hexahydrosiladifenidol has been researched along with piperidines in 58 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 14 (24.14) | 18.7374 |
1990's | 41 (70.69) | 18.2507 |
2000's | 3 (5.17) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Sastry, BV; Stephan, CC | 1 |
Aguilar, JS; Ballesta, JJ; Criado, M; Palmero, M; Reig, JA; Viniegra, S | 1 |
Kajimura, M; Reuben, MA; Sachs, G | 1 |
Bloom, JW; Halonen, M; Mahesh, VK; Nunan, LM; Palmer, JD; Yamamura, HI | 1 |
Fernandes, LB; Fryer, AD; Hirshman, CA | 1 |
Anderson, DJ; Connolly, T; McKinney, M; Miller, JH; Vella-Rountree, L | 1 |
Bagetta, G; Constanti, A | 1 |
Bindslev, N; Winding, B | 1 |
Daniel, EE; Janssen, LJ | 1 |
Jaiswal, N; Lambrecht, G; Malik, KU; Mutschler, E; Tacke, R | 1 |
Birdsall, NJ; Eveleigh, P; Hulme, EC; Pedder, EK; Poyner, D | 1 |
Jaiswal, N; Malik, KU | 1 |
Benedito, S; García-Sacristán, A; Hernández, M; Prieto, D; Rivera, L | 1 |
Richards, MH | 1 |
Yang, CM | 1 |
Baron, E; Boer, R; Eltze, M; Kromer, W | 1 |
Aasen, AJ; Feifel, R; Lambrecht, G; Mutschler, E; Rodrigues de Miranda, JF; Strohmann, C; Tacke, R | 1 |
Massi, M; Melchiorre, C; Perfumi, M; Polidori, C; Pompei, PL | 1 |
Camus, J; Christophe, J; Lambrecht, G; Mutschler, E; Strohmann, C; Tacke, R; Tastenoy, M; Waelbroeck, M | 1 |
Elzinga, CR; Roffel, AF; Zaagsma, J | 1 |
Lambrecht, G; Mutschler, E; Rettenmayr, NM; Rijntjes, NV; Rodrigues de Miranda, JF; Russel, FG; Strohmann, C; Tacke, R; van Ginneken, CA | 1 |
Hanack, C; Herawi, M; Kopp, R; Lambrecht, G; Moser, U; Mutschler, E; Pfeiffer, A; Tacke, R | 1 |
Lambrecht, G; Moser, U; Mutschler, E; Noelke, B; Pfeiffer, A; Rochlitz, H; Tacke, R | 1 |
Jackson, KN; Kachur, JF; Lowe, VC; Noronha-Blob, L; Sturm, BL | 1 |
Anderson, D; el-Fakahany, EE; Forray, C; McKinney, M | 1 |
Amrhein, CL; el-Fakahany, EE; Forray, C; Surichamorn, W | 1 |
Boddeke, H; Christophe, J; Feifel, R; Lambrecht, G; Mutschler, E; Strohmann, C; Tacke, R; Waelbroeck, M; Wagner-Röder, M; Zilch, H | 1 |
Fuder, H; Lambrecht, G; Melchiorre, C; Mutschler, E; Schöpf, J; Tacke, R; Unckell, J; Wesner, MT | 1 |
Camus, J; Choo, LK; Feifel, R; Lambrecht, G; Moser, U; Strohmann, C; Tacke, R; Tastenoy, M; Waelbroeck, M; Wagner-Röder, M | 1 |
Barnes, PJ; Mak, JC | 1 |
Camus, J; Christophe, J; Lambrecht, G; Linoh, H; Mutschler, E; Strohmann, C; Tacke, R; Tastenoy, M; Waelbroeck, M; Zilch, H | 1 |
Camus, J; Christophe, J; Waelbroeck, M; Winand, J | 1 |
Jaiswal, N; Lambrecht, G; Malik, KU; Mutschler, E | 1 |
Giraldo, E; Hammer, R; Ladinsky, H; Viganò, MA | 1 |
Akiba, I; Bujo, H; Kubo, T; Maeda, A; Mishina, M; Nakai, J; Numa, S | 1 |
Nilvebrant, L; Sparf, B | 1 |
Bali, JP; Baudiere, B; Giraldo, E; Ladinsky, H; Monferini, E | 1 |
Fuder, H; Kilbinger, H; Müller, H | 1 |
Mitchelson, F; Shen, A | 1 |
Elzinga, CR; Meurs, H; Roffel, AF; Zaagsma, J | 1 |
Dietrich, C; Kilbinger, H | 1 |
Boselli, C; Grana, E | 1 |
Peers, C; Reeve, HL; Vaughan, PF | 1 |
Classen, M; Schaffer, K; Schepp, W; Schusdziarra, V; Wegner, U; Weigert, N | 1 |
Robinson, NE; Wang, ZW; Yu, MF | 1 |
Gillman, TA; Mitchelson, F; Pennefather, JN | 1 |
Deirmengiant, C; Maslanski, JA; Patelt, J; Powelt, R | 1 |
Davenport, TA; Fukumoto, Y; Gousse, A; Kamai, T; Latifpour, J; Weiss, RM; Yoshida, M | 1 |
Garland, CJ; Hillier, K; Kerr, PM; Wallis, RM | 1 |
de la Vega, MT; Montano, JA; Nunez, A | 1 |
Bilezikian, JP; Huber, F; Robinson, RB; Steinberg, SF; Sun, LS; Vulliemoz, Y | 1 |
Levin, RJ; Przyborski, SA | 1 |
Hoover, DB; Neely, DA | 1 |
Baba, H; Goldstein, PA; Kohno, T; Okamoto, M; Shimoji, K; Yoshimura, M | 1 |
Chasserot-Golaz, S; Galzi, JL; Goeldner, M; Ilien, B; Weill, C | 1 |
Lau, WA; Mitchelson, FJ; Pennefather, JN | 1 |
Ishida, H; Ishikawa, Y; Skowronski, MT | 1 |
Aita, T; Ishihata, A; Katano, Y; Tezuka, A | 1 |
2 review(s) available for hexahydrosiladifenidol and piperidines
Article | Year |
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Pharmacology and second messenger interactions of cloned muscarinic receptors.
Topics: Animals; Atropine; Carbachol; Cell Line; Humans; Oxotremorine; Piperidines; Pirenzepine; Receptors, Muscarinic; Recombinant Proteins; Second Messenger Systems; Transfection | 1991 |
Pharmacology of hexahydro-difenidol, hexahydro-sila-difenidol and related selective muscarinic antagonists.
Topics: Animals; Humans; Parasympatholytics; Piperidines | 1989 |
56 other study(ies) available for hexahydrosiladifenidol and piperidines
Article | Year |
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Characterization of the subtype of muscarinic receptor coupled to the stimulation of phosphoinositide hydrolysis in 132-1N1 human astrocytoma cells.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Astrocytoma; Atropine; Carbachol; Diamines; Humans; Hydrolysis; Parasympathomimetics; Phosphatidylinositols; Piperidines; Pirenzepine; Receptors, Muscarinic; Scopolamine; Tumor Cells, Cultured | 1992 |
Muscarinic receptor subtypes in bovine adrenal medulla.
Topics: Adrenal Medulla; Animals; Atropine; Binding Sites; Binding, Competitive; Cattle; Cell Membrane; Dicyclomine; Muscarine; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Muscarinic | 1992 |
The muscarinic receptor gene expressed in rabbit parietal cells is the m3 subtype.
Topics: Animals; Atropine; Base Sequence; Blotting, Southern; Molecular Sequence Data; N-Methylscopolamine; Parietal Cells, Gastric; Piperidines; Pirenzepine; Polymerase Chain Reaction; Rabbits; Receptors, Muscarinic; RNA, Messenger; Scopolamine Derivatives | 1992 |
A minority of muscarinic receptors mediate rabbit tracheal smooth muscle contraction.
Topics: Animals; Atropine; Female; Male; Methacholine Chloride; Muscle Contraction; Muscle, Smooth; Myocardium; Parasympatholytics; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Rabbits; Radioligand Assay; Receptors, Muscarinic; Trachea | 1992 |
M2 muscarinic receptors inhibit isoproterenol-induced relaxation of canine airway smooth muscle.
Topics: Animals; Dogs; Drug Interactions; Isoproterenol; Methacholine Chloride; Muscle Relaxation; Muscle, Smooth; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Trachea | 1992 |
Pharmacological profiles for rat cortical M1 and M2 muscarinic receptors using selective antagonists: comparison with N1E-115 muscarinic receptors.
Topics: Animals; Cerebral Cortex; Cyclic AMP; Diamines; In Vitro Techniques; Muscarinic Antagonists; Parasympatholytics; Phenethylamines; Phosphatidylinositols; Piperidines; Pirenzepine; Rats; Receptors, Muscarinic; Tumor Cells, Cultured | 1991 |
Muscarinic inhibition of excitatory neurotransmission in guinea-pig olfactory cortex slices: weak antagonism by M3-muscarinic receptor antagonists.
Topics: Action Potentials; Animals; Carbachol; Cerebral Cortex; Evoked Potentials; Guinea Pigs; In Vitro Techniques; Olfactory Bulb; Parasympatholytics; Piperidines; Receptors, Muscarinic; Synaptic Transmission | 1991 |
Characterization of a muscarinic receptor controlling Cl- secretion in hen trachea.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Animals; Atropine; Bethanechol; Bethanechol Compounds; Bumetanide; Calcium Channels; Chickens; Chlorides; Dicyclomine; Female; In Vitro Techniques; Ion Channels; Kinetics; Mucous Membrane; Muscle, Smooth; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Trachea | 1990 |
Pre- and postjunctional muscarinic receptors in canine bronchi.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Bethanechol Compounds; Bronchi; Carbachol; Dogs; Electric Stimulation; In Vitro Techniques; Membrane Potentials; Microelectrodes; Muscle Contraction; Muscle, Smooth; Oxotremorine; Piperidines; Pirenzepine; Receptors, Muscarinic | 1990 |
Pharmacological characterization of the vascular muscarinic receptors mediating relaxation and contraction in rabbit aorta.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Animals; Antihypertensive Agents; Aorta, Abdominal; Arecoline; Atropine; Diamines; Endothelium, Vascular; Hexamethonium; Hexamethonium Compounds; Indomethacin; Male; Muscarinic Antagonists; Muscle Contraction; Muscle Relaxation; Norepinephrine; Parasympatholytics; Piperidines; Pirenzepine; Rabbits; Receptors, Muscarinic | 1991 |
Modulation of the structure-binding relationships of antagonists for muscarinic acetylcholine receptor subtypes.
Topics: Animals; Centrifugation; Cerebral Cortex; Cholic Acids; Digitonin; Gallamine Triethiodide; Heart; In Vitro Techniques; Lacrimal Apparatus; Membranes; Muscarinic Antagonists; Myocardium; Parasympatholytics; Piperidines; Pirenzepine; Rats; Structure-Activity Relationship | 1991 |
Methoctramine, a cardioselective antagonist: muscarinic receptor mediating prostaglandin synthesis in isolated rabbit heart.
Topics: 6-Ketoprostaglandin F1 alpha; Acetylcholine; Animals; Arachidonic Acid; Arachidonic Acids; Arecoline; Coronary Circulation; Diamines; Heart; Heart Rate; In Vitro Techniques; Isoproterenol; Male; Myocardium; Parasympatholytics; Piperidines; Prostaglandins; Rabbits; Receptors, Muscarinic | 1991 |
Distribution and function of cholinergic receptors in the sheep detrusor muscle.
Topics: Acetylcholine; Acetylcholinesterase; Animals; Atropine; Carbachol; Cholinesterase Inhibitors; Ganglia, Parasympathetic; Male; Muscle Contraction; Muscle, Smooth; Nerve Tissue Proteins; Piperidines; Pirenzepine; Receptors, Muscarinic; Sheep; Tetraisopropylpyrophosphamide; Urinary Bladder | 1991 |
Characterization of muscarinic receptors in dog tracheal smooth muscle cells.
Topics: Animals; Atropine; Carbachol; Diamines; Dogs; In Vitro Techniques; Kinetics; Muscle, Smooth; N-Methylscopolamine; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Scopolamine Derivatives; Trachea | 1991 |
Telenzepine inhibits electrically-stimulated, acetylcholine plus histamine-mediated acid secretion in the mouse isolated stomach by blockade of M1 muscarine receptors.
Topics: Acetylcholine; Alkaloids; Animals; Anti-Ulcer Agents; Electric Stimulation; Furans; Gastric Acid; Gastric Mucosa; Histamine; Mice; Muscarinic Antagonists; Naphthalenes; p-Methoxy-N-methylphenethylamine; Parasympatholytics; Piperidines; Pirenzepine; Stomach; Thiazepines; Vagus Nerve | 1991 |
Selective labelling of muscarinic M1 receptors in calf superior cervical ganglia by [3H](+/-)-telenzepine.
Topics: Animals; Binding, Competitive; Cattle; Ganglia; Half-Life; In Vitro Techniques; Male; Neck; Piperidines; Pirenzepine; Rabbits; Radioligand Assay; Receptors, Muscarinic; Tritium; Vas Deferens | 1991 |
Natriuresis, kaliuresis and antidiuresis induced by central carbachol injection are mediated by muscarinic M1 receptors.
Topics: Animals; Carbachol; Diamines; Diuresis; Dose-Response Relationship, Drug; Injections, Intraventricular; Male; Muscarinic Antagonists; Natriuresis; Piperidines; Potassium; Rats; Rats, Inbred Strains; Receptors, Muscarinic | 1991 |
Binding affinities of hexahydro-difenidol and hexahydro-sila-difenidol analogues at four muscarinic receptor subtypes: constitutional and stereochemical aspects.
Topics: Animals; Binding, Competitive; Brain; Humans; In Vitro Techniques; Kinetics; Myocardium; Pancreas; Piperidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Stereoisomerism; Structure-Activity Relationship; Tumor Cells, Cultured | 1991 |
Muscarinic M3 receptors mediate contraction of human central and peripheral airway smooth muscle.
Topics: Bronchi; Humans; In Vitro Techniques; Ipratropium; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Trachea | 1990 |
Pharmacokinetic properties of the antimuscarinic drug [3H]-hexahydro-sila-difenidol in the rat.
Topics: Administration, Oral; Anesthesia; Animals; Autoradiography; Bile; Injections, Intravenous; Male; Parasympatholytics; Piperidines; Rats; Rats, Inbred Strains; Tissue Distribution | 1990 |
Human gastric mucosa expresses glandular M3 subtype of muscarinic receptors.
Topics: Carbachol; Gastric Mucosa; Humans; In Vitro Techniques; N-Methylscopolamine; Parasympatholytics; Piperazines; Piperidines; Pirenzepine; Receptors, Muscarinic; Scopolamine Derivatives | 1990 |
Muscarinic receptors mediating acid secretion in isolated rat gastric parietal cells are of M3 type.
Topics: Animals; Gastric Acid; Parasympatholytics; Parietal Cells, Gastric; Piperazines; Piperidines; Radioligand Assay; Rats; Receptors, Muscarinic | 1990 |
In vitro and in vivo antimuscarinic effects of (-)cis 2,3-dihydro-3-(4-methylpiperazinylmethyl)-2-phenyl-1,5 benzothiazepin-4-(5H)one HCl (BTM-1086) in guinea pig peripheral tissues.
Topics: Animals; Atropine; Calcium; Female; Guinea Pigs; Heart Atria; Ileum; In Vitro Techniques; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Neurons; Parasympatholytics; Piperidines; Pirenzepine; Structure-Activity Relationship; Thiazepines; Tumor Cells, Cultured; Urinary Bladder; Vas Deferens | 1990 |
Characterization of the striatal M2 muscarinic receptor mediating inhibition of cyclic AMP using selective antagonists: a comparison with the brainstem M2 receptor.
Topics: Animals; Brain Stem; Corpus Striatum; Cyclic AMP; Diamines; Parasympatholytics; Piperidines; Pirenzepine; Rats; Receptors, Muscarinic | 1989 |
Inhibition of cyclic AMP formation in N1E-115 neuroblastoma cells is mediated by a non-cardiac M2 muscarinic receptor subtype.
Topics: Animals; Binding, Competitive; Cyclic AMP; Mice; Muscarinic Antagonists; N-Methylscopolamine; Neuroblastoma; Piperidines; Receptors, Muscarinic; Scopolamine Derivatives; Tumor Cells, Cultured | 1989 |
Affinity profiles of hexahydro-sila-difenidol analogues at muscarinic receptor subtypes.
Topics: Animals; Diamines; Female; Ganglia, Sympathetic; Guinea Pigs; Heart; Ileum; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Piperidines; Pirenzepine; Rabbits; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Vas Deferens | 1989 |
Different muscarine receptors mediate the prejunctional inhibition of [3H]-noradrenaline release in rat or guinea-pig iris and the contraction of the rabbit iris sphincter muscle.
Topics: Animals; Electric Stimulation; In Vitro Techniques; Iris; Kinetics; Methacholine Compounds; Muscle Contraction; Muscle, Smooth; Norepinephrine; Piperidines; Rabbits; Rats; Rats, Inbred Strains; Receptors, Muscarinic | 1989 |
Muscarinic receptor subtypes in human and guinea pig lung.
Topics: Adamantane; Adult; Aged; Animals; Atropine; Guinea Pigs; Humans; In Vitro Techniques; Lung; Middle Aged; Parasympatholytics; Piperidines; Pirenzepine; Protease Inhibitors; Quinuclidinyl Benzilate; Receptors, Muscarinic; Species Specificity | 1989 |
Binding and functional properties of antimuscarinics of the hexocyclium/sila-hexocyclium and hexahydro-diphenidol/hexahydro-sila-diphenidol type to muscarinic receptor subtypes.
Topics: Animals; Cells, Cultured; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Male; Muscle, Smooth; Myocardium; Pancreas; Parasympatholytics; Piperazines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Stereoisomerism; Structure-Activity Relationship | 1989 |
Different antagonist binding properties of rat pancreatic and cardiac muscarinic receptors.
Topics: Animals; Binding, Competitive; GTP-Binding Proteins; Kinetics; Male; Myocardium; N-Methylscopolamine; Pancreas; Parasympatholytics; Piperidines; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives; Type C Phospholipases | 1987 |
Contribution of M2 alpha and M2 beta muscarinic receptors to the action of cholinergic stimuli on prostaglandin synthesis and mechanical function in the isolated rabbit heart.
Topics: Acetylcholine; Animals; Arecoline; Dose-Response Relationship, Drug; Heart; In Vitro Techniques; Male; Parasympatholytics; Parasympathomimetics; Piperidines; Pirenzepine; Prostaglandins; Rabbits; Receptors, Muscarinic | 1988 |
Characterization of muscarinic receptors in guinea pig ileum longitudinal smooth muscle.
Topics: Animals; Binding, Competitive; Guinea Pigs; Ileum; In Vitro Techniques; Kinetics; Male; Muscle, Smooth; Myocardium; N-Methylscopolamine; Parasympatholytics; Phenoxybenzamine; Piperidines; Pirenzepine; Receptors, Muscarinic; Salivary Glands; Scopolamine Derivatives | 1988 |
Primary structure of porcine muscarinic acetylcholine receptor III and antagonist binding studies.
Topics: Amino Acid Sequence; Animals; Base Sequence; DNA, Recombinant; Glycosylation; Molecular Sequence Data; Muscarine; Oocytes; Piperidines; Pirenzepine; Protein Conformation; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; RNA, Messenger; Sequence Homology, Nucleic Acid; Swine; Xenopus laevis | 1988 |
Receptor binding profiles of some selective muscarinic antagonists.
Topics: Animals; Cerebral Cortex; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle, Smooth; Myocardial Contraction; Parasympatholytics; Parotid Gland; Piperidines; Pirenzepine; Procyclidine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Urinary Bladder | 1988 |
Characterization of the muscarinic receptor subtype in isolated gastric fundic cells of the rabbit.
Topics: Aminopyrine; Animals; Atropine; Carbachol; Gastric Fundus; Kinetics; Male; N-Methylscopolamine; Piperidines; Pirenzepine; Rabbits; Receptors, Muscarinic; Scopolamine Derivatives | 1987 |
Organ selectivity of hexahydrosiladifenidol in blocking pre- and postjunctional muscarinic receptors studied in guinea-pig ileum and rat heart.
Topics: Acetylcholine; Animals; Guinea Pigs; Heart; Ileum; In Vitro Techniques; Male; Muscle Contraction; Norepinephrine; Organ Specificity; Parasympatholytics; Piperidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic | 1985 |
Characterization of the muscarine receptor subtype on sympathetic nerve endings in the rat caudal artery.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Arteries; Atropine; Bis-Trimethylammonium Compounds; Carbachol; Female; In Vitro Techniques; Isoindoles; Male; Muscarinic Antagonists; Muscle, Smooth, Vascular; Nerve Endings; Parasympatholytics; Piperidines; Rats; Rats, Wistar; Receptors, Muscarinic; Sympathetic Nervous System; Tail; Trihexyphenidyl | 1994 |
No evidence for a role of muscarinic M2 receptors in functional antagonism in bovine trachea.
Topics: Animals; Bronchoconstrictor Agents; Cattle; Dose-Response Relationship, Drug; Gallamine Triethiodide; Histamine; In Vitro Techniques; Isoproterenol; Methacholine Chloride; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nicotinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Adrenergic, beta; Receptors, Muscarinic; Trachea | 1995 |
Prejunctional M1 and postjunctional M3 muscarinic receptors in the circular muscle of the guinea-pig ileum.
Topics: Acetylcholine; Animals; Choline; Female; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Neuromuscular Junction; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic | 1995 |
Mode of antagonism of methoctramine, AF-DX 116 and hexahydrosiladifenidol in guinea-pig left atrium and ileum: comparison of Schild and resultant analysis.
Topics: Animals; Diamines; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Myocardial Contraction; Parasympatholytics; Piperidines; Pirenzepine | 1995 |
Inhibition of N-type Ca2+ channel currents in human neuroblastoma (SH-SY5Y) cells by muscarine via stimulation of M3 receptors.
Topics: Brain Neoplasms; Calcium Channel Blockers; GTP-Binding Proteins; Humans; Muscarine; Muscarinic Agonists; Neuroblastoma; Parasympatholytics; Patch-Clamp Techniques; Pertussis Toxin; Piperidines; Receptors, Muscarinic; Tumor Cells, Cultured; Virulence Factors, Bordetella | 1995 |
Functional characterization of a muscarinic receptor stimulating gastrin release from rabbit antral G-cells in primary culture.
Topics: Animals; Arecoline; Atropine; Benzodiazepinones; Carbachol; Cell Adhesion; Cell Separation; Cells, Cultured; Gastrins; Immunohistochemistry; Male; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Pyloric Antrum; Rabbits; Receptors, Muscarinic | 1994 |
Prejunctional muscarinic autoreceptors on horse airway cholinergic nerves.
Topics: Acetylcholine; Animals; Atropine; Cholinergic Fibers; Electric Stimulation; Horses; In Vitro Techniques; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Trachea | 1995 |
Muscarinic receptors in rat uterus.
Topics: Alkaloids; Animals; Atropine; Binding, Competitive; Computer Simulation; Female; Furans; In Vitro Techniques; Ligands; Muscarinic Antagonists; Naphthalenes; Parasympatholytics; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Uterus | 1994 |
Assessment of the muscarinic receptor subtypes involved in pilocarpine-induced seizures in mice.
Topics: Animals; Atropine; Cerebral Ventricles; Injections, Intraventricular; Male; Mice; Parasympatholytics; Pilocarpine; Piperidines; Pirenzepine; Receptors, Muscarinic; Seizures | 1994 |
Diabetes-induced alterations in the properties of muscarinic cholinergic receptors in rat vas deferens.
Topics: Animals; Atropine; Binding, Competitive; Diabetes Mellitus, Experimental; Diamines; Insulin; Male; Parasympatholytics; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Up-Regulation; Vas Deferens | 1994 |
Characterization of muscarinic receptors mediating contractions of circular and longitudinal muscle of human isolated colon.
Topics: Alkaloids; Atropine; Carbachol; Carcinoma; Colon; Colonic Neoplasms; Dose-Response Relationship, Drug; Furans; Humans; In Vitro Techniques; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Naphthalenes; Piperidines; Pirenzepine | 1995 |
Carbachol stimulates inositol phosphate formation in rat thalamus slices through muscarinic M3-receptor activation.
Topics: Animals; Binding, Competitive; Carbachol; Dose-Response Relationship, Drug; Inositol Phosphates; Male; Muscarinic Agonists; Muscarinic Antagonists; Organ Culture Techniques; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic; Thalamus; Tritium | 1996 |
Muscarinic receptor heterogeneity in neonatal rat ventricular myocytes in culture.
Topics: Animals; Animals, Newborn; Carbachol; Cells, Cultured; Cyclic AMP; GTP-Binding Proteins; Heart Rate; Inositol Phosphates; Muscarinic Agonists; Muscarinic Antagonists; Myocardium; Pertussis Toxin; Piperidines; Rats; Receptor, Muscarinic M2; Receptors, Muscarinic; Signal Transduction; Stimulation, Chemical; Virulence Factors, Bordetella | 1996 |
Cholinergic modulation of electrogenic ion transport in different regions of the rat small intestine.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Analysis of Variance; Animals; Atropine; Bethanechol; Carbachol; Chlorides; Diamines; Duodenum; Ileum; Intestinal Mucosa; Ion Transport; Jejunum; Male; Muscarinic Agonists; Muscarinic Antagonists; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptor, Muscarinic M3; Receptors, Muscarinic; Structure-Activity Relationship; Tetrodotoxin | 1997 |
Differentiation of muscarinic receptors mediating negative chronotropic and vasoconstrictor responses to acetylcholine in isolated rat hearts.
Topics: Acetylcholine; Animals; Atropine; Coronary Vessels; Depression, Chemical; Diamines; Heart Rate; In Vitro Techniques; Male; Pertussis Toxin; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Vasoconstriction; Virulence Factors, Bordetella | 1997 |
Muscarinic facilitation of GABA release in substantia gelatinosa of the rat spinal dorsal horn.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Atropine; Carbachol; Diamines; Evoked Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Interneurons; Muscarinic Agonists; Neostigmine; Neurons; Parasympatholytics; Piperidines; Pirenzepine; Rats; Receptor, Muscarinic M1; Receptors, Muscarinic; Substantia Gelatinosa; Synaptic Transmission; Tetrodotoxin | 1998 |
Functional characterization and potential applications for enhanced green fluorescent protein- and epitope-fused human M1 muscarinic receptors.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Atropine; Binding, Competitive; Calcium; Cells, Cultured; DNA Primers; Epitopes; Flow Cytometry; Gene Expression; Green Fluorescent Proteins; Histidine; Humans; Indicators and Reagents; Kidney; Luminescent Proteins; Microscopy, Confocal; Muscarinic Antagonists; Mutagenesis, Site-Directed; Piperidines; Pirenzepine; Radioligand Assay; Receptor, Muscarinic M1; Receptors, Muscarinic; Recombinant Fusion Proteins; Tritium | 1999 |
Cholinergic facilitation of neurotransmission to the smooth muscle of the guinea-pig prostate gland.
Topics: Acetylcholine; Animals; Carbachol; Cholinergic Agonists; Electric Stimulation; Guinea Pigs; Male; Muscle Contraction; Muscle, Smooth; Piperidines; Prostate; Receptor, Muscarinic M1; Receptors, Muscarinic; Synaptic Transmission | 2000 |
Persistent increase in the amount of aquaporin-5 in the apical plasma membrane of rat parotid acinar cells induced by a muscarinic agonist SNI-2011.
Topics: Animals; Aquaporin 5; Aquaporins; Atropine; Calcium; Cell Membrane; Cells, Cultured; Inositol 1,4,5-Trisphosphate; Male; Membrane Proteins; Muscarinic Agonists; Parotid Gland; Piperidines; Quinuclidines; Rats; Rats, Wistar; Thiophenes | 2000 |
Aging-related alterations in the contractile responses to acetylcholine, muscarinic cholinoceptors and cholinesterase activities in jejunum and colon of the male Fischer 344 rats.
Topics: Acetylcholine; Aging; Animals; Atropine; Cholinesterases; Colon; Diamines; Dose-Response Relationship, Drug; Gastrointestinal Motility; In Vitro Techniques; Intestine, Large; Jejunum; Male; Muscarinic Antagonists; Muscle, Smooth; Piperidines; Pirenzepine; Rats; Rats, Inbred F344 | 2004 |