histamine and pirenzepine

histamine has been researched along with pirenzepine in 36 studies

Research

Studies (36)

TimeframeStudies, this research(%)All Research%
pre-199017 (47.22)18.7374
1990's16 (44.44)18.2507
2000's2 (5.56)29.6817
2010's1 (2.78)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Siergiejko, Z1
Biggs, DF; Yang, ZJ1
Ballabeni, V; Barocelli, E; Impicciatore, M; Lavezzo, A; Morini, G1
Baron, E; Boer, R; Eltze, M; Kromer, W1
Taché, Y; Walsh, JH; Yanagisawa, K; Yang, H1
Haga, T; Honda, N; Ichiyama, A; Kajimura, M; Kaneko, E1
O'Donnell, ME1
Cieszkowski, M; Konturek, SJ; Kromer, W; Szewczyk, K; Tasler, J1
Barrantes, MA; Blosser, JC; Manian, AA; McCreedy, SA; Palmer, GC1
Vatier, J1
Cook, PG; Hanson, CA; Risley, EA; Torchiana, ML; Wesley, CA; Westrick, BL; Wiese, SR; Williams, M1
Costa, E; Eva, C1
Lee, L; Smith, TL; Yamamura, HI1
Allescher, HD; Berezin, I; Daniel, EE; Jury, J1
Okada, T; Umeda, Y1
Ishii, K; Kato, R1
Ekelund, M; Håkanson, R; Vallgren, S1
Tanaka, C; Taniyama, K; Tsai, LH1
Rosenfeld, GC1
Bauer, P; Bonfils, S; Mignon, M; Vatier, J1
Búzás, G; Domuta, M; Puşcaş, I; Surányi, P1
Cotton, PB; Eugenides, N; Hobsley, M; Stockbrügger, RW1
Elzinga, CR; Meurs, H; Roffel, AF; Zaagsma, J1
Hamstra, JJ; Roffel, AF; Santing, RE; ten Berge, RE; Zaagsma, J1
Ehlert, FJ; Thomas, EA1
Célice-Pingaud, C; Farinotti, R; Mignon, M; Olivier, A; Riquet, W; Vatier, J1
Ehlert, FJ; Ostrom, RS2
Ehlert, FJ; Sawyer, GW1
Mitchelson, F; Shen, A1
Arai, H; Inoie, M; Marubuchi, S1
Arrang, JM; Morisset, S; Sahm, UG; Schwartz, JC; Tardivel-Lacombe, J; Traiffort, E1
Kajiyama, G; Kuruhara, Y; Okahara, S; Sumii, K; Tari, A; Yamauchi, R; Yonei, Y1
Shinomura, Y1

Reviews

1 review(s) available for histamine and pirenzepine

ArticleYear
[MI cholinergic receptors of gastric secretion: current status].
    Journal de pharmacologie, 1985, Volume: 16 Suppl 2

    Topics: Amino Acids; Animals; Atropine; Benzodiazepinones; Dogs; Gastric Acid; Gastric Emptying; Gastric Mucosa; Gastrins; Heart Rate; Histamine; Histamine Release; Molecular Conformation; Pirenzepine; Rats; Receptors, Muscarinic; Receptors, Nicotinic; Salivation; Somatostatin; Urinary Bladder; Vagus Nerve

1985

Trials

1 trial(s) available for histamine and pirenzepine

ArticleYear
Effect of pirenzepine on meal-stimulated acid secretion and gastrin release in normal man.
    Scandinavian journal of gastroenterology. Supplement, 1982, Volume: 72

    Topics: Adult; Benzodiazepinones; Eating; Gastric Acid; Gastrins; Histamine; Humans; Insulin; Male; Pentagastrin; Pirenzepine

1982

Other Studies

34 other study(ies) available for histamine and pirenzepine

ArticleYear
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
[The effect of muscarinic receptor blockers on non-specific bronchial reactivity in patients with bronchial asthma].
    Pneumonologia i alergologia polska, 1992, Volume: 60, Issue:11-12

    Topics: Adult; Asthma; Bronchial Provocation Tests; Bronchial Spasm; Choline; Female; Histamine; Humans; Ipratropium; Male; Pirenzepine

1992
Muscarinic-receptor functioning in tracheas from normal and ovalbumin-sensitive guinea pigs.
    Canadian journal of physiology and pharmacology, 1991, Volume: 69, Issue:6

    Topics: Aerosols; Animals; Asthma; Bethanidine; Electric Stimulation; Female; Gallamine Triethiodide; Guinea Pigs; Histamine; Hypersensitivity; In Vitro Techniques; Indomethacin; Methacholine Compounds; Ovalbumin; Pirenzepine; Propranolol; Receptors, Muscarinic; Trachea; Yohimbine

1991
Effects of two new pirenzepine analogs on the contractile response of the guinea-pig oesophageal muscularis mucosae to acetylcholine, bethanechol, histamine and high potassium.
    European journal of pharmacology, 1990, Apr-10, Volume: 179, Issue:1-2

    Topics: Acetylcholine; Animals; Atropine; Benzodiazepinones; Bethanechol; Bethanechol Compounds; Esophagus; Guinea Pigs; Histamine; Histamine Antagonists; Male; Muscle Contraction; Piperidines; Pirenzepine; Potassium; Pyrilamine; Receptors, Muscarinic

1990
Telenzepine inhibits electrically-stimulated, acetylcholine plus histamine-mediated acid secretion in the mouse isolated stomach by blockade of M1 muscarine receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 343, Issue:1

    Topics: Acetylcholine; Alkaloids; Animals; Anti-Ulcer Agents; Electric Stimulation; Furans; Gastric Acid; Gastric Mucosa; Histamine; Mice; Muscarinic Antagonists; Naphthalenes; p-Methoxy-N-methylphenethylamine; Parasympatholytics; Piperidines; Pirenzepine; Stomach; Thiazepines; Vagus Nerve

1991
Role of acetylcholine, histamine and gastrin in the acid response to intracisternal injection of TRH analog, RX 77368, in the rat.
    Regulatory peptides, 1990, Feb-04, Volume: 27, Issue:2

    Topics: Acetylcholine; Animals; Antibodies, Monoclonal; Cisterna Magna; Gastric Acid; Gastrins; Histamine; Injections, Intravenous; Male; Pirenzepine; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Thyrotropin-Releasing Hormone

1990
Carbachol-induced potentiation and inhibition of acid secretion by guinea pig gastric gland.
    European journal of pharmacology, 1990, Mar-13, Volume: 178, Issue:1

    Topics: Aminopyrine; Animals; Atropine; Binding, Competitive; Carbachol; Dose-Response Relationship, Drug; Gastric Acid; Gastric Mucosa; Guinea Pigs; Histamine; In Vitro Techniques; Male; N-Methylscopolamine; Parasympathomimetics; Pirenzepine; Receptors, Muscarinic; Scopolamine Derivatives

1990
Regulation of Na-K-Cl cotransport in endothelial cells by atrial natriuretic factor.
    The American journal of physiology, 1989, Volume: 257, Issue:1 Pt 1

    Topics: Acetylcholine; Animals; Aorta, Thoracic; Atrial Natriuretic Factor; Biological Transport; Cattle; Cells, Cultured; Chlorides; Cimetidine; Cyclic GMP; Endothelium, Vascular; Histamine; Kinetics; Norepinephrine; Pirenzepine; Potassium; Propranolol; Receptors, Adrenergic, beta; Receptors, Histamine H2; Receptors, Muscarinic; Second Messenger Systems; Sodium

1989
Comparison of telenzepine, pirenzepine and atropine on gastric acid and pepsin secretion in response to histamine, pentagastrin, bethanechol, sham-feeding and feeding.
    Digestion, 1989, Volume: 44, Issue:2

    Topics: Animals; Atropine; Bethanechol; Bethanechol Compounds; Dogs; Food; Gastric Acid; Gastric Fistula; Histamine; Parasympatholytics; Pentagastrin; Pepsin A; Pirenzepine; Stomach

1989
Correlation of activity of chlorpromazine and respective hydroxy, dimethoxy and sulphoxide analogues on dopamine, muscarinic, histamine and calmodulin sites of action.
    Xenobiotica; the fate of foreign compounds in biological systems, 1988, Volume: 18, Issue:3

    Topics: Adenylyl Cyclase Inhibitors; Animals; Binding Sites; Calmodulin; Cerebral Cortex; Chlorpromazine; Cyclic AMP; Dopamine; Histamine; Hypothalamus; Phosphoric Diester Hydrolases; Pirenzepine; Rats; Receptors, Dopamine; Receptors, Muscarinic; Spiperone; Sulfoxides

1988
Gastric antisecretory and pharmacologic properties of N,N-dimethyl-N'-(2-diisopropylaminoethyl)-N-(4,6-dimethyl-2-pyridyl)ur ea (L-634,366).
    Archives internationales de pharmacodynamie et de therapie, 1986, Volume: 281, Issue:1

    Topics: Animals; Anti-Ulcer Agents; Atropine; Benzodiazepinones; Blood Pressure; Cimetidine; Dogs; Female; Gastric Juice; Guinea Pigs; Heart Rate; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Male; Methylurea Compounds; Mice; Myocardial Contraction; Parasympathetic Nervous System; Pirenzepine; Rats; Stomach; Uterine Contraction

1986
Potassium ion facilitation of phosphoinositide turnover activation by muscarinic receptor agonists in rat brain.
    Journal of neurochemistry, 1986, Volume: 46, Issue:5

    Topics: Animals; Benzodiazepinones; Carbachol; Dioxolanes; Hippocampus; Histamine; Male; Norepinephrine; Oxotremorine; Phosphatidylinositols; Pirenzepine; Potassium; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1986
Effect of ethanol on receptor-stimulated phosphatidic acid and polyphosphoinositide metabolism in mouse brain.
    Life sciences, 1986, Nov-03, Volume: 39, Issue:18

    Topics: Animals; Brain Chemistry; Carbachol; Ethanol; Histamine; Hydrolysis; Male; Mice; Mice, Inbred C57BL; Norepinephrine; Phosphatidic Acids; Phosphatidylinositol Phosphates; Phosphatidylinositols; Phosphorus Radioisotopes; Pirenzepine; Receptors, Muscarinic

1986
Characteristics of canine lower esophageal sphincter: a new electrophysiological tool.
    The American journal of physiology, 1988, Volume: 255, Issue:4 Pt 1

    Topics: Animals; Carbachol; Cimetidine; Dogs; Electric Stimulation; Electrophysiology; Esophagus; Female; Histamine; In Vitro Techniques; Intercellular Junctions; Male; Microscopy, Electron; Muscle Contraction; Muscle, Smooth; Pirenzepine; Pyrilamine; Reference Values; Tetrodotoxin

1988
Inhibition of gastric acid secretion by human calcitonin gene-related peptide with picomolar potency in guinea-pig parietal cell preparations.
    Biochemical and biophysical research communications, 1987, Jul-31, Volume: 146, Issue:2

    Topics: Aminopyrine; Animals; Benzamides; Calcitonin Gene-Related Peptide; Cimetidine; Dose-Response Relationship, Drug; Gastric Acid; Guinea Pigs; Histamine; Male; Neuropeptides; Parietal Cells, Gastric; Pirenzepine

1987
Suppression by muscarinic M2 stimulation of the contractile mechanism via histamine H1 receptors in the longitudinal muscle of guinea pig ileum.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:2

    Topics: Animals; Atropine; Calcium; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Ileum; Male; Methacholine Chloride; Methacholine Compounds; Muscle Contraction; Phentolamine; Pirenzepine; Propranolol; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Temperature; Tetrodotoxin

1987
Effects of cimetidine, atropine and pirenzepine on basal and stimulated gastric acid secretion in the rat.
    European journal of pharmacology, 1987, Jun-19, Volume: 138, Issue:2

    Topics: Animals; Atropine; Cimetidine; Dose-Response Relationship, Drug; Gastric Acid; Histamine; Male; Monoamine Oxidase; Pentagastrin; Pirenzepine; Pupil; Rats; Rats, Inbred Strains

1987
gamma-Aminobutyric acid stimulates acid secretion from the isolated guinea pig stomach.
    The American journal of physiology, 1987, Volume: 253, Issue:5 Pt 1

    Topics: Animals; Bicuculline; gamma-Aminobutyric Acid; Gastric Acid; Gastric Mucosa; Guinea Pigs; Histamine; Male; Muscimol; Pirenzepine; Proglumide; Scopolamine; Stomach; Tetrodotoxin

1987
Pirenzepine (LS 519): a weak inhibitor of acid secretion by isolated rat parietal cells.
    European journal of pharmacology, 1982, Dec-17, Volume: 86, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Atropine; Benzodiazepinones; Bucladesine; Carbachol; Gastric Acid; Gastric Mucosa; Histamine; In Vitro Techniques; Pirenzepine; Rats

1982
[Pathogenesis, diagnosis and therapy of ulcer disease. Therapy. 3: Pharmacologic basis and therapy with pirenzepine].
    Die Medizinische Welt, 1983, Dec-02, Volume: 34, Issue:48

    Topics: Acetylcholine; Animals; Benzodiazepinones; Gastric Acid; Gastric Mucosa; Gastrins; Histamine; Humans; Pirenzepine; Rats; Stomach Ulcer

1983
Inhibition of gastric mucosa carbonic anhydrase by pirenzepine in patients with gastroduodenal ulcers.
    Arzneimittel-Forschung, 1981, Volume: 31, Issue:3

    Topics: Animals; Benzodiazepinones; Carbonic Anhydrase Inhibitors; Cattle; Duodenal Ulcer; Gastric Mucosa; Histamine; Humans; In Vitro Techniques; Peptic Ulcer; Piperazines; Pirenzepine; Stomach Ulcer

1981
Effect of two doses of pirenzepine on histamine-stimulated gastric acid secretion in man.
    Scandinavian journal of gastroenterology. Supplement, 1982, Volume: 72

    Topics: Adolescent; Adult; Benzodiazepinones; Dose-Response Relationship, Drug; Female; Gastric Acid; Histamine; Humans; Male; Middle Aged; Pirenzepine; Stimulation, Chemical

1982
No evidence for a role of muscarinic M2 receptors in functional antagonism in bovine trachea.
    British journal of pharmacology, 1995, Volume: 115, Issue:4

    Topics: Animals; Bronchoconstrictor Agents; Cattle; Dose-Response Relationship, Drug; Gallamine Triethiodide; Histamine; In Vitro Techniques; Isoproterenol; Methacholine Chloride; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nicotinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Adrenergic, beta; Receptors, Muscarinic; Trachea

1995
Dysfunction of muscarinic M2 receptors after the early allergic reaction: possible contribution to bronchial hyperresponsiveness in allergic guinea-pigs.
    British journal of pharmacology, 1995, Volume: 114, Issue:4

    Topics: Administration, Inhalation; Allergens; Animals; Asthma; Benzodiazepinones; Bronchial Hyperreactivity; Diamines; Disease Models, Animal; Electric Stimulation; Female; Gallamine Triethiodide; Guinea Pigs; Heart; Histamine; Hypersensitivity; In Vitro Techniques; Male; Muscarinic Antagonists; Muscle, Smooth; Neuromuscular Junction; Parasympatholytics; Pilocarpine; Piperidines; Pirenzepine; Receptors, Muscarinic; Trachea

1995
Involvement of the M2 muscarinic receptor in contractions of the guinea pig trachea, guinea pig esophagus, and rat fundus.
    Biochemical pharmacology, 1996, Mar-22, Volume: 51, Issue:6

    Topics: Adrenergic beta-Agonists; Animals; Colforsin; Cyclic AMP; Esophagus; Gastric Fundus; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Oxotremorine; Pertussis Toxin; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Serotonin; Trachea; Virulence Factors, Bordetella

1996
Effect on gastric secretion, gastrin and histamine release during and after long-term treatment by pirenzepine in dogs.
    Fundamental & clinical pharmacology, 1996, Volume: 10, Issue:2

    Topics: Animals; Anti-Ulcer Agents; Dogs; Eating; Gastric Acid; Gastric Mucosa; Gastrins; Histamine; Histamine Release; Male; Pepsin A; Pirenzepine; Receptors, Muscarinic

1996
M2 muscarinic receptor inhibition of agonist-induced cyclic adenosine monophosphate accumulation and relaxation in the guinea pig ileum.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 280, Issue:1

    Topics: Animals; Cyclic AMP; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Male; Muscarinic Agonists; Muscle Relaxation; Piperidines; Pirenzepine; Receptor, Muscarinic M2; Receptors, Muscarinic

1997
Contractile roles of the M2 and M3 muscarinic receptors in the guinea pig colon.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 284, Issue:1

    Topics: Animals; Colforsin; Colon; Cyclic AMP; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Oxotremorine; Pertussis Toxin; Piperidines; Pirenzepine; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Virulence Factors, Bordetella

1998
Muscarinic M2 receptor-mediated contraction in the guinea pig Taenia caeci: possible involvement of protein kinase C.
    Biochemical pharmacology, 1998, Dec-01, Volume: 56, Issue:11

    Topics: Animals; Cecum; Colforsin; Diphenylacetic Acids; Female; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Kinetics; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Parasympathomimetics; Piperidines; Pirenzepine; Protein Kinase C; Receptor, Muscarinic M2; Receptors, Muscarinic; Second Messenger Systems

1998
Histamine H2-receptor antagonism of T-593, an anti-ulcer agent: studies on aminopyrine accumulation in isolated canine gastric mucosal cells.
    Japanese journal of pharmacology, 1998, Volume: 78, Issue:3

    Topics: Aminopyrine; Animals; Anti-Ulcer Agents; Bucladesine; Carbachol; Carbon Radioisotopes; Cholinergic Agonists; Dogs; Dose-Response Relationship, Drug; Famotidine; Gastric Acid; Gastric Mucosa; Guanidines; Histamine; Histamine H2 Antagonists; Omeprazole; Pentagastrin; Pirenzepine; Ranitidine; Sulfones

1998
Atypical neuroleptics enhance histamine turnover in brain via 5-Hydroxytryptamine2A receptor blockade.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 288, Issue:2

    Topics: Animals; Antipsychotic Agents; Benzodiazepines; Brain; Catalepsy; Clozapine; Drug Interactions; Haloperidol; Histamine; Histamine Antagonists; Imidazoles; Male; Methylhistamines; Mice; Olanzapine; Pirenzepine; Receptor, Serotonin, 5-HT2A; Receptors, Histamine H3; Receptors, Serotonin; Serotonin Antagonists

1999
Comparison of functional antagonism between isoproterenol and M2 muscarinic receptors in guinea pig ileum and trachea.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 288, Issue:3

    Topics: Animals; Colforsin; Diphenylacetic Acids; Guinea Pigs; Histamine; Ileum; Isoproterenol; Muscle Relaxation; Oxotremorine; Pertussis Toxin; Piperidines; Pirenzepine; Receptor, Muscarinic M2; Receptors, Muscarinic; Trachea; Virulence Factors, Bordetella

1999
Effects of omeprazole and pirenzepine on enterochromaffin-like cells and parietal cells in rat stomach.
    Journal of gastroenterology, 2001, Volume: 36, Issue:6

    Topics: Animals; Anti-Ulcer Agents; Blotting, Northern; Drug Therapy, Combination; Enterochromaffin-like Cells; H(+)-K(+)-Exchanging ATPase; Histamine; Hydrogen-Ion Concentration; Male; Omeprazole; Parietal Cells, Gastric; Pirenzepine; Rats; Rats, Wistar; RNA, Messenger; Stomach

2001
Does pirenzepine suppress the undesirable effects of a proton pump inhibitor on enterochromaffin-like cells?
    Journal of gastroenterology, 2001, Volume: 36, Issue:6

    Topics: Animals; Anti-Ulcer Agents; Enterochromaffin-like Cells; Epidermal Growth Factor; Gastrins; Histamine; Humans; Male; Parietal Cells, Gastric; Pirenzepine; Proton Pump Inhibitors; Rats; RNA, Messenger; Stomach

2001