hexahydrosiladifenidol and piperidines

hexahydrosiladifenidol has been researched along with piperidines in 58 studies

Research

Studies (58)

TimeframeStudies, this research(%)All Research%
pre-199014 (24.14)18.7374
1990's41 (70.69)18.2507
2000's3 (5.17)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Sastry, BV; Stephan, CC1
Aguilar, JS; Ballesta, JJ; Criado, M; Palmero, M; Reig, JA; Viniegra, S1
Kajimura, M; Reuben, MA; Sachs, G1
Bloom, JW; Halonen, M; Mahesh, VK; Nunan, LM; Palmer, JD; Yamamura, HI1
Fernandes, LB; Fryer, AD; Hirshman, CA1
Anderson, DJ; Connolly, T; McKinney, M; Miller, JH; Vella-Rountree, L1
Bagetta, G; Constanti, A1
Bindslev, N; Winding, B1
Daniel, EE; Janssen, LJ1
Jaiswal, N; Lambrecht, G; Malik, KU; Mutschler, E; Tacke, R1
Birdsall, NJ; Eveleigh, P; Hulme, EC; Pedder, EK; Poyner, D1
Jaiswal, N; Malik, KU1
Benedito, S; García-Sacristán, A; Hernández, M; Prieto, D; Rivera, L1
Richards, MH1
Yang, CM1
Baron, E; Boer, R; Eltze, M; Kromer, W1
Aasen, AJ; Feifel, R; Lambrecht, G; Mutschler, E; Rodrigues de Miranda, JF; Strohmann, C; Tacke, R1
Massi, M; Melchiorre, C; Perfumi, M; Polidori, C; Pompei, PL1
Camus, J; Christophe, J; Lambrecht, G; Mutschler, E; Strohmann, C; Tacke, R; Tastenoy, M; Waelbroeck, M1
Elzinga, CR; Roffel, AF; Zaagsma, J1
Lambrecht, G; Mutschler, E; Rettenmayr, NM; Rijntjes, NV; Rodrigues de Miranda, JF; Russel, FG; Strohmann, C; Tacke, R; van Ginneken, CA1
Hanack, C; Herawi, M; Kopp, R; Lambrecht, G; Moser, U; Mutschler, E; Pfeiffer, A; Tacke, R1
Lambrecht, G; Moser, U; Mutschler, E; Noelke, B; Pfeiffer, A; Rochlitz, H; Tacke, R1
Jackson, KN; Kachur, JF; Lowe, VC; Noronha-Blob, L; Sturm, BL1
Anderson, D; el-Fakahany, EE; Forray, C; McKinney, M1
Amrhein, CL; el-Fakahany, EE; Forray, C; Surichamorn, W1
Boddeke, H; Christophe, J; Feifel, R; Lambrecht, G; Mutschler, E; Strohmann, C; Tacke, R; Waelbroeck, M; Wagner-Röder, M; Zilch, H1
Fuder, H; Lambrecht, G; Melchiorre, C; Mutschler, E; Schöpf, J; Tacke, R; Unckell, J; Wesner, MT1
Camus, J; Choo, LK; Feifel, R; Lambrecht, G; Moser, U; Strohmann, C; Tacke, R; Tastenoy, M; Waelbroeck, M; Wagner-Röder, M1
Barnes, PJ; Mak, JC1
Camus, J; Christophe, J; Lambrecht, G; Linoh, H; Mutschler, E; Strohmann, C; Tacke, R; Tastenoy, M; Waelbroeck, M; Zilch, H1
Camus, J; Christophe, J; Waelbroeck, M; Winand, J1
Jaiswal, N; Lambrecht, G; Malik, KU; Mutschler, E1
Giraldo, E; Hammer, R; Ladinsky, H; Viganò, MA1
Akiba, I; Bujo, H; Kubo, T; Maeda, A; Mishina, M; Nakai, J; Numa, S1
Nilvebrant, L; Sparf, B1
Bali, JP; Baudiere, B; Giraldo, E; Ladinsky, H; Monferini, E1
Fuder, H; Kilbinger, H; Müller, H1
Mitchelson, F; Shen, A1
Elzinga, CR; Meurs, H; Roffel, AF; Zaagsma, J1
Dietrich, C; Kilbinger, H1
Boselli, C; Grana, E1
Peers, C; Reeve, HL; Vaughan, PF1
Classen, M; Schaffer, K; Schepp, W; Schusdziarra, V; Wegner, U; Weigert, N1
Robinson, NE; Wang, ZW; Yu, MF1
Gillman, TA; Mitchelson, F; Pennefather, JN1
Deirmengiant, C; Maslanski, JA; Patelt, J; Powelt, R1
Davenport, TA; Fukumoto, Y; Gousse, A; Kamai, T; Latifpour, J; Weiss, RM; Yoshida, M1
Garland, CJ; Hillier, K; Kerr, PM; Wallis, RM1
de la Vega, MT; Montano, JA; Nunez, A1
Bilezikian, JP; Huber, F; Robinson, RB; Steinberg, SF; Sun, LS; Vulliemoz, Y1
Levin, RJ; Przyborski, SA1
Hoover, DB; Neely, DA1
Baba, H; Goldstein, PA; Kohno, T; Okamoto, M; Shimoji, K; Yoshimura, M1
Chasserot-Golaz, S; Galzi, JL; Goeldner, M; Ilien, B; Weill, C1
Lau, WA; Mitchelson, FJ; Pennefather, JN1
Ishida, H; Ishikawa, Y; Skowronski, MT1
Aita, T; Ishihata, A; Katano, Y; Tezuka, A1

Reviews

2 review(s) available for hexahydrosiladifenidol and piperidines

ArticleYear
Pharmacology and second messenger interactions of cloned muscarinic receptors.
    Biochemical pharmacology, 1991, Oct-09, Volume: 42, Issue:9

    Topics: Animals; Atropine; Carbachol; Cell Line; Humans; Oxotremorine; Piperidines; Pirenzepine; Receptors, Muscarinic; Recombinant Proteins; Second Messenger Systems; Transfection

1991
Pharmacology of hexahydro-difenidol, hexahydro-sila-difenidol and related selective muscarinic antagonists.
    Trends in pharmacological sciences, 1989, Volume: Suppl

    Topics: Animals; Humans; Parasympatholytics; Piperidines

1989

Other Studies

56 other study(ies) available for hexahydrosiladifenidol and piperidines

ArticleYear
Characterization of the subtype of muscarinic receptor coupled to the stimulation of phosphoinositide hydrolysis in 132-1N1 human astrocytoma cells.
    Cellular and molecular biology (Noisy-le-Grand, France), 1992, Volume: 38, Issue:7

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Astrocytoma; Atropine; Carbachol; Diamines; Humans; Hydrolysis; Parasympathomimetics; Phosphatidylinositols; Piperidines; Pirenzepine; Receptors, Muscarinic; Scopolamine; Tumor Cells, Cultured

1992
Muscarinic receptor subtypes in bovine adrenal medulla.
    Neurochemical research, 1992, Volume: 17, Issue:12

    Topics: Adrenal Medulla; Animals; Atropine; Binding Sites; Binding, Competitive; Cattle; Cell Membrane; Dicyclomine; Muscarine; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Muscarinic

1992
The muscarinic receptor gene expressed in rabbit parietal cells is the m3 subtype.
    Gastroenterology, 1992, Volume: 103, Issue:3

    Topics: Animals; Atropine; Base Sequence; Blotting, Southern; Molecular Sequence Data; N-Methylscopolamine; Parietal Cells, Gastric; Piperidines; Pirenzepine; Polymerase Chain Reaction; Rabbits; Receptors, Muscarinic; RNA, Messenger; Scopolamine Derivatives

1992
A minority of muscarinic receptors mediate rabbit tracheal smooth muscle contraction.
    American journal of respiratory cell and molecular biology, 1992, Volume: 6, Issue:3

    Topics: Animals; Atropine; Female; Male; Methacholine Chloride; Muscle Contraction; Muscle, Smooth; Myocardium; Parasympatholytics; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Rabbits; Radioligand Assay; Receptors, Muscarinic; Trachea

1992
M2 muscarinic receptors inhibit isoproterenol-induced relaxation of canine airway smooth muscle.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:1

    Topics: Animals; Dogs; Drug Interactions; Isoproterenol; Methacholine Chloride; Muscle Relaxation; Muscle, Smooth; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Trachea

1992
Pharmacological profiles for rat cortical M1 and M2 muscarinic receptors using selective antagonists: comparison with N1E-115 muscarinic receptors.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 257, Issue:3

    Topics: Animals; Cerebral Cortex; Cyclic AMP; Diamines; In Vitro Techniques; Muscarinic Antagonists; Parasympatholytics; Phenethylamines; Phosphatidylinositols; Piperidines; Pirenzepine; Rats; Receptors, Muscarinic; Tumor Cells, Cultured

1991
Muscarinic inhibition of excitatory neurotransmission in guinea-pig olfactory cortex slices: weak antagonism by M3-muscarinic receptor antagonists.
    European journal of pharmacology, 1991, May-30, Volume: 198, Issue:1

    Topics: Action Potentials; Animals; Carbachol; Cerebral Cortex; Evoked Potentials; Guinea Pigs; In Vitro Techniques; Olfactory Bulb; Parasympatholytics; Piperidines; Receptors, Muscarinic; Synaptic Transmission

1991
Characterization of a muscarinic receptor controlling Cl- secretion in hen trachea.
    The American journal of physiology, 1990, Volume: 258, Issue:6 Pt 1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Animals; Atropine; Bethanechol; Bethanechol Compounds; Bumetanide; Calcium Channels; Chickens; Chlorides; Dicyclomine; Female; In Vitro Techniques; Ion Channels; Kinetics; Mucous Membrane; Muscle, Smooth; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Trachea

1990
Pre- and postjunctional muscarinic receptors in canine bronchi.
    The American journal of physiology, 1990, Volume: 259, Issue:4 Pt 1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Bethanechol Compounds; Bronchi; Carbachol; Dogs; Electric Stimulation; In Vitro Techniques; Membrane Potentials; Microelectrodes; Muscle Contraction; Muscle, Smooth; Oxotremorine; Piperidines; Pirenzepine; Receptors, Muscarinic

1990
Pharmacological characterization of the vascular muscarinic receptors mediating relaxation and contraction in rabbit aorta.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 258, Issue:3

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Animals; Antihypertensive Agents; Aorta, Abdominal; Arecoline; Atropine; Diamines; Endothelium, Vascular; Hexamethonium; Hexamethonium Compounds; Indomethacin; Male; Muscarinic Antagonists; Muscle Contraction; Muscle Relaxation; Norepinephrine; Parasympatholytics; Piperidines; Pirenzepine; Rabbits; Receptors, Muscarinic

1991
Modulation of the structure-binding relationships of antagonists for muscarinic acetylcholine receptor subtypes.
    British journal of pharmacology, 1991, Volume: 103, Issue:2

    Topics: Animals; Centrifugation; Cerebral Cortex; Cholic Acids; Digitonin; Gallamine Triethiodide; Heart; In Vitro Techniques; Lacrimal Apparatus; Membranes; Muscarinic Antagonists; Myocardium; Parasympatholytics; Piperidines; Pirenzepine; Rats; Structure-Activity Relationship

1991
Methoctramine, a cardioselective antagonist: muscarinic receptor mediating prostaglandin synthesis in isolated rabbit heart.
    European journal of pharmacology, 1991, Jan-03, Volume: 192, Issue:1

    Topics: 6-Ketoprostaglandin F1 alpha; Acetylcholine; Animals; Arachidonic Acid; Arachidonic Acids; Arecoline; Coronary Circulation; Diamines; Heart; Heart Rate; In Vitro Techniques; Isoproterenol; Male; Myocardium; Parasympatholytics; Piperidines; Prostaglandins; Rabbits; Receptors, Muscarinic

1991
Distribution and function of cholinergic receptors in the sheep detrusor muscle.
    Journal of the autonomic nervous system, 1991, Jun-15, Volume: 34, Issue:2-3

    Topics: Acetylcholine; Acetylcholinesterase; Animals; Atropine; Carbachol; Cholinesterase Inhibitors; Ganglia, Parasympathetic; Male; Muscle Contraction; Muscle, Smooth; Nerve Tissue Proteins; Piperidines; Pirenzepine; Receptors, Muscarinic; Sheep; Tetraisopropylpyrophosphamide; Urinary Bladder

1991
Characterization of muscarinic receptors in dog tracheal smooth muscle cells.
    Journal of autonomic pharmacology, 1991, Volume: 11, Issue:1

    Topics: Animals; Atropine; Carbachol; Diamines; Dogs; In Vitro Techniques; Kinetics; Muscle, Smooth; N-Methylscopolamine; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Scopolamine Derivatives; Trachea

1991
Telenzepine inhibits electrically-stimulated, acetylcholine plus histamine-mediated acid secretion in the mouse isolated stomach by blockade of M1 muscarine receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 343, Issue:1

    Topics: Acetylcholine; Alkaloids; Animals; Anti-Ulcer Agents; Electric Stimulation; Furans; Gastric Acid; Gastric Mucosa; Histamine; Mice; Muscarinic Antagonists; Naphthalenes; p-Methoxy-N-methylphenethylamine; Parasympatholytics; Piperidines; Pirenzepine; Stomach; Thiazepines; Vagus Nerve

1991
Selective labelling of muscarinic M1 receptors in calf superior cervical ganglia by [3H](+/-)-telenzepine.
    European journal of pharmacology, 1991, Mar-19, Volume: 195, Issue:1

    Topics: Animals; Binding, Competitive; Cattle; Ganglia; Half-Life; In Vitro Techniques; Male; Neck; Piperidines; Pirenzepine; Rabbits; Radioligand Assay; Receptors, Muscarinic; Tritium; Vas Deferens

1991
Natriuresis, kaliuresis and antidiuresis induced by central carbachol injection are mediated by muscarinic M1 receptors.
    European journal of pharmacology, 1991, Mar-19, Volume: 195, Issue:1

    Topics: Animals; Carbachol; Diamines; Diuresis; Dose-Response Relationship, Drug; Injections, Intraventricular; Male; Muscarinic Antagonists; Natriuresis; Piperidines; Potassium; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1991
Binding affinities of hexahydro-difenidol and hexahydro-sila-difenidol analogues at four muscarinic receptor subtypes: constitutional and stereochemical aspects.
    European journal of pharmacology, 1991, Feb-25, Volume: 206, Issue:2

    Topics: Animals; Binding, Competitive; Brain; Humans; In Vitro Techniques; Kinetics; Myocardium; Pancreas; Piperidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Stereoisomerism; Structure-Activity Relationship; Tumor Cells, Cultured

1991
Muscarinic M3 receptors mediate contraction of human central and peripheral airway smooth muscle.
    Pulmonary pharmacology, 1990, Volume: 3, Issue:1

    Topics: Bronchi; Humans; In Vitro Techniques; Ipratropium; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Trachea

1990
Pharmacokinetic properties of the antimuscarinic drug [3H]-hexahydro-sila-difenidol in the rat.
    Naunyn-Schmiedeberg's archives of pharmacology, 1990, Volume: 342, Issue:2

    Topics: Administration, Oral; Anesthesia; Animals; Autoradiography; Bile; Injections, Intravenous; Male; Parasympatholytics; Piperidines; Rats; Rats, Inbred Strains; Tissue Distribution

1990
Human gastric mucosa expresses glandular M3 subtype of muscarinic receptors.
    Digestive diseases and sciences, 1990, Volume: 35, Issue:12

    Topics: Carbachol; Gastric Mucosa; Humans; In Vitro Techniques; N-Methylscopolamine; Parasympatholytics; Piperazines; Piperidines; Pirenzepine; Receptors, Muscarinic; Scopolamine Derivatives

1990
Muscarinic receptors mediating acid secretion in isolated rat gastric parietal cells are of M3 type.
    Gastroenterology, 1990, Volume: 98, Issue:1

    Topics: Animals; Gastric Acid; Parasympatholytics; Parietal Cells, Gastric; Piperazines; Piperidines; Radioligand Assay; Rats; Receptors, Muscarinic

1990
In vitro and in vivo antimuscarinic effects of (-)cis 2,3-dihydro-3-(4-methylpiperazinylmethyl)-2-phenyl-1,5 benzothiazepin-4-(5H)one HCl (BTM-1086) in guinea pig peripheral tissues.
    Life sciences, 1990, Volume: 46, Issue:17

    Topics: Animals; Atropine; Calcium; Female; Guinea Pigs; Heart Atria; Ileum; In Vitro Techniques; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Neurons; Parasympatholytics; Piperidines; Pirenzepine; Structure-Activity Relationship; Thiazepines; Tumor Cells, Cultured; Urinary Bladder; Vas Deferens

1990
Characterization of the striatal M2 muscarinic receptor mediating inhibition of cyclic AMP using selective antagonists: a comparison with the brainstem M2 receptor.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:2

    Topics: Animals; Brain Stem; Corpus Striatum; Cyclic AMP; Diamines; Parasympatholytics; Piperidines; Pirenzepine; Rats; Receptors, Muscarinic

1989
Inhibition of cyclic AMP formation in N1E-115 neuroblastoma cells is mediated by a non-cardiac M2 muscarinic receptor subtype.
    Brain research, 1989, Jul-31, Volume: 493, Issue:2

    Topics: Animals; Binding, Competitive; Cyclic AMP; Mice; Muscarinic Antagonists; N-Methylscopolamine; Neuroblastoma; Piperidines; Receptors, Muscarinic; Scopolamine Derivatives; Tumor Cells, Cultured

1989
Affinity profiles of hexahydro-sila-difenidol analogues at muscarinic receptor subtypes.
    European journal of pharmacology, 1989, Sep-01, Volume: 168, Issue:1

    Topics: Animals; Diamines; Female; Ganglia, Sympathetic; Guinea Pigs; Heart; Ileum; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Piperidines; Pirenzepine; Rabbits; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Vas Deferens

1989
Different muscarine receptors mediate the prejunctional inhibition of [3H]-noradrenaline release in rat or guinea-pig iris and the contraction of the rabbit iris sphincter muscle.
    Naunyn-Schmiedeberg's archives of pharmacology, 1989, Volume: 340, Issue:6

    Topics: Animals; Electric Stimulation; In Vitro Techniques; Iris; Kinetics; Methacholine Compounds; Muscle Contraction; Muscle, Smooth; Norepinephrine; Piperidines; Rabbits; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1989
Muscarinic receptor subtypes in human and guinea pig lung.
    European journal of pharmacology, 1989, May-19, Volume: 164, Issue:2

    Topics: Adamantane; Adult; Aged; Animals; Atropine; Guinea Pigs; Humans; In Vitro Techniques; Lung; Middle Aged; Parasympatholytics; Piperidines; Pirenzepine; Protease Inhibitors; Quinuclidinyl Benzilate; Receptors, Muscarinic; Species Specificity

1989
Binding and functional properties of antimuscarinics of the hexocyclium/sila-hexocyclium and hexahydro-diphenidol/hexahydro-sila-diphenidol type to muscarinic receptor subtypes.
    British journal of pharmacology, 1989, Volume: 98, Issue:1

    Topics: Animals; Cells, Cultured; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Male; Muscle, Smooth; Myocardium; Pancreas; Parasympatholytics; Piperazines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Stereoisomerism; Structure-Activity Relationship

1989
Different antagonist binding properties of rat pancreatic and cardiac muscarinic receptors.
    Life sciences, 1987, Nov-09, Volume: 41, Issue:19

    Topics: Animals; Binding, Competitive; GTP-Binding Proteins; Kinetics; Male; Myocardium; N-Methylscopolamine; Pancreas; Parasympatholytics; Piperidines; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives; Type C Phospholipases

1987
Contribution of M2 alpha and M2 beta muscarinic receptors to the action of cholinergic stimuli on prostaglandin synthesis and mechanical function in the isolated rabbit heart.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 247, Issue:1

    Topics: Acetylcholine; Animals; Arecoline; Dose-Response Relationship, Drug; Heart; In Vitro Techniques; Male; Parasympatholytics; Parasympathomimetics; Piperidines; Pirenzepine; Prostaglandins; Rabbits; Receptors, Muscarinic

1988
Characterization of muscarinic receptors in guinea pig ileum longitudinal smooth muscle.
    Molecular pharmacology, 1988, Volume: 33, Issue:6

    Topics: Animals; Binding, Competitive; Guinea Pigs; Ileum; In Vitro Techniques; Kinetics; Male; Muscle, Smooth; Myocardium; N-Methylscopolamine; Parasympatholytics; Phenoxybenzamine; Piperidines; Pirenzepine; Receptors, Muscarinic; Salivary Glands; Scopolamine Derivatives

1988
Primary structure of porcine muscarinic acetylcholine receptor III and antagonist binding studies.
    FEBS letters, 1988, Aug-01, Volume: 235, Issue:1-2

    Topics: Amino Acid Sequence; Animals; Base Sequence; DNA, Recombinant; Glycosylation; Molecular Sequence Data; Muscarine; Oocytes; Piperidines; Pirenzepine; Protein Conformation; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; RNA, Messenger; Sequence Homology, Nucleic Acid; Swine; Xenopus laevis

1988
Receptor binding profiles of some selective muscarinic antagonists.
    European journal of pharmacology, 1988, Jun-22, Volume: 151, Issue:1

    Topics: Animals; Cerebral Cortex; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle, Smooth; Myocardial Contraction; Parasympatholytics; Parotid Gland; Piperidines; Pirenzepine; Procyclidine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Urinary Bladder

1988
Characterization of the muscarinic receptor subtype in isolated gastric fundic cells of the rabbit.
    Biochemical pharmacology, 1987, Sep-15, Volume: 36, Issue:18

    Topics: Aminopyrine; Animals; Atropine; Carbachol; Gastric Fundus; Kinetics; Male; N-Methylscopolamine; Piperidines; Pirenzepine; Rabbits; Receptors, Muscarinic; Scopolamine Derivatives

1987
Organ selectivity of hexahydrosiladifenidol in blocking pre- and postjunctional muscarinic receptors studied in guinea-pig ileum and rat heart.
    European journal of pharmacology, 1985, Jul-11, Volume: 113, Issue:1

    Topics: Acetylcholine; Animals; Guinea Pigs; Heart; Ileum; In Vitro Techniques; Male; Muscle Contraction; Norepinephrine; Organ Specificity; Parasympatholytics; Piperidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1985
Characterization of the muscarine receptor subtype on sympathetic nerve endings in the rat caudal artery.
    European journal of pharmacology, 1994, Feb-03, Volume: 252, Issue:2

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Arteries; Atropine; Bis-Trimethylammonium Compounds; Carbachol; Female; In Vitro Techniques; Isoindoles; Male; Muscarinic Antagonists; Muscle, Smooth, Vascular; Nerve Endings; Parasympatholytics; Piperidines; Rats; Rats, Wistar; Receptors, Muscarinic; Sympathetic Nervous System; Tail; Trihexyphenidyl

1994
No evidence for a role of muscarinic M2 receptors in functional antagonism in bovine trachea.
    British journal of pharmacology, 1995, Volume: 115, Issue:4

    Topics: Animals; Bronchoconstrictor Agents; Cattle; Dose-Response Relationship, Drug; Gallamine Triethiodide; Histamine; In Vitro Techniques; Isoproterenol; Methacholine Chloride; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nicotinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Adrenergic, beta; Receptors, Muscarinic; Trachea

1995
Prejunctional M1 and postjunctional M3 muscarinic receptors in the circular muscle of the guinea-pig ileum.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 351, Issue:3

    Topics: Acetylcholine; Animals; Choline; Female; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Neuromuscular Junction; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic

1995
Mode of antagonism of methoctramine, AF-DX 116 and hexahydrosiladifenidol in guinea-pig left atrium and ileum: comparison of Schild and resultant analysis.
    Journal of autonomic pharmacology, 1995, Volume: 15, Issue:2

    Topics: Animals; Diamines; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Myocardial Contraction; Parasympatholytics; Piperidines; Pirenzepine

1995
Inhibition of N-type Ca2+ channel currents in human neuroblastoma (SH-SY5Y) cells by muscarine via stimulation of M3 receptors.
    Neuropharmacology, 1995, Volume: 34, Issue:3

    Topics: Brain Neoplasms; Calcium Channel Blockers; GTP-Binding Proteins; Humans; Muscarine; Muscarinic Agonists; Neuroblastoma; Parasympatholytics; Patch-Clamp Techniques; Pertussis Toxin; Piperidines; Receptors, Muscarinic; Tumor Cells, Cultured; Virulence Factors, Bordetella

1995
Functional characterization of a muscarinic receptor stimulating gastrin release from rabbit antral G-cells in primary culture.
    European journal of pharmacology, 1994, Nov-03, Volume: 264, Issue:3

    Topics: Animals; Arecoline; Atropine; Benzodiazepinones; Carbachol; Cell Adhesion; Cell Separation; Cells, Cultured; Gastrins; Immunohistochemistry; Male; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Pyloric Antrum; Rabbits; Receptors, Muscarinic

1994
Prejunctional muscarinic autoreceptors on horse airway cholinergic nerves.
    Life sciences, 1995, Volume: 56, Issue:25

    Topics: Acetylcholine; Animals; Atropine; Cholinergic Fibers; Electric Stimulation; Horses; In Vitro Techniques; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Trachea

1995
Muscarinic receptors in rat uterus.
    European journal of pharmacology, 1994, Sep-12, Volume: 262, Issue:3

    Topics: Alkaloids; Animals; Atropine; Binding, Competitive; Computer Simulation; Female; Furans; In Vitro Techniques; Ligands; Muscarinic Antagonists; Naphthalenes; Parasympatholytics; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Uterus

1994
Assessment of the muscarinic receptor subtypes involved in pilocarpine-induced seizures in mice.
    Neuroscience letters, 1994, Feb-28, Volume: 168, Issue:1-2

    Topics: Animals; Atropine; Cerebral Ventricles; Injections, Intraventricular; Male; Mice; Parasympatholytics; Pilocarpine; Piperidines; Pirenzepine; Receptors, Muscarinic; Seizures

1994
Diabetes-induced alterations in the properties of muscarinic cholinergic receptors in rat vas deferens.
    The Journal of urology, 1994, Volume: 152, Issue:3

    Topics: Animals; Atropine; Binding, Competitive; Diabetes Mellitus, Experimental; Diamines; Insulin; Male; Parasympatholytics; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Up-Regulation; Vas Deferens

1994
Characterization of muscarinic receptors mediating contractions of circular and longitudinal muscle of human isolated colon.
    British journal of pharmacology, 1995, Volume: 115, Issue:8

    Topics: Alkaloids; Atropine; Carbachol; Carcinoma; Colon; Colonic Neoplasms; Dose-Response Relationship, Drug; Furans; Humans; In Vitro Techniques; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Naphthalenes; Piperidines; Pirenzepine

1995
Carbachol stimulates inositol phosphate formation in rat thalamus slices through muscarinic M3-receptor activation.
    Neuroscience letters, 1996, Jul-26, Volume: 213, Issue:1

    Topics: Animals; Binding, Competitive; Carbachol; Dose-Response Relationship, Drug; Inositol Phosphates; Male; Muscarinic Agonists; Muscarinic Antagonists; Organ Culture Techniques; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic; Thalamus; Tritium

1996
Muscarinic receptor heterogeneity in neonatal rat ventricular myocytes in culture.
    Journal of cardiovascular pharmacology, 1996, Volume: 27, Issue:4

    Topics: Animals; Animals, Newborn; Carbachol; Cells, Cultured; Cyclic AMP; GTP-Binding Proteins; Heart Rate; Inositol Phosphates; Muscarinic Agonists; Muscarinic Antagonists; Myocardium; Pertussis Toxin; Piperidines; Rats; Receptor, Muscarinic M2; Receptors, Muscarinic; Signal Transduction; Stimulation, Chemical; Virulence Factors, Bordetella

1996
Cholinergic modulation of electrogenic ion transport in different regions of the rat small intestine.
    The Journal of pharmacy and pharmacology, 1997, Volume: 49, Issue:7

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Analysis of Variance; Animals; Atropine; Bethanechol; Carbachol; Chlorides; Diamines; Duodenum; Ileum; Intestinal Mucosa; Ion Transport; Jejunum; Male; Muscarinic Agonists; Muscarinic Antagonists; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptor, Muscarinic M3; Receptors, Muscarinic; Structure-Activity Relationship; Tetrodotoxin

1997
Differentiation of muscarinic receptors mediating negative chronotropic and vasoconstrictor responses to acetylcholine in isolated rat hearts.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 282, Issue:3

    Topics: Acetylcholine; Animals; Atropine; Coronary Vessels; Depression, Chemical; Diamines; Heart Rate; In Vitro Techniques; Male; Pertussis Toxin; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Vasoconstriction; Virulence Factors, Bordetella

1997
Muscarinic facilitation of GABA release in substantia gelatinosa of the rat spinal dorsal horn.
    The Journal of physiology, 1998, Apr-01, Volume: 508 ( Pt 1)

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Atropine; Carbachol; Diamines; Evoked Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Interneurons; Muscarinic Agonists; Neostigmine; Neurons; Parasympatholytics; Piperidines; Pirenzepine; Rats; Receptor, Muscarinic M1; Receptors, Muscarinic; Substantia Gelatinosa; Synaptic Transmission; Tetrodotoxin

1998
Functional characterization and potential applications for enhanced green fluorescent protein- and epitope-fused human M1 muscarinic receptors.
    Journal of neurochemistry, 1999, Volume: 73, Issue:2

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Atropine; Binding, Competitive; Calcium; Cells, Cultured; DNA Primers; Epitopes; Flow Cytometry; Gene Expression; Green Fluorescent Proteins; Histidine; Humans; Indicators and Reagents; Kidney; Luminescent Proteins; Microscopy, Confocal; Muscarinic Antagonists; Mutagenesis, Site-Directed; Piperidines; Pirenzepine; Radioligand Assay; Receptor, Muscarinic M1; Receptors, Muscarinic; Recombinant Fusion Proteins; Tritium

1999
Cholinergic facilitation of neurotransmission to the smooth muscle of the guinea-pig prostate gland.
    British journal of pharmacology, 2000, Volume: 130, Issue:5

    Topics: Acetylcholine; Animals; Carbachol; Cholinergic Agonists; Electric Stimulation; Guinea Pigs; Male; Muscle Contraction; Muscle, Smooth; Piperidines; Prostate; Receptor, Muscarinic M1; Receptors, Muscarinic; Synaptic Transmission

2000
Persistent increase in the amount of aquaporin-5 in the apical plasma membrane of rat parotid acinar cells induced by a muscarinic agonist SNI-2011.
    FEBS letters, 2000, Jul-21, Volume: 477, Issue:3

    Topics: Animals; Aquaporin 5; Aquaporins; Atropine; Calcium; Cell Membrane; Cells, Cultured; Inositol 1,4,5-Trisphosphate; Male; Membrane Proteins; Muscarinic Agonists; Parotid Gland; Piperidines; Quinuclidines; Rats; Rats, Wistar; Thiophenes

2000
Aging-related alterations in the contractile responses to acetylcholine, muscarinic cholinoceptors and cholinesterase activities in jejunum and colon of the male Fischer 344 rats.
    Experimental gerontology, 2004, Volume: 39, Issue:1

    Topics: Acetylcholine; Aging; Animals; Atropine; Cholinesterases; Colon; Diamines; Dose-Response Relationship, Drug; Gastrointestinal Motility; In Vitro Techniques; Intestine, Large; Jejunum; Male; Muscarinic Antagonists; Muscle, Smooth; Piperidines; Pirenzepine; Rats; Rats, Inbred F344

2004