric Juice; Gastric Mucosa; Histamine; Metiamide; Pentagastrin; Rats; Secretory Rate; Stimulation, Chemical; Stomach; Thiourea

1978
Inhibition of basal and stimulated gastric H+ and pepsin secretion in duodenal ulcer patients by metiamide, an H-2 histamine antagonist.
    The American journal of digestive diseases, 1976, Volume: 21, Issue:7

    Topics: Adolescent; Adult; Duodenal Ulcer; Female; Gastric Juice; Histamine; Humans; Hypoglycemia; Insulin; Male; Metiamide; Middle Aged; Pepsin A; Thiourea

1976
Further studies on histamine in spinal cord injury and post traumatic hyperemia.
    Surgical neurology, 1976, Volume: 5, Issue:2

    Topics: Animals; Chlorpheniramine; Haplorhini; Histamine; Hyperemia; Macaca mulatta; Regional Blood Flow; Spinal Cord; Spinal Cord Injuries; Thiourea

1976
Histamine receptors in the coronary circulation of the dog. Effects of mepyramine and metiamide on responses to histamine infusions.
    Circulation research, 1977, Volume: 40, Issue:6

    Topics: Animals; Coronary Circulation; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Histamine; Injections, Intra-Arterial; Metiamide; Myocardial Contraction; Pyridines; Pyrilamine; Receptors, Histamine; Thiourea; Time Factors

1977
Dimaprit, (S-[3-(N,N-dimethylamino)propyl]isothiourea). A highly specific histamine H2-receptor agonist. Part 2. Structure-activity considerations.
    Agents and actions, 1977, Volume: 7, Issue:1

    Topics: Histamine; Isomerism; Receptors, Histamine; Receptors, Histamine H2; Structure-Activity Relationship; Thiourea

1977
Histamine has no influence on the oxidative properties of ceruloplasmin.
    Biochemical pharmacology, 1977, May-15, Volume: 26, Issue:10

    Topics: Burimamide; Ceruloplasmin; Chemical Phenomena; Chemistry; Chlorides; Dianisidine; Histamine; Humans; In Vitro Techniques; Metiamide; Oxidation-Reduction; Phenylenediamines; Phosphates; Sodium Chloride; Thiourea

1977
Resistance to blockade of vasodepressor responses to tolazoline by chlorpheniramine and metiamide in rabbit hindlimb vasculature.
    Research communications in chemical pathology and pharmacology, 1977, Volume: 16, Issue:4

    Topics: Acetylcholine; Animals; Atropine; Blood Pressure; Chlorpheniramine; Drug Interactions; Hindlimb; Histamine; Isoproterenol; Metiamide; Propranolol; Rabbits; Regional Blood Flow; Thiourea; Tolazoline; Vasomotor System

1977
Influence of H1- and H2-receptor antagonists on the circulatory system and on the endogenous plasma histamine concentrations in dogs.
    Agents and actions, 1977, Volume: 7, Issue:1

    Topics: Animals; Blood Pressure; Burimamide; Dimethindene; Dogs; Female; Histamine; Male; Mesenteric Arteries; Respiration; Thiourea; Vascular Resistance

1977
The effect of metiamide in in vitro and in vivo canine models of type I hypersensitivity reactions.
    European journal of pharmacology, 1977, Jul-01, Volume: 44, Issue:1

    Topics: Airway Resistance; Animals; Ascaris; Asthma; Dogs; Histamine; Hypersensitivity, Immediate; In Vitro Techniques; Lung; Male; Metiamide; Thiourea; Time Factors

1977
Absence of blocking effect of burimamide and metiamide on positive chronotropic and inotropic responses to histamine in isolated dog atrium.
    Japanese journal of pharmacology, 1977, Volume: 27, Issue:2

    Topics: Alprenolol; Animals; Burimamide; Depression, Chemical; Desipramine; Diphenhydramine; Dogs; Dose-Response Relationship, Drug; Heart Atria; Heart Rate; Histamine; Histamine Antagonists; In Vitro Techniques; Metiamide; Myocardial Contraction; Norepinephrine; Receptors, Histamine; Stimulation, Chemical; Tetrodotoxin; Thiourea; Tripelennamine

1977
Histamine, histamine antagonists and regional blood flow.
    European journal of pharmacology, 1977, Aug-15, Volume: 44, Issue:4

    Topics: Animals; Blood Pressure; Cats; Drug Interactions; Female; Hemodynamics; Histamine; Male; Metiamide; Pyridines; Pyrilamine; Regional Blood Flow; Thiourea; Vascular Resistance

1977
Effect of the H2-receptor antagonist metiamide on carbachol- and histamine-induced gastric acid secretion in the Atlantic cod,Gadus morhua.
    Acta physiologica Scandinavica, 1976, Volume: 97, Issue:2

    Topics: Animals; Carbachol; Drinking; Drug Interactions; Fishes; Gastric Juice; Histamine; Metiamide; Secretory Rate; Sensory Receptor Cells; Thiourea

1976
Effects of metiamide on gastric acid hypersecretion, steatorrhea, and bone-marrow function in a patient with systemic mastocytosis.
    The New England journal of medicine, 1976, Nov-18, Volume: 295, Issue:21

    Topics: Agranulocytosis; Bone Marrow; Celiac Disease; Diarrhea; Gastric Juice; Histamine; Humans; Male; Metiamide; Middle Aged; Secretory Rate; Thiourea; Urticaria Pigmentosa

1976
In vitro anaphylaxis in guinea-pig skin: amplification by burimamide.
    The Journal of investigative dermatology, 1976, Volume: 67, Issue:6

    Topics: Anaphylaxis; Animals; Brocresine; Burimamide; Guinea Pigs; Histamine; Histidine Decarboxylase; In Vitro Techniques; Male; Skin; Thiourea

1976
Adenylate cyclase of the dog gastric mucosa: stimulation by histamine and inhibition by metiamide.
    Naunyn-Schmiedeberg's archives of pharmacology, 1976, Volume: 294, Issue:2

    Topics: Adenylyl Cyclases; Animals; Dogs; Female; Gastric Mucosa; Histamine; In Vitro Techniques; Metiamide; Pyrilamine; Thiourea

1976
Action of somatostatin and metiamide on gastric acid secretion from isolated bullfrog gastric mucosa.
    Research communications in chemical pathology and pharmacology, 1976, Volume: 13, Issue:1

    Topics: Animals; Depression, Chemical; Gastric Juice; Gastric Mucosa; Histamine; In Vitro Techniques; Metiamide; Pentagastrin; Rana catesbeiana; Somatostatin; Thiourea

1976
[Effect of histamine on the transport of non-electrolytes across the gastric mucosa of Rana esculenta].
    Bollettino della Societa italiana di biologia sperimentale, 1976, Apr-30, Volume: 52, Issue:7-8

    Topics: Animals; Biological Transport; Gastric Mucosa; Histamine; Rana esculenta; Thiourea

1976
Electrophysiological effects of burimamide and 16,16-dimethyl prostaglandin E2 on the canine gastric mucosa.
    Gastroenterology, 1975, Volume: 68, Issue:6

    Topics: Animals; Biological Transport, Active; Burimamide; Chlorides; Chlorine; Dogs; Electrophysiology; Female; Gastric Juice; Gastric Mucosa; Histamine; In Vitro Techniques; Male; Membrane Potentials; Prostaglandins E; Radioisotopes; Sodium; Sodium Radioisotopes; Thiourea

1975
An indirect sympathomimetic effect of burimamide on kitten isolated atria.
    British journal of pharmacology, 1975, Volume: 53, Issue:4

    Topics: Animals; Burimamide; Cats; Cocaine; Female; Heart Atria; Heart Rate; Histamine; In Vitro Techniques; Male; Metiamide; Myocardial Contraction; Norepinephrine; Propranolol; Reserpine; Stimulation, Chemical; Sympathomimetics; Thiourea; Tyramine

1975
Effects of metiamide on distribution of 14C-histamine in aortic smooth muscle.
    Archives internationales de pharmacodynamie et de therapie, 1975, Volume: 218, Issue:2

    Topics: Animals; Aorta, Thoracic; Female; Histamine; In Vitro Techniques; Male; Metiamide; Muscle Contraction; Muscle, Smooth; Rabbits; Thiourea; Time Factors

1975
Letter: H2-receptor antagonists for Z-E syndrome.
    The New England journal of medicine, 1976, Apr-29, Volume: 294, Issue:18

    Topics: Adult; Histamine; Humans; Male; Metiamide; Receptors, Drug; Thiourea; Zollinger-Ellison Syndrome

1976
Histamine increases cytosolic Ca2+ in HL-60 promyelocytes predominantly via H2 receptors with an unique agonist/antagonist profile and induces functional differentiation.
    Molecular pharmacology, 1992, Volume: 42, Issue:2

    Topics: Adenosine Triphosphate; Calcium; Cations; Cell Differentiation; Cyclic AMP; Cytosol; Dimaprit; Famotidine; Guanidines; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Imidazoles; Impromidine; Ion Channels; Leukemia, Experimental; Leukemia, Promyelocytic, Acute; Phosphatidylinositols; Receptors, Histamine H2; Stimulation, Chemical; Thiourea; Tumor Cells, Cultured

1992
A theoretical study concerning the mode of interaction of the histamine H2-agonist dimaprit.
    Journal of molecular graphics, 1992, Volume: 10, Issue:2

    Topics: Computer Simulation; Dimaprit; Electrophysiology; Histamine; Methylation; Models, Molecular; Molecular Conformation; Receptors, Histamine H2; Thiourea

1992
Effect of short-term treatment with gastrin and related peptides on gastrointestinal histamine H2-receptors.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:2

    Topics: Adenylyl Cyclases; Animals; Cimetidine; Digestive System; Dimaprit; Gastrins; Guinea Pigs; Histamine; In Vitro Techniques; Male; Pentagastrin; Receptors, Histamine H2; Sincalide; Thiourea

1992
Histamine receptors on human isolated pulmonary arterial muscle preparations: effects of endothelial cell removal and nitric oxide inhibitors.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 260, Issue:2

    Topics: Arginine; Burimamide; Chlorpheniramine; Cimetidine; Dimaprit; Endothelium, Vascular; Histamine; Humans; In Vitro Techniques; Indomethacin; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide; Nitroarginine; omega-N-Methylarginine; Pulmonary Artery; Receptors, Histamine; Serotonin; Tetraethylammonium; Tetraethylammonium Compounds; Thiourea

1992
Histamine N-methyltransferase controls the contractile response of guinea pig trachea to histamine.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 261, Issue:3

    Topics: Animals; Dimaprit; Dose-Response Relationship, Drug; Guanidines; Guinea Pigs; Histamine; Histamine N-Methyltransferase; Male; Muscle Contraction; Muscle, Smooth; Thiourea; Trachea

1992
Effects of histamine H1-, H2- and H3-receptor selective drugs on the mechanical activity of guinea-pig small and large intestine.
    British journal of pharmacology, 1991, Volume: 102, Issue:1

    Topics: Animals; Atropine; Dimaprit; Electric Stimulation; Guanidines; Guinea Pigs; Histamine; In Vitro Techniques; Intestine, Large; Intestine, Small; Male; Methacholine Compounds; Muscle Contraction; Muscle, Smooth; Pinacidil; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Stereoisomerism; Tetraethylammonium Compounds; Thiourea

1991
Theoretical analysis of the activity of dimaprit derivatives on the H2-receptor.
    Agents and actions. Supplements, 1991, Volume: 33

    Topics: Chemical Phenomena; Chemistry, Physical; Dimaprit; Electrochemistry; Histamine; Models, Molecular; Protons; Receptors, Histamine H2; Software; Thermodynamics; Thiourea

1991
Involvement of histamine in the mediation of the stress-induced release of alpha-melanocyte-stimulating hormone in male rats.
    Neuroendocrinology, 1991, Volume: 54, Issue:6

    Topics: Adrenocorticotropic Hormone; alpha-MSH; Animals; Bromocriptine; Dimaprit; Histamine; Male; Methylhistidines; Propranolol; Rats; Rats, Inbred Strains; Stress, Physiological; Thiourea

1991
Cyclic AMP generating systems in vertebrate retina: effects of histamine and an established retinal modulator, dopamine.
    Agents and actions, 1991, Volume: 33, Issue:1-2

    Topics: Adenylyl Cyclases; Animals; Cerebral Cortex; Chickens; Cimetidine; Colforsin; Cyclic AMP; Dimaprit; Dopamine; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistamines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Retina; Thiazoles; Thiourea

1991
Mechanism of action of H2-antagonists on histamine- or dimaprit-stimulated H2-receptors of spontaneously beating guinea-pig atrium.
    Agents and actions, 1990, Volume: 31, Issue:1-2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Cimetidine; Dimaprit; Famotidine; Female; Guinea Pigs; Heart; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Radioligand Assay; Ranitidine; Receptors, Histamine H2; Thiourea

1990
Influence of the endothelium on histamine-induced relaxation of rat middle cerebral arteries in vitro.
    Journal of cardiovascular pharmacology, 1991, Volume: 17, Issue:1

    Topics: Animals; Cerebral Arteries; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Histamine; Histamine H2 Antagonists; Kinetics; Male; Methylhistamines; Muscle Relaxation; Muscle, Smooth, Vascular; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H2; Receptors, Histamine H3; Thiourea

1991
Effects of thiourea tolerance on plasma histamine, and lung vascular permeability.
    Archives of toxicology, 1991, Volume: 65, Issue:7

    Topics: Animals; Capillary Permeability; Drug Tolerance; Histamine; Lung; Male; Pulmonary Edema; Rats; Rats, Inbred Strains; Thiourea

1991
Histamine induces endothelium-dependent relaxation of bovine retinal arteries.
    Investigative ophthalmology & visual science, 1991, Volume: 32, Issue:1

    Topics: Acetylcholine; Animals; Cattle; Cimetidine; Dimaprit; Endothelium, Vascular; Histamine; Muscle Relaxation; Pyridines; Pyrilamine; Receptors, Histamine; Retinal Artery; Tachyphylaxis; Thiourea

1991
Effect of histamine on human lymphocyte aggregation.
    Thrombosis research, 1991, Jan-15, Volume: 61, Issue:2

    Topics: Adult; Arachidonic Acid; Arachidonic Acids; Cell Aggregation; Dimaprit; Endothelium, Vascular; Histamine; Humans; In Vitro Techniques; Receptors, Histamine; T-Lymphocytes; Thiourea

1991
Vasomotor effect of histamine on pig and cattle coronary artery in vitro.
    Japanese journal of pharmacology, 1991, Volume: 55, Issue:3

    Topics: Animals; Cattle; Cimetidine; Coronary Vessels; Dimaprit; Diphenhydramine; Endothelium, Vascular; Histamine; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Swine; Thiourea

1991
Effect of histamine on tracheal mucosal perfusion, water content and airway smooth muscle in sheep.
    Respiration physiology, 1991, Volume: 84, Issue:2

    Topics: Animals; Atropine; Chlorpheniramine; Dimaprit; Female; Histamine; Lung Volume Measurements; Metiamide; Mucous Membrane; Muscle, Smooth; Receptors, Cholinergic; Receptors, Histamine H1; Receptors, Histamine H2; Regional Blood Flow; Sheep; Thiourea; Trachea; Water

1991
Involvement of calcium ions in the modulation of electrically-induced rat vas deferens contractions by histaminergic drugs.
    General pharmacology, 1991, Volume: 22, Issue:4

    Topics: Animals; Calcium; Cimetidine; Dimaprit; Diphenhydramine; Electric Stimulation; Histamine; In Vitro Techniques; Male; Muscle Contraction; Rats; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea; Vas Deferens; Verapamil

1991
GM-CSF in association with IL-1 triggers day-8 CFU-S into cell cycle: role of histamine.
    Journal of cellular physiology, 1991, Volume: 149, Issue:1

    Topics: Animals; Bone Marrow Cells; Cell Cycle; Cells, Cultured; Dimaprit; Female; Granulocyte-Macrophage Colony-Stimulating Factor; Hematopoietic Stem Cells; Histamine; Interleukin-1; Male; Mice; Mice, Inbred C57BL; S Phase; Spleen; Thiourea

1991
Histamine-induced vasodilations mediated by H1- and H2-receptors in isolated rat common carotid arteries.
    Heart and vessels, 1991, Volume: 6, Issue:4

    Topics: Acetylcholine; Animals; Carotid Arteries; Cimetidine; Dimaprit; Diphenhydramine; Dose-Response Relationship, Drug; Female; Histamine; In Vitro Techniques; Male; Pyridines; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Receptors, Histamine H2; Saponins; Thiourea; Vasodilation

1991
Theoretical studies on the histamine H2 receptor: construction of a receptor model based on the structural properties of dimaprit and N alpha-guanylhistamine.
    Molecular pharmacology, 1991, Volume: 40, Issue:6

    Topics: Computer Simulation; Dimaprit; Histamine; Kinetics; Models, Chemical; Models, Molecular; Receptors, Histamine H2; Thiourea

1991
Effects of thiourea on pulmonary vascular permeability and on lung and plasma histamine levels in rats.
    Toxicology letters, 1991, Volume: 57, Issue:3

    Topics: Age Factors; Animals; Capillary Permeability; Histamine; Lung; Male; Pulmonary Edema; Rats; Rats, Inbred Strains; Thiourea

1991
New role for histamine in interleukin-3-induced proliferation of hematopoietic stem cells.
    Journal of cellular physiology, 1990, Volume: 143, Issue:2

    Topics: Animals; Bone Marrow Cells; Cell Division; Cetirizine; Colony-Forming Units Assay; Dimaprit; Hematopoiesis; Hematopoietic Stem Cells; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Hydroxyzine; Imidazoles; In Vitro Techniques; Interleukin-3; Methylhistidines; Mice; Mice, Inbred C57BL; Thiourea

1990
Histamine stimulation of mucociliary activity in the rabbit maxillary sinus.
    The Annals of otology, rhinology, and laryngology, 1990, Volume: 99, Issue:8

    Topics: Animals; Atropine; Cilia; Cimetidine; Dimaprit; Female; Histamine; Histamine H2 Antagonists; Male; Maxillary Sinus; Mucociliary Clearance; Pyrilamine; Rabbits; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Muscarinic; Thiourea

1990
Histamine and abnormal automaticity in barium- and strophanthidin-treated sheep Purkinje fibers.
    Agents and actions, 1990, Volume: 31, Issue:1-2

    Topics: Animals; Barium; Dimaprit; Electrophysiology; Heart; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Membrane Potentials; Methylhistamines; Purkinje Fibers; Sheep; Strophanthidin; Thiourea

1990
Central cardiovascular responses of histamine and homodimaprit in normal and hypophysectomized rats.
    Agents and actions, 1990, Volume: 31, Issue:3-4

    Topics: Animals; Blood Pressure; Brain; Dimaprit; Hexamethonium; Hexamethonium Compounds; Histamine; Hypophysectomy; Kinetics; Male; Rats; Rats, Inbred Strains; Thiourea; Vasopressins

1990
Mechanism of action of doxepin in the treatment of chronic urticaria.
    Fundamental & clinical pharmacology, 1990, Volume: 4, Issue:2

    Topics: Adult; Aged; Animals; Atropine; Carbachol; Chronic Disease; Dimaprit; Doxepin; Female; Gastric Juice; Guinea Pigs; Heart; Histamine; Humans; In Vitro Techniques; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Pylorus; Pyrilamine; Rats; Thiourea; Urticaria

1990
H2 receptors mediate cyclical chloride secretion in guinea pig distal colon.
    The American journal of physiology, 1990, Volume: 258, Issue:6 Pt 1

    Topics: Animals; Bumetanide; Chlorides; Cimetidine; Colon; Dimaprit; Guinea Pigs; Histamine; In Vitro Techniques; Intestinal Mucosa; Kinetics; Male; Muscle, Smooth; Pyrilamine; Receptors, Histamine H2; Tetrodotoxin; Thiourea

1990
Antagonistic effect of naloxone on the hypertensive response of intraventricularly administered histamine.
    Agents and actions, 1990, Volume: 30, Issue:1-2

    Topics: Animals; Blood Pressure; Cimetidine; Dimaprit; Hemodynamics; Histamine; In Vitro Techniques; Injections, Intraventricular; Male; Naloxone; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Thiourea

1990
Endothelium and mechanical responses of isolated monkey pulmonary veins to histamine.
    The American journal of physiology, 1990, Volume: 259, Issue:4 Pt 2

    Topics: Animals; Dimaprit; Endothelium, Vascular; Famotidine; Hemoglobins; Histamine; In Vitro Techniques; Macaca; Methylene Blue; Pulmonary Veins; Pyridines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea; Vasoconstriction; Vasodilation

1990
Role of histamine in natural killer cell-mediated resistance against tumor cells.
    Journal of immunology (Baltimore, Md. : 1950), 1990, Dec-15, Volume: 145, Issue:12

    Topics: Animals; Cytotoxicity, Immunologic; Dimaprit; Histamine; Immunity, Cellular; Interleukin-2; Killer Cells, Natural; Lung Neoplasms; Melanoma, Experimental; Mice; Mice, Inbred Strains; Neoplasm Metastasis; Neoplasms, Experimental; Ranitidine; Receptors, Histamine H2; Thiourea

1990
Identification of two H3-histamine receptor subtypes.
    Molecular pharmacology, 1990, Volume: 38, Issue:5

    Topics: Animals; Binding Sites; Binding, Competitive; Brain Chemistry; Burimamide; Dimaprit; Guanidines; Guanosine 5'-O-(3-Thiotriphosphate); Histamine; Imidazoles; Impromidine; Male; Methylhistamines; Piperidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H3; Thiourea; Tritium

1990
Electrophysiological actions of histamine and H1-, H2-receptor antagonists in cardiac tissue.
    Agents and actions, 1986, Volume: 18, Issue:1-2

    Topics: 1-Methyl-3-isobutylxanthine; Action Potentials; Animals; Atrioventricular Node; Dimaprit; Guinea Pigs; Heart; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Imidazoles; Impromidine; In Vitro Techniques; Male; Rabbits; Thiourea

1986
Electrophysiological characterization of histamine receptor subtypes in mammalian heart preparations.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 334, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Action Potentials; Animals; Atrioventricular Node; Cimetidine; Dimaprit; Dimethindene; Guinea Pigs; Heart; Histamine; Histamine H1 Antagonists; Imidazoles; Impromidine; In Vitro Techniques; Male; Myocardial Contraction; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1986
Comparison of the interaction of the histamine H2-agonists [correction of H2-antagonists] histamine and dimaprit.
    Progress in clinical and biological research, 1989, Volume: 289

    Topics: Computer Simulation; Dimaprit; Electrochemistry; Histamine; Models, Molecular; Molecular Conformation; Receptors, Histamine H2; Thiourea

1989
Histamine H2-receptor mediated positive dromotropic effect in the canine atrioventricular node.
    Japanese journal of pharmacology, 1989, Volume: 49, Issue:3

    Topics: Animals; Atenolol; Atrioventricular Node; Cimetidine; Dimaprit; Diphenhydramine; Dogs; Female; Heart Conduction System; Histamine; Male; Norepinephrine; Receptors, Histamine H2; Stimulation, Chemical; Thiourea

1989
Antagonistic action of naloxone on central histamine receptors-stimulated corticosterone secretion in rats under stress.
    Agents and actions, 1989, Volume: 28, Issue:3-4

    Topics: Animals; Cimetidine; Corticosterone; Dimaprit; Histamine; Male; Methylhistamines; Naloxone; Pituitary-Adrenal System; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Restraint, Physical; Stress, Physiological; Thiourea

1989
Responses to histamine and selective H2-receptor agonists in lung parenchymal strips from normal and sensitized guinea-pigs.
    Agents and actions, 1989, Volume: 28, Issue:1-2

    Topics: Animals; Benzimidazoles; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Guanidines; Guinea Pigs; Histamine; Imidazoles; Impromidine; Isoproterenol; Lung; Male; Methylhistamines; Muscle Contraction; Muscle, Smooth; Receptors, Histamine H2; Thiourea

1989
Involvement of different receptors in the central and peripheral effects of histamine on intestinal motility in the rat.
    The Journal of pharmacy and pharmacology, 1989, Volume: 41, Issue:8

    Topics: Animals; Chlorpheniramine; Dimaprit; Gastrointestinal Motility; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Injections, Intraperitoneal; Injections, Intraventricular; Male; Methylhistamines; Rats; Rats, Inbred Strains; Receptors, Histamine; Thiourea

1989
Histamine modulates contraction and cyclic nucleotides in cultured rat mesangial cells. Differential effects mediated by histamine H1 and H2 receptors.
    The Journal of clinical investigation, 1985, Volume: 75, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Cell Movement; Cells, Cultured; Cyclic AMP; Cyclic GMP; Dimaprit; Glomerular Mesangium; Histamine; Kidney Glomerulus; Male; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1985
Histamine receptors coupled to [3H]cAMP accumulation in brain: pharmacological characterization in a vesicular preparation of guinea pig cortex.
    Molecular pharmacology, 1988, Volume: 33, Issue:1

    Topics: Adenosine Deaminase; Animals; Cerebral Cortex; Chlorpheniramine; Cimetidine; Cyclic AMP; Dimaprit; Egtazic Acid; Guinea Pigs; Histamine; In Vitro Techniques; Receptors, Histamine; Subcellular Fractions; Thiourea

1988
Phosphoinositides and cicletanine.
    Drugs under experimental and clinical research, 1988, Volume: 14, Issue:2-3

    Topics: Angiotensin II; Animals; Antihypertensive Agents; Aorta, Thoracic; Cells, Cultured; Dimaprit; Diuretics; Guinea Pigs; Histamine; Male; Muscle, Smooth, Vascular; Phenylephrine; Phosphatidylinositols; Pyridines; Pyrilamine; Thiourea

1988
Distortion of H2-antagonist equilibrium constants by uptake in rabbit gastric mucosal cells.
    Pharmacology, 1985, Volume: 30, Issue:4

    Topics: Aminopyrine; Animals; Cimetidine; Cyclic AMP; Dimaprit; Gastric Acid; Gastric Mucosa; Guanidines; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Pyrimidinones; Rabbits; Radioisotopes; Rubidium; Thiadiazoles; Thiourea

1985
Histamine H2 receptor antagonists may modify dog intestinal motility independently of their primary action on the H2 receptors.
    Pharmacological research communications, 1985, Volume: 17, Issue:3

    Topics: Acetylcholine; Animals; Blood Pressure; Ceruletide; Cimetidine; Dimaprit; Dogs; Female; Gastrointestinal Motility; Histamine; Histamine H2 Antagonists; Ileum; Imidazoles; Impromidine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Physalaemin; Ranitidine; Receptors, Histamine; Receptors, Histamine H2; Thiourea

1985
Histamine H2-receptor antagonistic action of N-(3-[3-(1-piperidinylmethyl)phenoxy]propyl)acetoxyacetamide hydrochloride (TZU-0460).
    Arzneimittel-Forschung, 1985, Volume: 35, Issue:4

    Topics: Animals; Cimetidine; Dimaprit; Dogs; Female; Gastric Acid; Guinea Pigs; Heart Atria; Heart Rate; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Male; Muscle Relaxation; Piperidines; Rats; Thiourea; Uterus

1985
The determination of receptor constants for histamine H2-agonists in the guinea-pig isolated right atrium using an irreversible H2-antagonist.
    British journal of pharmacology, 1986, Volume: 87, Issue:1

    Topics: Animals; Dimaprit; Dose-Response Relationship, Drug; Female; Guanidines; Guinea Pigs; Heart Rate; Histamine; Histamine H2 Antagonists; Imidazoles; Impromidine; In Vitro Techniques; Male; Methylhistamines; Receptors, Adrenergic, beta; Receptors, Histamine; Receptors, Histamine H2; Thiazoles; Thiourea

1986
Studies on histaminergic compounds, III. Synthesis and histamine H2-activity of a series of corresponding histamine and dimaprit analogues.
    Archiv der Pharmazie, 1986, Volume: 319, Issue:7

    Topics: Animals; Dimaprit; Female; Guinea Pigs; Histamine; Histamine H2 Antagonists; Male; Structure-Activity Relationship; Thiourea

1986
Histamine and histamine receptors: behavioral thermoregulation in the salamander Necturus maculosus.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1986, Volume: 85, Issue:1

    Topics: Animals; Body Temperature Regulation; Cimetidine; Dimaprit; Histamine; Histidine; Necturus; Pyridines; Pyrilamine; Receptors, Histamine; Thiourea

1986
Histaminergic stimulation of prolactin secretion mediated via H1- or H2-receptors: dependence on routes of administration.
    Neuroendocrinology, 1986, Volume: 44, Issue:1

    Topics: Animals; Cimetidine; Dimaprit; Histamine; Histamine H1 Antagonists; Male; Methylhistamines; Pituitary Gland, Anterior; Prolactin; Pyrilamine; Pyrimidinones; Rats; Receptors, Histamine; Thiazoles; Thiourea

1986
[Effect of a new H2 receptor antagonist, famotidine, on gastric secretion].
    Bollettino della Societa italiana di biologia sperimentale, 1986, Sep-30, Volume: 62, Issue:9

    Topics: Animals; Cats; Dimaprit; Dose-Response Relationship, Drug; Famotidine; Gastric Mucosa; Histamine; Histamine H2 Antagonists; Ranitidine; Rats; Thiazoles; Thiourea

1986
Chronotropic cardiac effects of histamine in the conscious dog with chronic atrioventricular block: interactions with the autonomic nervous system.
    Agents and actions, 1986, Volume: 19, Issue:3-4

    Topics: Adrenergic beta-Antagonists; Animals; Atrioventricular Node; Autonomic Nervous System; Blood Pressure; Dimaprit; Dogs; Drug Interactions; Electrocardiography; Female; Heart Block; Heart Conduction System; Heart Rate; Histamine; Male; Parasympatholytics; Thiourea

1986
The antianaphylactic action of histamine H2-receptor agonists in the guinea-pig isolated heart.
    British journal of pharmacology, 1987, Volume: 90, Issue:3

    Topics: Anaphylaxis; Animals; Cimetidine; Dimaprit; Female; Guinea Pigs; Heart; Heart Rate; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Male; Myocardial Contraction; Pyridines; Thiourea

1987
Famotidine and ranitidine: any difference in the duration of action?
    Pharmacological research communications, 1987, Volume: 19, Issue:1

    Topics: Animals; Cats; Dimaprit; Famotidine; Gastric Acid; Gastric Juice; Histamine; Histamine H2 Antagonists; Ranitidine; Rats; Thiazoles; Thiourea; Time Factors

1987
H1- and H2-receptor characterization in the tracheal circulation of sheep.
    British journal of pharmacology, 1988, Volume: 95, Issue:2

    Topics: Animals; Dimaprit; Female; Histamine; Histamine H2 Antagonists; Male; Muscle Tonus; Receptors, Histamine H2; Regional Blood Flow; Sheep; Thiourea; Trachea; Vagotomy; Vascular Resistance

1988
The effects of histamine and some related compounds on conditioned avoidance response in rats.
    Life sciences, 1985, Nov-25, Volume: 37, Issue:21

    Topics: Acetylcholine; Animals; Avoidance Learning; Dimaprit; Diphenhydramine; Dose-Response Relationship, Drug; Histamine; Histamine Antagonists; Hypothalamus; Injections, Intraventricular; Kinetics; Male; Methylhistamines; Pyrilamine; Rats; Rats, Inbred Strains; Scopolamine; Thiazoles; Thiourea

1985
Conjunctival immediate hypersensitivity: re-evaluation of histamine involvement in the vasopermeability response.
    Investigative ophthalmology & visual science, 1986, Volume: 27, Issue:1

    Topics: Albumins; Animals; Capillary Permeability; Cimetidine; Conjunctiva; Dimaprit; Dose-Response Relationship, Drug; Drug Combinations; Eyelids; Guinea Pigs; Histamine; Histamine Antagonists; Hypersensitivity, Immediate; Imidazoles; Impromidine; Male; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1986
Effects of H1 and H2 receptor agonists on nonspecific proliferative response of human peripheral blood lymphocytes.
    International archives of allergy and applied immunology, 1986, Volume: 79, Issue:3

    Topics: Cimetidine; Dimaprit; Diphenhydramine; Dose-Response Relationship, Drug; Histamine; Humans; Immunosuppressive Agents; Lymphocyte Activation; Methylhistamines; Phytohemagglutinins; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1986
Metronidazole and 5-aminosalicylic acid enhance the contractile activity of histaminergic agonists on the guinea-pig isolated ileum.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 236, Issue:3

    Topics: Aminosalicylic Acids; Animals; Cimetidine; Computers; Dimaprit; Dose-Response Relationship, Drug; Drug Synergism; Duodenum; Female; Guinea Pigs; Heart; Histamine; Ileum; In Vitro Techniques; Jejunum; Male; Mesalamine; Metronidazole; Muscle Contraction; Myenteric Plexus; Pyrilamine; Receptors, Histamine; Scopolamine; Tetrodotoxin; Thiourea

1986
Selective enhancement of histamine H1-receptor responses in guinea-pig ileal smooth muscle by 1,4-dithiothreitol.
    British journal of pharmacology, 1986, Volume: 87, Issue:1

    Topics: Acetylcholine; Animals; Dimaprit; Dithionitrobenzoic Acid; Dithiothreitol; Dose-Response Relationship, Drug; Female; Guanidines; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Thiourea

1986
Pharmacological activities of two new histamine analogs.
    Agents and actions, 1986, Volume: 18, Issue:1-2

    Topics: Animals; Cats; Dimaprit; Dose-Response Relationship, Drug; Gastric Acid; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Methylhistamines; Muscle Contraction; Receptors, Histamine H1; Structure-Activity Relationship; Thiourea

1986
Effects of Ca2+ ions on gastric acid secretion by the rat isolated stomach.
    Agents and actions, 1986, Volume: 18, Issue:1-2

    Topics: Adenylyl Cyclases; Animals; Calcium; Dimaprit; Dose-Response Relationship, Drug; Gastric Acid; Histamine; In Vitro Techniques; Male; Rats; Receptors, Histamine; Theophylline; Thiourea

1986
[Miosis induced by histamine injected into the anterior chamber of isolated pig eyes].
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1986, Volume: 7, Issue:1

    Topics: Animals; Anterior Chamber; Chlorpheniramine; Cimetidine; Dimaprit; Female; Histamine; In Vitro Techniques; Male; Pupil; Receptors, Histamine H2; Swine; Thiourea

1986
Participation of vascular H1-receptors in histaminergic relaxation of rabbit middle cerebral artery in vitro.
    Archives internationales de pharmacodynamie et de therapie, 1986, Volume: 283, Issue:2

    Topics: Animals; Cerebral Arteries; Cimetidine; Dimaprit; Drug Interactions; Histamine; In Vitro Techniques; Methylhistamines; Muscle Relaxation; Muscle, Smooth, Vascular; Phenethylamines; Pyrilamine; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Thiourea

1986
Studies on the desensitization of the central cardiovascular responses of histamine.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:3

    Topics: Animals; Blood Pressure; Brain; Cardiovascular System; Dimaprit; Heart Rate; Histamine; Imidazoles; Impromidine; Injections, Intraventricular; Male; Pyridines; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1986
Characterization with agonists of the histamine receptors mediating stimulation of gastric acid secretion in the Atlantic cod, Gadus morhua.
    Agents and actions, 1986, Volume: 19, Issue:1-2

    Topics: Animals; Cimetidine; Dimaprit; Female; Fishes; Gastric Acid; Histamine; Imidazoles; Impromidine; Male; Methylhistamines; Receptors, Histamine H2; Thiourea

1986
Hypotension and bradycardia elicited by histamine into the C1 area of the rostral ventrolateral medulla.
    European journal of pharmacology, 1987, Apr-14, Volume: 136, Issue:2

    Topics: Animals; Blood Pressure; Dimaprit; Heart Rate; Hemodynamics; Histamine; Injections; Male; Medulla Oblongata; Metiamide; Naphazoline; Phenoxybenzamine; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Thiourea

1987
Histamine receptors on rat ocular surface.
    Ophthalmic research, 1987, Volume: 19, Issue:4

    Topics: Animals; Capillary Permeability; Chlorpheniramine; Cimetidine; Conjunctiva; Dimaprit; Dose-Response Relationship, Drug; Drug Combinations; Histamine; Male; Rats; Rats, Inbred Strains; Receptors, Histamine; Thiourea

1987
Evidence for histaminergic arousal mechanisms in the hypothalamus of cat.
    Neuropharmacology, 1988, Volume: 27, Issue:2

    Topics: Animals; Arousal; Cats; Dimaprit; Female; Histamine; Histamine Antagonists; Histidine Decarboxylase; Hypothalamus; Hypothalamus, Posterior; Injections; Injections, Intraperitoneal; Male; Methylhistidines; Pyrilamine; Thiourea

1988
Characteristics of histamine receptors in the isolated and perfused canine coronary arteries.
    Archives internationales de pharmacodynamie et de therapie, 1987, Volume: 290, Issue:1

    Topics: Animals; Chlorpheniramine; Cimetidine; Coronary Vessels; Dimaprit; Dogs; Endothelium, Vascular; Female; Histamine; In Vitro Techniques; Male; Pyridines; Receptors, Histamine; Saponins; Thiourea; Vasoconstriction; Vasodilation

1987
Mucosal protective action of histamine against gastric lesions induced by HCl in rats: importance of antigastric motor activity mediated by H2-receptors.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:2

    Topics: Animals; Cimetidine; Dimaprit; Gastric Acid; Gastric Mucosa; Gastrointestinal Motility; Histamine; Hydrochloric Acid; Indomethacin; Male; Pyridines; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea; Tripelennamine

1988
Histaminergic regulation of prolactin secretion: involvement of tuberoinfundibular dopaminergic neurons.
    Neuroendocrinology, 1988, Volume: 48, Issue:2

    Topics: Animals; Cerebral Ventricles; Dimaprit; Dopamine; Histamine; Infusions, Intra-Arterial; Injections, Intraventricular; Male; Neurons; Prolactin; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Receptors, Histamine H2; Reference Values; Thiazoles; Thiourea

1988
Histaminergic regulation of prolactin secretion: involvement of serotoninergic neurons.
    Neuroendocrinology, 1988, Volume: 48, Issue:5

    Topics: Dimaprit; Histamine; Ketanserin; Methysergide; Neurons; Prolactin; Receptors, Dopamine; Receptors, Serotonin; Serotonin; Thiourea

1988
Histamine receptor effects on dissipation of an intracellular proton gradient of isolated gastric mucosal surface cells.
    Proceedings of the Society for Experimental Biology and Medicine. Society for Experimental Biology and Medicine (New York, N.Y.), 1987, Volume: 185, Issue:4

    Topics: Animals; Bicarbonates; Chlorides; Cimetidine; Dimaprit; Diphenhydramine; Gastric Acid; Gastric Mucosa; Histamine; Protons; Pyridines; Pyrilamine; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Sodium; Thiourea

1987
Comparing binding of histamine and H2-antagonist with their effects on gastric acid secretion.
    Biochimica et biophysica acta, 1987, Feb-20, Volume: 923, Issue:2

    Topics: Animals; Binding, Competitive; Gastric Acid; Gastric Mucosa; Histamine; Kinetics; Metiamide; Models, Biological; Rana catesbeiana; Receptors, Histamine; Thiourea

1987
Conservative and nonconservative inhibitors of gastric acid secretion.
    The American journal of physiology, 1987, Volume: 253, Issue:3 Pt 1

    Topics: Animals; Gastric Acid; Histamine; In Vitro Techniques; Metiamide; Nitrites; Rana catesbeiana; Stimulation, Chemical; Thiocyanates; Thiourea

1987
Enhanced adverse electrophysiologic effects of histamine after myocardial infarction in guinea pigs.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 232, Issue:2

    Topics: Action Potentials; Animals; Arrhythmias, Cardiac; Chlorpheniramine; Dimaprit; Electrophysiology; Guinea Pigs; Heart; Heart Rate; Histamine; Male; Myocardial Infarction; Thiourea

1985
Modulation of in vitro cellular immune response by histamine agonists or antagonists in murine species.
    Arzneimittel-Forschung, 1985, Volume: 35, Issue:1A

    Topics: Animals; Cell Line; Cell Survival; Chlorpheniramine; Chromium Radioisotopes; Cimetidine; Dimaprit; Diphenhydramine; Histamine; Histamine Antagonists; Imidazoles; Immunity, Cellular; Impromidine; Kinetics; Male; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Ranitidine; T-Lymphocytes, Cytotoxic; T-Lymphocytes, Regulatory; Thiourea

1985
Quantification of H2-agonism by clonidine and dimaprit in an adenylate cyclase assay.
    Agents and actions, 1985, Volume: 16, Issue:3-4

    Topics: Adenylyl Cyclases; Animals; Cimetidine; Clonidine; Dimaprit; Guinea Pigs; Histamine; In Vitro Techniques; Myocardium; Receptors, Histamine; Receptors, Histamine H2; Thiourea

1985
Histamine antagonists in the treatment of shock hyperglycemia in the rat.
    Annals of emergency medicine, 1985, Volume: 14, Issue:2

    Topics: Animals; Blood Glucose; Blood Pressure; Diphenhydramine; Drug Therapy, Combination; Histamine; Hyperglycemia; Isotonic Solutions; Liver Glycogen; Male; Metiamide; Rats; Rats, Inbred Strains; Ringer's Solution; Shock; Thiourea

1985
Effects in man of histamine H 2 -receptor blockade by burimamide.
    Lancet (London, England), 1972, Nov-25, Volume: 2, Issue:7787

    Topics: Adult; Gastric Juice; Histamine; Histamine H1 Antagonists; Humans; Imidazoles; Male; Parasympatholytics; Pentagastrin; Sensory Receptor Cells; Thiourea

1972
Studies on the mechanism of lymphocyte-mediated cytolysis. IV. Specificity of the histamine receptor on effector T cells.
    Journal of immunology (Baltimore, Md. : 1950), 1973, Volume: 111, Issue:2

    Topics: Animals; Ascitic Fluid; Cell Membrane; Chlorpheniramine; Cyclic AMP; Cyclizine; Diphenhydramine; Histamine; Histamine H1 Antagonists; Histamine Release; Imidazoles; Mast Cells; Mice; Mice, Inbred C57BL; Receptors, Drug; T-Lymphocytes; Thiourea

1973
Inhibition of histamine release by histamine controlled by H2 receptor.
    Nature, 1973, Aug-03, Volume: 244, Issue:5414

    Topics: Basophils; Cyclic AMP; Diphenhydramine; Feedback; Histamine; Histamine H1 Antagonists; Histamine Release; Humans; Hypersensitivity; Imidazoles; Leukocytes; Receptors, Drug; Thiourea

1973
Editorial: Gastric acid, ulcers, and H2-receptors.
    Lancet (London, England), 1974, Volume: 1, Issue:7859

    Topics: Binding, Competitive; Gastric Juice; Histamine; Histamine H1 Antagonists; Humans; Imidazoles; Parasympatholytics; Receptors, Drug; Stomach; Stomach Ulcer; Sulfides; Thiourea

1974
Mobilization of gastric mucosal histamine and gastric secretion after H2-receptor blockade.
    British journal of pharmacology, 1973, Volume: 49, Issue:4

    Topics: Animals; Biological Assay; Female; Gastric Juice; Gastric Mucosa; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine Release; Ileum; Imidazoles; Pentagastrin; Rats; Sulfides; Thiourea

1973
Presence of histamine H2-receptors in the guinea-pig pulmonary vascular bed.
    Pharmacology, 1973, Volume: 9, Issue:5

    Topics: Acetylcholine; Angiotensin II; Animals; Benzyl Compounds; Blood Pressure; Dose-Response Relationship, Drug; Ethylenediamines; Female; Guinea Pigs; Histamine; Histamine H1 Antagonists; Imidazoles; In Vitro Techniques; Lung; Male; Norepinephrine; Perfusion; Pulmonary Artery; Pulmonary Veins; Pyridines; Receptors, Drug; Serotonin; Thiourea

1973
Antagonism by burimamide of inhibitions induced by histamine in plexus-containing longitudinal muscle preparations from guinea-pig ileum.
    British journal of pharmacology, 1973, Volume: 48, Issue:2

    Topics: Animals; Atropine; Benzyl Compounds; Dose-Response Relationship, Drug; Electric Stimulation; Ethylenediamines; Guinea Pigs; Histamine; Histamine H1 Antagonists; Ileum; Imidazoles; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Pyridines; Receptors, Drug; Thiourea

1973
H2-receptor blockade and stimulation of histidine decarboxylase.
    Nature: New biology, 1973, Oct-03, Volume: 245, Issue:144

    Topics: Animals; Carbon Radioisotopes; Carboxy-Lyases; Enzyme Induction; Food; Gastric Mucosa; Histamine; Histamine H1 Antagonists; Histidine; Imidazoles; Male; Rats; Receptors, Drug; Stimulation, Chemical; Stomach; Thiourea

1973
Increase in histamine receptors on thymus-derived effector lymphocytes during the primary immune response to alloantigens.
    Nature, 1973, Aug-03, Volume: 244, Issue:5414

    Topics: Animals; Antigens, Neoplasm; Binding, Competitive; Chromium Radioisotopes; Cyclic AMP; Cytotoxicity Tests, Immunologic; Histamine; Histamine H1 Antagonists; Imidazoles; Immunity, Cellular; Immunization; Isoantigens; Mast-Cell Sarcoma; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Receptors, Drug; T-Lymphocytes; Thiourea

1973
Adenyl and guanyl cyclase in rabbit gastric mucosa.
    The American journal of physiology, 1973, Volume: 225, Issue:6

    Topics: Adenosine Triphosphate; Adenylyl Cyclases; Animals; Chromatography, Thin Layer; Fluorides; Gastric Mucosa; Guanylate Cyclase; Histamine; Histamine H1 Antagonists; Hydrogen-Ion Concentration; Imidazoles; In Vitro Techniques; Manganese; Pentagastrin; Rabbits; Thiourea; Time Factors

1973
Effect of histamine and its methyl derivatives on cyclic AMP metabolism in gastric mucosa and its blockade by an H2 receptor antagonist.
    The Journal of clinical investigation, 1974, Volume: 53, Issue:1

    Topics: Adenylyl Cyclases; Animals; Cell-Free System; Cyclic AMP; Dose-Response Relationship, Drug; Gastric Mucosa; Guinea Pigs; Histamine; Histamine H1 Antagonists; Imidazoles; Methylation; Thiourea

1974
Comparison of the antihistaminic effect of burimamide and mepyramine and their effect on the activity of histamine methyltransferase.
    Biochemical pharmacology, 1973, Nov-01, Volume: 22, Issue:21

    Topics: Animals; Benzyl Compounds; Brain; Carboxy-Lyases; Ethylenediamines; Guinea Pigs; Heart Atria; Histamine; Histamine H1 Antagonists; Histidine; Ileum; Imidazoles; In Vitro Techniques; Kinetics; Male; Methyltransferases; Monoamine Oxidase; Pyridines; Receptors, Drug; Stomach; Thiourea

1973
Proceedings: The effect of an H2-receptor antagonist on histamine-stimulated acid secretion by rat stomach in vitro.
    The Journal of physiology, 1973, Volume: 234, Issue:2

    Topics: Animals; Caffeine; Gastric Juice; Histamine; Histamine H1 Antagonists; Imidazoles; In Vitro Techniques; Isoproterenol; Pentagastrin; Propranolol; Rats; Reserpine; Secretory Rate; Stimulation, Chemical; Thiourea

1973
Blockade by burimamide of the effects of histamine and histamine analogs on cardiac contractility, phosphorylase activation and cyclic adenosine monophosphate.
    The Journal of pharmacology and experimental therapeutics, 1974, Volume: 188, Issue:1

    Topics: Adenylyl Cyclases; Animals; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Ethylamines; Guinea Pigs; Heart; Heparin; Histamine; Histamine H1 Antagonists; Imidazoles; In Vitro Techniques; Myocardium; Norepinephrine; Phosphorylases; Propranolol; Pyrazoles; Stimulation, Chemical; Theophylline; Thiourea; Time Factors; Triazoles

1974
Editorial: New antagonists excite an old histamine prospector.
    The New England journal of medicine, 1974, Mar-28, Volume: 290, Issue:13

    Topics: Animals; Arrhythmias, Cardiac; Cyclic AMP; Gastric Juice; Gastric Mucosa; Guinea Pigs; Heart; Heart Rate; Histamine; Histamine H1 Antagonists; Humans; Imidazoles; Myocardium; Peptic Ulcer; Rabbits; Receptors, Drug; Sulfides; Thiourea; Vagus Nerve

1974
Histamine H2-receptors in the sheep bronchus and cat trachea: the action of burimamide.
    British journal of pharmacology, 1973, Volume: 48, Issue:2

    Topics: Animals; Benzyl Compounds; Bronchi; Cats; Dose-Response Relationship, Drug; Ethylenediamines; Histamine; Histamine H1 Antagonists; Imidazoles; In Vitro Techniques; Isoproterenol; Methacholine Compounds; Muscle Contraction; Muscle, Smooth; Propranolol; Pyridines; Receptors, Drug; Sheep; Thiourea; Trachea

1973
Metiamide--an orally active histamine H2-receptor antagonist.
    Agents and actions, 1973, Volume: 3, Issue:3

    Topics: Administration, Oral; Animals; Dogs; Female; Gastric Juice; Gastric Mucosa; Guinea Pigs; Half-Life; Histamine; Histamine H1 Antagonists; Imidazoles; In Vitro Techniques; Injections, Intravenous; Pentagastrin; Rats; Receptors, Drug; Sulfides; Thiourea

1973
Studies on the mode of action of histamine H1- and H2-receptor antagonists on gastric histamine methyltransferase.
    Agents and actions, 1973, Volume: 3, Issue:3

    Topics: Animals; Carbon Radioisotopes; Dose-Response Relationship, Drug; Enzyme Activation; Gastric Mucosa; Histamine; Histamine H1 Antagonists; Imidazoles; In Vitro Techniques; Kinetics; Methylation; Methyltransferases; Osmolar Concentration; Phenothiazines; Pyloric Antrum; Receptors, Drug; Structure-Activity Relationship; Sulfides; Swine; Thiourea

1973
Similar actions of methylated histamines and histamine receptor antagonists on gastric histamine methyltransferase.
    Agents and actions, 1973, Volume: 3, Issue:3

    Topics: Animals; Gastric Mucosa; Histamine; Histamine H1 Antagonists; Imidazoles; In Vitro Techniques; Kinetics; Methylation; Methyltransferases; Receptors, Drug; Swine; Thiourea

1973
The influence of burimamide on 14C-histamine uptake and metabolism by guinea pig atrium and mouse neoplastic mast cells, in vitro.
    Agents and actions, 1973, Volume: 3, Issue:3

    Topics: Animals; Carbon Radioisotopes; Guinea Pigs; Heart Atria; Histamine; Histamine H1 Antagonists; Imidazoles; In Vitro Techniques; Mast Cells; Mast-Cell Sarcoma; Mice; Mice, Inbred Strains; Sarcoma, Experimental; Thiourea; Time Factors

1973
Effect of burimamide on histamine metabolism.
    Agents and actions, 1973, Volume: 3, Issue:3

    Topics: Animals; Benzyl Compounds; Carbon Radioisotopes; Ethylenediamines; Histamine; Histamine H1 Antagonists; Imidazoles; Mice; Pyridines; Thiourea; Time Factors

1973
Sulphur-methylene isosterism in the development of metiamide, a new histamine H2-receptor antagonist.
    Nature, 1974, Mar-01, Volume: 248, Issue:5443

    Topics: Animals; Binding, Competitive; Female; Histamine; Histamine H1 Antagonists; Hydrogen-Ion Concentration; Imidazoles; Kinetics; Myocardium; Receptors, Drug; Stereoisomerism; Structure-Activity Relationship; Sulfides; Thiourea; Uterus

1974
Inhibition of acid secretion in dog by metiamide, a histamine antagonist acting on H2 receptors.
    Gastroenterology, 1974, Volume: 66, Issue:4

    Topics: Animals; Atropine; Depression, Chemical; Dogs; Gastric Fistula; Gastric Juice; Glucose; Histamine; Histamine H1 Antagonists; Imidazoles; Liver Extracts; Pentagastrin; Receptors, Drug; Sulfides; Thiourea

1974
Action of Burimamide, a histamine antagonist, on acid secretion in vitro.
    The American journal of physiology, 1974, Volume: 226, Issue:4

    Topics: Animals; Cyclic AMP; Dogs; Gastric Juice; Gastric Mucosa; Histamine; Histamine H1 Antagonists; Imidazoles; Methacholine Compounds; Pentagastrin; Rana pipiens; Secretory Rate; Theophylline; Thiourea

1974
The effects of burimamide on gastric acid secretion and gastric mucosal blood flow in the anaesthetized cat.
    The Journal of physiology, 1974, Volume: 237, Issue:2

    Topics: Animals; Cats; Gastric Juice; Gastric Mucosa; Histamine; Histamine H1 Antagonists; Hydrogen-Ion Concentration; Imidazoles; Pentagastrin; Thiourea

1974
[Effect of metiamide, an antagonist of histamine H2-receptors, on gastric secretion (author's transl)].
    Przeglad lekarski, 1974, Volume: 31, Issue:2

    Topics: Animals; Bethanechol Compounds; Cats; Ceruletide; Female; Gastric Juice; Histamine; Histamine H1 Antagonists; Imidazoles; Male; Pentagastrin; Peptones; Receptors, Drug; Secretory Rate; Sulfides; Thiourea

1974
Actions of metiamide, an H2-histamine receptor antagonist, on gastric H+ and pepsin secretion in dogs.
    Gastroenterology, 1974, Volume: 67, Issue:1

    Topics: Animals; Bethanechol Compounds; Dogs; Gastric Juice; Gastric Mucosa; Glucose; Histamine; Histamine H1 Antagonists; Hydrogen-Ion Concentration; Imidazoles; Pentagastrin; Pepsin A; Receptors, Drug; Sulfides; Thiourea

1974
H2-receptors in peripheral blood vessels.
    Nature, 1974, May-24, Volume: 249, Issue:455

    Topics: Animals; Benzyl Compounds; Blood Vessels; Dogs; Ethylenediamines; Half-Life; Histamine; Histamine H1 Antagonists; Imidazoles; Pyridines; Radioisotopes; Receptors, Drug; Sulfides; Synovial Membrane; Thiourea; Vasomotor System; Xenon

1974
The inhibition of histamine uptake and metabolism by burimamide in the guinea-pig atrium and in mouse neoplastic mast cells, in vitro.
    British journal of pharmacology, 1973, Volume: 49, Issue:2

    Topics: Animals; Carbon Radioisotopes; Cell Line; Cells, Cultured; Electric Stimulation; Guinea Pigs; Heart Atria; Histamine; Histamine H1 Antagonists; Imidazoles; In Vitro Techniques; Mast Cells; Mice; Myocardium; Thiourea

1973
Proceedings: Effect of histamine H2-receptor antagonists on gastric secretion, circulation, and acid-base-balance in cats.
    Naunyn-Schmiedeberg's archives of pharmacology, 1974, Volume: 282, Issue:Suppl

    Topics: Acid-Base Equilibrium; Animals; Blood Pressure; Carbon Dioxide; Cats; Gastric Acidity Determination; Gastric Juice; Gastric Mucosa; Heart Rate; Hemodynamics; Histamine; Histamine H1 Antagonists; Imidazoles; Oxygen; Oxygen Consumption; Phenoxybenzamine; Receptors, Drug; Regional Blood Flow; Stomach; Sulfides; Thiourea

1974
Blockade by burimamide of the effects of histamine and histamine analogues on cardiac adenylate cyclase.
    The Journal of pharmacy and pharmacology, 1974, Volume: 26, Issue:5

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Guinea Pigs; Histamine; Histamine H1 Antagonists; Imidazoles; In Vitro Techniques; Myocardium; Pyrazoles; Thiourea; Triazoles

1974
Effects of burimamide, an antagonist of H-2 histamine receptors, in the gastric fistula dog.
    The American journal of digestive diseases, 1974, Volume: 19, Issue:9

    Topics: Animals; Chlorides; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Ethylamines; Fistula; Gastric Acidity Determination; Glucose; Histamine; Histamine H1 Antagonists; Hydrogen; Imidazoles; Pentagastrin; Pepsin A; Potassium; Pyrazoles; Receptors, Drug; Sodium; Stomach; Thiourea

1974
Investigations into the positive inotropic effect of clondine in isolated hearts.
    Naunyn-Schmiedeberg's archives of pharmacology, 1974, Volume: 282, Issue:2

    Topics: Action Potentials; Animals; Clonidine; Dose-Response Relationship, Drug; Electrocardiography; Female; Guinea Pigs; Heart; Heart Rate; Histamine; Histamine H1 Antagonists; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Perfusion; Pheniramine; Phentolamine; Phenyl Ethers; Propanolamines; Propylamines; Receptors, Drug; Stimulation, Chemical; Thiourea

1974
Proceedings: Failure of burimamide and (15S)-15-methyl prostaglandin E2 to prevent histamine-induced gastric mucosal hyperaemia in the rat.
    The Journal of physiology, 1974, Volume: 239, Issue:2

    Topics: Animals; Benzyl Compounds; Ethylenediamines; Gastric Juice; Gastric Mucosa; Histamine; Histamine H1 Antagonists; Hyperemia; Imidazoles; Prostaglandins; Pyridines; Rats; Thiourea

1974
The antagonism of the positive inotropic effect of histamine and noradrenaline by H1 and H2-receptor blocking agents.
    Agents and actions, 1974, Volume: 4, Issue:3

    Topics: Animals; Depression, Chemical; Dose-Response Relationship, Drug; Guinea Pigs; Heart Rate; Heart Ventricles; Histamine; Histamine H1 Antagonists; Imidazoles; In Vitro Techniques; Norepinephrine; Osmolar Concentration; Receptors, Drug; Sulfides; Thiourea

1974
The cardiovascular effects of histamine in laboratory animals.
    Agents and actions, 1974, Volume: 4, Issue:3

    Topics: Animals; Benzyl Compounds; Blood Pressure; Cats; Depression, Chemical; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Ethylenediamines; Guinea Pigs; Histamine; Histamine H1 Antagonists; Imidazoles; Phentolamine; Propranolol; Pyridines; Rabbits; Rats; Receptors, Drug; Species Specificity; Sulfides; Thiourea

1974
The presence of histamine H2-receptors in rabbit kidney.
    Archives internationales de pharmacodynamie et de therapie, 1974, Volume: 209, Issue:1

    Topics: Acetylcholine; Animals; Benzyl Compounds; Blood Pressure; Bradykinin; Diuresis; Dose-Response Relationship, Drug; Ethylenediamines; Female; Histamine; Histamine H1 Antagonists; Imidazoles; In Vitro Techniques; Kidney; Male; Perfusion; Pyridines; Rabbits; Receptors, Drug; Thiourea

1974
Effect of anaphylaxis and histamine, pyrilamine and burimamide on levels of cyclic AMP and cyclic GMP in guinea-pig lung.
    Research communications in chemical pathology and pharmacology, 1974, Volume: 8, Issue:4

    Topics: Analysis of Variance; Anaphylaxis; Animals; Antigen-Antibody Reactions; Benzyl Compounds; Carbon Radioisotopes; Cyclic AMP; Cyclic GMP; Ethylenediamines; Guinea Pigs; Histamine; Histamine H1 Antagonists; Humans; Imidazoles; In Vitro Techniques; Iodine Radioisotopes; Lung; Ovalbumin; Pyridines; Rabbits; Radioimmunoassay; Thiourea; Tritium

1974
Cardiovascular histamine receptors in the rabbit.
    The Australian journal of experimental biology and medical science, 1974, Volume: 52, Issue:Pt 3

    Topics: Animals; Atropine; Benzyl Compounds; Blood Pressure; Chemoreceptor Cells; Depression, Chemical; Dose-Response Relationship, Drug; Drug Synergism; Ethylenediamines; Female; Heart Rate; Histamine; Histamine H1 Antagonists; Imidazoles; Injections, Intravenous; Male; Pyridines; Rabbits; Stimulation, Chemical; Thiourea; Vagotomy; Vagus Nerve

1974
The role of histamine receptors in the stimulation of gastric acid secretion.
    The American journal of digestive diseases, 1974, Volume: 19, Issue:11

    Topics: Animals; Atropine; Bethanechol Compounds; Cats; Ceruletide; Gastrectomy; Gastric Juice; Gastric Mucosa; Histamine; Histamine H1 Antagonists; Imidazoles; Insulin; Pentagastrin; Peptones; Receptors, Drug; Sulfides; Thiourea

1974
A vasodepressor action of histamine mediated by H2-receptor activation.
    European journal of pharmacology, 1974, Volume: 29, Issue:1

    Topics: Animals; Benzyl Compounds; Blood Circulation; Depression, Chemical; Dose-Response Relationship, Drug; Ethylenediamines; Female; Gastric Juice; Guinea Pigs; Histamine; Histamine H1 Antagonists; In Vitro Techniques; Isoproterenol; Lung; Male; Perfusion; Pulmonary Artery; Pyridines; Receptors, Drug; Regional Blood Flow; Thiourea

1974
Inhibition of in vitro stimulated gastric acid secretion by a histamine H2-receptor antagonist, metiamide.
    European journal of pharmacology, 1974, Volume: 29, Issue:1

    Topics: Animals; Dose-Response Relationship, Drug; Gastric Juice; Gastric Mucosa; Histamine; Histamine H1 Antagonists; Imidazoles; In Vitro Techniques; Male; Pentagastrin; Rana temporaria; Rats; Stimulation, Chemical; Sulfides; Thiourea; Time Factors

1974
Proceedings: Histamine receptors in the cardiovascular system of the cat.
    British journal of pharmacology, 1974, Volume: 51, Issue:1

    Topics: Animals; Benzyl Compounds; Blood Pressure; Cardiovascular System; Cats; Dose-Response Relationship, Drug; Ethylenediamines; Histamine; Histamine H1 Antagonists; Imidazoles; Injections, Intravenous; Pyridines; Receptors, Drug; Sulfides; Thiourea

1974
The effect of histamine-H2-receptor-antagonists on gastric acid secretion, gastric mucosal blood flow and acid base balance in cats.
    Naunyn-Schmiedeberg's archives of pharmacology, 1974, Volume: 285, Issue:4

    Topics: Acid-Base Equilibrium; Animals; Benzyl Compounds; Bicarbonates; Carbon Dioxide; Cats; Chlorides; Ethylenediamines; Gastric Fistula; Gastric Juice; Gastric Mucosa; Histamine; Histamine H1 Antagonists; Hydrogen-Ion Concentration; Imidazoles; Oxygen; Partial Pressure; Phenoxybenzamine; Pyridines; Receptors, Drug; Regional Blood Flow; Sulfides; Thiourea

1974
Differentiation of H1- and H2-receptors mediating positive chrono- and inotropic responses to histamine on atrial preparations of the guinea-pig.
    Agents and actions, 1974, Volume: 4, Issue:4

    Topics: Animals; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Heart Atria; Heart Rate; Histamine; Histamine H1 Antagonists; Imidazoles; In Vitro Techniques; Male; Promethazine; Receptors, Drug; Stimulation, Chemical; Thiourea

1974
Cardiovascular effects of burimamide and metiamide.
    Agents and actions, 1974, Volume: 4, Issue:4

    Topics: Animals; Benzyl Compounds; Blood Pressure; Cats; Drug Interactions; Ethylenediamines; Gastric Fistula; Heart Rate; Hemodynamics; Histamine; Histamine H1 Antagonists; Imidazoles; Phenoxybenzamine; Pyridines; Receptors, Drug; Stimulation, Chemical; Sulfides; Thiourea

1974
Proceedings: Definition of the antagonistic action of burimamide and metiamide on the positive inotropic effect of histamine in isolated heart preparations.
    British journal of pharmacology, 1974, Volume: 52, Issue:3

    Topics: Animals; Burimamide; Electric Stimulation; Guinea Pigs; Heart; Histamine; Histamine H1 Antagonists; In Vitro Techniques; Metiamide; Stimulation, Chemical; Thiourea

1974
Effect of metiamide, a histamine antagonist of H2-receptors, on acid secretion of isolated canine stomach perfused with homologous blood.
    Pharmacology, 1974, Volume: 11, Issue:4

    Topics: Animals; Bethanechol Compounds; Carbon Dioxide; Depression, Chemical; Dogs; Gastric Juice; Gastric Mucosa; Histamine; Histamine H1 Antagonists; Hydrogen-Ion Concentration; Imidazoles; Injections, Intra-Arterial; Oxygen; Perfusion; Pressure; Receptors, Drug; Stimulation, Chemical; Stomach; Sulfides; Thiourea; Time Factors

1974
[Radioprotective action and possible mechanisms of action of some potential radiation-protective agents].
    Nauchnye doklady vysshei shkoly. Biologicheskie nauki, 1973, Volume: 113, Issue:5

    Topics: Animals; beta-Aminoethyl Isothiourea; Cysteamine; Histamine; Lipids; Mice; Oxidation-Reduction; Phospholipids; Polarography; Radiation Effects; Radiation-Protective Agents; Serotonin; Spectrometry, Fluorescence; Structure-Activity Relationship; Thiourea

1973
Effects of pulmonary irritants on DNA, ATPase activity, and histamine on rat lung.
    Proceedings of the Society for Experimental Biology and Medicine. Society for Experimental Biology and Medicine (New York, N.Y.), 1974, Volume: 146, Issue:1

    Topics: Adenosine Triphosphatases; Animals; DNA; Histamine; Lung; Male; Organ Size; Ozone; Phenylthiourea; Pulmonary Edema; Rats; Thiourea

1974
Increased production of cyclic AMP in gastric tissue by stimulation of histamine2 (H2)-receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1973, Volume: 279, Issue:1

    Topics: Animals; Binding, Competitive; Clonidine; Cyclic AMP; Diphenhydramine; Dose-Response Relationship, Drug; Gastric Mucosa; Guinea Pigs; Histamine; Imidazoles; In Vitro Techniques; Male; Rats; Receptors, Drug; Theophylline; Thiourea

1973
Histamine H1 and H2-receptors at a ganglionic synapse.
    Nature, 1973, Nov-16, Volume: 246, Issue:5429

    Topics: Action Potentials; Animals; Benzyl Compounds; Depression, Chemical; Drug Interactions; Electric Stimulation; Ethylenediamines; Ganglia, Spinal; Histamine; Histamine Antagonists; Imidazoles; In Vitro Techniques; Pyridines; Rabbits; Receptors, Drug; Synapses; Synaptic Transmission; Thiourea

1973
Definition and antagonism of histamine H 2 -receptors.
    Nature, 1972, Apr-21, Volume: 236, Issue:5347

    Topics: Animals; Benzyl Compounds; Blood Pressure; Cats; Dogs; Ethylenediamines; Female; Gastric Juice; Guinea Pigs; Heart Atria; Histamine; Histamine H1 Antagonists; Humans; Ileum; Imidazoles; In Vitro Techniques; Kinetics; Muscle Contraction; Muscle, Smooth; Pentagastrin; Pyridines; Rats; Receptors, Drug; Thiourea; Uterus

1972
The effect of burimamide on gastric secretion in man.
    The British journal of surgery, 1972, Volume: 59, Issue:11

    Topics: Depression, Chemical; Gastric Juice; Histamine; Histamine H1 Antagonists; Humans; Imidazoles; Pentagastrin; Secretory Rate; Stomach; Thiourea

1972
Secretin inhibition of gastrin-stimulated deoxyribonucleic acid synthesis.
    Gastroenterology, 1974, Volume: 67, Issue:4

    Topics: Animals; Autoradiography; Depression, Chemical; DNA; Duodenum; Gastric Juice; Gastric Mucosa; Histamine; Ileum; Imidazoles; Injections, Intraperitoneal; Male; Pentagastrin; Rats; Secretin; Stimulation, Chemical; Sulfides; Thiourea; Thymidine; Tritium

1974
Effect of H2 receptor antagonists on histidine decarboxylase activity in rat gastric mucosa.
    Biochemical pharmacology, 1974, Nov-01, Volume: 23, Issue:21

    Topics: Animals; Butanones; Carbon Radioisotopes; Carboxy-Lyases; Cycloheximide; Dactinomycin; Dose-Response Relationship, Drug; Female; Food; Gastric Mucosa; Histamine; Histidine; Imidazoles; In Vitro Techniques; Pentagastrin; Rats; Receptors, Drug; Stimulation, Chemical; Sulfides; Thiourea; Time Factors

1974
Stimulation of rat gastric adenylate cyclase by histamine and histamine analogues and blockade by burimamide.
    British journal of pharmacology, 1974, Volume: 52, Issue:1

    Topics: Adenylyl Cyclases; Animals; Burimamide; Histamine; In Vitro Techniques; Rats; Stimulation, Chemical; Stomach; Thiourea

1974
Effect of metiamide, a histamine H2-receptor antagonist, on gastric response to histamine, pentagastrin, insulin, and peptone meal in man.
    The American journal of digestive diseases, 1974, Volume: 19, Issue:7

    Topics: Adult; Depression, Chemical; Dose-Response Relationship, Drug; Duodenal Ulcer; Gastric Acidity Determination; Gastric Juice; Histamine; Humans; Imidazoles; Infusions, Parenteral; Insulin; Intubation, Gastrointestinal; Pentagastrin; Pepsin A; Peptones; Secretory Rate; Sulfides; Thiourea

1974
Evidence that the inhibitory effect of burimamide on gastric secretion is not due to decreased gastric mucosal blood flow.
    The Journal of physiology, 1973, Volume: 230, Issue:1

    Topics: Animals; Dogs; Female; Gastric Juice; Gastric Mucosa; Histamine; Imidazoles; Pentagastrin; Secretory Rate; Thiourea

1973
Some effects of histamine in the depolarized rat uterus.
    British journal of pharmacology, 1973, Volume: 49, Issue:3

    Topics: Acetates; Acetylcholine; Animals; Barium; Buffers; Calcium; Calcium Radioisotopes; Cell Membrane Permeability; Chelating Agents; Female; Glycols; Histamine; Hydrogen; Imidazoles; In Vitro Techniques; Isoproterenol; Muscle Contraction; Nitrites; Papaverine; Potassium; Propranolol; Rats; Receptors, Drug; Thiourea; Uterus

1973
Gastric secretion in the isolated stomach of the guinea-pig.
    The Journal of physiology, 1974, Volume: 237, Issue:2

    Topics: Animals; Gastric Mucosa; Guinea Pigs; Histamine; Imidazoles; In Vitro Techniques; Male; Pentagastrin; Theophylline; Thiocyanates; Thiourea

1974
Effect of histamine H-receptor blockade on fasting serum gastrin and fasting gastric acid secretion in the dog.
    Nature, 1974, Jun-14, Volume: 249, Issue:458

    Topics: Animals; Depression, Chemical; Gastric Juice; Gastric Mucosa; Gastrins; Histamine; Imidazoles; Receptors, Drug; Secretory Rate; Thiourea

1974
Effect of exposure to O3, SO2 and NO2 upon the lung histamine content of guinea pigs.
    The Bulletin of Tokyo Medical and Dental University, 1969, Volume: 16, Issue:2

    Topics: Animals; Gases; Guinea Pigs; Histamine; Lung; Male; Nitrogen Dioxide; Ozone; Sulfur Dioxide; Thiourea; Water

1969
Dentine in vivo impermeability to radioactively labeled prdnisolone.
    Oral surgery, oral medicine, and oral pathology, 1971, Volume: 31, Issue:1

    Topics: Administration, Topical; Animals; Anti-Inflammatory Agents; Carbon Isotopes; Cortisone; Dentin; Histamine; Prednisolone; Rats; Thiourea; Tooth Permeability; Tritium

1971
The effect of radioprotective compounds on the incorporation of tritiated thymidine into mammalian cells.
    International journal of radiation biology and related studies in physics, chemistry, and medicine, 1966, Volume: 10, Issue:4

    Topics: Animals; Autoradiography; beta-Aminoethyl Isothiourea; Bone Marrow; Bone Marrow Cells; Cell Division; Cysteamine; DNA; Histamine; Hypoxia; Intestinal Mucosa; Mice; Radiation; Radiation-Protective Agents; Sulfhydryl Compounds; Thiourea; Thymidine; Tritium

1966
The synthesis of zapotidine.
    Tetrahedron, 1967, Volume: 23, Issue:1

    Topics: Alkaloids; Chemistry, Organic; Histamine; Imidazoles; Organic Chemistry Phenomena; Sulfur; Thiourea

1967
Action of tricyclic antidepressants on cyclic AMP in mucosal cells from guinea pig stomach.
    European journal of pharmacology, 1984, Oct-01, Volume: 105, Issue:1-2

    Topics: Alprostadil; Amitriptyline; Animals; Antidepressive Agents, Tricyclic; Brain; Cyclic AMP; Dimaprit; Gastric Mucosa; Guinea Pigs; Histamine; In Vitro Techniques; Oxygen Consumption; Prostaglandins E; Receptors, Histamine; Theophylline; Thiourea

1984
Effects of histamine agonists and antagonists on luminol-dependent chemiluminescence of granulocytes.
    Agents and actions, 1984, Volume: 15, Issue:3-4

    Topics: Cimetidine; Dimaprit; Granulocytes; Histamine; Histamine Antagonists; Humans; In Vitro Techniques; Luminescent Measurements; Luminol; Pyridazines; Pyridines; Pyrilamine; Ranitidine; Thiourea

1984
The role of prostaglandins in histamine-induced gastric vasodilation in the dog.
    The Journal of pharmacology and experimental therapeutics, 1980, Volume: 213, Issue:1

    Topics: Acetazolamide; Animals; Anti-Inflammatory Agents; Arachidonic Acids; Dimaprit; Dogs; Drug Interactions; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Hydroxyzine; Male; Pharmaceutical Vehicles; Prostaglandins; Pyridines; Receptors, Histamine H1; Receptors, Histamine H2; Stomach; Thiourea; Time Factors; Vasodilation

1980
Effects of histamine on human isolated heart muscle: comparison with effects of noradrenaline.
    The Journal of pharmacy and pharmacology, 1980, Volume: 32, Issue:2

    Topics: Cimetidine; Dimaprit; Heart; Histamine; Humans; In Vitro Techniques; Myocardial Contraction; Norepinephrine; Propranolol; Pyrilamine; Receptors, Histamine H2; Thiourea

1980
Evaluation of the role of Histamine H1- and H2-receptors in cutaneous inflammation in the guinea-pig produced by histamine and mast cell degranulation.
    British journal of pharmacology, 1980, Volume: 69, Issue:4

    Topics: Animals; Cimetidine; Dimaprit; Guinea Pigs; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Inflammation; Male; Mast Cells; Mathematics; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Skin; Thiourea; Vasodilation

1980
Histamine inhibition of the in vitro induction of cytotoxic T-cell responses.
    Immunopharmacology, 1980, Volume: 2, Issue:3

    Topics: Animals; Cytotoxicity, Immunologic; Dimaprit; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Lymphocyte Culture Test, Mixed; Mice; T-Lymphocytes; Thiourea

1980
Gastrointestinal ulceration in the guinea pig in response to dimaprit, histamine, and H1- and H2-blocking agents.
    Digestive diseases and sciences, 1981, Volume: 26, Issue:4

    Topics: Animals; Cimetidine; Dimaprit; Diphenhydramine; Duodenal Ulcer; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Injections, Intramuscular; Injections, Intraperitoneal; Male; Receptors, Histamine H1; Receptors, Histamine H2; Stomach Ulcer; Thiourea

1981
Mesenteric vascular reactivity to histamine receptor agonists and antagonists.
    Digestive diseases and sciences, 1981, Volume: 26, Issue:5

    Topics: Adrenergic Agonists; Animals; Blood Flow Velocity; Dimaprit; Dogs; Dose-Response Relationship, Drug; Female; Furans; Hemodynamics; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Infusions, Intra-Arterial; Male; Mesentery; Oxygen Consumption; Ranitidine; Receptors, Histamine; Receptors, Histamine H1; Regional Blood Flow; Thiourea; Tripelennamine

1981
Impairment of pharmacological modulation of airways smooth muscle by a respiratory pathogen.
    The Journal of pharmacy and pharmacology, 1981, Volume: 33, Issue:7

    Topics: Airway Resistance; Animals; Bacterial Vaccines; Carbachol; Dimaprit; Haemophilus; Histamine; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Rats; Respiratory Tract Infections; Thiourea; Trachea

1981
Histamine-induced rise in core temperature of chloral-anaesthetized rats: mediation by H2-receptors located in the preopticus area of hypothalamus.
    Neuropharmacology, 1982, Volume: 21, Issue:1

    Topics: Animals; Body Temperature; Chloral Hydrate; Dimaprit; Guanidines; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Hypothalamus; Imidazoles; Impromidine; Male; Preoptic Area; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H2; Thiourea

1982
An inhibitory effect of histamine on the rat anococcygeus muscle.
    The Journal of pharmacy and pharmacology, 1982, Volume: 34, Issue:3

    Topics: Acetylcholine; Animals; Carbachol; Cimetidine; Dimaprit; Drug Interactions; Guanidines; Histamine; Imidazoles; Impromidine; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Pyrilamine; Rats; Thiourea

1982
Histamine suppresses in vitro synthesis of precursor (pro-C5) of the fifth complement component (C5) by mouse peritoneal macrophages.
    Journal of immunology (Baltimore, Md. : 1950), 1982, Volume: 129, Issue:1

    Topics: Animals; Antigens; Bucladesine; Cimetidine; Complement C5; Complement Inactivator Proteins; Dimaprit; Guinea Pigs; Hemolysis; Histamine; Histamine H2 Antagonists; Humans; Macrophages; Male; Mice; Mice, Inbred C57BL; Protein Precursors; Receptors, Histamine H2; Thiourea; Tripelennamine

1982
Apparent irreversible H2-receptor blocking and prolonged gastric antisecretory activities of 3-N-(3-[3-(1-piperidinomethyl)phenoxy]propyl) amino-4-amino-1,2,5-thiadiazole-1-oxide (L-643, 441).
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 224, Issue:3

    Topics: Animals; Cimetidine; Dimaprit; Dogs; Female; Furans; Gastric Juice; Guinea Pigs; Heart Rate; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Male; Ranitidine; Thiadiazoles; Thiourea

1983
Histamine receptors in primate gallbladder.
    Digestive diseases and sciences, 1983, Volume: 28, Issue:4

    Topics: Animals; Dimaprit; Dose-Response Relationship, Drug; Female; Gallbladder; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Papio; Pressure; Pyridines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1983
Histamine modulation of human neutrophil oxidative metabolism, locomotion, degranulation, and membrane potential changes.
    Journal of immunology (Baltimore, Md. : 1950), 1983, Volume: 130, Issue:4

    Topics: Carbocyanines; Chemotaxis, Leukocyte; Cytoplasmic Granules; Dimaprit; Glucuronidase; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Hydrogen Peroxide; Membrane Potentials; Muramidase; Neutrophils; Oxygen Consumption; Receptors, Histamine H1; Receptors, Histamine H2; Superoxides; Thiourea

1983
Evidence for histamine H1 and H2 receptors in guinea-pig oxyntic cells.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 227, Issue:1

    Topics: Animals; Carbonic Anhydrases; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Imidazoles; Impromidine; In Vitro Techniques; Methylhistamines; Parietal Cells, Gastric; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1983
Release of prolactin and luteinizing hormone by histamine agonists in ovariectomized, steroid-treated rats under ether anesthesia.
    Experimental brain research, 1983, Volume: 52, Issue:2

    Topics: Animals; Castration; Dimaprit; Female; Histamine; Histamine H1 Antagonists; Luteinizing Hormone; Methylhistamines; Metiamide; Pituitary Gland, Anterior; Prolactin; Pyridines; Pyrilamine; Rats; Thiourea

1983
The effect of histamine, H1 and H2 agonists, and H1 and H2 antagonists on postprandial pancreatic polypeptide release in dogs.
    Scandinavian journal of gastroenterology, 1983, Volume: 18, Issue:2

    Topics: Animals; Cimetidine; Dimaprit; Dogs; Food; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Pancreatic Polypeptide; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Secretory Rate; Thiazoles; Thiourea

1983
Intracellular study of effects of histamine on electrical behaviour of myenteric neurones in guinea-pig small intestine.
    The Journal of physiology, 1984, Volume: 355

    Topics: Action Potentials; Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Guinea Pigs; Histamine; Histamine Antagonists; In Vitro Techniques; Intestine, Small; Membrane Potentials; Myenteric Plexus; Neurons; Neurotransmitter Agents; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Serotonin; Thiourea

1984
Differences in the interaction of histamine H2 receptor antagonists and tricyclic antidepressants with adenylate cyclase from guinea pig gastric mucosa.
    Biochemical pharmacology, 1984, Nov-15, Volume: 33, Issue:22

    Topics: Adenylyl Cyclases; Animals; Antidepressive Agents, Tricyclic; Cell Membrane; Dimaprit; Gastric Fundus; Gastric Mucosa; Guinea Pigs; Histamine; Histamine H2 Antagonists; Iprindole; Kinetics; Receptors, Histamine H2; Thiourea

1984
Influence of histamine or dimaprit on histamine release induced by anti-ige from human whole blood.
    Agents and actions, 1980, Volume: 10, Issue:1 Pt 2

    Topics: Antibodies; Dimaprit; Histamine; Histamine Release; Humans; Immunoglobulin E; Receptors, Histamine; Receptors, Histamine H2; Thiourea

1980
Effects of the histamine H2-receptor agonists dimaprit and 4-methylhistamine on the central noradrenaline and serotonin system.
    Agents and actions, 1980, Volume: 10, Issue:1 Pt 2

    Topics: Animals; Behavior, Animal; Brain; Dimaprit; Female; Histamine; Hydroxyindoleacetic Acid; Methoxyhydroxyphenylglycol; Methylhistamines; Norepinephrine; Rats; Receptors, Histamine; Receptors, Histamine H2; Serotonin; Thiourea; Tranylcypromine

1980
Combination of cimetidine with other drugs for treatment of cancer.
    The New England journal of medicine, 1983, Mar-10, Volume: 308, Issue:10

    Topics: Aged; Animals; Cimetidine; Coumarins; Female; Guanidines; Histamine; Humans; Interferons; Male; Melanoma; Metiamide; Mice; Middle Aged; Neoplasms; Thiourea

1983
Enhancement of histamine synthesis in mouse skin by epinephrine.
    Life sciences, 1984, Oct-15, Volume: 35, Issue:16

    Topics: Animals; Dimaprit; Epinephrine; Guanidines; Histamine; Histamine Release; Kinetics; Male; Methylhistidines; Mice; Skin; Skin Physiological Phenomena; Thiourea

1984
Histamine H2 receptor desensitization in HL-60 human promyelocytic leukemia cells.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 231, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Cell Differentiation; Cell Line; Cimetidine; Cyclic AMP; Dimaprit; Dinoprostone; Dose-Response Relationship, Drug; Histamine; Humans; Leukemia, Myeloid, Acute; Prostaglandins E; Receptors, Histamine; Receptors, Histamine H2; Thiocarbamates; Thiourea

1984
Reciprocal H1- and H2-histamine receptors in guinea pig gallbladder.
    The Journal of surgical research, 1982, Volume: 33, Issue:2

    Topics: Animals; Dimaprit; Female; Gallbladder; Guinea Pigs; Histamine; Male; Muscle Contraction; Muscle, Smooth; Pyridines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1982
Rabbit mesenteric artery receptors formed by cold exposure mediating increased histamine-induced relaxation.
    Archives internationales de pharmacodynamie et de therapie, 1982, Volume: 256, Issue:2

    Topics: Animals; Cold Temperature; Dimaprit; Histamine; In Vitro Techniques; Mesenteric Arteries; Metiamide; Muscle, Smooth, Vascular; Phenylephrine; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Reserpine; Thiourea; Tripelennamine; Vasodilation

1982
Autacoid and autonomic reactivity of bovine and ovine bronchus: modifications by antigenic sensitization.
    Archives internationales de pharmacodynamie et de therapie, 1982, Volume: 258, Issue:1

    Topics: Animals; Bronchi; Carbachol; Cattle; Dimaprit; Dose-Response Relationship, Drug; Epinephrine; Histamine; In Vitro Techniques; Isoproterenol; Muscle Contraction; Phenylephrine; Serotonin; Sheep; Thiourea

1982
Histamine-induced inhibition of lymphocyte proliferation and lysosomal enzyme release from polymorphs may not be mediated via H1- or H2-receptors.
    Agents and actions, 1982, Volume: 12, Issue:5-6

    Topics: Dimaprit; Histamine; Humans; Lymphocyte Activation; Lysosomes; Metiamide; Phytohemagglutinins; Polymorphism, Genetic; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1982
The effect of histamine on the development of adjuvant arthritis in the rat.
    Agents and actions, 1982, Volume: 12, Issue:5-6

    Topics: Animals; Arthritis; Arthritis, Experimental; Dimaprit; Dose-Response Relationship, Drug; Female; Histamine; Metiamide; Pyridines; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea; Time Factors

1982
An investigation of the involvement of histaminergic systems in novelty-induced grooming in the mouse.
    Behavioral and neural biology, 1982, Volume: 35, Issue:4

    Topics: Animals; Arousal; Cimetidine; Dimaprit; Diphenhydramine; Dose-Response Relationship, Drug; Grooming; Histamine; Male; Mice; Pyridines; Receptors, Histamine; Thiourea

1982
Inhibition of phytohaemagglutinin-induced proliferation of human peripheral blood lymphocytes by histamine and histamine H1 and H2 agonists.
    Clinical and experimental immunology, 1983, Volume: 51, Issue:1

    Topics: Cell Division; Cells, Cultured; Dimaprit; Dose-Response Relationship, Drug; Histamine; Humans; Imidazoles; Impromidine; Lymphocytes; Methylhistamines; Phytohemagglutinins; Pyridines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea

1983
Histamine receptors in the human ureter.
    Pharmacological research communications, 1983, Volume: 15, Issue:2

    Topics: Chlorpheniramine; Dimaprit; Histamine; Humans; In Vitro Techniques; Metiamide; Muscle Contraction; Muscle, Smooth; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea; Ureter

1983
Vascular responses of the isolated perfused stomach of rabbit and rat to histamine.
    European journal of pharmacology, 1983, Apr-22, Volume: 89, Issue:1-2

    Topics: Animals; Dimaprit; Histamine; Histamine Antagonists; Male; Muscle, Smooth, Vascular; Rabbits; Rats; Receptors, Histamine H1; Receptors, Histamine H2; Species Specificity; Stomach; Thiourea; Vasodilator Agents

1983
The role of histamine receptors in the release of renin.
    British journal of pharmacology, 1983, Volume: 79, Issue:1

    Topics: Animals; Dimaprit; Dogs; Female; Histamine; Kidney; Male; Pyridines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Renal Circulation; Renin; Sodium Chloride; Thiourea

1983
Central H1- and H2-histaminergic stimulation of pituitary-adrenocortical response under stress in rats.
    Neuroendocrinology, 1983, Volume: 36, Issue:6

    Topics: Animals; Corticosterone; Dimaprit; Histamine; Histamine Antagonists; Male; Methylhistamines; Pituitary-Adrenal System; Pyridines; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Stress, Physiological; Thiourea

1983
Central histaminergic stimulation of pituitary--adrenocortical response in the rat.
    Life sciences, 1983, Sep-19, Volume: 33, Issue:12

    Topics: Animals; Cimetidine; Corticosterone; Dimaprit; Dose-Response Relationship, Drug; Histamine; Imidazoles; Impromidine; Male; Pituitary-Adrenal System; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1983
Effects of histamine receptor stimulation on regional myocardial blood flow.
    The American journal of physiology, 1983, Volume: 245, Issue:3

    Topics: Animals; Blood Pressure; Cimetidine; Coronary Circulation; Dimaprit; Diphenhydramine; Dogs; Female; Heart Rate; Histamine; Male; Microspheres; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea

1983
Studies on cutaneous vascular permeability in the rat: increases caused by histamine and histamine-like agents.
    Agents and actions, 1984, Volume: 14, Issue:1

    Topics: Animals; Capillary Permeability; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Histamine; Microcirculation; Pyrilamine; Rats; Regional Blood Flow; Skin; Thiourea

1984
Effect of histamine receptor agonists and antagonists on the uterine vasculature.
    Proceedings of the Society for Experimental Biology and Medicine. Society for Experimental Biology and Medicine (New York, N.Y.), 1984, Volume: 175, Issue:4

    Topics: Animals; Dimaprit; Female; Histamine; p-Methoxy-N-methylphenethylamine; Pyridines; Receptors, Histamine H1; Receptors, Histamine H2; Regional Blood Flow; Sheep; Thiourea; Uterus

1984
Studies on the effect of histamine in isolated human pulmonary arteries and veins.
    Acta pharmacologica et toxicologica, 1984, Volume: 54, Issue:2

    Topics: Aged; Dimaprit; Female; Histamine; Humans; In Vitro Techniques; Male; Methylhistamines; Middle Aged; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Phentolamine; Potassium; Pulmonary Artery; Pulmonary Veins; Pyrilamine; Thiourea

1984
Histamine action on guinea pig ileal mucosa.
    The American journal of physiology, 1984, Volume: 246, Issue:4 Pt 1

    Topics: Animals; Bicarbonates; Biological Transport, Active; Chlorides; Dimaprit; Electric Conductivity; Female; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Intestinal Mucosa; Male; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1984
Dibenamine enhancement of histamine-induced relaxation of the rabbit mesenteric artery.
    Artery, 1983, Volume: 11, Issue:6

    Topics: Animals; Cold Temperature; Dibenzylchlorethamine; Dimaprit; Drug Synergism; Histamine; Mesenteric Arteries; Muscle Contraction; Muscle Relaxation; Papaverine; Rabbits; Receptors, Histamine; Thiourea

1983
[Imidazolic H2-agonists: importance of 2-amino substitution for pharmacological activity].
    Bollettino della Societa italiana di biologia sperimentale, 1984, Apr-30, Volume: 60, Issue:4

    Topics: Animals; Biological Assay; Cats; Dimaprit; Gastric Acid; Guinea Pigs; Histamine; Methylhistamines; Muscle Relaxation; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Structure-Activity Relationship; Thiourea; Urinary Bladder

1984
A comparison of dimaprit, nordimaprit, methylamine and chloroquine as inhibitors of mitogen-induced lymphocyte activation.
    British journal of pharmacology, 1984, Volume: 83, Issue:1

    Topics: Cells, Cultured; Chloroquine; Chromium Radioisotopes; Concanavalin A; Dimaprit; Histamine; Humans; Lymphocyte Activation; Lymphocytes; Methylamines; Mitogens; Phytohemagglutinins; Thiourea; Thymidine

1984
Lack of an effect of drugs acting at histamine receptors on norepinephrine-induced relaxation of porcine coronary arteries.
    Archives internationales de pharmacodynamie et de therapie, 1984, Volume: 272, Issue:2

    Topics: Animals; Coronary Vessels; Dimaprit; Histamine; In Vitro Techniques; Muscle Relaxation; Muscle, Smooth, Vascular; Myocardial Contraction; Norepinephrine; Phenethylamines; Receptors, Histamine; Swine; Thiourea

1984
Specific activation of cyclic AMP-dependent protein kinase(s) by H2-histamine agonists in isolated gastric mucosal cells from guinea-pig.
    Biochimica et biophysica acta, 1980, May-22, Volume: 629, Issue:3

    Topics: Animals; Cimetidine; Cyclic AMP; Dimaprit; Diphenhydramine; Enzyme Activation; Gastric Mucosa; Guanidines; Guinea Pigs; Histamine; Imidazoles; Impromidine; In Vitro Techniques; Protein Kinases; Pyridines; Receptors, Histamine; Receptors, Histamine H2; Thiourea

1980
Histamine receptors on dispersed parathyroid cells from pathological human parathyroid tissue.
    The Journal of clinical endocrinology and metabolism, 1980, Volume: 51, Issue:6

    Topics: Cyclic AMP; Dimaprit; Dose-Response Relationship, Drug; Histamine; Histamine Antagonists; Humans; Hyperparathyroidism; In Vitro Techniques; Parathyroid Glands; Parathyroid Hormone; Receptors, Histamine H2; Thiourea

1980
Cardiac contractile and metabolic effects mediated via the myocardial H2-receptor adenylate cyclase system. Characterization of two new specific H2-receptor agonists, impromidine and dimaprit, in the guinea pig and human myocardium.
    Research in experimental medicine. Zeitschrift fur die gesamte experimentelle Medizin einschliesslich experimenteller Chirurgie, 1981, Volume: 179, Issue:1

    Topics: Adenylyl Cyclases; Animals; Cimetidine; Cyclic AMP; Dimaprit; Dose-Response Relationship, Drug; Female; Guanidines; Guinea Pigs; Histamine; Humans; Imidazoles; Impromidine; Isoproterenol; Metoprolol; Myocardial Contraction; Myocardial Infarction; Myocardium; Phosphoric Diester Hydrolases; Receptors, Histamine; Receptors, Histamine H2; Thiourea; Tyramine

1981
Cyclic AMP increase in canine parotid gland mediated by histamine H2-receptors.
    European journal of pharmacology, 1981, Dec-17, Volume: 76, Issue:4

    Topics: Animals; Cyclic AMP; Dimaprit; Dogs; Female; Histamine; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Parotid Gland; Pyridines; Receptors, Histamine; Receptors, Histamine H2; Thiourea

1981
Pharmacological interactions between ranitidine, cimetidine, metiamide and tiotidine at histamine H2-receptor sites in guinea-pig atria.
    Agents and actions, 1982, Volume: 12, Issue:1-2

    Topics: Animals; Cimetidine; Dimaprit; Drug Interactions; Furans; Guanidines; Guinea Pigs; Heart; Heart Rate; Histamine; In Vitro Techniques; Metiamide; Ranitidine; Receptors, Histamine; Receptors, Histamine H2; Thiazoles; Thiourea

1982
Interaction of histamine with gastric mucosal cells. Effect of histamine agonists on binding and biological response.
    Molecular pharmacology, 1982, Volume: 22, Issue:1

    Topics: Animals; Chemical Phenomena; Chemistry; Cyclic AMP; Dimaprit; Gastric Mucosa; Guinea Pigs; Histamine; In Vitro Techniques; Inosine Monophosphate; Kinetics; Male; Receptors, Histamine; Thiourea

1982
Inotropic and electrophysiological effects of histamine on human ventricular heart muscle.
    The Journal of physiology, 1982, Volume: 330

    Topics: Action Potentials; Adolescent; Adult; Aged; Animals; Child; Child, Preschool; Cyclic AMP; Dimaprit; Female; Guinea Pigs; Heart Ventricles; Histamine; Humans; Isoproterenol; Male; Middle Aged; Myocardial Contraction; Norepinephrine; Papillary Muscles; Receptors, Histamine H2; Stimulation, Chemical; Thionucleotides; Thiourea

1982
Histamine and serotonin suppression of lymphocyte response to phytohemagglutinin and allogeneic cells.
    Cellular immunology, 1984, Volume: 83, Issue:2

    Topics: Animals; Cimetidine; Dimaprit; Drug Antagonism; Female; Histamine; Lymphocyte Activation; Lymphocyte Culture Test, Mixed; Male; Metiamide; Mice; Mice, Inbred Strains; Phytohemagglutinins; Ranitidine; Serotonin; Thiourea

1984
Studies with specific agonists and antagonists of the role of histamine H1- and H2-receptor activation in the pathogenesis of gastric lesions in rats.
    Agents and actions, 1984, Volume: 14, Issue:2

    Topics: Aminopyridines; Animals; Atropine; Dimaprit; Drug Interactions; Female; Histamine; Pyridines; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Stomach Ulcer; Thiourea

1984
Role of histamine H1- and H2-receptors in myoelectric activity of small bowel in the dog.
    The American journal of physiology, 1980, Volume: 238, Issue:1

    Topics: Animals; Dogs; Gastrointestinal Motility; Histamine; Histamine Antagonists; Intestine, Small; Male; Methylhistamines; Metiamide; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea; Tripelennamine

1980
A question of the specificity of rabbit atrial chronotropic histamine receptors and agents which affect their activity.
    Journal of clinical pharmacology, 1980, Volume: 20, Issue:1

    Topics: Animals; Dimaprit; Female; Guinea Pigs; Heart Rate; Histamine; Male; Methylhistamines; Pyridines; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea; Time Factors

1980
Choledochal sphincter relaxation in response to histamine in the primate.
    The Journal of surgical research, 1980, Volume: 28, Issue:4

    Topics: Animals; Cholecystokinin; Dimaprit; Female; Gallbladder; Haplorhini; Histamine; Muscle, Smooth; Papio; Pressure; Pyridines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1980
Dimaprit inhibition of zymosan-stimulated beta-glucuronidase release from human granulocytes.
    Agents and actions, 1980, Volume: 10, Issue:1 Pt 2

    Topics: Adult; Dimaprit; Glucuronidase; Granulocytes; Histamine; Humans; In Vitro Techniques; Lysosomes; Metiamide; Neutrophils; Pyridines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea; Zymosan

1980
Cardiovascular and behavioural changes after i.c.v. infusions of histamine and agonists in conscious goat.
    Agents and actions, 1980, Volume: 10, Issue:1 Pt 2

    Topics: Animals; Behavior, Animal; Dimaprit; Female; Goats; Hemodynamics; Histamine; Injections, Intraventricular; Pyridines; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1980
Evidence for a role of endogenous histamine in central cardiovascular regulation: inhibition of histamine-N-methyltransferase by SKF 91488.
    The Journal of pharmacology and experimental therapeutics, 1981, Volume: 216, Issue:2

    Topics: Animals; Blood Pressure; Brain; Dimaprit; Heart Rate; Hemodynamics; Histamine; Histamine N-Methyltransferase; Male; Methyltransferases; Rats; Thiourea

1981
pH-dependent activity of H1- and H2-histamine receptors in guinea-pig gallbladder.
    The Journal of pharmacology and experimental therapeutics, 1981, Volume: 217, Issue:3

    Topics: Acetylcholine; Animals; Dimaprit; Female; Gallbladder; Guinea Pigs; Histamine; Hydrogen-Ion Concentration; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Potassium Chloride; Pyridines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1981
Vascular studies with histamine in vitro.
    Agents and actions, 1981, Volume: 11, Issue:1-2

    Topics: Animals; Blood Vessels; Cimetidine; Dimaprit; Hindlimb; Histamine; Histamine Antagonists; Male; Rats; Regional Blood Flow; Thiourea; Vasodilator Agents

1981
Hypothalamic superfusion with histamine agonists and antagonists modifies the pressor response to hypothalamic stimulation.
    Agents and actions, 1981, Volume: 11, Issue:1-2

    Topics: Animals; Blood Pressure; Cats; Dimaprit; Electric Stimulation; Histamine; Histamine Antagonists; Hypothalamus; Thiourea

1981
Lack of histamine involvement in parathyroid hormone hypotensive action.
    Pharmacology, 1981, Volume: 22, Issue:5

    Topics: Animals; Blood Pressure; Cimetidine; Dimaprit; Female; Histamine; Hypotension; Male; p-Methoxy-N-methylphenethylamine; Parathyroid Hormone; Peptide Fragments; Promethazine; Propranolol; Pyridines; Rats; Thiourea

1981
Effect of histamine H1- and H2-receptor agonists on gamma-aminobutyric acid (GABA) content in hypothalamus and striatum of the rat brain.
    Archivum immunologiae et therapiae experimentalis, 1980, Volume: 28, Issue:6

    Topics: Animals; Brain Chemistry; Corpus Striatum; Dimaprit; Female; gamma-Aminobutyric Acid; Histamine; Hypothalamus; Methylhistamines; Rats; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1980
Comparison of H2 receptor agonists in rabbit atria and aorta.
    Pharmacology, 1981, Volume: 22, Issue:4

    Topics: Animals; Aorta; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Female; Guanidines; Heart Atria; Heart Rate; Histamine; Imidazoles; Impromidine; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Rabbits; Receptors, Histamine; Receptors, Histamine H2; Thiourea

1981
Further experiments on the pharmacological actions of ergometrine.
    Bollettino della Societa italiana di biologia sperimentale, 1981, Jun-30, Volume: 57, Issue:12

    Topics: Animals; Cattle; Cimetidine; Coronary Vessels; Dimaprit; Ergonovine; Gastric Acid; Guinea Pigs; Histamine; Muscle Contraction; Pyrilamine; Rats; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1981
Characterization of neuronal and vascular histamine receptors mediating the salivary and vasodilator responses to histamine of the dog submandibular gland.
    The Tohoku journal of experimental medicine, 1981, Volume: 134, Issue:1

    Topics: Animals; Dimaprit; Dogs; Female; Histamine; Male; Pyridines; Receptors, Histamine; Regional Blood Flow; Salivation; Submandibular Gland; Thiourea; Vasodilation

1981
Cerebral circulation and histamine: 1. Participation of vascular H1- and H2-receptors in vasodilatory responses to carotid arterial infusion.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 1981, Volume: 1, Issue:1

    Topics: Animals; Blood-Brain Barrier; Carotid Artery, Internal; Cerebrovascular Circulation; Dimaprit; Glucose; Histamine; Injections, Intra-Arterial; Male; Pyridines; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea; Urea; Vasodilation

1981
Effect of histamine agonists and antagonists on the production of murine reaginic antibodies.
    International journal of immunopharmacology, 1981, Volume: 3, Issue:4

    Topics: Animals; Antibody Formation; Dimaprit; Histamine; Histamine Antagonists; Immunoglobulin E; Male; Methylhistamines; Metiamide; Mice; Reagins; Receptors, Histamine; Thiourea

1981
Changes in the response of guinea-pig airways in vivo and in vitro to cimetidine and propranolol during development.
    British journal of pharmacology, 1982, Volume: 75, Issue:3

    Topics: Aging; Airway Resistance; Animals; Bronchi; Cimetidine; Dimaprit; Female; Guanidines; Guinea Pigs; Histamine; In Vitro Techniques; Methylhistamines; Muscle Contraction; Propranolol; Receptors, Histamine; Receptors, Histamine H2; Thiourea; Trachea

1982
Hypothalamic superfusion with histamine agonists and antagonists modifies the pressor response to hypothalamic stimulation.
    Journal of autonomic pharmacology, 1981, Volume: 1, Issue:2

    Topics: Animals; Blood Pressure; Cats; Dimaprit; Electric Stimulation; Female; Histamine; Histamine Antagonists; Hypothalamus; Male; Methylhistamines; Metiamide; Sympathomimetics; Thiourea; Time Factors

1981
Effects of alkyl analogues of histamine and metiamide on the isolated guinea pig heart.
    Pharmacology, 1981, Volume: 22, Issue:2

    Topics: Animals; Female; Guinea Pigs; Heart; Heart Rate; Histamine; In Vitro Techniques; Male; Metiamide; Myocardial Contraction; Papillary Muscles; Thiourea

1981
Histamine H1- and H2-receptors in canine renal artery in vivo and in vitro.
    Revista espanola de fisiologia, 1981, Volume: 37, Issue:1

    Topics: Animals; Blood Flow Velocity; Blood Pressure; Diphenhydramine; Dogs; Dose-Response Relationship, Drug; Female; Heart Rate; Histamine; Male; Metiamide; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Renal Artery; Thiourea

1981
Influence of metiamide and atropine on acid and pepsin secretion in the anaesthetized Heidenhain cat.
    Agents and actions, 1981, Volume: 11, Issue:1-2

    Topics: Anesthesia; Animals; Atropine; Carbachol; Cats; Drug Interactions; Gastric Acid; Histamine; Male; Metiamide; Pentagastrin; Pepsin A; Salicylates; Thiourea

1981
Effects of histamine and antihistamines on the kinetics of carbon dioxide in the rat.
    Physiological chemistry and physics, 1981, Volume: 13, Issue:3

    Topics: Animals; Bicarbonates; Carbon Dioxide; Carbon Radioisotopes; Chlorpheniramine; Histamine; Kinetics; Metiamide; Radioisotope Dilution Technique; Rats; Rats, Inbred Strains; Thiourea

1981
Histamine content of tick attachment sites and the effects of H1 and H2 histamine antagonists on the expression of resistance.
    Annals of tropical medicine and parasitology, 1982, Volume: 76, Issue:2

    Topics: Animals; Dermacentor; Guinea Pigs; Histamine; Immunity, Innate; Male; Metiamide; Promethazine; Skin; Thiourea; Tick Infestations

1982
Does the histaminergic system mediate bombesin/GRP-induced suppression of food intake?
    The American journal of physiology, 1994, Volume: 267, Issue:6 Pt 2

    Topics: Animals; Behavior, Animal; Bombesin; Eating; Gastrin-Releasing Peptide; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Male; Methylhistamines; Motor Activity; Peptides; Piperidines; Rats; Rats, Sprague-Dawley; Satiation; Sincalide; Thiourea

1994
Inhibitory H3 receptors on sympathetic nerves of the pithed rat: activation by endogenous histamine and operation in spontaneously hypertensive rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 355, Issue:2

    Topics: Adrenergic Fibers; Animals; Blood Pressure; Decerebrate State; Electric Stimulation; Histamine; Histamine Agonists; Histamine Antagonists; Hypertension; Imidazoles; Male; Methylhistamines; Piperidines; Pyrimethamine; Rats; Rats, Wistar; Receptors, Histamine H3; Thiourea; Vagotomy; Vascular Resistance

1997
Some histamine-related compounds interacting with the benzylamine-oxidizing activity of rat white adipocytes.
    The Journal of pharmacy and pharmacology, 1997, Volume: 49, Issue:5

    Topics: Adipocytes; Amine Oxidase (Copper-Containing); Animals; Benzylamines; Cells, Cultured; Dialysis; Histamine; Male; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Oxidation-Reduction; Rats; Rats, Wistar; Structure-Activity Relationship; Thiourea

1997
Mutual interactions of the presynaptic histamine H3 and prostaglandin EP3 receptors on the noradrenergic terminals in the mouse brain.
    Neuroscience, 1997, Volume: 79, Issue:1

    Topics: Animals; Brain; Calcium; Cerebral Cortex; Dinoprostone; Electric Stimulation; Histamine; Histamine Agonists; Imidazoles; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Nerve Endings; Norepinephrine; Radioisotope Dilution Technique; Rats; Receptors, Adrenergic, alpha-2; Receptors, Histamine H3; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP3 Subtype; Thiourea; Tritium

1997
Identification of histamine H3 receptors in the tail artery from normotensive and spontaneously hypertensive rats.
    Journal of cardiovascular pharmacology, 1997, Volume: 29, Issue:6

    Topics: Adrenergic alpha-2 Receptor Antagonists; Animals; Arteries; Electric Stimulation; Histamine; Histamine Agonists; Imidazoles; Male; Norepinephrine; Piperidines; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Histamine H3; Sympathetic Fibers, Postganglionic; Thiourea; Yohimbine

1997
Comparison of the effects of histamine and N(alpha)-methylhistamine on neuronal function in the guinea-pig oesophagus and ileum.
    The Journal of pharmacy and pharmacology, 1997, Volume: 49, Issue:12

    Topics: Acetylcholine; Animals; Atropine; Dose-Response Relationship, Drug; Electric Stimulation; Esophagus; Guinea Pigs; Histamine; Histamine Antagonists; Ileum; Imidazoles; In Vitro Techniques; Methylhistamines; Muscle, Skeletal; Muscle, Smooth; Neurons; Neurons, Afferent; Pyrilamine; Receptors, Cholinergic; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P; Tetrodotoxin; Thiourea; Vagus Nerve

1997
Stimulation of pulmonary rapidly adapting receptors by inhaled wood smoke in rats.
    The Journal of physiology, 1998, Apr-15, Volume: 508 ( Pt 2)

    Topics: Animals; Bronchodilator Agents; Cyclooxygenase Inhibitors; Female; Free Radical Scavengers; Histamine; Indomethacin; Isoproterenol; Lung; Male; Mechanoreceptors; Neurons, Afferent; Rats; Rats, Sprague-Dawley; Smoke; Stimulation, Chemical; Thiourea

1998
Increase of acetylcholine release from cortex of freely moving rats by administration of histamine into the nucleus basalis magnocellularis.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1998, Volume: 47 Suppl 1

    Topics: Acetylcholine; Animals; Cerebral Cortex; Cimetidine; Electroencephalography; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Imidazoles; Male; Neurons; Rats; Rats, Wistar; Substantia Innominata; Telencephalon; Thiourea; Triprolidine

1998
Histamine inhibits the production of interleukin-12 through interaction with H2 receptors.
    The Journal of clinical investigation, 1998, Nov-15, Volume: 102, Issue:10

    Topics: Dinoprostone; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H2 Antagonists; Humans; Imidazoles; Interleukin-12; Interleukins; Monocytes; Ranitidine; Receptors, Histamine H2; RNA, Messenger; Thiourea; Triprolidine

1998
Histamine H3 receptor-mediated inhibition of noradrenaline release in the human brain.
    Fundamental & clinical pharmacology, 1999, Volume: 13, Issue:1

    Topics: Animals; Brain; Cerebral Cortex; Dimethindene; Electric Stimulation; Hippocampus; Histamine; Histamine Agonists; Histamine Antagonists; Humans; Imidazoles; Male; Mice; Mice, Inbred Strains; Norepinephrine; Piperidines; Ranitidine; Receptors, Histamine H3; Thiourea; Tritium

1999
Histaminergic and catecholaminergic interactions in the central regulation of vasopressin and oxytocin secretion.
    Endocrinology, 1999, Volume: 140, Issue:8

    Topics: Animals; Arginine Vasopressin; Blood Pressure; Cerebral Ventricles; Cimetidine; Epinephrine; Histamine; Histamine Agonists; Hypothalamus; Imidazoles; Infusions, Parenteral; Male; Methylhistamines; Norepinephrine; Oxytocin; Pituitary Gland, Posterior; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H2; Thiazoles; Thiourea

1999
Histamine H(3) receptor-mediated inhibition of endogenous acetylcholine release from the isolated, vascularly perfused rat stomach.
    European journal of pharmacology, 2000, Mar-24, Volume: 392, Issue:1-2

    Topics: Acetylcholine; Animals; Atropine; Gastric Mucosa; GTP-Binding Proteins; Histamine; Imidazoles; Male; Methylhistamines; Perfusion; Pertussis Toxin; Piperidines; Rats; Rats, Wistar; Receptors, Histamine H3; Thiourea; Vagus Nerve; Virulence Factors, Bordetella

2000
Mepyramine but not cimetidine or clobenpropit blocks pertussis toxin-induced histamine sensitization in rats.
    British journal of pharmacology, 2000, Volume: 129, Issue:8

    Topics: Animals; Blood Gas Analysis; Blood Pressure; Cimetidine; Drug Interactions; Histamine; Histamine Antagonists; Imidazoles; Male; Pertussis Toxin; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine; Thiourea; Virulence Factors, Bordetella

2000
Participation of GABAergic and histaminergic systems in inhibiting amygdaloid kindled seizures.
    Japanese journal of pharmacology, 2000, Volume: 82, Issue:1

    Topics: Amygdala; Animals; Bicuculline; Diazepam; gamma-Aminobutyric Acid; Histamine; Imidazoles; Kindling, Neurologic; Male; Muscimol; Rats; Rats, Wistar; Seizures; Thiourea; Valproic Acid

2000
Influence of different histamine receptor agonists and antagonists on apomorphine-induced licking behavior in rat.
    European journal of pharmacology, 2000, Sep-15, Volume: 404, Issue:1-2

    Topics: Animals; Apomorphine; Chlorpheniramine; Dimaprit; Diphenhydramine; Dopamine Agonists; Drug Interactions; Famotidine; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Male; Piperidines; Ranitidine; Rats; Rats, Sprague-Dawley; Stereotyped Behavior; Thiourea; Toluidines

2000
Cloning and characterization of a novel human histamine receptor.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 296, Issue:3

    Topics: Amino Acid Sequence; Cells, Cultured; Cloning, Molecular; Histamine; Histamine Agonists; Humans; Imidazoles; Molecular Sequence Data; Radioligand Assay; Receptors, Histamine; Receptors, Histamine H3; RNA, Messenger; Sequence Homology, Amino Acid; Thiourea; Tissue Distribution; Transfection

2001
Histamine H(3) receptor-mediated inhibition of depolarization-induced, dopamine D(1) receptor-dependent release of [(3)H]-gamma-aminobutryic acid from rat striatal slices.
    British journal of pharmacology, 2001, Volume: 133, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Calcium; Dopamine; Dopamine D2 Receptor Antagonists; gamma-Aminobutyric Acid; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; In Vitro Techniques; Male; Membrane Potentials; Neostriatum; Piperidines; Potassium; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Histamine H3; Reserpine; Sulpiride; Thiourea

2001
Effect of histamine H3-receptor antagonist clobenpropit on spatial memory of radial maze performance in rats.
    Acta pharmacologica Sinica, 2000, Volume: 21, Issue:10

    Topics: Animals; Brain; Histamine; Histamine Antagonists; Imidazoles; Injections, Intraventricular; Male; Maze Learning; Memory Disorders; Rats; Rats, Wistar; Scopolamine; Thiourea

2000
Dynamics of histamine H(3) receptor antagonists on brain histamine metabolism: do all histamine H(3) receptor antagonists act at a single site?
    European journal of pharmacology, 2001, Nov-16, Volume: 431, Issue:2

    Topics: Analysis of Variance; Animals; Binding Sites; Brain; Histamine; Histamine Antagonists; Imidazoles; Male; Methylhistamines; Mice; Pargyline; Piperidines; Rats; Receptors, Histamine H3; Thiourea

2001
Presynaptic H3 autoreceptors modulate histamine synthesis through cAMP pathway.
    Molecular pharmacology, 2002, Volume: 61, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Brain; Bucladesine; Colforsin; Cyclic AMP; Drug Interactions; Histamine; Imidazoles; In Vitro Techniques; Male; Piperidines; Potassium; Rats; Rats, Sprague-Dawley; Receptors, Histamine H3; Thionucleotides; Thiourea

2002
Molecular and pharmacological characterization of the mouse histamine H3 receptor.
    European journal of pharmacology, 2003, Apr-25, Volume: 467, Issue:1-3

    Topics: Alternative Splicing; Amino Acid Sequence; Animals; Brain; Calcium; Cells, Cultured; Chlorocebus aethiops; Cloning, Molecular; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Humans; Imidazoles; Mice; Molecular Sequence Data; Rats; Receptors, Histamine H3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sequence Homology; Thiourea

2003
Effects of endogenous histamine on seizure development of pentylenetetrazole-induced kindling in rats.
    Pharmacology, 2003, Volume: 69, Issue:1

    Topics: Animals; Dose-Response Relationship, Drug; Drug Synergism; Histamine; Histamine Release; Histidine; Imidazoles; Injections, Intraventricular; Kindling, Neurologic; Male; Methylhistidines; Pentylenetetrazole; Piperidines; Pyrilamine; Rats; Rats, Sprague-Dawley; Seizures; Thiourea

2003
Waking selective neurons in the posterior hypothalamus and their response to histamine H3-receptor ligands: an electrophysiological study in freely moving cats.
    Behavioural brain research, 2003, Sep-15, Volume: 144, Issue:1-2

    Topics: Action Potentials; Animals; Cats; Drug Administration Schedule; Electroencephalography; Electromyography; Electrooculography; Electrophysiology; Female; Geniculate Bodies; Hippocampus; Histamine; Histamine Agonists; Histamine Antagonists; Hypothalamus, Posterior; Imidazoles; Immunohistochemistry; Male; Methylhistamines; Neurons; Thiourea; Time Factors; Wakefulness

2003
Histamine induces cytoskeletal changes in human eosinophils via the H(4) receptor.
    British journal of pharmacology, 2003, Volume: 140, Issue:6

    Topics: Actins; Calcium; CD11b Antigen; Cell Size; Chemokine CCL11; Chemokines, CC; Chemotaxis; Clozapine; Cytoskeleton; Dose-Response Relationship, Drug; Eosinophils; Histamine; Histamine Agonists; Histamine Antagonists; Humans; Imidazoles; Pertussis Toxin; Piperidines; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Thiourea; Up-Regulation

2003
Histamine H3 receptors regulate vascular permeability changes in the skin of mast cell-deficient mice.
    International immunopharmacology, 2003, Volume: 3, Issue:12

    Topics: Animals; Capillary Permeability; Chlorpheniramine; Diphenhydramine; Evans Blue; Female; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Injections, Intradermal; Injections, Intravenous; Isothiuronium; Mast Cells; Mice; Mice, Mutant Strains; Piperidines; Receptors, Histamine H3; Skin; Thiourea; Tryptophan

2003
[Thiourea and acute histamine intoxication; relation between sensitivity to anaphylactic shock and to histamine shock during functional variations of the thyroid].
    Rassegna di neurologia vegetativa, 1950, Volume: 8, Issue:2

    Topics: Anaphylaxis; Drug-Related Side Effects and Adverse Reactions; Histamine; Psychoses, Substance-Induced; Shock; Thiourea; Thyroid Gland

1950
[Mechanisms of the effect of brain histamine on chronic epilepsy induced by pentylenetetrazole].
    Zhejiang da xue xue bao. Yi xue ban = Journal of Zhejiang University. Medical sciences, 2004, Volume: 33, Issue:3

    Topics: Animals; Brain; Chronic Disease; Dose-Response Relationship, Drug; Epilepsy; Histamine; Histidine; Imidazoles; Male; Pentylenetetrazole; Piperidines; Rats; Rats, Sprague-Dawley; Thiourea

2004
Cloning and expression of the mouse histamine H3 receptor: evidence for multiple isoforms.
    Journal of neurochemistry, 2004, Volume: 90, Issue:6

    Topics: Animals; Blotting, Northern; Brain; Chlorocebus aethiops; Cloning, Molecular; Competitive Bidding; COS Cells; Gene Expression; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; In Situ Hybridization; Iodine Radioisotopes; Isoenzymes; Mice; Piperidines; Radioligand Assay; Rats; Receptors, Histamine H3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiourea; Transfection

2004
H3 autoreceptors modulate histamine synthesis through calcium/calmodulin- and cAMP-dependent protein kinase pathways.
    Molecular pharmacology, 2005, Volume: 67, Issue:1

    Topics: Amino Acid Sequence; Animals; Brain; Calcium Channel Blockers; Calcium-Calmodulin-Dependent Protein Kinases; Cyclic AMP-Dependent Protein Kinase Type II; Cyclic AMP-Dependent Protein Kinases; Histamine; Histamine Agonists; Histidine Decarboxylase; Imidazoles; In Vitro Techniques; Male; Molecular Sequence Data; Peptide Fragments; Pertussis Toxin; Phosphorylation; Rats; Rats, Sprague-Dawley; Receptors, Histamine H3; Recombinant Proteins; Thiourea

2005
Inhibition of tryptase release from human colon mast cells by histamine receptor antagonists.
    Asian Pacific journal of allergy and immunology, 2005, Volume: 23, Issue:1

    Topics: Calcimycin; Cells, Cultured; Cimetidine; Colon; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Imidazoles; Ionophores; Mast Cells; Serine Endopeptidases; Serine Proteinase Inhibitors; Terfenadine; Thiourea; Tryptases

2005
Physiological role of the sodium-calcium exchanger in tracheal smooth muscle of guinea pig.
    Journal of muscle research and cell motility, 2004, Volume: 25, Issue:8

    Topics: Amiloride; Animals; Guinea Pigs; Histamine; Muscle, Smooth; Nifedipine; Sodium-Calcium Exchanger; Thiourea; Trachea

2004
Effects of intracerebroventricular administration of ultra low doses of histaminergic drugs on morphine state-dependent memory of passive avoidance in mice.
    Behavioural brain research, 2006, Jan-06, Volume: 166, Issue:1

    Topics: Analgesics, Opioid; Animals; Avoidance Learning; Behavior, Animal; Dose-Response Relationship, Drug; Drug Interactions; Histamine; Histamine Agents; Imidazoles; Injections, Intraventricular; Male; Memory; Mice; Morphine; Morphine Dependence; Pyrilamine; Reaction Time; Thiourea

2006
Histamine excites neonatal rat sympathetic preganglionic neurons in vitro via activation of H1 receptors.
    Journal of neurophysiology, 2006, Volume: 95, Issue:4

    Topics: Action Potentials; Animals; Animals, Newborn; Autonomic Fibers, Preganglionic; Barium; Dimaprit; Female; Ganglia, Sympathetic; Histamine; Histamine Agonists; Histamine H1 Antagonists; Imidazoles; In Vitro Techniques; Male; Membrane Potentials; Neurons; Patch-Clamp Techniques; Potassium; Rats; Rats, Inbred WKY; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiourea; Triprolidine

2006
Histamine increases sickle erythrocyte adherence to endothelium.
    British journal of haematology, 2006, Volume: 132, Issue:4

    Topics: Analysis of Variance; Anemia, Sickle Cell; Cell Adhesion; Cells, Cultured; Endothelial Cells; Endothelium, Vascular; Erythrocytes; Famotidine; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Imidazoles; Methylhistamines; P-Selectin; Piperidines; Pyrilamine; Stimulation, Chemical; Thiazoles; Thiourea; Venules

2006
Histaminergic neurons protect the developing hippocampus from kainic acid-induced neuronal damage in an organotypic coculture system.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2006, Jan-25, Volume: 26, Issue:4

    Topics: Animals; Cell Death; Cells, Cultured; Coculture Techniques; Convulsants; Hippocampus; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Hypothalamus, Anterior; Hypothalamus, Posterior; Imidazoles; Kainic Acid; Methylhistidines; Microscopy, Confocal; Neurons; Neuroprotective Agents; Organ Culture Techniques; Piperidines; Pyrilamine; Rats; Rats, Sprague-Dawley; Receptors, Histamine H1; Receptors, Histamine H3; Thiourea; Triprolidine

2006
Detection of multiple H3 receptor affinity states utilizing [3H]A-349821, a novel, selective, non-imidazole histamine H3 receptor inverse agonist radioligand.
    British journal of pharmacology, 2006, Volume: 148, Issue:5

    Topics: Animals; Binding, Competitive; Biphenyl Compounds; Cells, Cultured; Guanosine Diphosphate; Histamine; Histamine Agonists; Histamine Antagonists; Humans; Imidazoles; Methylhistamines; Models, Biological; Protein Binding; Radioligand Assay; Rats; Receptors, Histamine H3; Thiourea

2006
Constitutive activity of H3 autoreceptors modulates histamine synthesis in rat brain through the cAMP/PKA pathway.
    Neuropharmacology, 2006, Volume: 51, Issue:3

    Topics: Animals; Biphenyl Compounds; Brain; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; In Vitro Techniques; Male; Models, Biological; Nitriles; Piperidines; Potassium; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Histamine H3; Thiourea

2006
Pre-synaptic histamine H3 receptors regulate glutamate, but not GABA release in rat thalamus.
    Neuropharmacology, 2007, Volume: 52, Issue:2

    Topics: 4-Aminopyridine; Animals; Dose-Response Relationship, Drug; Drug Interactions; Evoked Potentials; gamma-Aminobutyric Acid; Glutamic Acid; Guanosine 5'-O-(3-Thiotriphosphate); Histamine; Histamine Antagonists; Imidazoles; In Vitro Techniques; Male; Methylhistamines; Pertussis Toxin; Presynaptic Terminals; Protein Binding; Rats; Rats, Wistar; Receptors, Histamine H3; Synaptosomes; Thalamus; Thiourea; Tritium

2007
The reverse mode of the Na(+)/Ca(2+) exchanger provides a source of Ca(2+) for store refilling following agonist-induced Ca(2+) mobilization.
    American journal of physiology. Lung cellular and molecular physiology, 2007, Volume: 292, Issue:2

    Topics: Acetylcholine; Animals; Caffeine; Calcium; Calcium Signaling; Cattle; Histamine; In Vitro Techniques; Muscle Contraction; Myocytes, Smooth Muscle; Potassium Chloride; Respiratory System; Serotonin; Sodium; Sodium-Calcium Exchanger; Thiourea

2007
[Reversing effect of histamine on neurotoxicity induced by beta-amyloid1-42].
    Zhejiang da xue xue bao. Yi xue ban = Journal of Zhejiang University. Medical sciences, 2007, Volume: 36, Issue:2

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Animals; Benzothiazoles; Diphenhydramine; Dose-Response Relationship, Drug; Histamine; Histamine H2 Antagonists; Histamine H3 Antagonists; Imidazoles; Neuroprotective Agents; PC12 Cells; Phenoxypropanolamines; Piperidines; Rats; Receptors, Histamine H2; Receptors, Histamine H3; Thiourea

2007
Functional coupling between the Na+/Ca2+ exchanger and nonselective cation channels during histamine stimulation in guinea pig tracheal smooth muscle.
    American journal of physiology. Lung cellular and molecular physiology, 2007, Volume: 293, Issue:1

    Topics: Animals; Cell Separation; Fluorescence; Guinea Pigs; Histamine; Imidazoles; In Vitro Techniques; Ion Channel Gating; Ion Channels; Isometric Contraction; Male; Meglumine; Models, Biological; Myocytes, Smooth Muscle; Sodium; Sodium-Calcium Exchanger; Thiourea; Trachea

2007
The plasma membrane Na+/Ca2+ exchange inhibitor KB-R7943 is also a potent inhibitor of the mitochondrial Ca2+ uniporter.
    British journal of pharmacology, 2007, Volume: 151, Issue:5

    Topics: Aequorin; Calcium; Calcium Channels; Cell Membrane; Cells, Cultured; Cytosol; Fluorescent Dyes; Fura-2; HeLa Cells; Histamine; Homeostasis; Humans; Inositol 1,4,5-Trisphosphate; Inositol 1,4,5-Trisphosphate Receptors; Membrane Potentials; Mitochondria; Sodium-Calcium Exchanger; Thiourea

2007
Histamine downregulates monocyte CCL2 production through the histamine H4 receptor.
    The Journal of allergy and clinical immunology, 2007, Volume: 120, Issue:2

    Topics: Calcium; Cells, Cultured; Chemokine CCL2; Chemotaxis, Leukocyte; Down-Regulation; Histamine; Histamine Agonists; Humans; Imidazoles; Indoles; Interferon-gamma; Matrix Metalloproteinase 1; Matrix Metalloproteinase 3; Matrix Metalloproteinase 8; Methylhistamines; Monocytes; Piperazines; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Thiourea; Up-Regulation

2007
Role of histamine in ghrelin-induced gastroprotection against acute gastric lesions.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 2007, Volume: 56 Suppl 1

    Topics: Animals; Anti-Ulcer Agents; Cytoprotection; Ethanol; Gastric Mucosa; Ghrelin; Histamine; Histamine Antagonists; Imidazoles; Male; Peptide Hormones; Ranitidine; Rats; Rats, Wistar; Regional Blood Flow; Thiourea

2007
The role of histamine in human mammary carcinogenesis: H3 and H4 receptors as potential therapeutic targets for breast cancer treatment.
    Cancer biology & therapy, 2008, Volume: 7, Issue:1

    Topics: Adult; Aged; Breast; Breast Neoplasms; Cell Movement; Cell Proliferation; Female; Histamine; Histidine Decarboxylase; Humans; Imidazoles; Middle Aged; Proliferating Cell Nuclear Antigen; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H3; Receptors, Histamine H4; Thiourea

2008
Comparison of the effect of an H(3)-inverse agonist on energy intake and hypothalamic histamine release in normal mice and leptin resistant mice with high fat diet-induced obesity.
    Behavioural brain research, 2008, Apr-09, Volume: 188, Issue:2

    Topics: Analysis of Variance; Animals; Behavior, Animal; Body Weight; Chromatography, High Pressure Liquid; Electrochemistry; Energy Intake; Fats; Histamine; Histamine H3 Antagonists; Hypothalamus; Imidazoles; Leptin; Male; Mice; Mice, Inbred C57BL; Microdialysis; Obesity; Thiourea; Time Factors

2008
Substance P is involved in the effect of histamine H3 receptor agonist, Sch 50971 on nasal allergic symptoms in mice.
    International immunopharmacology, 2008, Volume: 8, Issue:8

    Topics: Animals; Capsaicin; Cetirizine; Disease Models, Animal; Female; Histamine; Histamine Agonists; Histamine H1 Antagonists, Non-Sedating; Imidazoles; Mice; Mice, Inbred BALB C; Ovalbumin; Piperidines; Pyrrolidines; Receptors, Histamine H3; Rhinitis, Allergic, Perennial; Substance P; Thiourea

2008
Histamine H4 receptors modulate dendritic cell migration through skin--immunomodulatory role of histamine.
    Allergy, 2008, Volume: 63, Issue:10

    Topics: Animals; Cell Movement; Chemotaxis, Leukocyte; Dendritic Cells; Female; Guinea Pigs; Histamine; Histamine H3 Antagonists; Imidazoles; Immunologic Factors; Injections, Intradermal; Mice; Mice, Inbred BALB C; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H3; Receptors, Histamine H4; Skin; Thiourea

2008
The role of histamine 3 receptors in the control of food intake in a seasonal model of obesity: the Siberian hamster.
    Behavioural pharmacology, 2009, Volume: 20, Issue:2

    Topics: Animals; Body Temperature; Cell Line, Transformed; Cricetinae; Disease Models, Animal; Eating; Histamine; Imidazoles; Injections, Intraventricular; Motor Activity; Obesity; Phodopus; Photoperiod; Piperidines; Receptors, Histamine H3; Seasons; Thiourea; Transfection

2009
Withdrawal from repeated administration of morphine alters histamine-induced anxiogenic effects produced by intra-ventral hippocampal microinjection.
    Journal of psychopharmacology (Oxford, England), 2010, Volume: 24, Issue:6

    Topics: Analysis of Variance; Animals; Anxiety; Behavior, Animal; Hippocampus; Histamine; Histamine Antagonists; Imidazoles; Male; Microinjections; Morphine; Motor Activity; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Substance Withdrawal Syndrome; Thiourea

2010
The histamine H receptor as a new target for treatment of canine inflammatory skin diseases.
    Veterinary dermatology, 2009, Volume: 20, Issue:5-6

    Topics: Animals; Calcium; Cell Line; Dog Diseases; Dogs; Dose-Response Relationship, Drug; Female; Guanidines; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Indoles; Inflammation; Intercellular Signaling Peptides and Proteins; Male; Mastocytoma; Mice; Mice, Inbred BALB C; Peptides; Piperazines; Receptors, G-Protein-Coupled; Receptors, Histamine; Skin Diseases; Thiourea; Wasp Venoms

2009
Electrophysiological characterization of store-operated and agonist-induced Ca2+ entry pathways in endothelial cells.
    Pflugers Archiv : European journal of physiology, 2010, Volume: 460, Issue:1

    Topics: Barium; Calcium; Calcium Channels; Calcium Signaling; Calcium-Transporting ATPases; Cell Line; Endoplasmic Reticulum; Endothelial Cells; Enzyme Inhibitors; Histamine; Humans; Membrane Potentials; Nickel; Patch-Clamp Techniques; Sodium; Sodium-Calcium Exchanger; Thapsigargin; Thiourea; Time Factors; Transfection

2010
Beneficial interaction between clobenpropit and pyridoxine in prevention of electroshock-induced seizures in mice: lack of histaminergic mechanisms.
    Human & experimental toxicology, 2011, Volume: 30, Issue:1

    Topics: Animals; Anticonvulsants; Brain; Drug Interactions; Electroshock; Female; Histamine; Histamine H3 Antagonists; Histidine Decarboxylase; Imidazoles; Male; Mice; Pyridoxine; Seizures; Thiourea

2011
Histamine H3 receptor agonists decrease hypothalamic histamine levels and increase stereotypical biting in mice challenged with methamphetamine.
    Neurochemical research, 2011, Volume: 36, Issue:10

    Topics: Animals; Behavior, Animal; Central Nervous System Stimulants; Histamine; Histamine Agonists; Hypothalamus; Imidazoles; Male; Methamphetamine; Methylhistamines; Mice; Motor Activity; Piperidines; Random Allocation; Stereotyped Behavior; Thiourea

2011
Role of H4 receptor in histamine-mediated responses in human melanoma.
    Melanoma research, 2011, Volume: 21, Issue:5

    Topics: Cell Differentiation; Cell Growth Processes; Cell Line, Tumor; Guanidines; Histamine; Humans; Imidazoles; Immunohistochemistry; Indoles; Melanoma; Piperazines; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; RNA, Messenger; Skin Neoplasms; Thiourea

2011
Proxyfan acts as a neutral antagonist of histamine H3 receptors in the feeding-related hypothalamic ventromedial nucleus.
    British journal of pharmacology, 2012, Volume: 167, Issue:5

    Topics: Animals; Eating; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Male; Mice; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Histamine H3; Thiourea; Ventromedial Hypothalamic Nucleus

2012
Identification and pharmacological characterization of the histamine H3 receptor in cultured rat astrocytes.
    European journal of pharmacology, 2013, Nov-15, Volume: 720, Issue:1-3

    Topics: Animals; Animals, Newborn; Astrocytes; Binding, Competitive; Brain; Cells, Cultured; Ciprofloxacin; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Methylhistamines; Piperidines; Rats; Rats, Wistar; Receptors, Histamine H3; RNA, Messenger; Thiourea

2013
Role of histamine receptors in the effects of histamine on the production of reactive oxygen species by whole blood phagocytes.
    Life sciences, 2014, Mar-28, Volume: 100, Issue:1

    Topics: Benzimidazoles; Dimaprit; Guanidines; Histamine; Histamine Agonists; Humans; Male; Methylhistamines; Phagocytes; Reactive Oxygen Species; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H2; Receptors, Histamine H4; Thiourea

2014
Histamine H3 receptor antagonists display antischizophrenic activities in rats treated with MK-801.
    Journal of basic and clinical physiology and pharmacology, 2016, Sep-01, Volume: 27, Issue:5

    Topics: Animals; Antipsychotic Agents; Behavior, Animal; Disease Models, Animal; Dizocilpine Maleate; Histamine; Histamine H3 Antagonists; Imidazoles; Methylhistamines; Motor Activity; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Schizophrenia; Thiourea

2016
Histamine H
    British journal of pharmacology, 2017, Volume: 174, Issue:1

    Topics: Animals; Dose-Response Relationship, Drug; Guanidines; Histamine; Inflammation; Male; Mice; Neuralgia; Oxidative Stress; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Spinal Cord Injuries; Structure-Activity Relationship; Thiourea

2017
Natural amines inhibit activation of human plasmacytoid dendritic cells through CXCR4 engagement.
    Nature communications, 2017, 02-09, Volume: 8

    Topics: Amines; Ammonium Compounds; Animals; Dendritic Cells; Histamine; HIV; Humans; Imidazoles; Interferon Type I; Mice; Orthomyxoviridae; Receptors, CXCR4; Receptors, Histamine; Thiourea; TNF-Related Apoptosis-Inducing Ligand

2017
Intra-vermis H4 receptor agonist impairs performance in anxiety- and fear-mediated models.
    Brain research bulletin, 2017, Volume: 135

    Topics: Animals; Anxiety; Anxiety Disorders; Avoidance Learning; Cerebellar Vermis; Emotions; Fear; Guanidines; Histamine; Histamine H1 Antagonists; Male; Maze Learning; Memory; Memory Consolidation; Mice; Microinjections; Receptors, Histamine H4; Thiourea

2017
Visualization of the activation of the histamine H3 receptor (H3R) using novel fluorescence resonance energy transfer biosensors and their potential application to the study of H3R pharmacology.
    The FEBS journal, 2018, Volume: 285, Issue:12

    Topics: Bacterial Proteins; Biosensing Techniques; Cyclic AMP; Fluorescence Resonance Energy Transfer; Gene Expression; Green Fluorescent Proteins; HEK293 Cells; Histamine; Histamine Agonists; Histamine H3 Antagonists; Humans; Imidazoles; Kinetics; Luminescent Proteins; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Phosphorylation; Plasmids; Receptors, Histamine H3; Thiourea; Transfection; Tritium

2018
Disruption of histamine/H
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 2019, Volume: 70, Issue:2

    Topics: Animals; Cells, Cultured; Cicatrix; Collagen; Heart; Histamine; Imidazoles; Male; Mast Cells; Myocardial Infarction; Myofibroblasts; Rats; Rats, Wistar; Receptors, Histamine; Thiourea

2019
Histamine H
    European journal of pharmacology, 2020, Feb-05, Volume: 868

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic Neurons; Animals; Benzimidazoles; Clonidine; Disease Models, Animal; Guanidines; Histamine; Humans; Injections, Spinal; Locus Coeruleus; Male; Mice; Mice, Knockout; Microinjections; Neuralgia; Norepinephrine; Pain Management; Receptors, Histamine H4; Thiourea

2020