histamine and methylhistaprodifen

histamine has been researched along with methylhistaprodifen in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (12.50)18.2507
2000's6 (75.00)29.6817
2010's1 (12.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Detert, H; Elz, S; Kramer, K; Kühne, R; Pertz, HH; Schunack, W; ter Laak, AM1
Burckstummer, T; Buschauer, A; Dove, S; Elz, S; Pertz, HH; Schunack, W; Seifert, R; Wenzel-Seifert, K1
Elz, S; Kramer, K; Menghin, S; Pertz, HH; Schunack, W; Seifert, R1
Elz, S; Kramer, K; Malinowska, B; Piszcz, J; Schlicker, E; Schunack, W1
Bacciottini, L; Blandina, P; Cecchi, M; Mannaioni, PF; Passani, MB1
Elz, S; Kozłowska, H; Kramer, K; Kwolek, G; Malinowska, B; Pertz, HH; Schlicker, E; Schunack, W1
Elz, S; Pertz, HH; Schunack, W1
Tabarean, IV1

Reviews

1 review(s) available for histamine and methylhistaprodifen

ArticleYear
Structure-activity relationships of histamine H1-receptor agonists.
    Mini reviews in medicinal chemistry, 2004, Volume: 4, Issue:9

    Topics: Animals; Histamine; Histamine Agonists; Humans; Imidazoles; Methylhistamines; Structure-Activity Relationship

2004

Other Studies

7 other study(ies) available for histamine and methylhistaprodifen

ArticleYear
Histaprodifens: synthesis, pharmacological in vitro evaluation, and molecular modeling of a new class of highly active and selective histamine H(1)-receptor agonists.
    Journal of medicinal chemistry, 2000, Mar-23, Volume: 43, Issue:6

    Topics: Animals; Aorta; Endothelium, Vascular; Guinea Pigs; Histamine Agonists; Humans; Ileum; In Vitro Techniques; Male; Methylhistamines; Models, Molecular; Muscle Contraction; Muscle, Smooth; Protein Structure, Tertiary; Ranidae; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, Neurotransmitter; Rhodopsin; Structure-Activity Relationship; Vasoconstrictor Agents

2000
Multiple differences in agonist and antagonist pharmacology between human and guinea pig histamine H1-receptor.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 305, Issue:3

    Topics: Amino Acid Sequence; Animals; Binding Sites; Electrophoresis; GTP Phosphohydrolases; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Humans; Molecular Sequence Data; Protein Conformation; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Recombinant Proteins; Species Specificity; Tritium

2003
N(alpha)-imidazolylalkyl and pyridylalkyl derivatives of histaprodifen: synthesis and in vitro evaluation of highly potent histamine H(1)-receptor agonists.
    Journal of medicinal chemistry, 2003, Dec-04, Volume: 46, Issue:25

    Topics: Animals; Aorta; Endothelium, Vascular; Guinea Pigs; Histamine; Histamine Agonists; Ileum; Imidazoles; In Vitro Techniques; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Pyridines; Rats; Receptors, Histamine H1; Structure-Activity Relationship

2003
Histaprodifen, methylhistaprodifen, and dimethylhistaprodifen are potent H1-receptor agonists in the pithed and in the anaesthetized rat.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 359, Issue:1

    Topics: Anesthesia; Animals; Blood Pressure; Catecholamines; Decerebrate State; Enzyme Inhibitors; Heart Rate; Histamine; Histamine Agonists; Male; Methylhistamines; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Rats; Rats, Wistar; Vagotomy

1999
Cortical acetylcholine release elicited by stimulation of histamine H1 receptors in the nucleus basalis magnocellularis: a dual-probe microdialysis study in the freely moving rat.
    The European journal of neuroscience, 2001, Volume: 13, Issue:1

    Topics: Acetylcholine; Animals; Basal Nucleus of Meynert; Cerebral Cortex; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Histamine; Histamine H1 Antagonists; Male; Methylhistamines; Microdialysis; Potassium; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, Histamine H3; Tetrodotoxin

2001
Novel histaprodifen analogues as potent histamine H1-receptor agonists in the pithed and in the anaesthetized rat.
    Naunyn-Schmiedeberg's archives of pharmacology, 2001, Volume: 364, Issue:1

    Topics: Anesthesia; Animals; Blood Pressure; Cardiovascular System; Heart Rate; Histamine; Male; Methylhistamines; Rats; Rats, Wistar; Sympathomimetics; Vagotomy

2001
Functional pharmacology of H1 histamine receptors expressed in mouse preoptic/anterior hypothalamic neurons.
    British journal of pharmacology, 2013, Volume: 170, Issue:2

    Topics: Animals; Calcium; Cells, Cultured; Dose-Response Relationship, Drug; Fluorescent Dyes; Fura-2; Histamine; Histamine Agonists; Histamine H1 Antagonists; Hypothalamus, Anterior; Inhibitory Concentration 50; Methylhistamines; Mice; Mice, Inbred C57BL; Neurons; Patch-Clamp Techniques; Receptors, Histamine H1; Species Specificity

2013