hemicholinium 3 and ethylcholine aziridinium

hemicholinium 3 has been researched along with ethylcholine aziridinium in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19908 (53.33)18.7374
1990's4 (26.67)18.2507
2000's3 (20.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hanin, I; Kindel, G; Potter, PE; Tedford, CE1
Morio, Y; Yagasaki, O1
Chrobak, JJ; Spates, MJ; Stackman, RW; Walsh, TJ1
Dawson, TM; Dawson, VL; Filloux, FM; Wamsley, JK1
Fisher, A; Hanin, I1
Kelley, MC; Meyer, EM; Raizada, MK1
Cuello, AC; Maysinger, D; Tagari, PC1
Hanin, I; Leventer, SM; Roeske, WR; Vickroy, TW; Watson, M; Yamamura, HI1
Brake, WG; Pappas, BA1
Connell, TA; Weiss, B; Zhang, SP; Zhou, LW1
Estrada, C; Galea, E; Gómez, C; Martín, C1
Erickson, LC; Hanin, I; Santiago, LR1
Chen, SR; Pan, HL1
Bessho, T; Eguchi, J; Kawai, K; Mori, R; Saito, K; Takashina, K1
Inoue, H; Kuwagata, Y1

Reviews

1 review(s) available for hemicholinium 3 and ethylcholine aziridinium

ArticleYear
Potential animal models for senile dementia of Alzheimer's type, with emphasis on AF64A-induced cholinotoxicity.
    Annual review of pharmacology and toxicology, 1986, Volume: 26

    Topics: Aged; Aging; Aluminum; Alzheimer Disease; Animals; Aziridines; Choline; Disease Models, Animal; Haplorhini; Hemicholinium 3; Humans; Neuromuscular Blocking Agents; Neurotoxins; Parasympathetic Nervous System; Scopolamine

1986

Other Studies

14 other study(ies) available for hemicholinium 3 and ethylcholine aziridinium

ArticleYear
Inhibition of high affinity choline transport attenuates both cholinergic and non-cholinergic effects of ethylcholine aziridinium (AF64A).
    Brain research, 1989, May-22, Volume: 487, Issue:2

    Topics: Animals; Aziridines; Azirines; Biogenic Amines; Choline; Cholinergic Fibers; Hemicholinium 3; Hippocampus; Male; Neurotransmitter Uptake Inhibitors; Rats; Rats, Inbred Strains

1989
Effects of AF64A on cholinergic neurotransmission in the sixth abdominal ganglion of the cockroach.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1989, Volume: 94, Issue:1

    Topics: Abdomen; Acetylcholine; Action Potentials; Animals; Aziridines; Choline; Cockroaches; Electric Stimulation; Ganglia, Parasympathetic; Hemicholinium 3; Male; Microscopy, Electron; Synaptic Transmission

1989
Hemicholinium-3 prevents the working memory impairments and the cholinergic hypofunction induced by ethylcholine aziridinium ion (AF64A).
    Brain research, 1989, Dec-18, Volume: 504, Issue:2

    Topics: Animals; Aziridines; Choline; Cholinergic Fibers; Hemicholinium 3; Hippocampus; Injections, Intraventricular; Male; Memory Disorders; Rats; Rats, Inbred Strains

1989
Evidence for dopamine D-2 receptors on cholinergic interneurons in the rat caudate-putamen.
    Life sciences, 1988, Volume: 42, Issue:20

    Topics: Animals; Aziridines; Caudate Nucleus; Choline; Hemicholinium 3; Interneurons; Male; Putamen; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride

1988
Pharmacological characterization of high affinity choline transporters in primary neuronal cultures in rat brain.
    Neuropharmacology, 1988, Volume: 27, Issue:8

    Topics: Acetylcholine; Animals; Aziridines; Biological Transport, Active; Brain; Cells, Cultured; Choline; Choline O-Acetyltransferase; Hemicholinium 3; Male; Nerve Tissue Proteins; Neuromuscular Blocking Agents; Neurons; Rats; Rats, Inbred Strains; Synaptosomes

1988
Hemicholinium mustard derivatives: preliminary assessment of cholinergic neurotoxicity.
    Neurochemical research, 1986, Volume: 11, Issue:7

    Topics: Animals; Aziridines; Brain; Cerebral Cortex; Choline; Cholinergic Fibers; Corpus Striatum; Hemicholinium 3; Hippocampus; Injections, Intraventricular; Male; Mechlorethamine; Rats

1986
Regional differences in ethylcholine mustard aziridinium ion (AF64A)-induced deficits in presynaptic cholinergic markers for the rat central nervous system.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:3

    Topics: Animals; Aziridines; Azirines; Brain; Choline; Choline O-Acetyltransferase; Hemicholinium 3; Male; Neuromuscular Blocking Agents; Parasympathetic Nervous System; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Tritium

1985
Hemicholinium-3 (HC3) blocks the effects of ethylcholine mustard aziridinium (AF64A) in the developing rat.
    Brain research. Developmental brain research, 1994, Dec-16, Volume: 83, Issue:2

    Topics: Acetylcholine; Animals; Animals, Newborn; Aziridines; Behavior, Animal; Brain; Choline; Choline O-Acetyltransferase; Hemicholinium 3; Male; Rats

1994
Cholinergic lesions of mouse striatum induced by AF64A alter D2 dopaminergic behavior and reduce D2 dopamine receptors and D2 dopamine receptor mRNA.
    Neurochemistry international, 1993, Volume: 22, Issue:3

    Topics: Animals; Apomorphine; Aziridines; Behavior, Animal; Choline; Corpus Striatum; Dopamine; Glutamate Decarboxylase; Hemicholinium 3; Male; Mice; Mice, Inbred Strains; Parasympathetic Nervous System; Receptors, Dopamine D2; RNA, Messenger; Stereotyped Behavior; Toxins, Biological

1993
Direct cytotoxicity of ethylcholine mustard aziridinium in cerebral microvascular endothelial cells.
    Journal of neurochemistry, 1993, Volume: 60, Issue:4

    Topics: Animals; Aziridines; Biological Transport; Brain; Cattle; Cell Death; Cells, Cultured; Choline; Choline O-Acetyltransferase; Endothelium, Vascular; Hemicholinium 3; Humans; L-Lactate Dehydrogenase; Microcirculation; Neuroblastoma; Toxins, Biological; Tumor Cells, Cultured

1993
AF64A-induced changes in N-myc expression in the LA-N-2 human neuroblastoma cell line are modulated by choline and hemicholinium-3.
    Neurochemical research, 1998, Volume: 23, Issue:5

    Topics: Aziridines; Cell Division; Cell Survival; Choline; Gene Expression Regulation, Neoplastic; Hemicholinium 3; Humans; Kinetics; Neuroblastoma; Neuromuscular Blocking Agents; Proto-Oncogene Proteins c-myc; Tumor Cells, Cultured

1998
Spinal endogenous acetylcholine contributes to the analgesic effect of systemic morphine in rats.
    Anesthesiology, 2001, Volume: 95, Issue:2

    Topics: Acetylcholine; Analgesics, Opioid; Animals; Atropine; Aziridines; Carrier Proteins; Choline; Cholinergic Agents; Hemicholinium 3; Injections, Spinal; Male; Mecamylamine; Membrane Transport Proteins; Morphine; Muscarinic Antagonists; Nicotinic Antagonists; Pain Measurement; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Receptors, Nicotinic; Spinal Cord

2001
MKC-231, a choline uptake enhancer: (3) Mode of action of MKC-231 in the enhancement of high-affinity choline uptake.
    Journal of neural transmission (Vienna, Austria : 1996), 2008, Volume: 115, Issue:7

    Topics: Animals; Aziridines; Cell Membrane; Chlorocebus aethiops; Choline; COS Cells; Drug Interactions; Hemicholinium 3; Hippocampus; Male; Membrane Transport Proteins; Neurotransmitter Uptake Inhibitors; Protein Binding; Quinolines; Radioligand Assay; Rats; Rats, Wistar; Synaptosomes; Transfection; Tritium

2008
Effects of estrogen on AF64A-induced apoptosis in NG108-15 cells.
    Brain research, 2009, Nov-10, Volume: 1297

    Topics: Acetylcholine; Animals; Apoptosis; Aziridines; Cell Line, Tumor; Choline; Cholinergic Agents; Estradiol; Hemicholinium 3; Hybridomas; MAP Kinase Kinase 1; Mice; Neuromuscular Blocking Agents; Neurons; Neuroprotective Agents; Neurotoxins; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Rats; Receptors, Estrogen; Signal Transduction

2009