histamine has been researched along with methylhistaprodifen in 8 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (12.50) | 18.2507 |
2000's | 6 (75.00) | 29.6817 |
2010's | 1 (12.50) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Detert, H; Elz, S; Kramer, K; Kühne, R; Pertz, HH; Schunack, W; ter Laak, AM | 1 |
Burckstummer, T; Buschauer, A; Dove, S; Elz, S; Pertz, HH; Schunack, W; Seifert, R; Wenzel-Seifert, K | 1 |
Elz, S; Kramer, K; Menghin, S; Pertz, HH; Schunack, W; Seifert, R | 1 |
Elz, S; Kramer, K; Malinowska, B; Piszcz, J; Schlicker, E; Schunack, W | 1 |
Bacciottini, L; Blandina, P; Cecchi, M; Mannaioni, PF; Passani, MB | 1 |
Elz, S; Kozłowska, H; Kramer, K; Kwolek, G; Malinowska, B; Pertz, HH; Schlicker, E; Schunack, W | 1 |
Elz, S; Pertz, HH; Schunack, W | 1 |
Tabarean, IV | 1 |
1 review(s) available for histamine and methylhistaprodifen
Article | Year |
---|---|
Structure-activity relationships of histamine H1-receptor agonists.
Topics: Animals; Histamine; Histamine Agonists; Humans; Imidazoles; Methylhistamines; Structure-Activity Relationship | 2004 |
7 other study(ies) available for histamine and methylhistaprodifen
Article | Year |
---|---|
Histaprodifens: synthesis, pharmacological in vitro evaluation, and molecular modeling of a new class of highly active and selective histamine H(1)-receptor agonists.
Topics: Animals; Aorta; Endothelium, Vascular; Guinea Pigs; Histamine Agonists; Humans; Ileum; In Vitro Techniques; Male; Methylhistamines; Models, Molecular; Muscle Contraction; Muscle, Smooth; Protein Structure, Tertiary; Ranidae; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, Neurotransmitter; Rhodopsin; Structure-Activity Relationship; Vasoconstrictor Agents | 2000 |
Multiple differences in agonist and antagonist pharmacology between human and guinea pig histamine H1-receptor.
Topics: Amino Acid Sequence; Animals; Binding Sites; Electrophoresis; GTP Phosphohydrolases; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Humans; Molecular Sequence Data; Protein Conformation; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Recombinant Proteins; Species Specificity; Tritium | 2003 |
N(alpha)-imidazolylalkyl and pyridylalkyl derivatives of histaprodifen: synthesis and in vitro evaluation of highly potent histamine H(1)-receptor agonists.
Topics: Animals; Aorta; Endothelium, Vascular; Guinea Pigs; Histamine; Histamine Agonists; Ileum; Imidazoles; In Vitro Techniques; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Pyridines; Rats; Receptors, Histamine H1; Structure-Activity Relationship | 2003 |
Histaprodifen, methylhistaprodifen, and dimethylhistaprodifen are potent H1-receptor agonists in the pithed and in the anaesthetized rat.
Topics: Anesthesia; Animals; Blood Pressure; Catecholamines; Decerebrate State; Enzyme Inhibitors; Heart Rate; Histamine; Histamine Agonists; Male; Methylhistamines; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Rats; Rats, Wistar; Vagotomy | 1999 |
Cortical acetylcholine release elicited by stimulation of histamine H1 receptors in the nucleus basalis magnocellularis: a dual-probe microdialysis study in the freely moving rat.
Topics: Acetylcholine; Animals; Basal Nucleus of Meynert; Cerebral Cortex; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Histamine; Histamine H1 Antagonists; Male; Methylhistamines; Microdialysis; Potassium; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, Histamine H3; Tetrodotoxin | 2001 |
Novel histaprodifen analogues as potent histamine H1-receptor agonists in the pithed and in the anaesthetized rat.
Topics: Anesthesia; Animals; Blood Pressure; Cardiovascular System; Heart Rate; Histamine; Male; Methylhistamines; Rats; Rats, Wistar; Sympathomimetics; Vagotomy | 2001 |
Functional pharmacology of H1 histamine receptors expressed in mouse preoptic/anterior hypothalamic neurons.
Topics: Animals; Calcium; Cells, Cultured; Dose-Response Relationship, Drug; Fluorescent Dyes; Fura-2; Histamine; Histamine Agonists; Histamine H1 Antagonists; Hypothalamus, Anterior; Inhibitory Concentration 50; Methylhistamines; Mice; Mice, Inbred C57BL; Neurons; Patch-Clamp Techniques; Receptors, Histamine H1; Species Specificity | 2013 |