Compounds > histamine

histamine and 6,7-dichloro 3-(4-methylpiperazin-1-yl)quinoxalin-2(1h)-one

histamine has been researched along with 6,7-dichloro 3-(4-methylpiperazin-1-yl)quinoxalin-2(1h)-one in 3 studies

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (66.67)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Adami, M; Coruzzi, G; de Esch, IJ; Guaita, E; Hanzer, A; Leurs, R; Lim, HD; Smits, RA; Zuiderveld, OP1
Adami, M; Broeker, J; Coruzzi, G; de Esch, IJ; Guaita, E; Haaksma, E; Leurs, R; Sansuk, K; Smits, RA; Zuiderveld, OP1
Bessembinder, K; de Esch, IJ; Kuhne, S; Leurs, R; Lim, HD; Smits, RA; van der Meer, T; Wijtmans, M; Zuiderveld, OP1

Other Studies

3 other study(ies) available for histamine and 6,7-dichloro 3-(4-methylpiperazin-1-yl)quinoxalin-2(1h)-one

ArticleYear
Fragment based design of new H4 receptor-ligands with anti-inflammatory properties in vivo.
    Journal of medicinal chemistry, 2008, Apr-24, Volume: 51, Issue:8

    Topics: Anti-Inflammatory Agents; Drug Design; Humans; Ligands; Magnetic Resonance Spectroscopy; Models, Molecular; Receptors, Histamine; Spectrometry, Mass, Electrospray Ionization; Structure-Activity Relationship

2008
Discovery of quinazolines as histamine H4 receptor inverse agonists using a scaffold hopping approach.
    Journal of medicinal chemistry, 2008, Dec-25, Volume: 51, Issue:24

    Topics: Animals; Anti-Inflammatory Agents; Chemistry, Pharmaceutical; Drug Design; Histamine Agonists; Humans; Hydrogen-Ion Concentration; Inhibitory Concentration 50; Kinetics; Models, Chemical; Models, Molecular; Molecular Conformation; Quinazolines; Rats; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4

2008
Ligand based design of novel histamine Hâ‚„ receptor antagonists; fragment optimization and analysis of binding kinetics.
    Bioorganic & medicinal chemistry letters, 2012, Jan-01, Volume: 22, Issue:1

    Topics: Animals; Biological Availability; Chemistry, Pharmaceutical; Drug Design; Histamine Antagonists; Humans; Hypersensitivity; Inhibitory Concentration 50; Kinetics; Ligands; Mice; Models, Chemical; Models, Molecular; Molecular Conformation; Rats; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Structure-Activity Relationship; Time Factors

2012