haloperidol has been researched along with sb 277011 in 14 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 8 (57.14) | 29.6817 |
| 2010's | 4 (28.57) | 24.3611 |
| 2020's | 2 (14.29) | 2.80 |
| Authors | Studies |
|---|---|
| Jadhav, A; Kerns, E; Nguyen, K; Shah, P; Sun, H; Xu, X; Yan, Z; Yu, KR | 1 |
| Kabir, M; Kerns, E; Nguyen, K; Shah, P; Sun, H; Wang, Y; Xu, X; Yu, KR | 1 |
| Kabir, M; Kerns, E; Neyra, J; Nguyen, K; Nguyễn, ÐT; Shah, P; Siramshetty, VB; Southall, N; Williams, J; Xu, X; Yu, KR | 1 |
| Itkin, M; Kabir, M; Mathé, EA; Nguyễn, ÐT; Padilha, EC; Shah, P; Shinn, P; Siramshetty, V; Wang, AQ; Williams, J; Xu, X; Yu, KR; Zhao, T | 1 |
| Ashby, CR; Hagan, JJ; Middlemiss, DN; Minabe, Y; Stemp, G | 1 |
| Ashby, CR; Gardner, EL; Hagan, JJ; Hayes, R; Liu, X; Middlemiss, DN; Paul, M; Stemp, G; Vorel, SR | 1 |
| Gál, K; Gyertyán, I | 2 |
| Cummins, R; Gnoffo, Z; Kew, JN; Roberts, C | 1 |
| Bespalov, A; Gross, G; Harich, S; Jongen-Rêlo, AL; Schoemaker, H; van Gaalen, M | 1 |
| Gyertyán, I; Sághy, K | 1 |
| Agai-Csongor, E; Bugovics, G; Domány, G; Fazekas, K; Gyertyán, I; Horváth, A; Kiss, B; Laszlovszky, I; Némethy, Z; Schmidt, E; Szombathelyi, Z | 1 |
| Davoodi, N; Langlois, X; te Riele, P | 1 |
| Ananthan, S; Głowacka, U; Kosmowska, B; Ossowska, K; Wardas, J | 1 |
1 review(s) available for haloperidol and sb 277011
| Article | Year |
|---|---|
Using in vitro ADME data for lead compound selection: An emphasis on PAMPA pH 5 permeability and oral bioavailability.
Topics: Administration, Oral; Animals; Betamethasone; Biological Availability; Caco-2 Cells; Cell Membrane Permeability; Cells, Cultured; Dexamethasone; Dogs; Dose-Response Relationship, Drug; Humans; Hydrogen-Ion Concentration; Madin Darby Canine Kidney Cells; Mice; Molecular Structure; Neural Networks, Computer; Ranitidine; Rats; Structure-Activity Relationship; Verapamil | 2022 |
13 other study(ies) available for haloperidol and sb 277011
| Article | Year |
|---|---|
Highly predictive and interpretable models for PAMPA permeability.
Topics: Artificial Intelligence; Caco-2 Cells; Cell Membrane Permeability; Humans; Models, Biological; Organic Chemicals; Regression Analysis; Support Vector Machine | 2017 |
Predictive models of aqueous solubility of organic compounds built on A large dataset of high integrity.
Topics: Drug Discovery; Organic Chemicals; Pharmaceutical Preparations; Solubility | 2019 |
Retrospective assessment of rat liver microsomal stability at NCATS: data and QSAR models.
Topics: Animals; Computer Simulation; Databases, Factual; Drug Discovery; High-Throughput Screening Assays; Liver; Machine Learning; Male; Microsomes, Liver; National Center for Advancing Translational Sciences (U.S.); Pharmaceutical Preparations; Quantitative Structure-Activity Relationship; Rats; Rats, Sprague-Dawley; Retrospective Studies; United States | 2020 |
Acute and chronic administration of the selective D(3) receptor antagonist SB-277011-A alters activity of midbrain dopamine neurons in rats: an in vivo electrophysiological study.
Topics: Action Potentials; Administration, Oral; Animals; Cell Count; Dogs; Dopamine Antagonists; Dose-Response Relationship, Drug; Haloperidol; Injections, Intravenous; Male; Mesencephalon; Neurons; Nitriles; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Substantia Nigra; Tegmentum Mesencephali; Tetrahydroisoquinolines | 2000 |
Dopamine D3 receptor antagonism inhibits cocaine-seeking and cocaine-enhanced brain reward in rats.
Topics: Animals; Behavior, Animal; Brain; Catalepsy; Cocaine; Cocaine-Related Disorders; Conditioning, Operant; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Electric Stimulation; Electrodes, Implanted; Haloperidol; Male; Nitriles; Quinolines; Rats; Rats, Long-Evans; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Reinforcement, Psychology; Reward; Secondary Prevention; Self Administration; Spatial Behavior; Tetrahydroisoquinolines | 2002 |
Dopamine D3 receptor ligands show place conditioning effect but do not influence cocaine-induced place preference.
Topics: Animals; Avoidance Learning; Benzazepines; Benzopyrans; Cocaine; Conditioning, Classical; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Haloperidol; Indans; Male; Naphthalenes; Nitriles; Oxazines; Piperazines; Pyrrolidines; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Reinforcement, Psychology; Reward; Spatial Behavior; Substance-Related Disorders; Tetrahydroisoquinolines; Tetrahydronaphthalenes | 2003 |
Dopamine D3 as well as D2 receptor ligands attenuate the cue-induced cocaine-seeking in a relapse model in rats.
Topics: Animals; Brain; Cocaine-Related Disorders; Cues; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Extinction, Psychological; Haloperidol; Male; Nitriles; Piperazines; Rats; Rats, Long-Evans; Receptors, Dopamine D2; Receptors, Dopamine D3; Reinforcement, Psychology; Self Administration; Social Facilitation; Sucrose; Tetrahydroisoquinolines | 2006 |
Dopamine D3 receptor modulation of dopamine efflux in the rat nucleus accumbens.
Topics: Animals; Antipsychotic Agents; Clozapine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Electric Stimulation; Haloperidol; Male; Nitriles; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulpiride; Tetrahydroisoquinolines; Tetrahydronaphthalenes | 2006 |
Habituation deficits induced by metabotropic glutamate receptors 2/3 receptor blockade in mice: reversal by antipsychotic drugs.
Topics: Amino Acids; Animals; Antipsychotic Agents; Cognition Disorders; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Habituation, Psychophysiologic; Haloperidol; Male; Methamphetamine; Mice; Motor Activity; Nitriles; Receptors, Metabotropic Glutamate; Tetrahydroisoquinolines; Xanthenes | 2007 |
The selective dopamine D3 receptor antagonists, SB 277011-A and S 33084 block haloperidol-induced catalepsy in rats.
Topics: Animals; Benzopyrans; Catalepsy; Haloperidol; Male; Nitriles; Pyrroles; Rats; Rats, Wistar; Receptors, Dopamine D3; Tetrahydroisoquinolines | 2007 |
Subnanomolar dopamine D3 receptor antagonism coupled to moderate D2 affinity results in favourable antipsychotic-like activity in rodent models: I. neurochemical characterisation of RG-15.
Topics: Amisulpride; Animals; CHO Cells; Cricetinae; Cricetulus; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Haloperidol; Humans; Inhibitory Concentration 50; Male; Mice; Nitriles; Prolactin; Pyridines; Rats; Rats, Wistar; Receptors, Dopamine D3; Sulfonamides; Sulpiride; Tetrahydroisoquinolines | 2008 |
Examining dopamine D3 receptor occupancy by antipsychotic drugs via [3H]7-OH-DPAT ex vivo autoradiography and its cross-validation via c-fos immunohistochemistry in the rat brain.
Topics: Animals; Antipsychotic Agents; Autoradiography; Benzodiazepines; Clozapine; Dopamine Antagonists; Haloperidol; Indoles; Islands of Calleja; Male; Nitriles; Olanzapine; Piperidines; Proto-Oncogene Proteins c-fos; Radiography; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydroisoquinolines; Tetrahydronaphthalenes | 2014 |
Pramipexole at a Low Dose Induces Beneficial Effect in the Harmaline-induced Model of Essential Tremor in Rats.
Topics: Amisulpride; Animals; Anti-Dyskinesia Agents; Benzothiazoles; Disease Models, Animal; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Essential Tremor; Haloperidol; Harmaline; Imidazoles; Male; Movement; Nitriles; Pramipexole; Pyridines; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulpiride; Tetrahydroisoquinolines; Tetrahydronaphthalenes; Treatment Outcome | 2016 |