histamine has been researched along with colforsin in 209 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 66 (31.58) | 18.7374 |
1990's | 103 (49.28) | 18.2507 |
2000's | 32 (15.31) | 29.6817 |
2010's | 8 (3.83) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Noma, A; Ono, K; Tareen, FM; Yoshida, A | 1 |
Kamei, C; Mukai, T; Tasaka, K | 1 |
Classen, M; Roithmaier, S; Seidler, U; Silen, W | 1 |
Boeynaems, JM; Côte, S; Hekimian, G; Van Sande, J | 1 |
Felíu, JE; Herias, M; Olea, J; Pereda, C; Rossi, I | 1 |
Amiel, C; Friedlander, G; Herman, P; Huy, PT | 1 |
Wilson, SP | 1 |
Fukaya, T; Koizumi, H; Kumakiri, M; Ohkawara, A; Ueda, T; Yasui, C | 1 |
Classen, M; Offermanns, S; Rosenthal, W; Schepp, W; Schmidtler, J; Schusdziarra, V | 1 |
Gespach, C; Hanson, PJ; McKenna, P; Williams, JM | 1 |
Gadsby, DC; Horie, M; Hwang, TC; Nairn, AC | 1 |
Fischer, MJ; Janssen, LH; Nijkamp, FP; van Oosterhout, AJ | 1 |
Pahapill, PA; Schlichter, LC | 1 |
Boswell, CA; Joris, I; Majno, G; Ostrom, KA | 1 |
Asano, K; Iizuka, H; Ito, F; Takahashi, H; Tamura, T; Tsutsui, M | 1 |
Nowak, JZ; Sek, B | 2 |
Koren, R; Liberman, A; Narinsky, R; Novogrodsky, A; Ravid, A; Rotem, C | 1 |
Malinowska, DH | 1 |
Classen, M; Schepp, W; Schmidtler, J; Schusdziarra, V; Tatge, C | 1 |
Classen, M; Fürlinger, C; Janczewska, I; Schepp, W; Schmidtler, J; Schusdziarra, V; Weigert, N | 1 |
Heim, HK; Oestmann, A; Sewing, KF | 2 |
Jachno, K; Johnston, MJ; Marley, PD; Thomson, KA | 1 |
Beil, W; Bersimbaev, R; Sewing, KF | 1 |
Chew, CS; Petropoulos, AC | 1 |
Cuthbert, AW; Pickles, RJ | 1 |
Forte, JG; Reenstra, WW | 1 |
Donaldson, J; Hill, SJ; Kendall, DA | 1 |
Fukaya, T; Koizumi, H; Ohkawara, A; Osawa, Y; Ueda, T; Yasui, C | 1 |
Asher, VA; Goldenring, JR; Lewis, JJ; Modlin, IM | 2 |
Iizuka, H; Takahashi, H; Tamura, T; Tsutsui, M | 1 |
Fraser, G; Long, S; Sandle, GI; Warhurst, G | 1 |
Kristersson, A; Mazzoni, L; Morley, J; Sanjar, S; Schaeublin, E | 1 |
Greene, RW; Haas, HL | 1 |
Coffey, RJ; Goldenring, JR; Lewis, JJ; Modlin, IM | 1 |
Reutter, K; Ruoff, HJ; Schepp, W | 1 |
Bickel, M; Herling, AW | 1 |
Alvarez, R; Amirian, DA; Chen, MC; Soll, AH; Toomey, M | 1 |
Greeff, K; Schmitt, M | 1 |
Black, EW; Strada, SJ; Thompson, WJ | 1 |
Beuckelmann, D; Böhm, M; Brown, L; Erdmann, E; Feiler, G; Kemkes, B; Lorenz, B; Näbauer, M | 1 |
Böhm, M; Brown, L; Diet, F; Eichhorn, M; Erdmann, E; Kemkes, B; Näbauer, M; Pieske, B | 1 |
Black, EW; Cornwell, TL; Lincoln, TM; Strada, SJ; Thompson, WJ | 1 |
Kelly, E; Koenig, SM; Leff, AR; Mitchell, RW; Popovich, KJ; White, SR | 1 |
Seidler, U; Sewing, KF | 1 |
Ciarrocchi, A; Fernández, E; Michelangeli, F; Ruiz, MC | 1 |
Ballantyne, GH; Modlin, IM; Zdon, MJ; Zucker, KA | 1 |
Bowman, BF; Stull, JT; Taylor, DA | 1 |
Saari, JT; Schuschke, DA | 1 |
Danilov, SM; Grigorian, GY; Repin, VS; Resink, TJ; Tkachuk, VA; Voino-Yasenetskaya, TA | 1 |
Nowak, JZ; Sek, B; Szkiel, B | 1 |
Albinus, M; Armbruckner, L; Klein, S; Maier, R | 1 |
Donaldson, J; Hall, IP; Hill, SJ | 1 |
Ducroc, R; Garzon, B; Geloso, JP; Hervatin, F; Moreau, E | 1 |
Carson, MR; Shasby, DM; Shasby, SS | 1 |
Mitsuhashi, M; Mitsuhashi, T; Payan, DG | 1 |
Bhalla, RC; Sharma, RV | 1 |
Bunn, SJ; Livett, BG; Wan, DC | 1 |
Brown, MR; Chew, CS | 1 |
Lohse, MJ; Puurunen, J; Schwabe, U | 1 |
Baba, A; Iwata, H; Nishiuchi, Y; Uemura, A | 1 |
Brown, JK; Madison, JM | 1 |
Bali, JP; Choquet, A; Galleyrand, JC; Magous, R | 1 |
Foreman, JC; Norris, DB; Rising, TJ; Webber, SE | 1 |
Chiba, T; Park, J; Yamada, T | 1 |
Michelangeli, F; Pelacca, A; Rodríguez, CL; Ruiz, MC | 1 |
Bhoola, KD; Gadd, AL | 1 |
Baba, A; Iwata, H; Nishiuchi, Y; Tatsuno, T; Uemura, A | 1 |
Nowak, JZ; Sebastjanska, A; Sek, B | 1 |
Adrian, TE; Lewis, JJ; Modlin, IM; Zdon, MJ | 1 |
Chew, CS | 3 |
Burton, JL; Creveling, CR; Daly, JW; Hollingsworth, EB; McNeal, ET; Williams, RJ | 1 |
Goldie, RG; Papadimitriou, JM; Paterson, JW; Rigby, PJ; Self, HM; Spina, D | 1 |
Rosenfeld, GC | 1 |
Fredholm, BB; Jonzon, B; Lindström, K | 1 |
Forte, JG; Okamoto, C; Reichstein, BJ | 1 |
Kimura, A; Nakagawa, H; Ohuchi, T; Oka, M | 1 |
Markstein, R; Palacios, JM; Pazos, A | 1 |
Condorelli, M; Marone, G; Triggiani, M; Vigorita, S | 1 |
Forte, JG; Urushidani, T | 1 |
Adrian, TE; Ballantyne, GH; Modlin, IM; Zdon, MJ; Zucker, KA | 1 |
Classen, M; Heim, HK; Ruoff, HJ; Schepp, W; Schneider, J; Schusdziarra, V | 1 |
Box, RJ; Portenier, M; Staehelin, M | 1 |
Corvol, P; Ménard, J; Mizrahi, J; Pinet, F | 1 |
Feldman, R; Motulsky, HJ; Smith, D; Terman, BI | 1 |
Satake, T; Suzuki, K; Suzuki, R; Takagi, K; Tsukawaki, M | 1 |
Kelley, G; Rasmussen, H; Takuwa, N; Takuwa, Y | 1 |
Contreras-Rodríguez, JL; de la Garza, MC; García-Sáinz, JA; Nájera-Alvarado, A | 1 |
Palmer, JM; Wood, JD; Zafirov, DH | 1 |
Dhawan, BN; Dhawan, KN; Gulati, A; Shukla, R; Srimal, RC | 1 |
Dale, MM; Obianime, W | 1 |
Daly, JW; Padgett, W; Seamon, KB | 1 |
Hersey, SJ; Miller, M; Norris, SH | 1 |
Hamabe, S; Himeno, S; Kitani, T; Kurokawa, M; Kuroshima, T; Moriwaki, K; Saito, R; Shinomura, Y; Takahashi, S; Tarui, S | 1 |
Chang, J; Dervinis, A; Hand, JM; Lewis, AJ; Schwalm, S | 1 |
Holian, O; Nyhus, LM | 1 |
Ekblad, EB; Licko, V | 1 |
Daly, JW; Sugio, K | 1 |
Diarra, A; Gallo-Payet, N; Garneau, L; Sauvé, R; Wang, R | 1 |
Finkbeiner, WE; Mrsny, RJ; Shen, BQ; Widdicombe, JH; Wine, JJ | 1 |
Lajas, AI; Pariente, JA; Salido, GM | 1 |
Absood, A; Maruno, K; Said, SI | 1 |
Lelkes, PI; Manolopoulos, VG; Samet, MM | 1 |
Rembold, CM; Stull, JT; Van Riper, DA; Weaver, BA | 1 |
Arilla, E; Puebla, L | 1 |
Brandi, ML; Fiorelli, G; Pioli, P; Rechler, MM; Yang, YW | 1 |
Goldenring, JR; Hidaka, H; Ishikawa, T; Mamiya, N; Modlin, IM; Natsume, A; Tsunoda, Y; Usuda, N; Yasui, K | 1 |
Arima, N; Chiba, T; Kinoshita, Y; Nakamura, A; Yamashita, Y | 1 |
Esteva, F; Lanas, AI; Nerín, J; Sáinz, R | 1 |
Greger, R; Gruenert, DC; Hug, T; Koslowsky, T; Kunzelmann, K | 1 |
Hall, IP; Hill, SJ; McCreath, G | 1 |
Kobayashi, S; Tanaka, T; Tani, S | 1 |
Fleissner, S; Heimann-Weitschat, I; Lindstaedt, R; Schmidt, J; Szelenyi, I | 1 |
den Hertog, A; Duin, M; Hoiting, B; Nelemans, A; Sipma, H | 1 |
Alexander, SP; Curtis, AR; Hill, SJ; Kendall, DA | 1 |
Baram, D; Hershkoviz, R; Lider, O; Mekori, YA; Miron, S; Reshef, T | 1 |
Beil, W; Bersimbaev, RI; Gandjour, A; Heim, HK; Sewing, KF | 1 |
Ellis, JL; Fernandes, LB; Undem, BJ | 1 |
Cohen, AJ; Fishman, JB; Silbiger, SR; Stoff, JS | 1 |
Abiko, Y; Yazawa, K | 1 |
Classen, M; Dehne, K; Offermanns, S; Rosenthal, W; Schepp, W; Schmidtler, J | 1 |
Abad, MJ; Acosta, A; Michelangeli, F; Ruiz, MC | 1 |
Becker, I; Huber, W; Peskar, BM; Schenck, U; Schepp, W; Trautmann, M | 1 |
Lindsley, K; Moy, A; Shasby, DM; Shasby, S; Sheldon, R | 1 |
Arrang, JM; Leurs, R; Ruat, M; Schwartz, JC; Tardivel-Lacombe, J; Traiffort, E | 1 |
Crowe, SE; Perdue, MH | 1 |
Hashimoto, Y; Iizuka, H; Ishida-Yamamoto, A; Takahashi, H | 1 |
Horie, M; James, AF; Sasayama, S; Watanuki, M; Xie, LH | 1 |
Ehlert, FJ; Thomas, EA | 2 |
Alewijnse, AE; Leurs, R; Roovers, E; Smit, MJ; Timmerman, H; van de Vrede, Y | 1 |
Harrisss, DR; Hill, SJ; Marsh, KA | 1 |
Bissonnette, EY | 1 |
Benishin, CG; Hirsh, AJ; Jones, RL; Man, SF; Pang, PK | 1 |
Bianchi, BR; Chiou, W; Lin, CW; Magnuson, SR; Wu-Wong, JR | 1 |
Baldi, A; Davio, C; Lemos, B; Mladovan, A; Rivera, E; Shayo, C | 1 |
Arilla, E; Puebla, L; Rodríguez-Martín, E | 1 |
Celuch, SM | 1 |
Elzinga, CR; Hoiting, BH; Kuipers, R; Meurs, H; Schuiling, M; Zaagsma, J | 1 |
Fredberg, JJ; Heyder, J; Hubmayr, RD; Moller, W; Panettieri, RA; Planus, E; Shore, SA; Wang, N | 1 |
Aihara, M; Anai, M; Asano, T; Fukushima, Y; Funaki, M; Inukai, K; Katagiri, H; Matsuhashi, N; Ogihara, T; Oka, Y; Saitoh, T; Sugano, K; Yazaki, Y | 1 |
Chiba, S; Furukawa, Y; Hirose, M; Yamazaki, K | 1 |
Fertel, RH; Wood, JD; Xia, Y | 1 |
Camello, C; Camello, PJ; Gonzalez, A; Lajas, AI; Pariente, JA | 1 |
Warashina, A | 1 |
Cantabrana, B; Hidalgo, A; Perez-Vallina, JR; Revuelta, MP | 1 |
Ehlert, FJ; Sawyer, GW | 1 |
Butler, K; Del Valle, J; Hare, B; Hoeltzel, M; Todisco, A; Wang, LD; Wang, M | 1 |
Crowe, SE; Luthra, GK; Perdue, MH | 1 |
Gibson, WJ; Pinnock, RD; Young, JM; Young, KW | 1 |
Honjo, H; Kodama, I; Satake, K; Shibata, S; Takagi, K; Toyama, J | 1 |
Bolz, SS; Pohl, U | 1 |
Beales, IL; Calam, J | 1 |
Ehlert, FJ; Ostrom, RS | 2 |
Khan, MM; Poluektova, LY | 1 |
Baldi, A; Barbosa, M; Brodsky, A; Davio, C; Lardo, M; Lemos Legnazzi, B; Morelli, A; Rivera, E; Sanchez Avalos, JC; Shayo, C | 1 |
Goldstein, JL; Layden, TJ; Moyer, MP; Nataraja, SG; Rao, MC; Sahi, J | 1 |
Kuba, K; Nowak, JZ; Woldan-Tambor, A; Zawilska, JB | 1 |
Chugun, A; Gomi, H; Hara, Y; Kaigo, H; Kondo, H; Minami, I; Nishimura, H; Watanabe, H | 1 |
Bachmann, O; Gregor, M; Lamprecht, G; Seidler, U; Siegel, WK; Sonnentag, T; Weichert, A | 1 |
Mitchelson, F; Shen, A | 1 |
Ikeda, K; Makimoto, H; Mayumi, T; Mizuguchi, H; Nakagawa, S; Utoguchi, N | 1 |
Ehlert, F; Sawyer, G | 1 |
Benovic, JL; Billington, CK; Hall, IP; Mundell, SJ; Panettieri, RA; Parent, JL; Penn, RB | 1 |
Barth, H; Vischer, UM; Wollheim, CB | 1 |
Blandizzi, C; Colucci, R; Del Tacca, M; Tognetti, M | 1 |
Abdulkadir, O; Gunter-Smith, PJ; Hammonds-Odie, L; Scanlon, M; Terrell, R | 1 |
Ezeamuzie, CI | 1 |
Carmosino, M; Gobin, R; Mannucci, R; Nicchia, GP; Procino, G; Svelto, M; Valenti, G; Verbavatz, JM | 1 |
Bessard, G; Bréant, D; Caron, F; Corompt, E; Devillier, P | 1 |
Arima, N; Hamada, T; Kimura, S; Murata, Y; Nomaguchi, M; Sasaguri, Y; Tanimoto, A; Xu, H | 1 |
Michelangeli, F; Pérez, JF; Ruiz, MC | 1 |
Blanco, I; Gomez-Ramirez, J; Ortiz, J | 1 |
Koda, H; Mizumura, K | 1 |
Bergoc, R; Cricco, G; Darvas, Z; Falus, A; Fitzsimons, C; Hegyesi, H; Kovács, P; Lázár-Molnár, E; Martin, G; Pállinger, E; Rivera, ES; Tóth, S | 1 |
Basta-Kaim, A; Budziszewska, B; Jaworska-Feil, L; Kubera, M; Lasoń, W; Leśkiewicz, M; Tetich, M | 1 |
Esbenshade, TA; Hancock, AA; Kang, CH; Krueger, KM; Masters, JN; Miller, TR; Roch, JM; Witte, DG | 1 |
Aihara, T; Furutani, K; Ichikawa, A; Nakamura, E; Ohtsu, H; Okabe, S; Tanaka, S | 1 |
Advenier, C; Cortijo, J; Mata, M; Morcillo, EJ; Naline, E; Sarria, B | 1 |
Hool, LC | 1 |
Jan, CR; Liu, CP | 1 |
Boterman, M; Elzinga, CR; Eppens, PB; Meurs, H; Wagemakers, D; Zaagsma, J | 1 |
El-Hajj, H; Oriowo, MA | 1 |
Bakke, O; Barois, N; Hagelsteen, K; Haraldsen, G; Johansen, FE; Øynebråten, I | 1 |
Li, X; Rosado, JA; Woodard, GE | 1 |
Arrang, JM; Chabret, C; Gbahou, F; Humbert-Claude, M; Tardivel-Lacombe, J; Vincent, L | 1 |
Ballmann, M; Naim, HY; Stanke, F; Tümmler, B; van Barneveld, A | 1 |
Arias-Montaño, JA; Garduño-Torres, B | 1 |
Carmosino, M; Mannucci, R; Procino, G; Svelto, M; Tamma, G; Valenti, G | 1 |
Han, S; Meeks, MK; Rembold, CM; Ripley, ML | 1 |
Awad, H; Cardounel, AJ; Chen, Z; Christofi, FL; Cooke, H; Guzman, J; Hassanain, HH; Javed, A; Palmer, J; Suntres, Z; Xue, J; Yu, JG | 1 |
Rembold, CM | 1 |
Akiyama, K; Kajiwara, K; Morishima, H; Yanagihara, Y | 1 |
Bevan, S; Foster, AF; Nicolson, TA; Richards, CD | 1 |
Alvarez, E; Cairrão, E; Morgado, M; Santos-Silva, AJ; Verde, I | 1 |
Chow, RH; McDonald, ML; Mircheff, AK; Nakamura, T; Schechter, JE; Selvam, S; Wang, Y; Yiu, SC | 1 |
Cid, LP; Flores, CA; Sepúlveda, FV | 1 |
Bertelsen, LS; Frankson, M; Keely, SJ; Kelly, OB; Mroz, MS; Toumi, F; Ward, JB | 1 |
Bekkali, N; Benninga, MA; Bijlsma, PB; de Jonge, HR; Desjeux, JF; Taminiau, JA; van den Wijngaard, RM; van der Steeg, AF | 1 |
Lelliott, A; Nikkar-Esfahani, A; Offer, J; Orchard, P; Roberts, RE | 1 |
Arrang, JM; Gbahou, F; Rouleau, A | 1 |
DeBiasio, JV; Musch, MW; Newman, SJ; Ruhnke, I; Steiner, JM; Suchodolski, JS | 1 |
Baudenbacher, FJ; Brophy, CM; Cheung-Flynn, J; Hocking, KM; Komalavilas, P; Putumbaka, G; Venkatraman, S | 1 |
Hendriksen, CFM; Hoonakker, ME; Sloots, A; van der Maas, L; Verhagen, LM | 1 |
2 review(s) available for histamine and colforsin
Article | Year |
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Development of acid secretory function in the rat stomach: sensitivity to secretagogues and corticosterone.
Topics: Animals; Animals, Newborn; Bucladesine; Carbachol; Colforsin; Corticosterone; Dose-Response Relationship, Drug; Gastric Acid; Guanidines; Histamine; Imidazoles; Impromidine; Male; Pentagastrin; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Stomach | 1989 |
Functional role of M2 muscarinic receptors in the guinea pig ileum.
Topics: Animals; Colforsin; Cyclic AMP; Guinea Pigs; Heart; Histamine; Ileum; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Oxotremorine; Pertussis Toxin; Piperidines; Rats; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Signal Transduction; Submandibular Gland; Virulence Factors, Bordetella | 1995 |
207 other study(ies) available for histamine and colforsin
Article | Year |
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Synergistic action of cyclic GMP on catecholamine-induced chloride current in guinea-pig ventricular cells.
Topics: Animals; Catecholamines; Cells, Cultured; Chlorides; Colforsin; Cyclic AMP; Cyclic GMP; Guinea Pigs; Heart Ventricles; Histamine; Ion Channels; Isoproterenol; Membrane Potentials; Milrinone; Myocardium; Pyridones | 1992 |
Histamine-induced depolarization and the cyclic AMP--protein kinase A system in isolated guinea pig adipocytes.
Topics: 1-Methyl-3-isobutylxanthine; Adipose Tissue; Alprostadil; Animals; Carbazoles; Colforsin; Cyclic AMP; Electrophysiology; Epididymis; Guinea Pigs; Histamine; In Vitro Techniques; Indoles; Insulin; Isoproterenol; Male; Membrane Potentials; Protein Kinase C; Protein Kinases; Pyrroles; Rats; Rats, Wistar | 1992 |
Influence of acid secretory state on Cl(-)-base and Na(+)-H+ exchange and pHi in isolated rabbit parietal cells.
Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Aminopyrine; Animals; Carrier Proteins; Chlorides; Colforsin; Extracellular Space; Gastric Acid; Histamine; Hydrogen-Ion Concentration; Omeprazole; Parietal Cells, Gastric; Rabbits; Rest; Sodium-Hydrogen Exchangers | 1992 |
H2 receptor-mediated responses of aortic endothelial cells to histamine.
Topics: Animals; Aorta; Cell Membrane Permeability; Cells, Cultured; Colforsin; Cyclic AMP; Drug Combinations; Endothelium, Vascular; Histamine; Histamine Antagonists; Ranitidine; Receptors, Histamine H2 | 1992 |
Fructose 2,6-bisphosphate levels and modulation of glycolysis by histamine, cholecystokinin, and forskolin in isolated rabbit gastric glands.
Topics: 3-O-Methylglucose; Animals; Colforsin; Cyclic AMP; Fructosediphosphates; Gastric Mucosa; Glucose; Glycolysis; Histamine; In Vitro Techniques; Kinetics; Lactates; Methylglucosides; Pepsinogens; Phosphofructokinase-2; Phosphotransferases; Rabbits; Sincalide | 1992 |
Ion transport by primary cultures of Mongolian gerbil middle ear epithelium.
Topics: Amiloride; Animals; Arginine Vasopressin; Biological Transport; Bradykinin; Cell Membrane; Cell Membrane Permeability; Cells, Cultured; Chlorides; Colforsin; Cyclic AMP; Dinoprostone; Ear, Middle; Epithelium; Gerbillinae; Glucagon; Histamine; Indomethacin; Isoproterenol; Male; Mannitol; Microscopy, Electron; Parathyroid Hormone; Sodium | 1992 |
Vasoactive intestinal peptide is a secretagogue in bovine chromaffin cells pretreated with pertussis toxin.
Topics: Adenylate Cyclase Toxin; Adrenal Medulla; Animals; Catecholamines; Cattle; Cells, Cultured; Colforsin; Cyclic AMP; Histamine; Pertussis Toxin; Phosphatidylinositols; Second Messenger Systems; Vasoactive Intestinal Peptide; Virulence Factors, Bordetella | 1992 |
Adenylate cyclase induces intracellular calcium increase in single human epidermal keratinocytes measured by fluorescence microscopy using Fura 2-AM.
Topics: Adenosine; Adenylyl Cyclases; Bucladesine; Calcium; Cells, Cultured; Colforsin; Epinephrine; Fluorescent Dyes; Fura-2; Histamine; Humans; Intracellular Fluid; Keratinocytes; Microscopy, Fluorescence | 1992 |
Pertussis toxin reverses prostaglandin E2- and somatostatin-induced inhibition of rat parietal cell H(+)-production.
Topics: Adenosine Diphosphate; Adenylate Cyclase Toxin; Aminopyrine; Animals; Colforsin; Dinoprostone; Female; GTP-Binding Proteins; Histamine; Parietal Cells, Gastric; Pertussis Toxin; Protons; Rats; Rats, Inbred Strains; Somatostatin; Virulence Factors, Bordetella | 1992 |
Protein kinase C inhibits histamine H2 receptor-mediated stimulation of cyclic AMP content in the human gastric cancer cell line HGT-1.
Topics: Cell Line; Cholera Toxin; Colforsin; Cyclic AMP; Histamine; Histamine H2 Antagonists; Humans; Protein Kinase C; Receptors, Histamine H2; Stomach Neoplasms; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1992 |
Role of GTP-binding proteins in the regulation of mammalian cardiac chloride conductance.
Topics: Acetylcholine; Adenylate Cyclase Toxin; Adrenergic beta-Agonists; Animals; Carbachol; Cells, Cultured; Chloride Channels; Chlorides; Colforsin; Cyclic AMP; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; Heart; Histamine; Ion Channels; Isoproterenol; Membrane Proteins; Myocardium; Pertussis Toxin; Phosphorylation; Propranolol; Receptors, Adrenergic, beta; Receptors, Muscarinic; Time Factors; Virulence Factors, Bordetella | 1992 |
Effect of albumin on adenylate cyclase receptor-related signal transduction of human peripheral blood mononuclear cells.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Colforsin; Cyclic AMP; Drug Interactions; Enzyme Activation; Histamine; Humans; Hydrogen-Ion Concentration; Isoproterenol; Monocytes; Serum Albumin; Signal Transduction | 1992 |
Modulation of potassium channels in intact human T lymphocytes.
Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Calcium; Colforsin; Cyclic AMP; Cytoplasm; Dinoprostone; Electric Stimulation; Histamine; Humans; Isoproterenol; Potassium Channels; T-Lymphocytes; Temperature | 1992 |
Acute endothelial cell contraction in vitro: a comparison with vascular smooth muscle cells and fibroblasts.
Topics: Actin Cytoskeleton; Animals; Aorta; Bradykinin; Cattle; Colforsin; Culture Techniques; Cytochalasin B; Endothelium; Fibroblasts; Histamine; Muscle Contraction; Muscle, Smooth, Vascular; Rats; Serotonin; Thrombin; Vasoconstriction | 1992 |
Desensitization of the epidermal adenylate cyclase system: agonists and phorbol esters desensitize by independent mechanisms.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine; Adenosine Triphosphate; Adenylate Cyclase Toxin; Adenylyl Cyclases; Alkaloids; Animals; Cholera Toxin; Colforsin; Cyclic AMP; Epidermis; Epinephrine; Histamine; Isoquinolines; Pertussis Toxin; Piperazines; Receptors, Adrenergic, beta; Receptors, Histamine; Skin; Staurosporine; Swine; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella | 1991 |
Cyclic AMP generating systems in vertebrate retina: effects of histamine and an established retinal modulator, dopamine.
Topics: Adenylyl Cyclases; Animals; Cerebral Cortex; Chickens; Cimetidine; Colforsin; Cyclic AMP; Dimaprit; Dopamine; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistamines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Retina; Thiazoles; Thiourea | 1991 |
1,25-dihydroxyvitamin D3 and agents that increase intracellular adenosine 3',5'-monophosphate synergistically inhibit the mitogenic stimulation of human lymphocytes.
Topics: 1-Methyl-3-isobutylxanthine; Adenosine Monophosphate; Binding Sites; Calcitriol; Cells, Cultured; Cholera Toxin; Colforsin; Cyclic AMP; Dinoprostone; Drug Synergism; Histamine; Humans; In Vitro Techniques; Lymphocyte Activation; Lymphocytes | 1990 |
Cl- channel blockers inhibit acid secretion in rabbit parietal cells.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Anthracenes; Atropine; Carbachol; Chloride Channels; Cimetidine; Colforsin; Gastric Acid; Gastric Mucosa; Histamine; In Vitro Techniques; Ion Channels; Kinetics; Membrane Proteins; ortho-Aminobenzoates; Rabbits | 1990 |
Effect of substance P and neurokinin A on rat parietal cell function.
Topics: Aminopyrine; Animals; Biological Transport; Bucladesine; Carbachol; Cell Separation; Colforsin; Cyclic AMP; Female; Histamine; In Vitro Techniques; Kinetics; Neurokinin A; Parietal Cells, Gastric; Rats; Rats, Inbred Strains; Substance P | 1990 |
GLP-1-(7-36) amide, -(1-37), and -(1-36) amide: potent cAMP-dependent stimuli of rat parietal cell function.
Topics: 1-Methyl-3-isobutylxanthine; Aminopyrine; Animals; Biological Transport; Bucladesine; Carbachol; Colforsin; Cyclic AMP; Female; Gastric Acid; Glucagon; Glucagon-Like Peptide 1; Glucagon-Like Peptides; Histamine; In Vitro Techniques; Inositol Phosphates; Kinetics; Parietal Cells, Gastric; Peptide Fragments; Peptides; Pertussis Toxin; Rats; Rats, Inbred Strains; Virulence Factors, Bordetella | 1991 |
Effects of histamine and activators of the cyclic AMP system on protein synthesis in and release of high molecular weight glycoproteins from isolated gastric non-parietal cells.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Bucladesine; Cell Separation; Chromatography, Gel; Colforsin; Cyclic AMP; Gastric Mucosa; Glycoproteins; Histamine; In Vitro Techniques; Molecular Weight; Protein Biosynthesis; Ranitidine; Swine | 1991 |
Histamine-induced increases in cyclic AMP levels in bovine adrenal medullary cells.
Topics: 1-Methyl-3-isobutylxanthine; Adrenal Medulla; Animals; Calcium; Cattle; Cells, Cultured; Chromaffin System; Colforsin; Cyclic AMP; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Radioimmunoassay; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3 | 1991 |
Signal transduction pathway in gastric mucous cells.
Topics: Adenylyl Cyclases; Animals; Calcium; Carbachol; Cell Membrane; Cholera Toxin; Colforsin; Cytosol; Dinoprost; Dinoprostone; Dose-Response Relationship, Drug; Enzyme Activation; Gastric Mucosa; Guinea Pigs; Histamine; In Vitro Techniques; Kinetics; Phosphatidylserines; Protein Kinase C; Protein Kinases; Signal Transduction; Tetradecanoylphorbol Acetate | 1991 |
Thapsigargin potentiates histamine-stimulated HCl secretion in gastric parietal cells but does not mimic cholinergic responses.
Topics: Aminopyrine; Animals; Calcium; Carbachol; Colforsin; Cyclic AMP; Drug Synergism; Gastric Acid; Gastric Mucosa; Histamine; In Vitro Techniques; Rabbits; Receptors, Cholinergic; Terpenes; Tetradecanoylphorbol Acetate; Thapsigargin | 1991 |
Relation of anion secretory activity to intracellular Ca2+ in response to lysylbradykinin and histamine in a cultured human colonic epithelium.
Topics: Acetazolamide; Calcimycin; Calcium; Carbachol; Cell Line; Cells, Cultured; Colforsin; Colon; Digitonin; Drug Interactions; Epithelial Cells; Epithelium; Fura-2; Histamine; Humans; Intestinal Mucosa; Kallidin; Kinetics; Spectrometry, Fluorescence; Sulfonamides | 1991 |
Isolation of H+,K(+)-ATPase-containing membranes from the gastric oxyntic cell.
Topics: 4-Nitrophenylphosphatase; Adenosine Triphosphatases; Animals; Cell Fractionation; Cell Membrane; Centrifugation, Density Gradient; Cimetidine; Colforsin; Female; Gastric Mucosa; H(+)-K(+)-Exchanging ATPase; Histamine; Indicators and Reagents; Kinetics; Male; Molecular Weight; Parietal Cells, Gastric; Rabbits | 1990 |
Discriminatory effects of forskolin and EGTA on the indirect cyclic AMP responses to histamine, noradrenaline, 5-hydroxytryptamine, and glutamate in guinea-pig cerebral cortical slices.
Topics: Animals; Cerebral Cortex; Colforsin; Cyclic AMP; Egtazic Acid; Glutamates; Glutamic Acid; Guinea Pigs; Histamine; In Vitro Techniques; Inositol Phosphates; Neurotransmitter Agents; Norepinephrine; Phorbol 12,13-Dibutyrate; Serotonin | 1990 |
Effects of histamine on protein and glycoprotein production of isolated pig gastric mucosal cells.
Topics: 16,16-Dimethylprostaglandin E2; Acetylglucosamine; Animals; Colforsin; Gastric Mucosa; Glycoproteins; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Leucine; Protein Biosynthesis; Pyrilamine; Ranitidine; Receptors, Histamine H1; Receptors, Histamine H2; Swine; Tritium | 1990 |
Adenylate cyclase induces intracellular Ca2+ increase in single human epidermal keratinocytes of the epidermal sheet as measured by digital imaging microscopy using Fura 2-AM.
Topics: Adenosine; Adenylyl Cyclases; Albuterol; Calcium; Cells, Cultured; Colforsin; Epinephrine; Fura-2; Histamine; Humans; Keratinocytes; Microscopy, Fluorescence; Propranolol | 1991 |
Effects of epidermal growth factor on signal transduction in rabbit parietal cells.
Topics: Aminopyrine; Animals; Benzofurans; Buffers; Calcium; Carbachol; Colforsin; Cyclic AMP; Cytosol; Epidermal Growth Factor; Fluorescent Dyes; Fura-2; Gastric Acid; Histamine; In Vitro Techniques; Intrinsic Factor; Kinetics; Parietal Cells, Gastric; Phosphorylation; Proteins; Rabbits; Signal Transduction | 1990 |
Adenylate cyclase system in fetal rat keratinizing epidermal cells (FRSK cells) and SV40-transformed human keratinocytes.
Topics: Adenosine; Adenylyl Cyclases; Animals; Blotting, Northern; Cell Line; Cell Line, Transformed; Cholera Toxin; Colforsin; Cyclic AMP; Dinoprostone; Epinephrine; Histamine; Humans; Keratinocytes; Rats; RNA, Messenger; Simian virus 40 | 1990 |
A cAMP-activated chloride channel in the plasma membrane of cultured human gastric cells (HGT-1).
Topics: Adenocarcinoma; Bucladesine; Cell Membrane; Cell Membrane Permeability; Chloride Channels; Colforsin; Cyclic AMP; Electrophysiology; Histamine; Humans; Membrane Proteins; ortho-Aminobenzoates; Parietal Cells, Gastric; Stomach Neoplasms; Tumor Cells, Cultured | 1990 |
Increased airway reactivity in the guinea-pig follows exposure to intravenous isoprenaline.
Topics: Airway Resistance; Animals; Atropine; Blood Platelets; Bombesin; Bronchodilator Agents; Colforsin; Dopamine; Epinephrine; Guinea Pigs; Histamine; Injections, Intravenous; Isoproterenol; Male; Norepinephrine; Platelet Activating Factor; Propranolol; Rabbits; Vagotomy; Vagus Nerve | 1990 |
Effects of histamine on dentate granule cells in vitro.
Topics: Action Potentials; Adenylyl Cyclases; Animals; Colforsin; Hippocampus; Histamine; In Vitro Techniques; Membrane Potentials; Rats; Rats, Inbred Strains | 1990 |
Inhibition of parietal cell H+ secretion by transforming growth factor alpha: a possible autocrine regulatory mechanism.
Topics: Aminopyrine; Animals; Bicarbonates; Buffers; Carbachol; Cell Separation; Colforsin; Histamine; Hydrogen; Parietal Cells, Gastric; Pertussis Toxin; Transforming Growth Factors; Virulence Factors, Bordetella | 1990 |
Histamine content and release of isolated rat gastric mucosal cells.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Carbachol; Colforsin; Diterpenes; Gastric Mucosa; Histamine; Histamine Release; In Vitro Techniques; Rats | 1985 |
The stimulatory effect of forskolin on gastric acid secretion in rats.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Carbachol; Cimetidine; Colforsin; Dose-Response Relationship, Drug; Gastric Acid; Histamine; Male; Rats; Rats, Inbred Strains; Stimulation, Chemical; Time Factors | 1986 |
Prostanoid inhibition of canine parietal cells.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Aminopyrine; Animals; Carbachol; Cells, Cultured; Colforsin; Cyclic AMP; Dinoprostone; Dogs; Enprostil; Histamine; Parietal Cells, Gastric; Prostaglandins E; Prostaglandins E, Synthetic; Stimulation, Chemical | 1986 |
Interaction of phosphodiesterase inhibitors triamterene, papaverine, theophylline, IBMX and amrinone with other positive inotropic acting substances on isolated guinea-pig atria.
Topics: 1-Methyl-3-isobutylxanthine; Amrinone; Animals; Colforsin; Drug Interactions; Electric Stimulation; Guinea Pigs; Heart Rate; Histamine; In Vitro Techniques; Male; Metaproterenol; Myocardial Contraction; Papaverine; Phosphodiesterase Inhibitors; Stimulation, Chemical; Theophylline; Triamterene | 1987 |
Relationships of secretagogue-induced cAMP accumulation and acid secretion in elutriated rat gastric parietal cells.
Topics: 1-Methyl-3-isobutylxanthine; 3',5'-Cyclic-AMP Phosphodiesterases; Aminopyrine; Animals; Chromatography, High Pressure Liquid; Colforsin; Cyclic AMP; Fluorescence; Gastric Acid; Gastric Mucosa; Histamine; In Vitro Techniques; Isoproterenol; Male; Microscopy, Electron; Radioimmunoassay; Rats; Rats, Inbred Strains | 1988 |
Reduction of beta-adrenoceptor density and evaluation of positive inotropic responses in isolated, diseased human myocardium.
Topics: 1-Methyl-3-isobutylxanthine; Adult; Bucladesine; Calcium; Cardiac Output, Low; Cardiotonic Agents; Colforsin; Digitoxin; Digoxin; Dobutamine; Histamine; Humans; In Vitro Techniques; Middle Aged; Myocardial Contraction; Myocardium; Receptors, Adrenergic, beta; Stimulation, Chemical | 1988 |
Positive inotropic effects in isolated ventricular myocardium from non-failing and terminally failing human hearts.
Topics: 1-Methyl-3-isobutylxanthine; Adult; Bucladesine; Calcium; Cardiomyopathy, Dilated; Cardiotonic Agents; Colforsin; Coronary Disease; Female; Histamine; Humans; In Vitro Techniques; Male; Middle Aged; Myocardial Contraction; Papillary Muscles | 1988 |
Fura 2 analysis of cytosolic calcium regulation in elutriated rat gastric parietal cells.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Benzofurans; Calcium; Carbachol; Colforsin; Cytosol; Fluorescent Dyes; Fura-2; Histamine; Homeostasis; In Vitro Techniques; Kinetics; Male; Molecular Weight; Parietal Cells, Gastric; Phosphoproteins; Phosphorylation; Rats; Rats, Inbred Strains; Spectrometry, Fluorescence | 1989 |
Beta-adrenergic relaxation of dog trachealis: contractile agonist-specific interaction.
Topics: 1-Methyl-3-isobutylxanthine; Acetylcholine; Adrenergic beta-Agonists; Animals; Bucladesine; Colforsin; Dogs; Histamine; In Vitro Techniques; Isoproterenol; Muscle Contraction; Muscle, Smooth; Potassium Chloride; Serotonin; Trachea | 1989 |
Ca2+-dependent and -independent secretagogue action on gastric mucus secretion in rabbit mucosal explants.
Topics: Acetylcholine; Acetylglucosamine; Animals; Atropine; Calcimycin; Calcium; Calmodulin; Colforsin; Dinoprostone; Gastric Fundus; Gastric Mucosa; Glycoproteins; Histamine; Male; Molecular Weight; Organ Culture Techniques; Pentagastrin; Pyloric Antrum; Rabbits; Sulfonamides; Tetradecanoylphorbol Acetate | 1989 |
Role of Ca2+ in H+ transport by rabbit gastric glands studied with A23187 and BAPTA, an incorporated Ca2+ chelator.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Acetylcholine; Aminopyrine; Benzofurans; Calcimycin; Calcium; Chelating Agents; Colforsin; Egtazic Acid; Fura-2; Gastric Acid; Gastric Mucosa; Histamine; Kinetics | 1989 |
cAMP- and calcium-mediated modulation of intrinsic factor secretion in isolated rabbit gastric glands.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Calcimycin; Calcium; Carbachol; Colforsin; Cyclic AMP; Histamine; In Vitro Techniques; Intrinsic Factor; Parietal Cells, Gastric; Pentagastrin; Rabbits | 1989 |
Cytoplasmic Ca2+ is a primary determinant for myosin phosphorylation in smooth muscle cells.
Topics: Animals; Calcium; Cattle; Colforsin; Cyclic AMP; Cyclic GMP; Cytoplasm; Ethers; Histamine; In Vitro Techniques; Ionomycin; Muscle, Smooth; Myosins; Phosphorylation; Serotonin; Trachea | 1989 |
Histamine-mediated vasoconstriction and cAMP levels in coronary arteries of the isolated rabbit heart.
Topics: Animals; Blood Pressure; Colforsin; Coronary Vessels; Cyclic AMP; Female; Heart; Histamine; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Myocardial Contraction; Myocardium; Perfusion; Rabbits; Theophylline; Vasoconstriction | 1989 |
Synergistic potentiation of polyphosphoinositide breakdown by adenylate cyclase coupled receptors in human endothelial cells.
Topics: Adenylyl Cyclases; Bucladesine; Cells, Cultured; Cholera Toxin; Colforsin; Drug Synergism; Endothelium, Vascular; Histamine; Humans; Isoproterenol; Phosphatidylinositols; Receptors, Cyclic AMP; Signal Transduction | 1989 |
Histamine-mediated regulation of cAMP levels and inositol phosphate metabolism in isolated rabbit retina.
Topics: Animals; Carbachol; Colforsin; Cyclic AMP; Histamine; In Vitro Techniques; Inositol Phosphates; Rabbits; Receptors, Histamine H1; Retina | 1989 |
The possible role of histamine-mediated cAMP formation as a link between H2-receptor stimulation and ultrastructural changes in guinea-pig oxyntic cells.
Topics: Animals; Colforsin; Cyclic AMP; Guanosine Triphosphate; Guinea Pigs; Histamine; In Vitro Techniques; Microtubules; Parietal Cells, Gastric; Ranitidine; Receptors, Histamine H2; Tubulin | 1989 |
Inhibition of histamine-stimulated inositol phospholipid hydrolysis by agents which increase cyclic AMP levels in bovine tracheal smooth muscle.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenine; Albuterol; Animals; Bucladesine; Cattle; Colforsin; Cyclic AMP; Histamine; Histamine Antagonists; Hydrolysis; In Vitro Techniques; Inositol Phosphates; Muscle, Smooth; Phosphodiesterase Inhibitors; Pyrrolidinones; Rolipram; Sugar Phosphates; Trachea; Vasoactive Intestinal Peptide | 1989 |
Pancreastatin: a novel peptide inhibitor of parietal cell signal transduction.
Topics: Aminopyrine; Animals; Calcium; Carbachol; Chromogranin A; Colforsin; Cyclic AMP; Histamine; In Vitro Techniques; Pancreatic Hormones; Parietal Cells, Gastric; Pertussis Toxin; Rabbits; Signal Transduction; Spectrometry, Fluorescence; Virulence Factors, Bordetella | 1989 |
Histamine and inositol phosphate accumulation in endothelium: cAMP and a G protein.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Cells, Cultured; Colforsin; Cyclic AMP; Endothelium, Vascular; Female; GTP-Binding Proteins; Histamine; Humans; Inositol Phosphates; Kinetics; Pregnancy; Theophylline; Umbilical Veins | 1989 |
Multiple signaling pathways of histamine H2 receptors. Identification of an H2 receptor-dependent Ca2+ mobilization pathway in human HL-60 promyelocytic leukemia cells.
Topics: Calcium; Calcium Channel Blockers; Cell Differentiation; Cholera Toxin; Colforsin; Cyclic AMP; Dimethyl Sulfoxide; Dinoprostone; Histamine; Humans; Inositol 1,4,5-Trisphosphate; Isoproterenol; Kinetics; Leukemia, Promyelocytic, Acute; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Receptors, Histamine H2; Signal Transduction; Tumor Cells, Cultured | 1989 |
Regulation of cytosolic free Ca2+ concentration in vascular smooth muscle cells by A- and C-kinases.
Topics: Benzofurans; Calcium; Colforsin; Cytosol; Fluorescent Dyes; Fura-2; Histamine; Humans; Image Processing, Computer-Assisted; Muscle, Smooth, Vascular; Osmolar Concentration; Phorbol Esters; Protein Kinase C; Protein Kinases; Umbilical Veins; Vasopressins | 1989 |
Effects of phorbol esters and forskolin on basal and histamine-induced accumulation of inositol phosphates in cultured bovine adrenal chromaffin cells.
Topics: Adrenal Medulla; Animals; Cattle; Cells, Cultured; Cimetidine; Colforsin; Epinephrine; Histamine; Inositol Phosphates; Kinetics; Norepinephrine; Phorbol Esters; Pyrilamine; Sugar Phosphates; Tetradecanoylphorbol Acetate | 1989 |
Histamine increases phosphorylation of 27- and 40-kDa parietal cell proteins.
Topics: Animals; Calcium; Colforsin; Cyclic AMP; Cytoskeleton; Gastric Mucosa; Histamine; Molecular Weight; Phosphoproteins; Polyethylene Glycols; Rabbits; Solubility; Time Factors | 1987 |
Interactions between intracellular cyclic AMP and agonist-induced inositol phospholipid breakdown in isolated gastric mucosal cells of the rat.
Topics: Animals; Bucladesine; Carbachol; Cimetidine; Colforsin; Cyclic AMP; Dibutyryl Cyclic GMP; Enzyme Activation; Histamine; In Vitro Techniques; Inositol Phosphates; Male; Parietal Cells, Gastric; Phorbol Esters; Phosphodiesterase Inhibitors; Protein Kinase C; Pyrrolidinones; Rats; Rats, Inbred Strains; Rolipram; Sugar Phosphates | 1987 |
Mechanism of excitatory amino acid-induced accumulation of cyclic AMP in hippocampal slices: role of extracellular chloride.
Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Aminobutyrates; Animals; Bromides; Chlorides; Colforsin; Cyclic AMP; Fluorides; Furosemide; Guinea Pigs; Hippocampus; Histamine; Male | 1988 |
Differential inhibitory effects of forskolin, isoproterenol, and dibutyryl cyclic adenosine monophosphate on phosphoinositide hydrolysis in canine tracheal smooth muscle.
Topics: Animals; Bucladesine; Colforsin; Dogs; Histamine; Hydrolysis; Isoproterenol; Methacholine Chloride; Methacholine Compounds; Muscle Contraction; Muscle, Smooth; Phosphatidylinositols; Trachea | 1988 |
[Is forskolin a stimulant of gastric secretion?].
Topics: Aminopyridines; Animals; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Gastric Acid; Gastrins; Histamine; Parietal Cells, Gastric; Rabbits; Rats | 1988 |
A study of the H2-receptor for histamine stimulating adenylate cyclase in homogenates of guinea-pig lung parenchyma.
Topics: Adenylyl Cyclases; Animals; Cimetidine; Colforsin; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Lung; Male; Propranolol; Pyrilamine; Receptors, Histamine; Receptors, Histamine H2 | 1986 |
Mechanisms for direct inhibition of canine gastric parietal cells by somatostatin.
Topics: Aminopyrine; Animals; Carbachol; Cell Membrane; Cell Separation; Colforsin; Cyclic AMP; Dogs; Histamine; In Vitro Techniques; Kinetics; Parietal Cells, Gastric; Pentagastrin; Pertussis Toxin; Phosphates; Phosphatidylinositols; Receptors, Neurotransmitter; Receptors, Somatostatin; Somatostatin; Virulence Factors, Bordetella | 1987 |
Somatostatin inhibition of secretagogue and forskolin-stimulated gastric acid secretion.
Topics: Acetylcholine; Animals; Bufo marinus; Colforsin; Gastric Acid; Gastric Mucosa; Histamine; In Vitro Techniques; Indomethacin; Kinetics; Somatostatin | 1988 |
Modulation of guinea-pig lung adenylate cyclase by ovalbumin sensitization.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Bradykinin; Colforsin; Dose-Response Relationship, Drug; Guanosine Triphosphate; Guinea Pigs; Histamine; Immunoglobulin G; Lung; Male; Ovalbumin; Sodium Fluoride | 1988 |
Inhibition by forskolin of excitatory amino acid-induced accumulation of cyclic AMP in guinea pig hippocampal slices.
Topics: Adenosine; Amino Acids; Animals; Aspartic Acid; Chlorides; Colforsin; Cyclic AMP; Cysteine; Drug Interactions; Ethylmaleimide; Glutamates; Glutamic Acid; Guanosine Triphosphate; Guinea Pigs; Hippocampus; Histamine; Male; N-Methylaspartate; Neurotransmitter Agents; Veratridine | 1988 |
Histamine dependent cyclic AMP generating system in rabbit CNS: interaction with neuroregulators and forskolin.
Topics: Animals; Central Nervous System; Cerebral Cortex; Colforsin; Cyclic AMP; Histamine; In Vitro Techniques; Neurotransmitter Agents; Rabbits; Retina | 1988 |
Pancreastatin: a novel peptide inhibitor of parietal cell secretion.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Aminopyrine; Animals; Carbachol; Chromogranin A; Colforsin; Histamine; In Vitro Techniques; Pancreatic Hormones; Parietal Cells, Gastric; Peptides; Rabbits; Somatostatin | 1988 |
Parietal cell protein kinases. Selective activation of type I cAMP-dependent protein kinase by histamine.
Topics: Adenylyl Cyclase Inhibitors; Animals; Azides; Colforsin; Cyclic AMP; Diterpenes; Enzyme Activation; Histamine; Kinetics; Molecular Weight; Parietal Cells, Gastric; Protein Kinases; Rabbits; Subcellular Fractions | 1985 |
Biochemical characterization of a filtered synaptoneurosome preparation from guinea pig cerebral cortex: cyclic adenosine 3':5'-monophosphate-generating systems, receptors, and enzymes.
Topics: 2-Chloroadenosine; 3',5'-Cyclic-AMP Phosphodiesterases; Acetylcholinesterase; Adenosine; Adenylyl Cyclases; Animals; Butyrylcholinesterase; Cerebral Cortex; Colforsin; Cyclic AMP; Diterpenes; Dose-Response Relationship, Drug; Filtration; Guinea Pigs; Histamine; Microscopy, Electron; Norepinephrine; Receptors, Adrenergic, beta; Receptors, Cell Surface; Receptors, Histamine H2; Receptors, Purinergic; Synaptosomes | 1985 |
Influence of the epithelium on responsiveness of guinea-pig isolated trachea to contractile and relaxant agonists.
Topics: Acetylcholine; Animals; Asthma; Autoradiography; Carbachol; Cimetidine; Colforsin; Dose-Response Relationship, Drug; Epithelium; Female; Guinea Pigs; Histamine; In Vitro Techniques; Iodocyanopindolol; Isoproterenol; Kinetics; Male; Muscle Contraction; Nitroglycerin; Pindolol; Potassium; Receptors, Adrenergic, beta; Theophylline; Trachea | 1986 |
Prostaglandin E2 inhibition of secretagogue-stimulated [14C]aminopyrine accumulation in rat parietal cells: a model for its mechanism of action.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Aminopyrine; Animals; Bucladesine; Carbon Radioisotopes; Colforsin; Dinoprostone; Dose-Response Relationship, Drug; GTP-Binding Proteins; Histamine; In Vitro Techniques; Isoproterenol; Male; Models, Biological; Parasympathetic Nervous System; Parietal Cells, Gastric; Pertussis Toxin; Prostaglandins E; Rats; Rats, Inbred Strains; Virulence Factors, Bordetella | 1986 |
Effect of adenosine receptor agonists and other compounds on cyclic AMP accumulation in forskolin-treated hippocampal slices.
Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adenylyl Cyclases; Animals; Colforsin; Cyclic AMP; Deoxyadenosines; Dideoxyadenosine; Dinoprostone; Dose-Response Relationship, Drug; Enzyme Activation; Hippocampus; Histamine; Isoproterenol; Male; Phenylisopropyladenosine; Prostaglandins E; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Purinergic; Theophylline; Xanthines | 1986 |
Effect of ethanol on acid secretion by isolated gastric glands from rabbit.
Topics: Adenosine Triphosphatases; Adenylyl Cyclases; Aminopyrine; Animals; Cell Membrane; Cell Membrane Permeability; Colforsin; Ethanol; Gastric Acid; Gastric Fundus; Gastric Mucosa; Histamine; In Vitro Techniques; Intracellular Membranes; Parietal Cells, Gastric; Protons; Rabbits | 1986 |
Effect of age on the formation of cyclic nucleotides in guinea-pig tracheal smooth muscle in response to pharmacological agents.
Topics: Aging; Alprostadil; Animals; Carbachol; Cholera Toxin; Colforsin; Cyclic AMP; Cyclic GMP; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Male; Muscle, Smooth; Nitroprusside; Potassium; Trachea | 1986 |
Serotonin-1C sites in the choroid plexus are not linked in a stimulatory or inhibitory way to adenylate cyclase.
Topics: Adenylyl Cyclases; Animals; Binding, Competitive; Cerebral Cortex; Choroid Plexus; Colforsin; Cyclic AMP; Dopamine; Ergolines; Hippocampus; Histamine; Kinetics; Mianserin; Rats; Receptors, Serotonin; Serotonin; Swine | 1986 |
Adenosine receptors on human lymphocytes.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Alprostadil; Binding Sites; Colforsin; Cyclic AMP; Deoxyadenosines; Dideoxyadenosine; Histamine; Humans; In Vitro Techniques; Isoproterenol; Lymphocytes; Manganese; Neutrophils; Receptors, Purinergic; Theophylline; Vidarabine | 1986 |
Stimulation-associated redistribution of H+-K+-ATPase activity in isolated gastric glands.
Topics: Adenosine Triphosphatases; Animals; Carbachol; Cell Compartmentation; Colforsin; Cyclic AMP; Female; Gastric Juice; Gastric Mucosa; Glucosides; H(+)-K(+)-Exchanging ATPase; Histamine; Hydrogen-Ion Concentration; Male; Metiamide; Microsomes; Oligomycins; Potassium; Rabbits; Time Factors | 1987 |
Prostaglandin inhibition of acid is cAMP dependent.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Aminopyrine; Animals; Cholera Toxin; Colforsin; Cyclic AMP; Ethylmaleimide; Gastric Acid; Histamine; In Vitro Techniques; Parietal Cells, Gastric; Prostaglandins E; Rabbits | 1987 |
A calmodulin antagonist inhibits histamine-stimulated acid production by isolated rat parietal cells.
Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Aminopyrine; Animals; Bucladesine; Calmodulin; Colforsin; Gastric Acid; H(+)-K(+)-Exchanging ATPase; Histamine; Hydrogen-Ion Concentration; In Vitro Techniques; Oligomycins; Parietal Cells, Gastric; Potassium; Rats; Receptors, Histamine H2; Sulfonamides | 1987 |
Similarities in cAMP responses between murine lymphoid cell lines and subsets of mouse lymphocytes.
Topics: Animals; Cell Line; Colforsin; Cyclic AMP; Dinoprostone; Drug Synergism; Enzyme Activation; Histamine; Isoproterenol; Lymphocytes; Mice; Prostaglandins E; Protein Kinases | 1987 |
Role of cyclic AMP in renin secretion by human transfected juxtaglomerular cells.
Topics: Bucladesine; Cell Transformation, Viral; Cells, Cultured; Cimetidine; Colforsin; Cyclic AMP; Histamine; Humans; Isoproterenol; Juxtaglomerular Apparatus; Renin; Simian virus 40; Transfection | 1986 |
Regulation of hormone-stimulated cyclic AMP accumulation in intact human mononuclear leukocytes by blood plasma.
Topics: Adenosine Triphosphate; Adenylate Cyclase Toxin; Alprostadil; Cold Temperature; Colforsin; Cyclic AMP; GTP-Binding Proteins; Histamine; Humans; Isoproterenol; Lymphocytes; Monocytes; Virulence Factors, Bordetella | 1986 |
Relaxant effects of forskolin on guinea pig tracheal smooth muscle.
Topics: Animals; Colforsin; Cyclic AMP; Differential Threshold; Ethanol; Guinea Pigs; Histamine; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Respiration; Trachea | 1987 |
Protein phosphorylation changes in bovine carotid artery smooth muscle during contraction and relaxation.
Topics: Angiotensin II; Animals; Calcium; Carotid Arteries; Cattle; Colforsin; Cytoplasm; Diglycerides; Histamine; Muscle Contraction; Muscle Proteins; Muscle Relaxation; Muscle, Smooth, Vascular; Phorbol Esters; Phosphoproteins; Phosphorylation; Potassium; Trachea | 1988 |
Effects of histamine on the metabolism of isolated rat hepatocytes: roles of H1- and H2-histamine receptors.
Topics: Animals; Calcium; Colforsin; Gluconeogenesis; Histamine; Hypothyroidism; Liver; Liver Glycogen; Pertussis Toxin; Rats; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Tetradecanoylphorbol Acetate; Urea; Virulence Factors, Bordetella | 1987 |
Transduction of aminergic and peptidergic signals in enteric neurones of the guinea-pig.
Topics: Action Potentials; Animals; Biogenic Amines; Colforsin; Guinea Pigs; Histamine; In Vitro Techniques; Myenteric Plexus; Neurons; Peptides; Serotonin; Time Factors | 1987 |
Cholecystokinin, carbachol, gastrin, histamine, and forskolin increase [Ca2+]i in gastric glands.
Topics: Aminoquinolines; Animals; Atropine; Calcium; Carbachol; Colforsin; Dibutyryl Cyclic GMP; Fluorescent Dyes; Gastric Mucosa; Gastrins; Histamine; Male; Pepsinogens; Rabbits; Sincalide; Spectrometry, Fluorescence | 1986 |
Differential effects of extracellular calcium removal and nonspecific effects of Ca2+ antagonists on acid secretory activity in isolated gastric glands.
Topics: Aminopyrine; Animals; Calcium; Carbachol; Carbon Radioisotopes; Colforsin; Egtazic Acid; Exocrine Glands; Gastric Acid; Gastric Juice; Gastric Mucosa; Histamine; In Vitro Techniques; Kinetics; Male; Rabbits | 1985 |
Evidence for the involvement of histamine in the regulation of blood-brain barrier permeability.
Topics: Animals; Blood-Brain Barrier; Colforsin; Diterpenes; Dogs; Female; Fluorescein; Fluoresceins; Histamine; Histamine Antagonists; Male; Methylhistamines; Metiamide; Pyrilamine; Time Factors | 1985 |
Phorbol myristate acetate causes in guinea-pig lung parenchymal strip a maintained spasm which is relatively resistant to isoprenaline.
Topics: Aminophylline; Animals; Colforsin; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Lung; Male; Muscle Contraction; Muscle, Smooth; Nitroprusside; Phorbols; Tetradecanoylphorbol Acetate | 1985 |
Activation of cyclic AMP-generating systems in brain membranes and slices by the diterpene forskolin: augmentation of receptor-mediated responses.
Topics: Adenylyl Cyclases; Animals; Brain; Cerebral Cortex; Colforsin; Cyclic AMP; Diterpenes; Dose-Response Relationship, Drug; Histamine; Isoproterenol; Male; Neurotransmitter Agents; Norepinephrine; Rats; Vasoactive Intestinal Peptide | 1982 |
Forskolin: a new biochemical tool for studying gastric secretion.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Animals; Antihypertensive Agents; Bufo marinus; Cimetidine; Colforsin; Cyclic AMP; Diterpenes; Gastric Juice; Gastric Mucosa; Histamine; Isoproterenol; Kinetics; Oxygen Consumption; Rabbits; Sodium Fluoride | 1983 |
Forskolin-induced cyclic AMP production and gastric acid secretion in dispersed rabbit parietal cells: novel evidence for a major role of cyclic AMP in acid release.
Topics: Animals; Cells, Cultured; Colforsin; Cyclic AMP; Diterpenes; Dose-Response Relationship, Drug; Drug Synergism; Gastric Acid; Gastric Acidity Determination; Histamine; Parietal Cells, Gastric; Rabbits; Time Factors | 1983 |
Bronchodilating activity of forskolin in vitro and in vivo.
Topics: Acetylcholine; Anaphylaxis; Animals; Bronchodilator Agents; Chlorpheniramine; Colforsin; Diterpenes; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Muscle, Smooth; SRS-A; Trachea | 1984 |
Forskolin action on histamine stimulated adenylyl cyclase in parietal cells of rat and guinea pig.
Topics: Adenylyl Cyclases; Animals; Cimetidine; Colforsin; Diterpenes; Enzyme Activation; Epinephrine; Guinea Pigs; Histamine; Kinetics; Male; Parietal Cells, Gastric; Rats; Rats, Inbred Strains | 1984 |
Invariant relation between total acid secretion and secretagogue exposure: secretory dynamics in bullfrog.
Topics: Animals; Colforsin; Diterpenes; Gastric Juice; Gastric Mucosa; Histamine; In Vitro Techniques; Rana catesbeiana; Secretory Rate | 1984 |
Effect of forskolin on alterations of vascular permeability induced with bradykinin, prostaglandin E1, adenosine, histamine and carrageenin in rats.
Topics: Adenosine; Alprostadil; Animals; Bradykinin; Bromelains; Capillary Permeability; Carrageenan; Colforsin; Diterpenes; Dose-Response Relationship, Drug; Edema; Foot Diseases; Histamine; Indomethacin; Male; Prostaglandins E; Rats; Rats, Inbred Strains; Skin | 1983 |
Histamine-evoked Ca2+ oscillations in HeLa cells are sensitive to methylxanthines but insensitive to ryanodine.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Biological Clocks; Caffeine; Calcium; Colforsin; HeLa Cells; Histamine; Humans; Inositol 1,4,5-Trisphosphate; Inositol Phosphates; Intracellular Fluid; Ruthenium Red; Ryanodine; Theophylline | 1994 |
Calu-3: a human airway epithelial cell line that shows cAMP-dependent Cl- secretion.
Topics: Bradykinin; Bumetanide; Calcimycin; Cell Line; Cell Membrane; Cell Membrane Permeability; Chloride Channels; Chlorides; Colforsin; Cyclic AMP; Cystic Fibrosis Transmembrane Conductance Regulator; Cytoplasmic Granules; Desmosomes; Epithelium; Histamine; Humans; Intercellular Junctions; Isoproterenol; Kinetics; Lung Neoplasms; Membrane Proteins; Methacholine Chloride; Microscopy, Electron; Nystatin; Ouabain; Sodium; Trypsin; Tumor Cells, Cultured | 1994 |
Stimulatory effect of histamine on cyclic AMP formation in chick pineal gland.
Topics: 1-Methyl-3-isobutylxanthine; Adenine; Analysis of Variance; Animals; Carbon Radioisotopes; Chickens; Colforsin; Cyclic AMP; Dimaprit; Guinea Pigs; Hippocampus; Histamine; Histamine Agonists; In Vitro Techniques; Kinetics; Male; Methylhistamines; Pineal Gland; Ranitidine; Rats; Rats, Wistar; Thiazoles; Tritium | 1994 |
Histamine and the cAMP pathway in the guinea-pig pancreas.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Amylases; Animals; Colforsin; Cyclic AMP; Guinea Pigs; Histamine; Pancreas; Vasoactive Intestinal Peptide | 1995 |
VIP inhibits basal and histamine-stimulated proliferation of human airway smooth muscle cells.
Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Carbazoles; Cell Cycle; Cell Division; Cell Line; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; DNA; Dose-Response Relationship, Drug; Glucagon; Histamine; Histamine Antagonists; Humans; Indoles; Kinetics; Muscle, Smooth; Pyrroles; Thymidine; Trachea; Vasoactive Intestinal Peptide | 1995 |
Regulation of the adenylyl cyclase signaling system in various types of cultured endothelial cells.
Topics: 1-Methyl-3-isobutylxanthine; Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Bucladesine; Cattle; Cells, Cultured; Cholera Toxin; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Endothelium, Vascular; GTP-Binding Proteins; Histamine; Humans; Isoproterenol; Phosphoric Diester Hydrolases; Signal Transduction; Swine; Virulence Factors, Bordetella | 1995 |
Myosin light chain kinase phosphorylation in swine carotid artery contraction and relaxation.
Topics: Animals; Calcium; Carotid Artery, Common; Colforsin; Histamine; In Vitro Techniques; Kinetics; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Myosin-Light-Chain Kinase; Myosins; Peptide Mapping; Phosphates; Phosphopeptides; Phosphorus Radioisotopes; Phosphorylation; Potassium Chloride; Swine | 1995 |
Exogenous histamine increases the somatostatin receptor/effector system in the rat frontoparietal cortex.
Topics: Animals; Binding, Competitive; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Frontal Lobe; Histamine; Parietal Lobe; Radioimmunoassay; Rats; Rats, Wistar; Receptors, Somatostatin; Somatostatin | 1995 |
Cyclic adenosine monophosphate stimulates insulin-like growth factor binding protein-4 and its messenger ribonucleic acid in a clonal endothelial cell line.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Blotting, Northern; Bone and Bones; Bucladesine; Carrier Proteins; Cattle; Cell Line; Colforsin; Culture Media, Conditioned; Cyclic AMP; Endothelium; Glycosylation; Histamine; Immunosorbent Techniques; Insulin-Like Growth Factor Binding Protein 4; Kinetics; Parathyroid Glands; RNA, Messenger | 1993 |
Inhibition of acid secretion in gastric parietal cells by the Ca2+/calmodulin-dependent protein kinase II inhibitor KN-93.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Benzylamines; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Cimetidine; Colforsin; Cyclic AMP; Gastric Acid; H(+)-K(+)-Exchanging ATPase; Histamine; Hydrogen-Ion Concentration; In Vitro Techniques; Kinetics; Microscopy, Electron; Parietal Cells, Gastric; Protein Kinase Inhibitors; Rabbits; Sulfonamides | 1993 |
Homologous desensitization of histamine H2 receptors in the human gastric carcinoma cell line MKN-45.
Topics: 1-Methyl-3-isobutylxanthine; Cell Line; Cimetidine; Colforsin; Cyclic AMP; Dinoprostone; Dose-Response Relationship, Drug; Histamine; Histamine H2 Antagonists; Humans; Kinetics; Receptors, Histamine H2; Sodium Fluoride; Stomach Neoplasms; Tumor Cells, Cultured | 1993 |
Non-steroidal anti-inflammatory drugs and prostaglandin effects on pepsinogen secretion by dispersed human peptic cells.
Topics: Acetylcholine; Adolescent; Adult; Anti-Inflammatory Agents, Non-Steroidal; Aspirin; Colforsin; Dinoprostone; Drug Synergism; Female; Gastric Mucosa; Histamine; Humans; Ibuprofen; In Vitro Techniques; Male; Middle Aged; Pepsinogens; Prostaglandin D2; Stimulation, Chemical | 1995 |
cAMP-dependent activation of ion conductances in bronchial epithelial cells.
Topics: Bronchi; Chlorides; Colforsin; Cyclic AMP; Electric Conductivity; Epithelium; Histamine; Humans; Ions; Isoproterenol | 1994 |
Agonist-induced desensitization of histamine H1 receptor-mediated inositol phospholipid hydrolysis in human umbilical vein endothelial cells.
Topics: Alkaloids; Cells, Cultured; Colforsin; Endothelium, Vascular; Histamine; Humans; Hydrolysis; Indoles; Nitroprusside; Phorbol 12,13-Dibutyrate; Phosphatidylinositols; Receptors, Histamine H1; Sodium Fluoride; Staurosporine; Umbilical Veins | 1994 |
Secretion of intrinsic factor from cultured rat gastric chief cells.
Topics: Animals; Blotting, Western; Calcimycin; Calcium; Carbachol; Cells, Cultured; Centrifugation, Density Gradient; Chromatography, Affinity; Colforsin; Cyclic AMP; Electrophoresis, Polyacrylamide Gel; Gastric Mucosa; Histamine; Immunoenzyme Techniques; Immunohistochemistry; Intrinsic Factor; Kidney; Liver; Rabbits; Rats; Sincalide; Spleen; Submandibular Gland; Tetragastrin; Tissue Distribution; Transcobalamins | 1994 |
Histamine increases anti-CD3 induced IL-5 production of TH2-type T cells via histamine H2-receptors.
Topics: Animals; CD3 Complex; Cells, Cultured; Colforsin; Cyclic AMP; Cytokines; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Indicators and Reagents; Interleukin-4; Interleukin-5; Male; Mice; Mice, Inbred Strains; Receptors, Histamine H2; Spleen; T-Lymphocytes, Helper-Inducer | 1994 |
Regulation of histamine- and UTP-induced increases in Ins(1,4,5)P3, Ins (1,3,4,5)P4 and Ca2+ by cyclic AMP in DDT1 MF-2 cells.
Topics: Adenylyl Cyclases; Animals; Calcium; Cell Line; Colforsin; Cricetinae; Cyclic AMP; Histamine; Inositol 1,4,5-Trisphosphate; Inositol Phosphates; Isoproterenol; Male; Mesocricetus; Muscle, Smooth; Receptors, Histamine H1; Receptors, Purinergic P2; Type C Phospholipases; Uridine Triphosphate; Vas Deferens | 1995 |
A1 adenosine receptor inhibition of cyclic AMP formation and radioligand binding in the guinea-pig cerebral cortex.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Binding, Competitive; Cerebral Cortex; Colforsin; Cyclic AMP; Guinea Pigs; Histamine; In Vitro Techniques; Phenylisopropyladenosine; Phosphatidylinositols; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Purines; Radioligand Assay; Receptors, Purinergic P1; Sulfonamides; Vasodilator Agents; Xanthines | 1994 |
Inhibition of T cell adhesion to extracellular matrix glycoproteins by histamine: a role for mast cell degranulation products.
Topics: Animals; Bucladesine; Calcium; CD4-Positive T-Lymphocytes; Cell Adhesion; Cell Adhesion Molecules; Cell Degranulation; Colforsin; Down-Regulation; Extracellular Matrix Proteins; Fibronectins; Histamine; Humans; Integrins; Laminin; Mast Cells; Rats; Rats, Inbred Lew; Receptors, Histamine H2; Second Messenger Systems | 1994 |
Effects of prostaglandins on [Ca2+]i and adenylate cyclase activity in isolated porcine gastric mucous cells.
Topics: Adenylyl Cyclases; Animals; Atropine; Bucladesine; Calcium; Carbachol; Cells, Cultured; Colforsin; Gastric Mucosa; Histamine; Prostaglandins; Proteins; Ranitidine; Swine | 1994 |
Potentiation of nonadrenergic noncholinergic relaxation of human isolated bronchus by selective inhibitors of phosphodiesterase isozymes.
Topics: Atropine; Bronchi; Colforsin; Electric Stimulation; Histamine; Humans; In Vitro Techniques; Indomethacin; Isoenzymes; Molsidomine; Muscle Relaxation; Nitroprusside; Phosphodiesterase Inhibitors; Propranolol; Purinones; Pyrrolidinones; Rolipram | 1994 |
Defective glomerular beta-adrenergic signal transmission in spontaneously diabetic rats.
Topics: Animals; Blood Glucose; Colforsin; Cyclic AMP; Diabetes Mellitus, Type 1; Dinoprostone; Histamine; Isoproterenol; Kidney Glomerulus; Rats; Rats, Inbred BB; Rats, Mutant Strains; Receptors, Adrenergic, beta; Signal Transduction | 1994 |
Modulation by histamine of the delayed outward potassium current in guinea-pig ventricular myocytes.
Topics: Animals; Calcium Channels; Colforsin; Electrophysiology; Guinea Pigs; Heart; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Myocardium; Potassium; Potassium Channels; Protein Kinases; Sodium | 1993 |
Stimulation of rat parietal cell function by histamine and GLP-1-(7-36) amide is mediated by Gs alpha.
Topics: Adenosine Diphosphate; Adenylyl Cyclases; Aminopyrine; Animals; Cell Membrane; Cell Separation; Cells, Cultured; Cholera Toxin; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Electrophoresis, Polyacrylamide Gel; Female; Glucagon; Glucagon-Like Peptide 1; Glucagon-Like Peptides; GTP-Binding Proteins; Histamine; Kinetics; Molecular Weight; Parietal Cells, Gastric; Peptide Fragments; Rats; Rats, Wistar | 1994 |
Nonparallel secretion of pepsinogen and acid by gastric oxyntopeptic cells of the toad (Bufo marinus).
Topics: Animals; Bufo marinus; Carbachol; Cimetidine; Colforsin; Esophagus; Gastric Acid; Gastric Mucosa; Histamine; In Vitro Techniques; Intestinal Mucosa; Kinetics; Microscopy, Electron; Mucous Membrane; Omeprazole; Parietal Cells, Gastric; Pepsin A; Pepsinogens; Time Factors | 1993 |
Leukotriene B4 and C4 production in isolated rat gastric mucosal cells.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Arachidonic Acid; Bucladesine; Calcimycin; Cell Separation; Colforsin; Diglycerides; Female; Gastric Mucosa; Histamine; In Vitro Techniques; Interleukin-1; Interleukin-2; Kinetics; Leukotriene B4; Leukotriene C4; Lipoxygenase Inhibitors; N-Formylmethionine Leucyl-Phenylalanine; Pentagastrin; Phenothiazines; Platelet Activating Factor; Rats; Rats, Wistar; Tetradecanoylphorbol Acetate | 1993 |
Role of myosin light-chain phosphorylation in endothelial cell retraction.
Topics: Aminophylline; Animals; Azepines; Blood Platelets; Cell Membrane Permeability; Cells, Cultured; Colforsin; Cyclic AMP; Egtazic Acid; Electrophoresis, Polyacrylamide Gel; Endothelium, Vascular; Histamine; Humans; Kinetics; Myosin-Light-Chain Kinase; Myosins; Peptide Fragments; Peptide Mapping; Phosphorylation; Pulmonary Artery; Swine; Umbilical Veins | 1993 |
Guinea pig histamine H1 receptor. II. Stable expression in Chinese hamster ovary cells reveals the interaction with three major signal transduction pathways.
Topics: Animals; Arachidonic Acid; Calcium; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Guinea Pigs; HeLa Cells; Histamine; Humans; Hydrolysis; Intracellular Membranes; Osmolar Concentration; Phosphatidylinositols; Receptors, Histamine H1; Signal Transduction | 1994 |
Anti-immunoglobulin E-stimulated ion transport in human large and small intestine.
Topics: Antibodies, Anti-Idiotypic; Cells, Cultured; Colforsin; Cromolyn Sodium; Electric Stimulation; Histamine; Humans; Immunoglobulin E; Intestinal Absorption; Intestinal Mucosa; Intestine, Large; Intestine, Small; Ion Transport; Mast Cells; Piroxicam; Pyrilamine; Receptors, Histamine H1; Tetrodotoxin | 1993 |
Activators of protein kinase C but not of phospholipase C modulate adenylate cyclase-responses of normal pig epidermis.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine; Adenylyl Cyclases; Animals; Bradykinin; Cell Division; Cholera Toxin; Colforsin; Cyclic AMP; Diglycerides; Dinoprostone; Enzyme Activation; Enzyme Inhibitors; Epidermal Cells; Epidermal Growth Factor; Epidermis; Epinephrine; Histamine; Isoquinolines; Keratinocytes; Piperazines; Protein Kinase C; Swine; Tetradecanoylphorbol Acetate; Thrombin; Type C Phospholipases | 1995 |
Endothelin-1 inhibits L-type Ca currents enhanced by isoproterenol in guinea-pig ventricular myocytes.
Topics: Animals; Calcium Channel Blockers; Calcium Channels; Colforsin; Cyclic AMP; Endothelins; Guinea Pigs; Heart Ventricles; Histamine; Isoproterenol; Membrane Potentials; Myocardium; Receptors, Endothelin | 1996 |
Involvement of the M2 muscarinic receptor in contractions of the guinea pig trachea, guinea pig esophagus, and rat fundus.
Topics: Adrenergic beta-Agonists; Animals; Colforsin; Cyclic AMP; Esophagus; Gastric Fundus; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Oxotremorine; Pertussis Toxin; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Serotonin; Trachea; Virulence Factors, Bordetella | 1996 |
Two distinct pathways for histamine H2 receptor down-regulation. H2 Leu124 --> Ala receptor mutant provides evidence for a cAMP-independent action of H2 agonists.
Topics: 1-Methyl-3-isobutylxanthine; Amino Acid Sequence; Animals; Base Sequence; CHO Cells; Cholera Toxin; Colforsin; Cricetinae; Cyclic AMP; DNA Primers; Dose-Response Relationship, Drug; Down-Regulation; Gene Expression; Guanidines; Histamine; Histamine Agonists; Histamine H2 Antagonists; Iodine Radioisotopes; Kinetics; Molecular Sequence Data; Mutagenesis, Site-Directed; Point Mutation; Polymerase Chain Reaction; Protein Structure, Secondary; Radioligand Assay; Rats; Receptors, Histamine H2; Recombinant Proteins; RNA, Messenger; Transfection | 1996 |
Desensitization of muscarinic receptor-coupled inositol phospholipid hydrolysis in human detrusor cultured smooth cells.
Topics: Carbachol; Cells, Cultured; Colforsin; Histamine; Humans; Inositol Phosphates; Muscarinic Agonists; Muscle, Smooth; Nitroprusside; Receptors, Muscarinic; Sodium Fluoride; Urinary Bladder | 1996 |
Histamine inhibits tumor necrosis factor alpha release by mast cells through H2 and H3 receptors.
Topics: Animals; Antibody Specificity; Colforsin; Cyclic AMP; Cyclooxygenase Inhibitors; Cytotoxins; Dinoprostone; Dose-Response Relationship, Drug; Histamine; Macrophages, Peritoneal; Male; Mast Cells; Rats; Rats, Sprague-Dawley; Receptors, Histamine H2; Receptors, Histamine H3; Sensitivity and Specificity; Time Factors; Tumor Necrosis Factor-alpha | 1996 |
Calcium mobilization and isometric tension in bovine tracheal smooth muscle: effects of salbutamol and histamine.
Topics: Albuterol; Aniline Compounds; Animals; Bronchodilator Agents; Calcium; Cattle; Colforsin; Electrophysiology; Fluorescent Dyes; Histamine; Isometric Contraction; Male; Muscle Relaxation; Muscle, Smooth; Sodium; Trachea; Xanthenes | 1996 |
Human astrocytoma U138MG cells express predominantly type-A endothelin receptor.
Topics: Astrocytoma; Base Sequence; Binding, Competitive; Cell Membrane; Colforsin; Cyclic AMP; DNA Primers; Endocytosis; Endothelin Receptor Antagonists; Endothelins; Guanylyl Imidodiphosphate; Histamine; Humans; Isoproterenol; Ligands; Molecular Sequence Data; Phosphatidylinositols; Polymerase Chain Reaction; Protein Binding; Pyrimidines; Receptor, Endothelin A; Receptors, Endothelin; RNA, Messenger; Sulfonamides; Tumor Cells, Cultured | 1996 |
Histamine receptors in neoplastic transformation: studies in human cell lines.
Topics: Analysis of Variance; Binding Sites; Cell Transformation, Neoplastic; Cholera Toxin; Colforsin; Cyclic AMP; Dinoprostone; Histamine; Histamine Agonists; Humans; Lethal Dose 50; Oxytocics; Phosphatidylinositols; Receptors, Histamine H1; Receptors, Histamine H2; Signal Transduction; Tumor Cells, Cultured; Type C Phospholipases | 1996 |
Hippocampal somatostatin receptors and modulation of adenylyl cyclase activity in histamine-treated rats.
Topics: Adenylyl Cyclases; Animals; Cerebral Ventricles; Cimetidine; Colforsin; Dose-Response Relationship, Drug; Guanylyl Imidodiphosphate; Hippocampus; Histamine; Injections, Intraperitoneal; Injections, Intraventricular; Kinetics; Pyrilamine; Rats; Rats, Wistar; Receptors, Somatostatin; Somatostatin; Time Factors | 1996 |
Possible participation of histamine H3 receptors in the modulation of noradrenaline release from rat spinal cord slices.
Topics: Animals; Colforsin; Desipramine; Dose-Response Relationship, Drug; Female; Histamine; Male; Norepinephrine; Phentolamine; Radioligand Assay; Rats; Rats, Wistar; Receptors, Histamine H3; Spinal Cord | 1995 |
Modulation of agonist-induced phosphoinositide metabolism, Ca2+ signalling and contraction of airway smooth muscle by cyclic AMP-dependent mechanisms.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic beta-Agonists; Animals; Calcium; Cattle; Cells, Cultured; Cholinergic Agents; Colforsin; Cyclic AMP; Histamine; Isoproterenol; Methacholine Chloride; Muscle Contraction; Muscle, Smooth; Phosphatidylinositols; Signal Transduction; Trachea | 1996 |
Pharmacological activation changes stiffness of cultured human airway smooth muscle cells.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Acetylcholine; Actins; Bradykinin; Bronchodilator Agents; Bucladesine; Carbachol; Cells, Cultured; Colforsin; Collagen; Cytoskeleton; Dinoprostone; Histamine; Humans; Isoproterenol; Kinetics; Magnetics; Muscarinic Agonists; Muscle Contraction; Muscle, Smooth; Myosins; Potassium Chloride; Substance P; Time Factors; Trachea | 1996 |
Interaction between the two signal transduction systems of the histamine H2 receptor: desensitizing and sensitizing effects of histamine stimulation on histamine-dependent cAMP production in Chinese hamster ovary cells.
Topics: Animals; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Dogs; Histamine; Histamine Agonists; Indoles; Maleimides; Receptors, Histamine H2; Recombinant Proteins; Signal Transduction; Tetradecanoylphorbol Acetate | 1996 |
Zatebradine inhibits tachycardia induced by bronchodilators without affecting respiratory resistance in dogs.
Topics: Airway Resistance; Aminophylline; Animals; Benzazepines; Bronchodilator Agents; Cardiotonic Agents; Colforsin; Cyclic AMP; Dogs; Female; Heart Rate; Histamine; Isoproterenol; Male; Procaterol; Tachycardia | 1997 |
Suppression of cAMP formation by adenosine in myenteric ganglia from guinea-pig small intestine.
Topics: Adenosine; Adenosine Deaminase; Animals; Colforsin; Cyclic AMP; Drug Antagonism; Ganglia; Guinea Pigs; Histamine; Intestine, Small; Male; Myenteric Plexus; Purinergic P1 Receptor Agonists; Serotonin; Signal Transduction; Stimulation, Chemical; Substance P | 1997 |
Histamine does not potentiate cyclic AMP-mediated amylase secretion in the guinea-pig pancreatic acinar cells.
Topics: Amylases; Animals; Colforsin; Cyclic AMP; Female; Guinea Pigs; Histamine; In Vitro Techniques; Male; Pancreas; Vasoactive Intestinal Peptide | 1997 |
Involvement of protein kinase C in homologous desensitization of histamine-evoked secretory responses in rat chromaffin cells.
Topics: Animals; Calcium; Carcinogens; Catecholamines; Chromaffin Cells; Colforsin; Cyclic AMP-Dependent Protein Kinases; Cyclic GMP; Cytoplasmic Granules; Desensitization, Immunologic; Enzyme Inhibitors; GTP-Binding Proteins; Histamine; Indoles; Male; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Rats, Wistar; Receptors, Histamine H1; Stimulation, Chemical | 1997 |
Effect of Rp diastereoisomer of adenosine 3',5' cyclic-monophosphothioate on the cAMP-dependent relaxation of smooth muscle.
Topics: Animals; Colforsin; Cyclic AMP; Drug Interactions; Enzyme Inhibitors; Female; Histamine; Muscle Relaxation; Papaverine; Phosphodiesterase Inhibitors; Potassium Chloride; Pyrrolidinones; Rats; Rats, Wistar; Rolipram; Stereoisomerism; Thionucleotides; Uterine Contraction; Uterus; Vanadates; Vinca Alkaloids | 1997 |
Contractile roles of the M2 and M3 muscarinic receptors in the guinea pig colon.
Topics: Animals; Colforsin; Colon; Cyclic AMP; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Oxotremorine; Pertussis Toxin; Piperidines; Pirenzepine; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Virulence Factors, Bordetella | 1998 |
Activation of the human histamine H2 receptor is linked to cell proliferation and c-fos gene transcription.
Topics: Cell Division; Cell Line; Cimetidine; Cloning, Molecular; Colforsin; Cyclic AMP; Enzyme Activation; Epidermal Growth Factor; Epinephrine; Genes, fos; Genes, Reporter; Histamine; Humans; Inositol 1,4,5-Trisphosphate; Kinetics; Luciferases; Promoter Regions, Genetic; Protein Kinase C; Proto-Oncogene Proteins c-fos; Receptors, Histamine H2; Recombinant Fusion Proteins; Signal Transduction; Staurosporine; Tetradecanoylphorbol Acetate; Transcription, Genetic; Transfection | 1997 |
Mast cell mediated ion transport in intestine from patients with and without inflammatory bowel disease.
Topics: Animals; Antibodies, Anti-Idiotypic; Colforsin; Colitis, Ulcerative; Crohn Disease; Histamine; Histamine H1 Antagonists; Humans; Immunoglobulin E; In Vitro Techniques; Intestinal Mucosa; Ion Transport; Mast Cells; Pyrilamine; Rabbits | 1997 |
Dual effects of histamine and substance P on intracellular calcium levels in human U373 MG astrocytoma cells: role of protein kinase C.
Topics: Animals; Astrocytoma; Brain Neoplasms; Calcium; Cerebellum; Colforsin; Cyclic AMP; Enzyme Inhibitors; Fluorescent Dyes; Fura-2; Guinea Pigs; HeLa Cells; Histamine; Humans; Inositol Phosphates; Protein Kinase C; Pyrilamine; Substance P; Thapsigargin; Tritium; Tumor Cells, Cultured | 1998 |
Relaxant effects of NKH477, a new water-soluble forskolin derivative, on guinea-pig tracheal smooth muscle: the role of Ca2+-activated K+ channels.
Topics: Animals; Bronchodilator Agents; Calcium; Colforsin; Cyclic AMP; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nifedipine; Peptides; Potassium; Potassium Channels; Solubility; Trachea; Water | 1998 |
Indomethacin enhances endothelial NO release--evidence for a role of PGI2 in the autocrine control of calcium-dependent autacoid production.
Topics: Autocrine Communication; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic GMP; Cyclooxygenase Inhibitors; Endothelium, Vascular; Epoprostenol; Feedback; Histamine; Humans; Indomethacin; Nitric Oxide; Umbilical Veins | 1997 |
Interleukin 1 beta and tumour necrosis factor alpha inhibit acid secretion in cultured rabbit parietal cells by multiple pathways.
Topics: Animals; Benzoquinones; Calcimycin; Carbachol; Cells, Cultured; Colforsin; Depression, Chemical; Dose-Response Relationship, Drug; Enzyme Inhibitors; Gastric Acid; Gastrins; Histamine; Interleukin-1; Ionophores; Lactams, Macrocyclic; Nicotinic Agonists; Parietal Cells, Gastric; Pertussis Toxin; Protein-Tyrosine Kinases; Quinones; Rabbits; Rifabutin; Tumor Necrosis Factor-alpha; Virulence Factors, Bordetella | 1998 |
M2 muscarinic receptors inhibit forskolin- but not isoproterenol-mediated relaxation in bovine tracheal smooth muscle.
Topics: Animals; Cattle; Colforsin; Cyclic AMP; Diphenylacetic Acids; Histamine; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Oxotremorine; Piperidines; Receptor, Muscarinic M2; Receptors, Muscarinic; Trachea | 1998 |
Protein kinase A inhibitors reverse histamine-mediated regulation of IL-5 secretion.
Topics: Animals; Bucladesine; Cell Line; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Histamine; Histamine Release; Interleukin-5; Isoquinolines; Mice; T-Lymphocytes, Helper-Inducer; Thionucleotides | 1998 |
Forskolin induces U937 cell line differentiation as a result of a sustained cAMP elevation.
Topics: Antigens, Neoplasm; Cell Differentiation; Cell Division; Cell Line; Chemotaxis; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Genes, myc; Histamine; Humans; Oxidation-Reduction; Tumor Cells, Cultured | 1998 |
Cl- transport in an immortalized human epithelial cell line (NCM460) derived from the normal transverse colon.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Alprostadil; Bacterial Toxins; Biological Transport; Cell Line, Transformed; Chlorides; Colforsin; Colon; Cyclic AMP; Cyclic GMP; Cystic Fibrosis Transmembrane Conductance Regulator; Enterotoxins; Escherichia coli; Escherichia coli Proteins; Fluorescent Dyes; Histamine; Humans; Intestinal Mucosa; Models, Biological; Phorbol 12,13-Dibutyrate; Reproducibility of Results; Reverse Transcriptase Polymerase Chain Reaction; Transcription, Genetic | 1998 |
A synergistic interaction between histamine and vasoactive intestinal peptide (VIP) on cyclic AMP production in the chick pineal gland.
Topics: Amino Acid Sequence; Animals; Chickens; Colforsin; Cyclic AMP; Drug Synergism; Histamine; Isoproterenol; Molecular Sequence Data; Pineal Gland; Retina; Vasoactive Intestinal Peptide | 1998 |
Diazepam potentiates the positive inotropic effects of histamine and forskolin in guinea-pig papillary muscles.
Topics: Anesthetics, Intravenous; Animals; Colforsin; Cyclic AMP; Diazepam; Drug Interactions; Guinea Pigs; Histamine; Myocardial Contraction; Papillary Muscles; Stimulation, Chemical | 1998 |
Different acid secretagogues activate different Na+/H+ exchanger isoforms in rabbit parietal cells.
Topics: Aminopyrine; Animals; Biological Transport; Carbachol; Cells, Cultured; Colforsin; Cytochalasin D; Gastric Acid; Guanidines; Histamine; Imidazoles; Kinetics; Omeprazole; Parietal Cells, Gastric; Rabbits; Sodium-Hydrogen Exchangers; Sulfones; Time Factors | 1998 |
Muscarinic M2 receptor-mediated contraction in the guinea pig Taenia caeci: possible involvement of protein kinase C.
Topics: Animals; Cecum; Colforsin; Diphenylacetic Acids; Female; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Kinetics; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Parasympathomimetics; Piperidines; Pirenzepine; Protein Kinase C; Receptor, Muscarinic M2; Receptors, Muscarinic; Second Messenger Systems | 1998 |
Comparison of functional antagonism between isoproterenol and M2 muscarinic receptors in guinea pig ileum and trachea.
Topics: Animals; Colforsin; Diphenylacetic Acids; Guinea Pigs; Histamine; Ileum; Isoproterenol; Muscle Relaxation; Oxotremorine; Pertussis Toxin; Piperidines; Pirenzepine; Receptor, Muscarinic M2; Receptors, Muscarinic; Trachea; Virulence Factors, Bordetella | 1999 |
Different reactions of aortic and venular endothelial cell monolayers to histamine on macromolecular permeability: role of cAMP, cytosolic Ca2+ and F-actin.
Topics: Actins; Animals; Aorta; Calcium; Capillary Permeability; Cattle; Cells, Cultured; Colforsin; Cyclic AMP; Endothelium, Vascular; Histamine; Humans; Intracellular Membranes; Ionomycin; Ionophores; Macromolecular Substances; Osmolar Concentration; Venules | 1999 |
Pertussis toxin increases isoproterenol induced relaxation in field-stimulated ileum.
Topics: Animals; Colforsin; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Histamine; Histamine Agonists; Ileum; In Vitro Techniques; Isoproterenol; Male; Muscarinic Agonists; Muscle Contraction; Muscle Relaxation; Oxotremorine; Pertussis Toxin; Sympathomimetics; Virulence Factors, Bordetella | 1999 |
Inflammatory and contractile agents sensitize specific adenylyl cyclase isoforms in human airway smooth muscle.
Topics: Adenylyl Cyclases; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Cells, Cultured; Cholinergic Agonists; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Free Radical Scavengers; GTP-Binding Protein alpha Subunits, Gs; Histamine; Humans; Isoenzymes; Muscle, Smooth; Receptors, Adrenergic, beta-2; Respiratory System; Signal Transduction; Vasoconstrictor Agents | 1999 |
Regulated von Willebrand factor secretion is associated with agonist-specific patterns of cytoskeletal remodeling in cultured endothelial cells.
Topics: Actins; Adenosine; ADP Ribose Transferases; Biological Transport; Botulinum Toxins; Calcimycin; Calcium; Cell Size; Cells, Cultured; Colchicine; Colforsin; Cyclic AMP; Cytochalasin B; Cytochalasin D; Cytoplasmic Granules; Endothelium, Vascular; Epinephrine; GTPase-Activating Proteins; Histamine; Humans; Ionophores; Microtubules; Myosins; Nucleic Acid Synthesis Inhibitors; Sympathomimetics; Thrombin; Umbilical Veins; Vasodilator Agents; von Willebrand Factor | 2000 |
Histamine H(3) receptors mediate inhibition of noradrenaline release from intestinal sympathetic nerves.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 4-Aminopyridine; Adrenergic alpha-Antagonists; Animals; Calcium; Colforsin; Dose-Response Relationship, Drug; Ethylmaleimide; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Ileum; In Vitro Techniques; Intestinal Mucosa; Intestines; Male; Muscle, Smooth; Myenteric Plexus; Nifedipine; Norepinephrine; omega-Conotoxins; Pertussis Toxin; Phenols; Receptors, Histamine H3; Rolipram; Sympathetic Nervous System; Tetradecanoylphorbol Acetate; Tetraethylammonium; Tetrodotoxin; Virulence Factors, Bordetella; Yohimbine | 2000 |
A primary culture of guinea pig gallbladder epithelial cells that is responsive to secretagogues.
Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Adenosine Triphosphate; Animals; Anions; Biological Transport; Calcium; Calcium Channel Blockers; Cells, Cultured; Cholecystokinin; Colforsin; Cyclic AMP; Dinoprostone; Epithelial Cells; Gallbladder; Gastrointestinal Agents; Guinea Pigs; Histamine; Ionomycin; Ionophores; Male; ortho-Aminobenzoates; Secretin; Vasoactive Intestinal Peptide | 2000 |
Requirement of additional adenylate cyclase activation for the inhibition of human eosinophil degranulation by phosphodiesterase IV inhibitors.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenylyl Cyclases; Adult; Albuterol; Benzamides; Cell Degranulation; Colforsin; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Cyclohexanecarboxylic Acids; Dinoprostone; Dose-Response Relationship, Drug; Enzyme Activation; Eosinophil Peroxidase; Eosinophils; Histamine; Humans; Nitriles; Peroxidases; Phosphodiesterase Inhibitors; Pyridines; Rolipram; Superoxides; Theophylline | 2001 |
Histamine treatment induces rearrangements of orthogonal arrays of particles (OAPs) in human AQP4-expressing gastric cells.
Topics: Animals; Aquaporin 4; Aquaporins; Cell Line; Colforsin; Dimerization; Epithelial Cells; Freeze Fracturing; Histamine; Humans; Microscopy, Electron; Osmosis; Particle Size; Rats; Stomach; Transfection | 2001 |
Relaxation and modulation of cyclic AMP production in response to atrial natriuretic peptides in guinea pig tracheal smooth muscle.
Topics: Adenylyl Cyclases; Animals; Apamin; Atrial Natriuretic Factor; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Glyburide; Guanylate Cyclase; Guinea Pigs; Histamine; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Natriuretic Peptide, C-Type; Nitroprusside; Oxadiazoles; Peptide Fragments; Peptides; Phosphodiesterase Inhibitors; Potassium Channel Blockers; Quinoxalines; Rolipram; Trachea | 2001 |
Histamine increases the expression of LOX-1 via H2 receptor in human monocytic THP-1 cells.
Topics: Bucladesine; Cell Differentiation; Colforsin; CREB-Binding Protein; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cytokines; Dinoprostone; Enzyme Inhibitors; Gene Expression Regulation; Histamine; Humans; Isoquinolines; Macrophages; Monocytes; Nuclear Proteins; Promoter Regions, Genetic; Prostaglandin D2; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, LDL; Receptors, Oxidized LDL; RNA, Messenger; Scavenger Receptors, Class E; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Trans-Activators; Tumor Cells, Cultured; Up-Regulation | 2001 |
Simultaneous measurement and imaging of intracellular Ca(2+) and H(+) transport in isolated rabbit gastric glands.
Topics: Animals; Biological Transport; Calcium; Carbachol; Colforsin; Gastric Acid; Histamine; Hydrogen; In Vitro Techniques; Intracellular Membranes; Osmolar Concentration; Oxazoles; Parietal Cells, Gastric; Rabbits | 2001 |
Presynaptic H3 autoreceptors modulate histamine synthesis through cAMP pathway.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Brain; Bucladesine; Colforsin; Cyclic AMP; Drug Interactions; Histamine; Imidazoles; In Vitro Techniques; Male; Piperidines; Potassium; Rats; Rats, Sprague-Dawley; Receptors, Histamine H3; Thionucleotides; Thiourea | 2002 |
Sensitization to mechanical stimulation by inflammatory mediators and by mild burn in canine visceral nociceptors in vitro.
Topics: Animals; Bradykinin; Burns; Colforsin; Dinoprostone; Dogs; Histamine; Hot Temperature; Inflammation Mediators; Nociceptors; Phorbol 12,13-Dibutyrate; Physical Stimulation; Protons; Viscera | 2002 |
Inhibition of human primary melanoma cell proliferation by histamine is enhanced by interleukin-6.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Bucladesine; Cell Division; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Gene Expression; Guanidines; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Imidazoles; Interleukin-6; Isoquinolines; Melanoma; Polymerase Chain Reaction; Receptors, Interleukin-6; Skin Neoplasms; Sulfonamides; Tumor Cells, Cultured | 2002 |
Chlorpromazine inhibits the glucocorticoid receptor-mediated gene transcription in a calcium-dependent manner.
Topics: Animals; Antipsychotic Agents; Calcimycin; Calcium; Calcium Channel Blockers; Cell Line; Cell Line, Transformed; Chloramphenicol O-Acetyltransferase; Chlorpromazine; Clozapine; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Estrenes; Fibroblasts; Gene Expression Regulation; Genes, Reporter; Haloperidol; Histamine; Histamine H1 Antagonists; Ionophores; Mammary Tumor Virus, Mouse; Mice; Nifedipine; Phorbol Esters; Phosphodiesterase Inhibitors; Protein Kinase C; Protein Kinase C-alpha; Pyrilamine; Pyrrolidinones; Raclopride; Receptors, Glucocorticoid; Remoxipride; Sulfonamides; Sulpiride; Tetradecanoylphorbol Acetate; Thionucleotides; Transcription, Genetic; Type C Phospholipases | 2002 |
Differential activation of dual signaling responses by human H1 and H2 histamine receptors.
Topics: Calcium Signaling; Cell Line; Colforsin; Cyclic AMP; Dimaprit; Histamine; Histamine Agonists; Humans; Kinetics; Receptors, Histamine H1; Receptors, Histamine H2; Recombinant Proteins; Signal Transduction; Transfection | 2003 |
Crucial role of histamine for regulation of gastric acid secretion ascertained by histidine decarboxylase-knockout mice.
Topics: Animals; Carbachol; Colforsin; Female; Gastric Acid; Gastrins; Histamine; Histidine Decarboxylase; Hydrogen-Ion Concentration; Male; Mice; Mice, Inbred ICR; Mice, Knockout; Theophylline | 2003 |
Effects of ouabain on human bronchial muscle in vitro.
Topics: Acetylcholine; Bronchi; Calcium; Calcium Channel Blockers; Colforsin; Cromakalim; Histamine; Humans; In Vitro Techniques; Inositol Phosphates; Isoproterenol; Membrane Potentials; Muscle Relaxation; Muscle, Smooth; Nitroprusside; Ouabain; Protein Kinase C; Sodium Potassium Chloride Symporter Inhibitors; Sodium-Hydrogen Exchangers; Sodium-Potassium-Exchanging ATPase; Time Factors; Vasoconstrictor Agents; Vasodilator Agents | 2003 |
Differential regulation of the slow and rapid components of guinea-pig cardiac delayed rectifier K+ channels by hypoxia.
Topics: Animals; Cardiotonic Agents; Colforsin; Delayed Rectifier Potassium Channels; Guinea Pigs; Histamine; Hypoxia; Isoproterenol; Myocardium; Oxidation-Reduction; Potassium Channels; Potassium Channels, Voltage-Gated; Protein Kinase C; Protein Kinase C beta; Sulfhydryl Compounds; Time Factors | 2004 |
Effect of carvedilol on Ca2+ movement and cytotoxicity in human MG63 osteosarcoma cells.
Topics: Adenylyl Cyclases; Calcium; Calcium Channels; Calcium Signaling; Carbazoles; Carvedilol; Cell Compartmentation; Cell Line, Tumor; Cell Proliferation; Cell Survival; Colforsin; Dose-Response Relationship, Drug; Endoplasmic Reticulum; Estrenes; Fluorescence; Fura-2; Histamine; Histamine Antagonists; Humans; Inositol 1,4,5-Trisphosphate; Manganese; Osteosarcoma; Phorbol Esters; Propanolamines; Protein Kinase C; Pyrrolidinones; Tetrazolium Salts; Thapsigargin; Time Factors; Type C Phospholipases | 2004 |
Potentiation of beta-adrenoceptor function in bovine tracheal smooth muscle by inhibition of protein kinase C.
Topics: Adrenergic beta-Agonists; Animals; Cattle; Colforsin; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Histamine; In Vitro Techniques; Indoles; Isoproterenol; Maleimides; Methacholine Chloride; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Protein Kinase C; Receptors, Adrenergic, beta; Trachea | 2005 |
Effect of chronic exposure to cold on isoprenaline-induced cAMP accumulation and relaxation in the rat aorta.
Topics: Acclimatization; Animals; Aorta; Blood Pressure; Bucladesine; Cold Temperature; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Histamine; Isoproterenol; Male; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Vasodilation | 2006 |
Characterization of a novel chemokine-containing storage granule in endothelial cells: evidence for preferential exocytosis mediated by protein kinase A and diacylglycerol.
Topics: Cells, Cultured; Chemokine CCL2; Chemokine CXCL1; Chemokines; Chemokines, CXC; Colforsin; Cyclic AMP-Dependent Protein Kinases; Cytoplasmic Granules; Diglycerides; Dose-Response Relationship, Immunologic; Endothelium, Vascular; Exocytosis; Histamine; Humans; Intercellular Signaling Peptides and Proteins; Protein Kinase C; rab GTP-Binding Proteins; rab27 GTP-Binding Proteins | 2005 |
Characteristics of the renal C-type natriuretic peptide receptor in hypertrophied and developing rat kidney.
Topics: Animals; Atrial Natriuretic Factor; Binding Sites; Binding, Competitive; Colforsin; Cyclic AMP; Histamine; Hypertrophy; Kidney; Kidney Glomerulus; Kinetics; Male; Natriuretic Peptide, C-Type; Nephrectomy; Peptide Fragments; Rats; Rats, Inbred WKY; Receptors, Atrial Natriuretic Factor; Serotonin | 2005 |
Compared pharmacology of human histamine H3 and H4 receptors: structure-activity relationships of histamine derivatives.
Topics: Binding, Competitive; Colforsin; Cyclic AMP; DNA, Complementary; Histamine; Histamine H2 Antagonists; Humans; Imidazoles; In Vitro Techniques; Kidney; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H3; Receptors, Histamine H4; Recombinant Proteins; Structure-Activity Relationship; Transfection | 2006 |
Ex vivo biochemical analysis of CFTR in human rectal biopsies.
Topics: Adolescent; Adult; Biopsy; Carbachol; Child; Child, Preschool; Colforsin; Cysteine; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Electrophysiology; Histamine; Humans; Immunoprecipitation; In Vitro Techniques; Intestinal Mucosa; Isotope Labeling; Middle Aged; Rectum; Sulfur Radioisotopes | 2006 |
Homologous down-regulation of histamine H3 receptors in rat striatal slices.
Topics: Animals; Arsenicals; Binding, Competitive; Colforsin; Corpus Striatum; Cyclic AMP; Down-Regulation; Endocytosis; Enzyme Inhibitors; Histamine; Histamine Agonists; Imidazoles; Male; Organ Culture Techniques; Piperidines; Radioligand Assay; Rats; Rats, Wistar; Receptor Aggregation; Receptors, Histamine H3 | 2006 |
Trafficking and phosphorylation dynamics of AQP4 in histamine-treated human gastric cells.
Topics: Animals; Aquaporin 4; Cell Membrane; Colforsin; Cyclic AMP-Dependent Protein Kinases; Endocytosis; Endosomes; Exocytosis; Histamine; Humans; Parietal Cells, Gastric; Phosphorylation; Protein Transport; Rats; Transfection; Vesicular stomatitis Indiana virus | 2007 |
Longer muscle lengths recapitulate force suppression in swine carotid artery.
Topics: Analysis of Variance; Animals; Carotid Artery, Common; Colforsin; Dose-Response Relationship, Drug; Histamine; HSP20 Heat-Shock Proteins; In Vitro Techniques; Muscle, Smooth, Vascular; Myosin-Light-Chain Kinase; Phosphorylation; Potassium Chloride; Swine; Vasoconstriction; Vasoconstrictor Agents; Vasodilation; Vasodilator Agents | 2007 |
Cyclic AMP signaling contributes to neural plasticity and hyperexcitability in AH sensory neurons following intestinal Trichinella spiralis-induced inflammation.
Topics: Animals; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Dideoxyadenosine; Dinoprostone; Guinea Pigs; Histamine; Imidazoles; In Vitro Techniques; Intestinal Mucosa; Leukotriene B4; Lysine; Male; Membrane Potentials; Muscle, Smooth; Neuronal Plasticity; Neurons, Afferent; Nitric Oxide; Peroxidase; Signal Transduction; Substance P; Thiobarbituric Acid Reactive Substances; Trichinella spiralis; Trichinellosis; Tryptases | 2007 |
Force suppression and the crossbridge cycle in swine carotid artery.
Topics: Actin Cytoskeleton; Actins; Animals; Biomechanical Phenomena; Bridged Bicyclo Compounds, Heterocyclic; Carotid Artery, Common; Colforsin; Histamine; Histamine Agents; HSP20 Heat-Shock Proteins; In Vitro Techniques; Muscle, Smooth, Vascular; Phosphorylation; Swine; Thiazolidines; Vasoconstriction | 2007 |
Ligation of Toll-like receptor 3 differentially regulates M2 and M3 muscarinic receptor expression and function in human airway smooth muscle cells.
Topics: 2-Aminopurine; Bronchial Hyperreactivity; Calcium Signaling; Cells, Cultured; Chloroquine; Colforsin; Cyclic AMP; eIF-2 Kinase; Gene Expression Regulation; Histamine; Humans; Leukotriene D4; Membrane Proteins; Muscarinic Antagonists; Myocytes, Smooth Muscle; Poly I-C; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Histamine H1; Receptors, Leukotriene; Signal Transduction; Toll-Like Receptor 3 | 2008 |
Prostaglandin E2 sensitizes primary sensory neurons to histamine.
Topics: Animals; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Dinoprostone; Dose-Response Relationship, Drug; Drug Interactions; Ganglia, Spinal; Histamine; Histamine Agonists; Inositol 1,4,5-Trisphosphate; Isoquinolines; Models, Biological; Neurons, Afferent; Protein Kinase Inhibitors; Rats; Rats, Sprague-Dawley; Rats, Wistar; Sulfonamides; Time Factors | 2007 |
PDE4 and PDE5 regulate cyclic nucleotides relaxing effects in human umbilical arteries.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Colforsin; Cyclic AMP; Cyclic GMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Cyclic Nucleotide Phosphodiesterases, Type 5; Dipyridamole; Female; Guanylate Cyclase; Histamine; Humans; In Vitro Techniques; Isoenzymes; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Naphthyridines; Nitroprusside; Phosphodiesterase 4 Inhibitors; Phosphodiesterase 5 Inhibitors; Pyrimidines; Reverse Transcriptase Polymerase Chain Reaction; Rolipram; Serotonin; Umbilical Arteries; Vasodilator Agents | 2008 |
Cytopathology and exocrine dysfunction induced in ex vivo rabbit lacrimal gland acinar cell models by chronic exposure to histamine or serotonin.
Topics: Actins; Animals; beta-N-Acetylhexosaminidases; Calcium; Carbachol; Cells, Cultured; Cholinergic Agonists; Colforsin; Cytosol; Dose-Response Relationship, Drug; Dynactin Complex; Epithelial Cells; Female; Fluorescent Antibody Technique, Indirect; Histamine; Lacrimal Apparatus; Lacrimal Apparatus Diseases; Microscopy, Confocal; Microtubule-Associated Proteins; Rabbits; Serotonin | 2009 |
Strain-dependent differences in electrogenic secretion of electrolytes across mouse colon epithelium.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Barium; Bumetanide; Carbachol; Colforsin; Colon; Cyclic AMP; Electrolytes; Feces; Histamine; Histamine Antagonists; Intestinal Mucosa; Large-Conductance Calcium-Activated Potassium Channel alpha Subunits; Mice; Mice, Inbred C57BL; Mice, Inbred Strains; Muscarinic Antagonists; Potassium; Receptors, Histamine H1; Receptors, Muscarinic; Sodium-Potassium-Chloride Symporters; Solute Carrier Family 12, Member 2; Water | 2010 |
Chronic regulation of colonic epithelial secretory function by activation of G protein-coupled receptors.
Topics: Adenocarcinoma; Calcium; Carbachol; Cell Line, Tumor; Chlorides; Colforsin; Colonic Neoplasms; Epithelial Cells; Histamine; Humans; Patch-Clamp Techniques; Protein Kinase C; Receptor, Muscarinic M3; Receptors, G-Protein-Coupled; Thapsigargin | 2011 |
The role of rectal chloride secretion in childhood constipation.
Topics: 1-Methyl-3-isobutylxanthine; Amiloride; Biopsy; Carbachol; Child; Chlorides; Cholinergic Agonists; Colforsin; Constipation; Cystic Fibrosis Transmembrane Conductance Regulator; Defecation; Female; Hirschsprung Disease; Histamine; Histamine Agonists; Humans; Male; Phosphodiesterase Inhibitors; Rectum; Sodium Channel Blockers | 2011 |
The role of extracellular-signal regulate kinase (ERK) in the regulation of airway tone in porcine isolated peripheral bronchioles.
Topics: Animals; Bronchioles; Carbachol; Colforsin; Cyclooxygenase Inhibitors; Endothelin-1; Extracellular Signal-Regulated MAP Kinases; Histamine; In Vitro Techniques; Mitogen-Activated Protein Kinase Kinases; Muscle Relaxation; Muscle, Smooth; Potassium Channels; Prostaglandin-Endoperoxide Synthases; Protein Kinase C; Receptors, Adrenergic, beta; Swine | 2012 |
The histamine autoreceptor is a short isoform of the H₃ receptor.
Topics: Animals; Arachidonic Acid; Autoreceptors; Brain; Calcimycin; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Guanosine 5'-O-(3-Thiotriphosphate); Histamine; Imidazoles; In Vitro Techniques; Male; Methylhistamines; Protein Isoforms; Rats; Rats, Wistar; Receptors, Histamine H3 | 2012 |
Adapter-modified Ussing chamber enables evaluation of endoscopically-obtained colonic biopsy samples from cats and dogs.
Topics: Animals; Biopsy; Cat Diseases; Cats; Colforsin; Colonic Diseases; Colonoscopy; Dog Diseases; Dogs; Electric Conductivity; Female; Glucose; Histamine; Male; Phlorhizin; Serotonin; Specimen Handling | 2012 |
Role of cyclic nucleotide-dependent actin cytoskeletal dynamics:Ca(2+)](i) and force suppression in forskolin-pretreated porcine coronary arteries.
Topics: Actin Cytoskeleton; Actin Depolymerizing Factors; Actins; Animals; Biomechanical Phenomena; Calcium; Cell Adhesion Molecules; Colforsin; Coronary Vessels; Histamine; HSP20 Heat-Shock Proteins; Intracellular Space; Microfilament Proteins; Muscle Contraction; Myosin Light Chains; Nucleotides, Cyclic; Paxillin; Phosphoproteins; Phosphorylation; Sus scrofa | 2013 |
Reporter cell lines for detection of pertussis toxin in acellular pertussis vaccines as a functional animal-free alternative to the in vivo histamine sensitization test.
Topics: Animals; Biological Assay; Cell Line; CHO Cells; Colforsin; Cricetulus; Cyclic AMP; Founder Effect; Genes, Reporter; Histamine; Humans; Luciferases; Luminescent Measurements; Myocytes, Smooth Muscle; Pertussis Toxin; Pertussis Vaccine; Rats; Response Elements; Sensitivity and Specificity; Vaccines, Acellular | 2017 |