hexahydrosiladifenidol and methoctramine

hexahydrosiladifenidol has been researched along with methoctramine in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19903 (17.65)18.7374
1990's13 (76.47)18.2507
2000's1 (5.88)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bonner, TI; Brann, MR; Buckley, CM; Buckley, NJ1
Ehlert, FJ; Esqueda, EE; Gerstin, EH; Griffin, MT1
Kovacs, I; Roeske, WR; Varga, EV; Waite, SL; Yamamura, HI1
Sastry, BV; Stephan, CC1
Anderson, DJ; Connolly, T; McKinney, M; Miller, JH; Vella-Rountree, L1
Jaiswal, N; Lambrecht, G; Malik, KU; Mutschler, E; Tacke, R1
Jaiswal, N; Malik, KU1
Yang, CM1
Massi, M; Melchiorre, C; Perfumi, M; Polidori, C; Pompei, PL1
Anderson, D; el-Fakahany, EE; Forray, C; McKinney, M1
Boddeke, H; Christophe, J; Feifel, R; Lambrecht, G; Mutschler, E; Strohmann, C; Tacke, R; Waelbroeck, M; Wagner-Röder, M; Zilch, H1
Boselli, C; Grana, E1
Davenport, TA; Fukumoto, Y; Gousse, A; Kamai, T; Latifpour, J; Weiss, RM; Yoshida, M1
Levin, RJ; Przyborski, SA1
Hoover, DB; Neely, DA1
Baba, H; Goldstein, PA; Kohno, T; Okamoto, M; Shimoji, K; Yoshimura, M1
Aita, T; Ishihata, A; Katano, Y; Tezuka, A1

Other Studies

17 other study(ies) available for hexahydrosiladifenidol and methoctramine

ArticleYear
Antagonist binding properties of five cloned muscarinic receptors expressed in CHO-K1 cells.
    Molecular pharmacology, 1989, Volume: 35, Issue:4

    Topics: Animals; Cell Line; Cloning, Molecular; Cricetinae; Humans; Kinetics; N-Methylscopolamine; Parasympatholytics; Rats; Receptors, Muscarinic; Scopolamine Derivatives

1989
Stimulation of cyclic AMP accumulation and phosphoinositide hydrolysis by M3 muscarinic receptors in the rat peripheral lung.
    Biochemical pharmacology, 1996, Aug-23, Volume: 52, Issue:4

    Topics: Animals; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Hydrolysis; Lung; Male; Oxotremorine; Phosphatidylinositols; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic

1996
Pharmacological comparison of the cloned human and rat M2 muscarinic receptor genes expressed in the murine fibroblast (B82) cell line.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 284, Issue:2

    Topics: Amino Acid Sequence; Animals; Carbachol; Cloning, Molecular; Cyclic AMP; Humans; Mice; Molecular Sequence Data; Muscarinic Agonists; Muscarinic Antagonists; Phosphatidylinositols; Radioligand Assay; Rats; Receptors, Muscarinic; Sequence Alignment; Sequence Homology, Amino Acid; Signal Transduction; Species Specificity

1998
Characterization of the subtype of muscarinic receptor coupled to the stimulation of phosphoinositide hydrolysis in 132-1N1 human astrocytoma cells.
    Cellular and molecular biology (Noisy-le-Grand, France), 1992, Volume: 38, Issue:7

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Astrocytoma; Atropine; Carbachol; Diamines; Humans; Hydrolysis; Parasympathomimetics; Phosphatidylinositols; Piperidines; Pirenzepine; Receptors, Muscarinic; Scopolamine; Tumor Cells, Cultured

1992
Pharmacological profiles for rat cortical M1 and M2 muscarinic receptors using selective antagonists: comparison with N1E-115 muscarinic receptors.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 257, Issue:3

    Topics: Animals; Cerebral Cortex; Cyclic AMP; Diamines; In Vitro Techniques; Muscarinic Antagonists; Parasympatholytics; Phenethylamines; Phosphatidylinositols; Piperidines; Pirenzepine; Rats; Receptors, Muscarinic; Tumor Cells, Cultured

1991
Pharmacological characterization of the vascular muscarinic receptors mediating relaxation and contraction in rabbit aorta.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 258, Issue:3

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Animals; Antihypertensive Agents; Aorta, Abdominal; Arecoline; Atropine; Diamines; Endothelium, Vascular; Hexamethonium; Hexamethonium Compounds; Indomethacin; Male; Muscarinic Antagonists; Muscle Contraction; Muscle Relaxation; Norepinephrine; Parasympatholytics; Piperidines; Pirenzepine; Rabbits; Receptors, Muscarinic

1991
Methoctramine, a cardioselective antagonist: muscarinic receptor mediating prostaglandin synthesis in isolated rabbit heart.
    European journal of pharmacology, 1991, Jan-03, Volume: 192, Issue:1

    Topics: 6-Ketoprostaglandin F1 alpha; Acetylcholine; Animals; Arachidonic Acid; Arachidonic Acids; Arecoline; Coronary Circulation; Diamines; Heart; Heart Rate; In Vitro Techniques; Isoproterenol; Male; Myocardium; Parasympatholytics; Piperidines; Prostaglandins; Rabbits; Receptors, Muscarinic

1991
Characterization of muscarinic receptors in dog tracheal smooth muscle cells.
    Journal of autonomic pharmacology, 1991, Volume: 11, Issue:1

    Topics: Animals; Atropine; Carbachol; Diamines; Dogs; In Vitro Techniques; Kinetics; Muscle, Smooth; N-Methylscopolamine; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Scopolamine Derivatives; Trachea

1991
Natriuresis, kaliuresis and antidiuresis induced by central carbachol injection are mediated by muscarinic M1 receptors.
    European journal of pharmacology, 1991, Mar-19, Volume: 195, Issue:1

    Topics: Animals; Carbachol; Diamines; Diuresis; Dose-Response Relationship, Drug; Injections, Intraventricular; Male; Muscarinic Antagonists; Natriuresis; Piperidines; Potassium; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1991
Characterization of the striatal M2 muscarinic receptor mediating inhibition of cyclic AMP using selective antagonists: a comparison with the brainstem M2 receptor.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:2

    Topics: Animals; Brain Stem; Corpus Striatum; Cyclic AMP; Diamines; Parasympatholytics; Piperidines; Pirenzepine; Rats; Receptors, Muscarinic

1989
Affinity profiles of hexahydro-sila-difenidol analogues at muscarinic receptor subtypes.
    European journal of pharmacology, 1989, Sep-01, Volume: 168, Issue:1

    Topics: Animals; Diamines; Female; Ganglia, Sympathetic; Guinea Pigs; Heart; Ileum; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Piperidines; Pirenzepine; Rabbits; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Vas Deferens

1989
Mode of antagonism of methoctramine, AF-DX 116 and hexahydrosiladifenidol in guinea-pig left atrium and ileum: comparison of Schild and resultant analysis.
    Journal of autonomic pharmacology, 1995, Volume: 15, Issue:2

    Topics: Animals; Diamines; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Myocardial Contraction; Parasympatholytics; Piperidines; Pirenzepine

1995
Diabetes-induced alterations in the properties of muscarinic cholinergic receptors in rat vas deferens.
    The Journal of urology, 1994, Volume: 152, Issue:3

    Topics: Animals; Atropine; Binding, Competitive; Diabetes Mellitus, Experimental; Diamines; Insulin; Male; Parasympatholytics; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Up-Regulation; Vas Deferens

1994
Cholinergic modulation of electrogenic ion transport in different regions of the rat small intestine.
    The Journal of pharmacy and pharmacology, 1997, Volume: 49, Issue:7

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Analysis of Variance; Animals; Atropine; Bethanechol; Carbachol; Chlorides; Diamines; Duodenum; Ileum; Intestinal Mucosa; Ion Transport; Jejunum; Male; Muscarinic Agonists; Muscarinic Antagonists; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptor, Muscarinic M3; Receptors, Muscarinic; Structure-Activity Relationship; Tetrodotoxin

1997
Differentiation of muscarinic receptors mediating negative chronotropic and vasoconstrictor responses to acetylcholine in isolated rat hearts.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 282, Issue:3

    Topics: Acetylcholine; Animals; Atropine; Coronary Vessels; Depression, Chemical; Diamines; Heart Rate; In Vitro Techniques; Male; Pertussis Toxin; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Vasoconstriction; Virulence Factors, Bordetella

1997
Muscarinic facilitation of GABA release in substantia gelatinosa of the rat spinal dorsal horn.
    The Journal of physiology, 1998, Apr-01, Volume: 508 ( Pt 1)

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Atropine; Carbachol; Diamines; Evoked Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Interneurons; Muscarinic Agonists; Neostigmine; Neurons; Parasympatholytics; Piperidines; Pirenzepine; Rats; Receptor, Muscarinic M1; Receptors, Muscarinic; Substantia Gelatinosa; Synaptic Transmission; Tetrodotoxin

1998
Aging-related alterations in the contractile responses to acetylcholine, muscarinic cholinoceptors and cholinesterase activities in jejunum and colon of the male Fischer 344 rats.
    Experimental gerontology, 2004, Volume: 39, Issue:1

    Topics: Acetylcholine; Aging; Animals; Atropine; Cholinesterases; Colon; Diamines; Dose-Response Relationship, Drug; Gastrointestinal Motility; In Vitro Techniques; Intestine, Large; Jejunum; Male; Muscarinic Antagonists; Muscle, Smooth; Piperidines; Pirenzepine; Rats; Rats, Inbred F344

2004